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1) Enantiomeric Diketopiperazines: Getting Insight of the Impact of the Configuration to the Conformation, Nanoimage, u-PA Inhibition and Anti-metastatic Activity (ChemMedComm) Tuesday March 31st 2015
Feng Wang, Shan Li, Yuji Wang, Haimei Zhu, Xiaoyi Zhang, Ming Zhao, Jianhui Wu, Shiqi Peng

2) Chemical genomics reveals novel biological activity of 1,2,3-dithiazoles as potent and reversible melanin synthesis inhibitors (ChemMedComm) Tuesday March 31st 2015
Panayiotis Andreas Koutentis, Paris Skourides, Oleg Alekseevich Rakitin, Anna Charalambous, Maria Koyioni, Ioanna Antoniades, Sophia Michaelidou, Iro Eleftheriou, Stanislav A Amelichev, Lidia S konstantinova, Despoina Pegeioti

3) Correction: Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday March 31st 2015
Taha M. A. Eldebss, Sobhi M. Gomha, Mohamed M. Abdulla, Reem K. Arafa

4) Structure-Based Virtual Screening for Fragment-Like Ligands of the G Protein-Coupled Histamine H4 Receptor (ChemMedComm) Monday March 30th 2015
Enade P. Istyastono, Albert J. Kooistra, Henry Vischer, Martien Kuijer, Luc Roumen, Saskia Nijmeijer, Rogier Smits, Iwan de Esch, Rob Leurs, Chris de Graaf

5) Novel synthesis of fluorochrome-coupled zoledronate with preserved functional activity on gamma/delta T cells and tumor cells (ChemMedComm) Monday March 30th 2015
Vijayanand Chandrasekaran, Shirin Kalyan, Valentina Biehl, Marcus Lettau, Patrik Theodor Nerdal, Hans-Heinrich Oberg, Daniela Wesch, Thisbe K Lindhorst, Dieter Kabelitz

6) Discovery of 2-(5,6-dimethoxypyridin-3-yl)-4-(2,4,6-trifluorobenzyl)-2H-pyrido[2,3-e][1,2,4]thiadiazin-3(4H)-one 1,1-dioxide (HTL6641), a dual orexin receptor antagonist with differentiated pharmacodynamic properties.[dagger] (ChemMedComm) Monday March 30th 2015
John Andrew Christopher, Sarah Aves, Jason Brown, James Errey, Suki Klair, Christopher Langmead, Oliver Mace, Richard Mould, Jayesh Patel, Ben Tehan, Andrei Zhukov, Fiona Marshall, Miles Congreve

7) Design of pyrazolo-pyrimidines as 11β-HSD1 inhibitors through optimisation of molecular electrostatic potential (ChemMedComm) Monday March 30th 2015
Graeme Robb, Scott Boyd, Christopher Davies, Alexander Dossetter, Frederick W Goldberg, Paul D Kemmitt, James Scott, John Swales

8) Concise Synthesis of Spergualin-Inspired Molecules With Broad-Spectrum Antibiotic Activity (ChemMedComm) Monday March 30th 2015
Victoria Assimon, Hao Shao, Sylvie Garneau-Tsodikova, Jason E. Gestwicki

9) 4-methyl-coumarins with cytotoxic activity against T24 and RT4 human bladder cancer cell lines (ChemMedComm) Thursday March 26th 2015
DAMIANA DA ROCHA VIANNA, LEILA Ruschel, FABRICIA Dietrich, Fabricio Figueiro, Fernanda Morrone, Romulo F. S. Canto, Flavia Corvello, Alice Velho, Allan Crestani, Helder Teixeira, Gilsane Lino von Poser, Ana Maria Oliveira Battastini, Vera Eifler-Lima

10) Tantalising technology (ChemMedComm) Tuesday March 24th 2015
Derek Lowe

11) Synthesis of a new HYNIC-DAPI derivative for labelling with 99mTechnetium and its in vitro evaluation in an FRTL5 cell line (ChemMedComm) Monday March 23rd 2015
Sandra Ferl, Gerd Wunderlich, Rene Smits, Alexander Hoepping, Anne Naumann, Jorg Kotzerke

12) Interactive articles in MedChemComm - connecting readers to a wealth of data and information (ChemMedComm) Thursday March 19th 2015
Richard Kelly

