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1) Discovery of Novel Guanidinophenylpyrazole Human Acrosin Inhibitors by Molecular Hybridization (ChemMedComm) Monday July 28th 2014
Juntao Zhao, Nuannuan Sun, Yue Gao, Diya Lv, Yang Liu, Yan Jiang, Guoqiang Dong, Qianqian Chen, Wei Li, Youjun Zhou, Ju Zhu, Jiaguo Lv, Chunquan Sheng

2) Osthol and curcumin as inhibitors of human Pgp and multidrug efflux pumps of Staphylococcus aureus: Reversing the resistance against frontline antibacterial drugs (ChemMedComm) Wednesday July 23rd 2014
Prashant Joshi, Samsher Singh, Abubakar Wani, Sadhana Sharma, Shreyans K Jain, Baljinder Singh, Bishan Gupta, Naresh Satti, S Koul, Inshad A Khan, Ajay Kumar, Sandip Bibishan Bharate, Ram A Vishwakarma

3) A novel surface-coated nanocarrier for efficient encapsulation and delivery of Camptothecin to cells (ChemMedComm) Wednesday July 23rd 2014
Rie Wakabayashi, Ryutaro Ishiyama, Noriho Kamiya, Masahiro Goto

4) A Critical Evaluation of Pyrrolo[2,3-d]pyrimidine-4-amines as Plasmodium falciparum Apical Membrane Antigen 1 (AMA1) Inhibitors (ChemMedComm) Wednesday July 23rd 2014
Shane Devine, San Lim, Indu Chandrashekaran, Christopher MacRaild, Damien Drew, Cael Debono, Raymond Lam, Robin Anders, James Beeson, Martin Scanlon, Peter J. Scammells, Ray Norton

5) Gold compounds as aquaporin inhibitors: new opportunities for therapy and imaging (ChemMedComm) Tuesday July 22nd 2014
Andreia de Almeida, Graca Soveral, Angela Casini

6) Diversity-Oriented Synthesis for Novel, Selective and Drug-like Inhibitors for a Phosphatase from Mycobacterium Tuberculosis (ChemMedComm) Tuesday July 22nd 2014
Rongjun He, Yunpeng Bai, Zhi-Hong Yu, Li Wu, Andrea M. Gunawan, Zhong-Yin Zhang

7) Gold(I) compounds with lansoprazole-type ligands: synthesis, characterization and anticancer properties in vitro (ChemMedComm) Monday July 21st 2014
Maria Serratrice, Benoit Bertrand, Esmee F. J. Janssen, Eline Hemelt, Antonio Zucca, Fabio Cocco, Maria A. Cinellu, Angela Casini

8) Synthesis of a novel series of 2,3,4-trisubstituted oxazolidines designed by isosteric replacement or rigidification of the structure and cytotoxic evaluation (ChemMedComm) Monday July 21st 2014
Saulo Andrade, Claudia Teixeira, Jonas Ramos, Marcela Lopes, Rodrigo Padua, Monica Oliveira, Elaine Souza-Fagundes, Ricardo Alves

9) Anaplastic lymphoma kinase (ALK) inhibitors: a review of design and discovery (ChemMedComm) Monday July 21st 2014
Wen-Chieh Wang, Hui-Yi Shiao, Chieh-Chien Lee, Ka-Shu Fung, Hsing-Pang Hsieh

10) Structure-based approaches towards identification of fragments for the low-druggability ATAD2 bromodomain (ChemMedComm) Tuesday July 15th 2014
Apirat Chaikuada, Andrew Petros, Oleg Fedorov, Jing Xu, Stefan Knapp

11) Carbohydrates themed issue (ChemMedComm) Tuesday July 15th 2014
Sylvie Garneau-Tsodikova, Timor Baasov

12) Beyond substrate analogues: new inhibitor chemotypes for glycosyltransferases (ChemMedComm) Friday July 11th 2014
Lauren Tedaldi, Gerd K. Wagner

