Discovery of 3-Alkoxyamino-5-(pyridin-2-ylamino)pyrazine-2-carbonitriles as Selective, Orally Bioavailable CHK1 Inhibitors
(Journal of Medicinal Chemistry)
Friday October 19th 2012
Author(s): Michael Lainchbury, Thomas P. Matthews, Tatiana McHardy, Kathy J. Boxall, Michael I. Walton, Paul D. Eve, Angela Hayes, Melanie R. Valenti, Alexis K. de Haven Brandon, Gary Box, G. Wynne Aherne, John C. Reader, Florence I. Raynaud, Suzanne A. Eccles, Michelle D. Garrett, Ian Collins,
DOI:10.1021/jm3012933
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