13) Insights into a defined secondary binding region on β-adrenoceptors and putative roles in ligand binding and drug design (ChemMedComm) Thursday March 12th 2015
Marvin Antonio Soriano-Ursua, Jose G Trujillo-Ferrara, Jose A Arias-Montano, Rafael Villalobos-Molina

14) Synthesis and evaluation of anticancer activity of novel andrographolide derivatives (ChemMedComm) Monday March 9th 2015
Devendar Ponnam, Lakshma Nayak V, Dharmendra Yadav, Niranjana Kumar Arigari, Kotesh Kumar Jonnala, Satya Srinivas KVN, Sridhar Balasubramanian, Feroz Khan, Pandu Sastry Kakaraparthi, Ramakrishna Sistla

15) Contributors to 'New Talent: Asia-Pacific' (ChemMedComm) Monday March 9th 2015


16) Membrane-interacting properties of the functionalised fatty acid moiety of muraymycin antibiotics (ChemMedComm) Friday March 6th 2015
Oliver Ries, Christian Carnarius, Claudia Steinem, Christian Ducho

17) In silico study on aging and reactivation processes of tabun conjugated AChE (ChemMedComm) Monday March 2nd 2015
Nellore Bhanu Chandar, Rabindranath Lo, Manoj K Kesharwani, Bishwajit Ganguly

18) Design, synthesis and biological evaluation of thiourea and nicotinamide-containing sorafenib analogs as antitumor agents (ChemMedComm) Monday March 2nd 2015
Xiangkai Kong, Zeyu Yao, Zuopeng He, Wen-Fang Xu, Jianwen Yao

19) Novel non-substrate modulators of the transmembrane efflux pump P-glycoprotein (ABCB1) (ChemMedComm) Friday February 27th 2015
Soren Krawczyk, Christiane Baumert, Josef Molnar, Christoph Ritter, Jens Hopner, Charlotte Kloft, Andreas Hilgeroth

20) Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday February 17th 2015
Taha Eldebss, Sobhi Gomha, Mohamed Abdalla, Reem Arafa

21) Matrix-immobilized yeast for large-scale production of recombinant human lactoferrin (ChemMedComm) Tuesday February 17th 2015
Chun Loong Ho, In Young Hwang, Kathy Loh, Matthew Chang

22) Synthesis and evaluation of amide, sulfonamide and urea - benzisoxazole derivatives as potential atypical antipsychotics (ChemMedComm) Friday February 13th 2015
Yin Chen, Yu Lan, Xudong Cao, Xiangqing Xu, Juecheng Zhang, Minquan Yu, Xin Liu, Bifeng Liu, Guisen Zhang

23) Synthesis and protective effect of new ligustrazine derivatives against CoCl2-induced neurotoxicity in differentiated PC12 cells. Part 2 (ChemMedComm) Thursday February 12th 2015
Bing Xu, Yan Gong, Xin Xu, Chenze Zhang, Yuzhong Zhang, Fuhao Chu, Hongbing Liu, Penglong Wang, Haimin Lei

24) BODIPY appended copper(II) complexes of curcumin showing mitochondria targeted remarkable photocytotoxicity in visible light (ChemMedComm) Thursday February 12th 2015
Akhil R Chakravarty, Arnab Bhattacharyya, Akanksha Dixit, Koushambi Mitra, Samya Banerjee, Anjali A Karande

25) Synthesis and biological evaluation of novel [capital Delta]2-isoxazoline fused cyclopentane derivatives as potential antimicrobial and anticancer agents (ChemMedComm) Wednesday February 11th 2015
Nagendra Babu Bathini, Santosh Kumar Prajapti, Shweta Shrivastava, Umesh Bihade, Ajay Kumar Gupta, V.G. M Naidu, Uttam Chand Banerjee

26) Evaluation of the anti-inflammatory/chondroprotective activity of aldose reductase inhibitors in human chondrocyte cultures (ChemMedComm) Wednesday February 4th 2015
Annamaria Panico, Rosanna Maccari, Venera Cardile, Sergio Avondo, Lucia Crasci, Rosaria Ottana