13) Benzylidene-linked thiohydantoin derivatives as inhibitors of tyrosinase and melanogenesis: Importance of β-phenyl-α,β-unsaturated carbonyl functionality (ChemMedComm) Wednesday July 2nd 2014
Hye Rim Kim, Hye Jin Lee, Yeon Ja Choi, Yun Jung Park, Youngwoo Woo, Seong Jin Kim, Min Hi Park, Hee Won Lee, Pusoon Chun, H.Y. Chung, Hyung Ryong Moon

14) N-Arylalkylbenzo[d]thiazole-2-carboxamides as anti-mycobacterial agents: Design, new methods of synthesis and biological evaluation (ChemMedComm) Monday June 30th 2014
Asit Kumar Chakraborti, Parth Shah, Tejas Dhameliya, Rohit Bansal, Manesh Nautiyal, Damodara Naidu Kommi, Pradeep S. Jadhavar, Jonnalagadda Padma Sridevi, Yogeeswari Sriram, Dharmarajan Sriram

15) Triazole containing novobiocin and biphenyl amides as Hsp90 C-terminal inhibitors (ChemMedComm) Friday June 27th 2014
Jinbo Zhao, Huiping Zhao, Jessica A. Hall, Douglas Brown, Eileen Brandes, Joseph Bazzill, Patrick T. Grogan, Chitra Subramanian, George Vielhauer, Mark S. Cohen, Brian S. J. Blagg

16) Mechanism of forming trimer, self-assembling nano-particle and inhibiting tumor growth of small molecule CIPPCT (ChemMedComm) Wednesday June 25th 2014
Fengxiang Du, Xiaoyi Zhang, Shan Li, Yaonan Wang, Meiqing Zheng, Yuji Wang, Shurui Zhao, Jianhui Wu, Lin Gui, Ming Zhao, Shiqi Peng

17) Prekinamycin and an Isosteric-Isoelectronic Analogue Exhibit Comparable Cytotoxicity Towards K562 Human Leukemia Cells (ChemMedComm) Wednesday June 25th 2014
Gary I Dmitrienko, Glenn Abbott, Brian Hasinoff, Xing Wu, Vladimir Birman, zhufeng zhao, Lei Guo

18) In vitro selection of a peptide aptamer that potentiates inhibition of cyclin-dependent kinase by purvalanol (ChemMedComm) Wednesday June 25th 2014
Wei Wang, Yoshinori Hirano, Takanori Uzawa, Mingzhe Liu, Makoto Taiji, Yoshihiro Ito

19) Optimization of the anti-cancer activity of phopshotidylinositol-3 kinase pathway inhibitor PITENIN-1: switching a thiourea with 1,2,3-triazole (ChemMedComm) Tuesday June 24th 2014
Yadagiri Kommagalla, Sinziana Cornea, Robert Riehle, Vladimir Torchilin, Alexei Degterev, Cherupi Ramana

20) Imidazolium derived ionic salts induce inhibition of cancerous cell growth through apoptosis (ChemMedComm) Tuesday June 24th 2014
Sanjay Malhotra, Vineet Kumar, Christian E Velez Gerena, Beatriz Zayas

21) Identification of Tanshinone IIA as a Natural Monoacylglycerol Lipase Inhibitor by Combined in silico and in vitro Approach (ChemMedComm) Monday June 23rd 2014
Jianhua Liu, Ruolin Yang, Yang Lu

22) Evaluation of Functional Groups as Acetyl-Lysine Mimetics for BET Bromodomain Inhibition (ChemMedComm) Monday June 23rd 2014
Phillip Patrick Sharp, Jean-Marc Garnier, David C.S. Huang, Christopher J Burns