27) Inhibition of Insulin Amyloid Fibrillization by Glyco-Acridines: In vitro and in silico study (ChemMedComm) Wednesday February 4th 2015
Quan Van Vuong, Zuzana Bednarikova, Andrea Antosova, Huy Dinh Quoc Pham, Katarina Siposova, Nguyen Anh Tuan, Mai Suan Li, Zuzana Gazova

28) Application of QM/MM and QM methods to investigate histone deacetylase 8 (ChemMedComm) Monday February 2nd 2015
Duangkamol Gleeson, M. Paul Gleeson

29) Structure-Based Design, Synthesis by Click Chemistry and in Vivo Activity of Highly Selective A3 Adenosine Receptor Agonists (ChemMedComm) Monday February 2nd 2015
Dilip Tosh, Silvia Paoletta, Zhoumou Chen, Steven Crane, John Lloyd, Zhan-Guo Gao, Elizabeth Gizewski, John Auchampach, Daniela Salvemini, Kenneth A. Jacobson

30) Synthesis and evaluation of a series of resveratrol analogues as potent anticancer agents that target tubulin (ChemMedComm) Friday January 30th 2015
Nikhil Reddy Madadi, Hongliang Zong, Amit Ketkar, Zhen Chen, Narsimha Penthala, Venumadhav Janganati, Shobanbabu Bommagani, Robert Eoff, Monica Guzman, Peter Crooks

31) Design, Facile Synthesis and Anthelmintic Activity of New O-Substituted 6-Methoxybenzothiazole-2-carbamates (ChemMedComm) Tuesday January 27th 2015
A. Mohsen M.E. Omar, Omaima M. Aboulwafa, Doaa A. E. Issa, May M.S. El-Shokrofy, May E. Amr, Ibrahim M. El-Ashmawy

32) BEYOND THE AFFINITY FOR PROTEIN KINASE C: EXPLORING 2-PHENYL-3-HYDROXYPROPYL PIVALATE ANALOGUES AS C1 DOMAIN-TARGETING LIGANDS (ChemMedComm) Monday January 26th 2015
Daniela Rossi, Virpi Talman, Gustav Boije, Annamaria Marra, pietro Picconi, Rita Nasti, Massimo Serra, ANN JIHYAE, Marialaura Amadio, Alessia Pascale, Jeewoo Lee, Raimo Tuominen, Jari Yli-Kauhaluoma, Simona Collina

33) Correction: Identification of tris-(phenylalkyl)amines as new selective h5-HT2B receptor antagonists (ChemMedComm) Friday January 23rd 2015
Shashikanth Ponnala, Nirav Kapadia, Wayne Wesley Harding

34) Identification of Camphor Derivatives as Novel M2 Ion Channel Inhibitors of Influenza A Virus (ChemMedComm) Monday January 19th 2015
Xin Zhao, Zhen-Wei Zhang, Wei Cui, Shengwei Chen, Yang Zhou, Jianghong Dong, Yanling Jie, Junting Wan, Yong Xu, Wenhui Hu

35) O-Benzoyl Pyridine Aldoxime and Amidoxime Derivatives: Novel Efficient DNA Photo-Cleavage Agents (ChemMedComm) Thursday January 15th 2015
PARASKEVI KARAMTZIOTI, ASTERIOS PAPASTERGIOU, JOHN G. STEFANAKIS, ALEXANDROS E. KOUMBIS, IOANNA ANASTASIOU, MARIA KOFFA, KONSTANTINA C. FYLAKTAKIDOU

36) Nature of the Charged Head Group Dictates the Anticancer Potential of Lithocholic Acid-Tamoxifen Conjugates For Breast Cancer Therapy (ChemMedComm) Wednesday January 14th 2015
Kavita Yadav, Priyanshu Bhargava, Sandhya Bansal, Manish Singh, Siddhi Gupta, Geeta Sandhu, Sandeep Kumar, Vedagopuram Sreekanth, Avinash Bajaj

37) Targeted Photoresponsive TiO2-Coumarin nanoconjugate for efficient Combination therapy in MDA-MB-231 breast cancer cells: Synergic effect of Photodynamic Therapy (PDT) and Anticancer drug Chlorambucil (ChemMedComm) Wednesday January 14th 2015
Moumita Ganguly, Sourav K. Mukhopadhyay, Karthik S, Sharabani Barman, Pradeep N.D. Singh