23) Benzothiazolyl Substituted Iminothiazolidinones and Benzamido-oxothiazolidines as Potent and Partly Selective Aldose Reductase Inhibitors (ChemMedComm) Friday June 20th 2014
Jamshed Iqbal, Aamer Saeed, Yildiz Tehseen, Humera Raffique, Norbert Furtmann, J Bajorath, Ulrich Floerke

24) Conformational Analysis of Peramivir Reveals Critical Differences Between Free and Enzyme-Bound States (ChemMedComm) Thursday June 19th 2014
Michele R Richards, Michael G Brant, Martin Boulanger, Christopher W. Cairo, Jeremy E Wulff

25) Understanding the Structural Requirements of Hybrid (S)-6-((2-(4-Phenylpiperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-1-ol and its Analogs as D2/D3 Receptor Ligands: A Three-Dimensional Quantitative Structure-Activity Relationship (3D QSAR) Investigation (ChemMedComm) Thursday June 19th 2014
Gyan Prakash Modi, Horrick Sharma, Prashant Suresh Kharkar, Aloke K. Dutta

26) Characterization of a selective inhibitor for matrix metalloproteinase-8 (MMP-8) (ChemMedComm) Wednesday June 18th 2014
Derong Ding, Katerina Lichtenwalter, Hualiang Pi, Shahriar Mobashery, Mayland Chang

27) Synthesis of Hybrid Anticancer Agents Based on Kinase and Histone Deacetylase Inhibitors (ChemMedComm) Wednesday June 18th 2014
Hiren Patel, Irina Chuckowree, Peter Coxhead, Matthew Guille, Minghua Wang, Alexandra Zuckerman, Robin Williams, Mariangela Librizzi, Ronald Paranal, James Bradner, John Spencer

28) Inhibitors of the human neuraminidase enzymes (ChemMedComm) Wednesday June 18th 2014
Christopher W. Cairo

29) A fundamental view of enthalpy-entropy compensation (ChemMedComm) Tuesday June 17th 2014
Ulf Ryde

30) NMR and Molecular recognition. The application of ligand-based NMR methods to monitor molecular interactions (ChemMedComm) Tuesday June 17th 2014
Unione Luca, Galante Silvia, Diaz Dolores, Javier Canada, Jesus Barbero

31) A versatile acid-labile linker for antibody-drug conjugates (ChemMedComm) Tuesday June 17th 2014
Mathew Finniss, Kevin Chu, Charles Bowerman, James Luft, Zishan Haroon, J. M. Desimone

32) Theoretical and experimental investigation on clarithromycin, erythromycin A and azithromycin and descladinosyl derivatives of clarithromycin and azithromycin with 3-O substitution as anti-bacterial agents (ChemMedComm) Wednesday June 11th 2014
Jill Barber, Biljana Arsic, Abida Awan, Richard Brennan, Juan Aguilar, Ruth Ledder, Andrew J McBain, Andrew Charles Regan

33) Branched α-D-mannopyranosides; a new class of potent FimH antagonists (ChemMedComm) Wednesday June 11th 2014
Tihomir Tomasic, Said Rabbani, Martina Gobec, Irena Mlinaric Rascan, Crtomir Podlipnik, B Ernst, Marko Anderluh

34) Species differences in drug plasma protein binding (ChemMedComm) Tuesday June 10th 2014
Nicola Colclough, Linette Ruston, J. Matthew Wood, Philip A. MacFaul

35) Synthesis of 3'-Deoxy-3'-fluorothymidine (FLT) 5'-O-Glucuronide: A Reference Standard for Imaging Studies with [18F]FLT (ChemMedComm) Tuesday June 3rd 2014
Bernard Thomas Golding, Suzannah Harnor, Tommy Rennison, Martin Galler, Celine Cano, Roger J Griffin, David Newell

36) Recognition of diazirine-modified O-GlcNAc by human O-GlcNAcase (ChemMedComm) Monday June 2nd 2014
Andrea Rodriguez, Jennifer Kohler

37) Multivalent Amino Sugars to Recognize Different TAR RNA Conformations (ChemMedComm) Friday May 30th 2014
Dev P Arya, Patrick Kellish, Mirko Hennig, Meredith Newby, Todd Mack, Sunil Kumar

38) Exploring the meaning of sugar configuration in a supramolecular environment: Comparison of six octyl glycoside micelles by ITC and NMR spectroscopy (ChemMedComm) Friday May 30th 2014
Thisbe K Lindhorst, Jorn Schmidt-Lassen

39) Synthesis, complex stability and small animal PET imaging of a novel 64Cu-labelled cryptand molecule (ChemMedComm) Friday May 30th 2014
Christian Foerster, James Christopher Knight, Melinda Wuest, Brendan Rowan, Suzanne E. Lapi, Angelo J. Amoroso, Peter G Edwards, Frank Wuest

40) Synthesis and biological evaluation of panitumumab-IRDye800 conjugate as a fluorescence imaging probe for EGFR-expressing cancers (ChemMedComm) Friday May 30th 2014
Sibaprasad Bhattacharyya, Nimit Patel, Ling Wei, Lisa A Riffle, Joseph D Kalen, G Craig Hill, Paula M Jacobs, Kurt R Zinn, Eben Rosenthal

41) Tetracycline analogues with a selective inhibitory effect on HIF-1α (ChemMedComm) Friday May 30th 2014
Y. Bendiabdellah, K. M. Rahman, B. Uranchimeg, K. S. Nahar, D. Antonow, R. H. Shoemaker, G. Melillo, G. Zinzalla, D. E. Thurston

42) Synthesis, chiral resolution, absolute configuration assignment and pharmacological evaluation of a series of melatoninergic ligands (ChemMedComm) Wednesday May 28th 2014
Mohamed Ettaoussi, Basile Peres, Christian Jarry, Olivier Nosjean, Jean Boutin, Arnaud Gohier, Clotilde Mannoury la Cour, Daniel Caignard, Philippe Delagrange, Pascal Berthelot, Said Yous

43) A practical glycosyltransferase assay for the identification of new inhibitor chemotypes (ChemMedComm) Friday May 23rd 2014
Lauren Tedaldi, Andrew Evitt, Niina Goos, Jingqian Jiang, Gerd K. Wagner

44) Synthesis of Isoxazole Moiety Containing Ferrocene Derivatives and Preliminarily in vitro Anticancer Activity (ChemMedComm) Thursday May 22nd 2014
Yong Jianping, Can-Zhong Lu, Xiao-Yuan Wu

45) Structure of the Cannabinoid Receptor 1: Homology Modeling of Its Inactive State and Enrichment Study Based on CB1 Antagonist Docking (ChemMedComm) Tuesday May 20th 2014
Haining Liu, Ronak Patel, Robert J. Doerksen

46) When Proteins Start to Make Sense: Fine-tuning Aminoglycosides for PTC Suppression Therapy (ChemMedComm) Friday May 16th 2014
Moran Shalev, Timor BAASOV

47) [small omega]-Heteroarylalkylcarbamates as inhibitors of fatty acid amide hydrolase (FAAH) (ChemMedComm) Friday May 16th 2014
Tobias Terwege, Helmut Dahlhaus, Walburga Hanekamp, M Lehr

48) Small-Molecule Phosphodiesterase Probes: Discovery of Potent and Selective CNS-Penetrable Quinazoline Inhibitors of PDE1 (ChemMedComm) Friday May 16th 2014
John M Humphrey, Eddie Yang, Christopher W. am Ende, Eric Arnold, Jenna Head, Stephen Jenkinson, Spiros Liras, jayvardhan Pandit, Brian Samas, Frank Menniti, Felix Vajdos, Lorraine Lebel

49) Multivalent Glycoconjugates as Vaccines and Potential Drug Candidates (ChemMedComm) Friday May 16th 2014
Rainer Haag, Sumati Bhatia, Mathias Dimde