38) Radiosynthesis of high affinity fluorine-18 labeled GnRH peptide analogues: in vitro studies and in vivo assessment of brain uptake in rats (ChemMedComm) Monday January 12th 2015
Dag Erlend Olberg, Sven H Hausner, Nadine Bauer, Jo Klaveness, Bard Indrevoll, Finn Olav Levy, Kjetil Wessel Andressen, Marie Dahl, Julie L. Sutcliffe, Ira Haraldsen

39) Design, synthesis and biological activity of 4′-[(benzimidazol-1-yl)methyl] biphenyl-2-sulphonamides as dual angiotensin II and endothelin A receptor antagonists (ChemMedComm) Monday January 12th 2015
Liping Hao, Weizhe Xue, Xiaofeng Han, Xing He, Jun Zhang, Zhiming Zhou

40) Activity Based Probes as Molecular Tools for Biomarker Discovery (ChemMedComm) Friday January 9th 2015
Luis Carvalho, Susana Dias Lucas, Eduardo Ruivo, Rui Moreira

41) Cytotoxic potential of di-spirooxindolo/acenaphthoquino andrographolide derivatives against MCF7 cell lines (ChemMedComm) Thursday January 8th 2015
Debanjana Chakraborty, Arindam Maitya, Chetan Kumar Jain, Abhijit Hazra, Yogesh Pandharinath Bharitkar, Tarun Jha, Hemanta Majumder, Susanta Roy Choudhury, Nirup Bikash Mondal

42) Dimethylaminoethyl Methacrylate Copolymer-siRNA nanoparticles for silencing therapeutically relevant gene in macrophages (ChemMedComm) Monday January 5th 2015
Ratnesh Jain, Prajakta Dandekar, Brigitta Loretz, Marcus Koch, C-M. lehr

43) Structure-activity relationship study on senktide for development of novel potent neurokinin-3 receptor selective agonists (ChemMedComm) Monday January 5th 2015
Ryosuke Misu, Koki Yamamoto, Ai Yamada, Taro Noguchi, Hiroaki Ohno, Takashi Yamamura, Hiroaki Okamura, Fuko Matsuda, Satoshi Ohkura, Shinya Oishi, Nobutaka Fujii

44) Synthesis and biological evaluation of pentanedioic acid derivatives as farnesyltransferase inhibitors (ChemMedComm) Monday January 5th 2015
liuqing Yang, wei liu, Hanbin Mei, yuan Zhang, Xiaojuan Yu, yufang xu, Honglin Li, Jin Huang, Zhenjiang Zhao

45) Recent discoveries and developments of Androgen Receptor based therapy for Prostate Cancer (ChemMedComm) Monday January 5th 2015
Ramakrishnan Elancheran, V.L Maruthanila, M Ramanathan, S Kabilan, R Devi, A Kunnumakara, Jibon Kotoky

46) Chemical space is big. Really big (ChemMedComm) Monday January 5th 2015
Derek Lowe

47) Discovery of Highly Potent Triazole Antifungal Agents with Piperdine-oxadiazole Side Chains (ChemMedComm) Wednesday December 24th 2014
Xiaomeng He, Yan Jiang, Yongqiang Zhang, Shanchao Wu, Guoqiang Dong, Na Liu, Yang Liu, Jianzhong Yao, Zhenyuan Miao, Yan Wang, Wannian Zhang, Chunquan Sheng

48) The Natural Product Brartemicin is a High Affinity Ligand for the Carbohydrate-Recognition Domain of the Macrophage Receptor Mincle (ChemMedComm) Tuesday December 23rd 2014
Kristian Mark Jacobsen, Ulrik Keiding, Lise Lindkvist Clement, Eva Susanne Schaffert, Neela Rambaruth, Mogens Johannsen, Kurt Drickamer, Thomas Bjornskov Poulsen

49) Inhibition of Influenza H5N1 invasion by modified heparin derivatives (ChemMedComm) Tuesday December 23rd 2014
Mark A. Skidmore, Anna Kajaste-Rudnitski, Nicola Wells, Scott Guimond, Timothy Rudd, Eliza Vicenzi, Edwin Yates

50) Pyrrole- and indole-containing tranylcypromine derivatives as novel lysine-specific demethylase 1 inhibitors active on cancer cells (ChemMedComm) Tuesday December 23rd 2014
Veronica Rodriguez, Sergio Valente, Stefano Rovida, Dante Rotili, Giulia Stazi, Alessia Lucidi, Giuseppe Ciossani, Andrea Mattevi, Oronza Botrugno, Paola Dessanti, Ciro Mercurio, Paola Vianello, Saverio Minucci, mario varasi, Antonello Mai

51) Enantiomeric resolution of [(2,2-diphenyl-1,3-dioxolan-4-yl)methyl](2-phenoxyethyl)amine, a potent α 1 and 5HT1A receptors ligand: an In Vitro and Computational Study (ChemMedComm) Tuesday December 23rd 2014
Livio Brasili, Silvia Franchini, Annamaria Baraldi, Claudia Sorbi, Federica Pellati, Elena Cichero, Umberto M. Battisti, Piero Angeli, Antonio Cilia

52) Synthesis and relationship of stability and biological activity of new DSS and TMP conjugates (ChemMedComm) Monday December 22nd 2014
Yewei Sun, Zicheng Tan, Zhibin Liang, Liang Wang, Luchen Shan, Pei Yu, Simon MingYuen Lee, Yuqiang Wang

53) Synthesis and antibacterial activity of trivalent ultrashort Arg-Trp-based antimicrobial peptides (AMPs) (ChemMedComm) Monday December 22nd 2014
Barbara C. Hoffknecht, H. Bauke Albada, Marina Sturm, Pascal Prochnow, Julia E. Bandow, Nils Metzler-Nolte

54) Non-nucleoside anti-HBV agents: Advances in structural optimization and mechanism of action investigations (ChemMedComm) Tuesday December 16th 2014
Na Liu, Diwakar Rai, Fabao Zhao, Haiyong Jia, Peng Zhan, Xinyong Liu

55) Discovery of a new class of histone deacetylase inhibitors with a novel zinc binding group (ChemMedComm) Tuesday December 16th 2014
Youxuan Li, Patrick M. Woster

56) The chemistry and pharmacology of privileged pyrroloquinazolines (ChemMedComm) Monday December 15th 2014
Bo Chao, Bingbing X Li, Xiangshu Xiao

57) Synthesis of six mexiletine derivatives with isoindolines attached as potential antioxidants and their evaluation as cardioprotective agents (ChemMedComm) Monday December 15th 2014
W Roy Jackson, Anh Chau, Grant Drummond, Bevyn Jarrott, Alyson Miller, Kamani Subasinghe, Christina Yan Ru Tan, Paul J White, Christine E Wright, James Ziogas

58) Solid- and solution-phase-based library of 2β-methyl substituted penicillin derivatives. Effects on growth inhibition of tumor cell lines (ChemMedComm) Monday December 15th 2014
Dora B. Boggian, Patricia Cornier, Ernesto Mata, Viviana Blanck, Mariano Cardenas, LP Roguin

59) Identification of tris-(phenylalkyl)amines as new selective h5-HT2B receptor antagonists (ChemMedComm) Monday December 15th 2014
Wayne Harding, Shashikanth Ponnala, Nirav Kapadia

60) Photoswitching property of hairpin ODNs with azobenzene derivatives in the loop (ChemMedComm) Monday December 15th 2014
Li Wu, Ya Wu, Hongwei Jin, Liangren Zhang, Yujian He, XinJing Tang

61) Synthesis and evaluation of 6-methylcoumarin derivatives as potent and selective Monoamine Oxidase B inhibitors (ChemMedComm) Monday December 15th 2014
Jin-Shuai Lan, Long-Fei Pan, Sai-Sai Xie, Xiao-Bing Wang, Ling-Yi Kong

62) Naturally occurring FANCF-Hes1 complex inhibitors from Wrightia religiosa (ChemMedComm) Thursday December 11th 2014
Midori A. Arai, Kenji Uemura, Nozomi Hamahiga, Naoki Ishikawa, Takashi Koyano, Thaworn Kowithayakorn, Tagrid Kaddar, Madeleine Carreau, Masami Ishibashi