50) Synthesis of Cyclohexapeptides as Antimalarial and Anti-trypanosomal Agents (ChemMedComm) Friday May 16th 2014
Stella Pena, Catherine Fagundez, Andrea Medeiros, Marcelo Comini, Laura Scarone, Diver Sellanes, E Manta, Judit Tulla-Puche, Fernando Albericio, Lindsay Stewart, Vanessa Yardley, Gloria Serra

51) Carbohydrate Antigen Delivery by Water Soluble Copolymers as Potential Anti-cancer Vaccines (ChemMedComm) Friday May 16th 2014
Qian Qin, Zhaojun Yin, Philip Bentley, Xuefei Huang

52) New trends in aminoglycosides use (ChemMedComm) Thursday May 15th 2014
Marina Fosso Yatchang, Yijia Li, Sylvie Garneau-Tsodikova

53) Protein-protein interactions of ASPP2: an emerging therapeutic target (ChemMedComm) Wednesday May 14th 2014
Anat Iosub-Amir, Assaf Friedler

54) Ugi 4-CR Synthesis of γ- and [small delta]-Lactams (ChemMedComm) Wednesday May 14th 2014
Alexander Domling, Eberhardt Herdtweck, Ting Zhao, George Liao, andre Boltjes

55) Synthesis and Evaluation of Artesunate-Indoloquinoline Hybrids as Antimalarial Drug Candidates (ChemMedComm) Monday May 12th 2014
Ning Wang, Kathryn Jean Wicht, Elkhabiry Shaban, Ngoc Anh Tran, Ming-Qi Wang, Ikuya Hayashi, Md.Imran Hossain, Yoshihiko Takemasa, Marcel Kaiser, Ibrahim Sayed, Timothy J Egan, Tsutomu Inokuchi

56) Anti-bacterial glycosyl triazoles - Identification of an N-acetylglucosamine derivative with bacteriostatic activity against Bacillus (ChemMedComm) Thursday May 8th 2014
Helene Kuhn, Danielle Gutelius, Eimear Black, Christina Nadolny, Amit Basu, Christopher W Reid

57) Synthesis, characterization and evaluation of the substituent effect on the amoebicide activity of new hydrazones derivatives (ChemMedComm) Thursday May 8th 2014
Yanis Toledano, Ruth Melendrez-Luevano, Marisol Navarro-Olivarria, Juan Carlos Garcia-Ramos, Marcos Flores-Alamo, Luis Ortiz-Frade, Lena Ruiz-Azuara, Blanca M. Cabrera Vivas

58) Investigation of novel ropinirole analogues: Synthesis, pharmacological evaluation and computational analysis of dopamine D2 receptor functionalized congeners and homobivalent ligands (ChemMedComm) Tuesday May 6th 2014
Manuela Jorg, Agnieszka Kaczor, Frankie Mak, Kiew Ching Lee, Antti Poso, Neil Miller, Peter J. Scammells, Ben Capuano

59) Synthesis and biological evaluation of novel bivalent β-carbolines as potential antitumor agents (ChemMedComm) Tuesday May 6th 2014
Qifeng Wu, Zhushuang Bai, Qin Ma, Wenxi Fan, Liang Guo, Guoxian Zhang, Liqin Qiu, Huijuan Yu, guang shao, Rihui Cao

60) Synthesis and evaluation of a series of quinolinyl trans-cyanostilbene analogs as anticancer agents (ChemMedComm) Tuesday May 6th 2014
Narsimha Penthala, Venumadhav Janganati, Shobanbabu Bommagani, Peter Crooks

61) Design, Synthesis, and Evaluation of 4- and 5-Substituted o-(Octanesulfonamido)benzoic Acids as Inhibitors of Glycerol-3-Phosphate Acyltransferase (ChemMedComm) Tuesday May 6th 2014
Victor K Outlaw, Edward Wydysh, Aravinda Vadlamundi, Susan Medghalchi, CA Townsend

62) Synthesis and Antiproliferative Evaluation of 9-Methoxy- 6-(piperazin-1-yl)-11H-indeno[1,2-c]quinoline-11-one Derivatives. Part 4. (ChemMedComm) Tuesday May 6th 2014
Chih-Hua Tseng, CC Tzeng, Chien-Chih Chiu, Chiao-Li Yang, Pei-Jung Lu, Chon-Kit Chou, Chun-Yen Liu, Yeh-Long Chen

63) Antifungal Amphiphilic Aminoglycosides (ChemMedComm) Thursday May 1st 2014
Tom Chang, Jon Takemoto

64) Metabolism of a novel Skepinone L- like p38 mitogen-activated protein kinase inhibitor (ChemMedComm) Monday April 28th 2014
Kirsten Storch, matthias gehringer, Benjamin Baur, Stefan Laufer

65) Selective Inhibition of Bacterial Topoisomerase I by alkynyl-bisbenzimidazoles (ChemMedComm) Friday April 25th 2014
Dev P Arya, Nihar Ranjan, Geraldine Fulcrand, Ada King, Joseph Brown, X. Jiang, Fenfei Leng

66) A Mechanistic Study on the α-N-acetylgalactosaminidase from E. meningosepticum: A Family 109 Glycoside Hydrolase (ChemMedComm) Friday April 25th 2014
Saswati Chakladar, Saeideh Shamsi Kazem Abadi, Andrew J Bennet

67) Neoglycosylation and neoglycorandomization: Enabling tools for the discovery of novel glycosylated bioactive probes and early stage leads (ChemMedComm) Wednesday April 23rd 2014
Randal Goff, Jon S Thorson

68) Surface plasmon resonance for the characterization of bacterial polysaccharide antigens: a review (ChemMedComm) Wednesday April 23rd 2014
Francesco Berti, Barbara Brogioni

69) Synthesis, enantiomeric separation and docking studies on spiropiperidine analogues as ligands of nociceptin/orphanin FQ receptor (ChemMedComm) Wednesday April 23rd 2014
Livio Brasili, Umberto M. Battisti, Sandra Corrado, Claudia Sorbi, Andrea Cornia, Annalisa Tait, Davide Malfacini, Maria C Cerlesi, Girolamo Calo

70) Response of osteoblast-like MG63 on neoglycosylated collagen matrices (ChemMedComm) Wednesday April 23rd 2014
Laura Russo, Antonella Sgambato, Paolo Giannoni, Rodolfo Quarto, Simone Vesentini, Alfonso Gautieri, Laura Cipolla

71) Thiazole-based aminopyrimidines and N-phenylpyrazolines as potent antimicrobial agents. Synthesis and biological evaluation (ChemMedComm) Wednesday April 16th 2014
Prof. Athina Geronikaki, Konstantinos Liaras, Jasmina Glamocilija, Ana Ciric, Marina Sokovic

72) Bioactivity of surface tethered Osteogenic Growth Peptide motifs (ChemMedComm) Wednesday April 16th 2014
silvia panseri, Laura Russo, Monica Montesi, Francesca Taraballi, Carla Cunha, Maurilio Marcacci, Laura Cipolla

73) New glycopolymers as multivalent systems for lectin recognition (ChemMedComm) Wednesday April 16th 2014
VALESSA BARBIER, Michele Fiore, Nathalie Berthet, Olivier Renaudet

74) The role of modern drug discovery in the fight against neglected and tropical diseases (ChemMedComm) Wednesday April 16th 2014
Jeremy N. Burrows, Richard L. Elliott, Takushi Kaneko, Charles E. Mowbray, David Waterson

75) Synthesis of 4′-deoxy-4′-fluoro neamine and 4′-deoxy-4′-fluoro 4′-epi neamine (ChemMedComm) Tuesday April 15th 2014
Stephen Hanessian, Oscar M. Saavedra, Miguel A. Vilchis-Reyes, Ana M. Llaguno-Rueda