63) Correction: Design and chemoproteomic functional characterization of a chemical probe targeted to bromodomains of BET family proteins (ChemMedComm) Monday December 8th 2014
Jiang Wu, Julia Shin, Cara M. M. Williams, Kieran F. Geoghegan, Stephen W. Wright, David C. Limburg, Parag Sahasrabudhe, Paul D. Bonin, Bruce A. Lefker, Simeon J. Ramsey

64) Relating Caco-2 permeability to molecular properties using block relevance analysis (ChemMedComm) Monday December 8th 2014
Tim Potter, G Caron, Giuseppe Ermondi, Gayle Newbury

65) Design, synthesis and biological evaluation of imidazopyridine/imidazopyrimidine-benzimidazole conjugates as potential anticancer agents (ChemMedComm) Wednesday December 3rd 2014
Ahmed Kamal, Bharath Kumar G, Lakshma Nayak V, Santhosh Reddy Vangala, Anver Basha Shaik, Rajender Rajender, Kashi Reddy Methuku

66) Synthesis and cytostatic activity of 7-arylsulfanyl-7-deazapurine bases and ribonucleosides (ChemMedComm) Tuesday December 2nd 2014
Martin Klecka, Lenka Slavetinska, Eva Tloustova, Petr Dzubak, Marian Hajduch, Michal Hocek

67) Synthesis of 17-membered azalides from a 16-membered macrolide utilizing amide-selective silane reduction (ChemMedComm) Tuesday December 2nd 2014
Atsushi Seki, Toshihiro Mori, Kouji Sasaki, Yoshiaki Takahashi, Toshiaki Miyake, Yuzuru Akamatsu

68) 3-(2,6-Dichloro-benzyloxy)-11-oxo-olean-12-ene-29-oic acid, a semisynthetic derivative of glycyrrhetic acid: Synthesis, antiproliferative, apoptotic and anti-angiogenesis activity (ChemMedComm) Monday December 1st 2014
Rajni Sharma, Santosh Guru, Shreyans K Jain, Anup S Pathania, Ram A Vishwakarma, Shashi Bhushan, Sandip Bibishan Bharate

69) Discovery of novel 5-fluoro-N2,N4-diphenylpyrimidine-2,4-diamines as potent inhibitors against CDK2 and CDK9 (ChemMedComm) Friday November 28th 2014
Jiadi Gao, Cheng Fang, Zhiyan Xiao, Li Huang, Chin Ho Chen, Li-Ting Wang, Kuo-Hsiung Lee

70) Recent advances in molecular imaging probes for β-amyloid plaques (ChemMedComm) Tuesday November 25th 2014
Masahiro Ono, Hideo Saji

71) Design, synthesis and evaluation of QD-DTC-BisBiotin Nanobioconjugate as a potential Optical-SPECT imaging agent (ChemMedComm) Friday November 21st 2014
Narmada Bag, Rashi Mathur, Sweta Singh, Firasat Hussain, Ramprakash Chauhan, krishna Chuttani, Anil K Mishra

72) 4-Thiazolidinone derivatives as potent antimicrobial agents: microwave-assisted synthesis, biological evaluation and docking studies (ChemMedComm) Wednesday November 19th 2014
Eleni Pitta, Evangelia Tsolaki, Athina Geronikaki, Jovana Petrovic, Jasmina Glamoclija, Marina Sokovic, Emmanuele Crespan, Giovanni Maga, Shome S. Bhunia, Anil K. Saxena

73) Evaluation of aromatic 6-substituted thienopyrimidines as scaffolds against parasites that cause trypanosomiasis, leishmaniasis, and malaria. (ChemMedComm) Friday November 14th 2014
Jennifer Woodring, Gautam Patel, Jessey Erath, Ranjan Behera, Patricia Lee, Susan Leed, Ana Rodriguez, Richard Sciotti, Kojo Mensa-Wilmot, Michael Pollastri

74) Exclusive Formation of Imino [4+4] cycloaddition Products with Biologically Relevant Amines: Plausible Candidates of Acrolein Biomarkers and Biofunctional Modulators (ChemMedComm) Friday November 14th 2014
Ayumi Tsutsui, Ambara R. Pradipta, Elena Saigitbatalova, Almira Kurbangalieva, Katsunori Tanaka