Sophie Le Trionairre, Alexis Perry, Bartosz Szczesny, Szabo Csaba, Paul Winyard, Jacqueline Whatmore, Mark E. Wood, Matt Whiteman

77) Synthesis, Antiribosomal and Antibacterial Activity of 4'-O-Glycopyranosyl Paromomycin Aminoglycoside Antibiotics (ChemMedComm) Monday April 7th 2014
Weiwei Chen, Takahiko Matsushita, Dimitri Shcherbakov, Heithem Boukari, Andrea Vasella, Erik Bottger, D Crich

78) Dimerization hot spots in the structure of human Hsp90 (ChemMedComm) Friday April 4th 2014
Giulio Rastelli

79) N1-Linked Melatonin Dimers as Bivalent Ligands Targeting Dimeric Melatonin Receptors (ChemMedComm) Friday April 4th 2014
Anne-Sophie Journe, Samy A.M. Habib, Bala R. Dodda, Mina N.F. Morcos, Mirna S. Sadek, Sarah A.A. Tadros, Paula Witt-Enderby, Ralf Jockers, Darius Paul Zlotos

80) A full conformational characterization of antiandrogen cortexolone-17α-propionate and related compounds through theoretical calculations and nuclear magnetic resonance spectroscopy (ChemMedComm) Friday April 4th 2014
Patrizia Ferraboschi, Laura Legnani, Giuseppe Celasco, Luigi Moro, Laura Ragonesi, Diego Colombo

81) Design and synthesis of membrane-targeting antibiotics: from peptides- to aminosugar-based antimicrobial cationic amphiphiles (ChemMedComm) Thursday April 3rd 2014
Ido M. Herzog, Micha Fridman

82) Elucidating structural features of an entirely carbohydrate cancer vaccine construct employing circular dichroism and fluorescent labeling (ChemMedComm) Tuesday April 1st 2014
Kevin R. Trabbic, Ravindra A. De Silva, Peter R. Andreana

83) Novel inhibitors of breast cancer relevant kinases Brk and HER2 (ChemMedComm) Monday March 31st 2014
Kazem Ahmed Mahmoud, Tom Wersig, Inna Slynko, Frank Totzke, Christoph Schachtele, Markus Oelze, Wolfgang Sippl, Christoph Ritter, Andreas Hilgeroth

84) Novel phthalimide derivatives with TNF-α and IL-1β expression inhibitory and apoptotic inducer properties (ChemMedComm) Friday March 28th 2014
Lucas Cunha Duarte Coelho, Marcos Verissimo de Oliveira Cardoso, Diogo Rodrigo Magalhaes Moreira, Paulo Andre Teixeira de Moraes Gomes, Gevanio Bezerra de Oliveira Filho, Suellen Melo Tiburcio Cavalcanti, Lucianna Rabelo Pessoa Siqueira, Miria de Oliveira Barbosa, Arsenio Rodrigues Oliveira, Elizabeth Fernanda de Oliveira Borba, Teresinha Goncalves Silva, Belinda Kaskow, Mahdad Karimi, Lawrence J Abraham, Ana Cristina Lima Leite

85) Discovery and SAR study of a sulfonamide hydroxamic acid inhibitor for the botulinum neurotoxin serotype A light chain (ChemMedComm) Friday March 28th 2014
Nicholas Salzameda, Alexander Burtea

86) Design of glycosyltransferase inhibitors targeting human O-GlcNAc Transferase (OGT) (ChemMedComm) Friday March 21st 2014
Shuai Wang, David L Shen, Dominique Lafont, Anne-Sophie Vercoutter-Edouart, Marlene Mortuaire, Yun Shi, Ofelia Maniti, Agnes Girard-Egrot, Tony Lefebvre, B Mario Pinto, David Vocadlo, Sebastien Vidal

87) Synthesis and Antimicrobial Activities of His(2-aryl)-Arg and Trp-His(2-aryl) Classes of Dipeptidomimetics (ChemMedComm) Friday March 21st 2014
Amit Mahindra, Krishna Kumar Sharma, Dinesh Rathore, Shabana Khan, Melissa Jacobs, R Jain

88) Synthesis of iminosugar derivatives presenting naphthyl and alkylamine interacting groups and binding to somatostatin receptors (ChemMedComm) Thursday March 20th 2014
Stephen Barron, Paul Murphy

89) Specific chemical changes leading to consistent potency increases in structurally diverse active compounds (ChemMedComm) Thursday March 20th 2014
Dilyana Dimova, Dagmar Stumpfe, J Bajorath

90) Discovery of small molecule inhibitors targeting the SUMO-SIM interaction using a protein interface consensus approach (ChemMedComm) Tuesday March 18th 2014
Arnout Voet, Akihiro Ito, Mikako Hirohama, Seiji Matsuoka, Naoya Tochio, Takanori Kigawa, Minoru Yoshida, Kam Y.J. Zhang

91) Scaffold hopping of potential anti-tumor agents by WEGA: a shape-based approach (ChemMedComm) Tuesday March 18th 2014
Hu Ge, Yu Wang, Wenxia Zhao, Wei Lin, Xin Yan, Jun Xu

92) Two diseases, one approach: multitarget drug discovery in Alzheimer's and neglected tropical diseases (ChemMedComm) Monday March 17th 2014
Federica Prati, Elisa Uliassi, Maria Laura Bolognesi

93) Repurposing human Aurora kinase inhibitors as leads for anti-protozoan drug discovery. (ChemMedComm) Monday March 17th 2014
Gautam Patel, Norma Roncal, Patricia Lee, Susan Leed, Jessey Erath, Ana Rodriguez, Richard Sciotti, Michael Pollastri

94) Introduction of polar groups on the naphthalene scaffold of molecular tongs inhibiting wild-type and mutated HIV-1 protease dimerization (ChemMedComm) Monday March 17th 2014
Sandrine Ongeri, Roberto Fanelli, Ana-Sofia Ressurreicao, Laure Dufau, Jean-Louis Soulier, Anamaria Vidu, Nicolo Tonali, Guillaume Bernadat, Michele Reboud-Ravaux

95) Conformational Properties of Cholic Acid, a Lead Compound at the Crossroads of Bile Acid Inspired Drug Discovery. (ChemMedComm) Monday March 17th 2014
Antimo Gioiello, Francesco Venturoni, Sara Tamimi, Chiara Custodi, Roberto Pellicciari, Antonio Macchiarulo

96) Combretastatin A-4 Inspired Novel 2-Aryl-3-arylamino-imidazo-pyridines/pyrazines as Tubulin Polymerization Inhibitors, Antimitotic and Anticancer Agents (ChemMedComm) Monday March 17th 2014
Sankar Kumar Guchhait, Nitesh Sanghai, Vaibhav Jain, Ranjan Preet, Somnath Kandekar, Sarita Das, Neha Trivedi, Purusottam Mohapatra, Garima Priyadarshani, Maneesh Kashyap, Dipon Das, Shakti Ranjan Sathapathy, Sumit Siddharth, Chanakya N. Kundu, Prasad. V. Bharatam

97) Design, synthesis and biological evaluation of novel trimethylpyrazine-2-carbonyloxy-cinnamic acids as potent cardiovascular agents (ChemMedComm) Wednesday March 12th 2014
Hongfei Chen, Guoning Li, Peng Zhan, Hong Li, Shouxun Wang, Xinyong Liu

98) Sulfonium Ions as Inhibitors of the Mycobacterial Galactofuranosyltransferase GlfT2 (ChemMedComm) Wednesday March 12th 2014
Jing Li, Todd L Lowary

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