75) Cytotoxic Peptide Conjugates of Dinuclear Arene Ruthenium Trithiolato Complexes (ChemMedComm) Wednesday November 12th 2014
Federico Giannini, Marco Bartoloni, Lydia E. H. Paul, Georg Suss-Fink, Jean-Louis Reymond, Julien Furrer

76) Novel β-carboline-quinazolinone hybrid as inhibitor of Leishmania donovani Trypanothione Reductase: Synthesis, molecular docking and bioevaluation (ChemMedComm) Tuesday November 4th 2014
Shikha S. Chauhan, Shashi pandey, Rahul Shivahare, Karthik Ramalingam, Shagun Krishna, Preeti Vishwakarma, M. I. Siddiqi, Suman Gupta, Neena Goyal, PMS Chauhan

77) Potent chemical chaperone compounds for GM1-gangliosidosis: N-substituted (+)-conduramine F-4 derivatives (ChemMedComm) Tuesday November 4th 2014
Shinichi Kuno, Katsumi Higaki, Atsushi Takahashi, Eiji Namba, Seiichiro Ogawa

78) Decorated 6,6',7,7'-tetrahydro-1H,1'H-2,3'-biindole scaffold as promising candidate for recognition of CDK2 allosteric site (ChemMedComm) Monday November 3rd 2014
Maria Teresa Sciortino, Angela Scala, Antonio Rescifina, Ivana Colao, Gabriel Siracusano, Antonino Mazzaglia, Ugo Chiacchio, Giovanni Grassi

79) Virtual screening for novel Atg5-Atg16 complex inhibitors for autophagy modulation (ChemMedComm) Monday November 3rd 2014
Elizabeth Robinson, Euphemia Leung, Anna Matuszek, Niels Krogsgaard-Larsen, Daniel Furkert, Margaret A Brimble, Alan Richardson, Johannes Reynisson

80) Antimicrobial spine-bone cement with caffeic acid phenethyl ester for controlled release formulation and in vivo biological assessments (ChemMedComm) Monday November 3rd 2014
Hye Sun Lee, Jeong Ho Chang

81) Design, synthesis and anticancer mechanistic studies of linked azoles (ChemMedComm) Friday October 31st 2014
Amirul Islam, Yuqi Zhang, Yao Wang, Shelli Renee McAlpine

82) Probing cytochrome P450-mediated activation with a truncated azinomycin analogue (ChemMedComm) Wednesday October 22nd 2014
Victoria Vinader, Maria Sadiq, Mark Sutherland, Mengying Huang, Paul Loadman, Lina Elsalem, Steve Shnyder, Hongjuan Cui, Kamyar Afarinkia, Mark Searcey, L H Patterson, Klaus Pors

83) Study of a D-proline peptidomimetic inhibitor of melanoma and endothelial cells invasion through activity towards MMP-2 and MMP-9 (ChemMedComm) Tuesday October 21st 2014
Francesca Bianchini, Chiara Calugi, Jessica Ruzzolini, Gloria Menchi, Lido Calorini, Antonio Guarna, Andrea Trabocchi

84) Polymeric Micelles for Hydrogen Sulfide Delivery (ChemMedComm) Tuesday October 21st 2014
Urara Hasegawa, Andre J van der Vlies

85) Synthesis and Biological Evaluation of novel derivatives of Gambogenic acid as Anticancer Agent (ChemMedComm) Friday October 17th 2014
Liqin He, Peng Huang, Zhong Hu, Xiaoshan Wang, Yaxian Wu

86) Synthesis, 3D pharmacophore, QSAR and docking studies of novel quinazoline derivatives with nitric oxide release moiety as preferential COX-2 inhibitors (ChemMedComm) Friday October 17th 2014
Doaa Boshra Farag, Nahla Ahmed Farag, Ahmed Esmat, Sally A. Abuelezz, Eman Abdel-Salam Ibrahim, Dalal A. Abou El Ella

87) Synthesis, Structure-Activity Relationship, and Mechanistic Investigation of Lithocholic Acid Amphiphiles for Colon Cancer Therapy (ChemMedComm) Wednesday October 15th 2014
Manish Singh, Sandhya Bansal, Somanath Kundu, Priyanshu Bhargava, Ashima Singh, Rajender Motiani, Radhey Shyam, Vedagopuram Sreekanth, Sagar Sengupta, Avinash Bajaj

88) Towards understanding cell penetration by stapled peptides (ChemMedComm) Tuesday October 14th 2014
Qian Chu, Raymond E. Moellering, Gerard J. Hilinski, Young-Woo Kim, Tom N. Grossmann, Johannes T.-H. Yeh, Gregory L. Verdine

89) Synthesis of new betulinic acid-peptide conjugates and in vivo and in silico studies of the influence of peptide moieties on the triterpenoid core activity (ChemMedComm) Monday October 13th 2014
Valentine Nenajdenko, Anastasiya Govdi, Nadezhda Sokolova, Irina Sorokina, Sergey Vasilevsky, Dmitry Baev, Tatyana Tolstikova, Victor Mamatyuk, Dmitry Fadeev

90) Poly-α,β-aspartyl-Arg-Gly-Asp-Phe: A novel polymeric nanomedicine (ChemMedComm) Monday October 13th 2014
Shuangling Chen, Yuji Wang, Shan Li, Yaonan Wang, Ming Zhao, Haimei Zhu, Jianhui Wu, Shiqi Peng

91) Synthesis and biological evaluation of a new class of quinazolinone azoles as potential antimicrobial agents and their interactions with calf thymus DNA and Human Serum Albumin (ChemMedComm) Wednesday October 8th 2014
Cheng-He Zhou, Li-Ping Peng, Nagarajan Sangaraiah, RASHEED SYED

92) Synthesis and Evaluation of Phenoxymethylbenzamide Analogues as Anti-Trypanosomal Agents (ChemMedComm) Wednesday October 8th 2014
Richard James Payne, Alexandra Manos-Turvey, Emma Watson, Vicky Mary Avery, Amy Jones, Melissa Sykes, Jonathan D. Baell, Marcel Kaiser

93) Polypharmacology Modelling Using Proteochemometrics (PCM): Recent Methodological Developments, Applications to Target Families, and Future Prospects (ChemMedComm) Tuesday October 7th 2014
Isidro Cortes-Ciriano, Qurrat ul Ain, Vigneshwari Subramanian, Bart Lenselink, Oscar Mendez-Lucio, AP IJzerman, Gerd Wohlfahrt, Peteris Prusis, Therese E Malliavin, Gerard van Westen, Andreas Bender

94) Can we use the epigenetic bioactivity of caloric restriction and phytochemicals to promote healthy ageing? (ChemMedComm) Friday October 3rd 2014
nadine helene martinet, adeline thomas, Stephane Poulain, Michael Christodoulou, Bertrand Philippe, rachid benhida, Daniele Passarella, melita vidakovic, daumantas matulis, maija .lahtela-kakkonen, eva Bartova, christophe blanquart, E. Mikros, nikolas fokialakis

95) Elucidation of shanorellin biosynthetic pathway and functional analysis of associated enzymes (ChemMedComm) Thursday October 2nd 2014
Michio Sato, Haruka Yamada, Kinya Hotta, Kenji Watanabe

96) Synthesis and biological evaluation of a series of aryl triazoles as firefly luciferase inhibitors (ChemMedComm) Tuesday September 30th 2014
Haixiu Bai, Peng Zhu, Wenxiao Wu, Jing Li, Zhao Ma, Wei Zhang, Yanna Cheng, Lupei Du, Minyong Li

97) Discovery of novel Sphingosine Kinase 1 inhibitors via structure-based hierarchical virtual screening (ChemMedComm) Tuesday September 30th 2014
Xiaojian Wang, Chenbin Sun, Liang Fang, Dali Yin

98) Discovery of mitochondria-targeting berberine derivatives as inhibitors of proliferation, invasion and migration against rat C6 and human U87 glioma cells (ChemMedComm) Tuesday September 30th 2014
Shengnan Fu, Yanqi Xie, Juo Tuo, Yalong Wang, Wenbo Zhu, Sihan Wu, Guangmei Yan, Haiyan Hu

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This week's C&EN

Shining a Light on Erectile Disfunction

Analytical Chemists Met in Graz


Mitch Andre Garcia's Chem Feeds 2008-present

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