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1) Synthesis of fusidic acid bioisosteres as antiplasmodial agents and molecular docking studies in the binding site of elongation factor-G (ChemMedComm) Tuesday October 13th 2015
Gurminder Kaur, Kawaljit Singh, Elumalai Pavadai, Mathew Njoroge, Marlene Espinoza-Moraga, Carmen De Kock, Peter J. Smith, Sergio Wittlin, Kelly Chibale

2) Patterns of Biofilm Structure and Formation Kinetics among Acinetobacter baumannii Clinical Isolates with Different Antibiotic Resistance Profiles (ChemMedComm) Tuesday October 13th 2015
Elias Dahdouh, Belen Orgaz, Rosa Gomez-Gil, Jesus Mingorance, Ziad Daoud, Monica Suarez, Carmen SanJose

3) Molecular Basis for Resistance Against Phosphonate Antibiotics and Herbicides (ChemMedComm) Monday October 12th 2015
Jonathan Chekan, Dillon P Cogan, Satish Nair

4) Thermoresponsive fluorinated small-molecule drugs: a new concept for efficient localized chemotherapy. (ChemMedComm) Thursday October 8th 2015
Paul Dyson, Catherine Clavel, Patrycja Nowak-Sliwinska, Emilia Paunescu

5) In silico-driven multicomponent synthesis of 4,5- and 1,5-disustituted imidazoles as indoleamine 2,3-dioxygenase inhibitors (ChemMedComm) Thursday October 8th 2015
Silvia Fallarini, Alberto Massarotti, Alessandro Gesu, Sara Giovarruscio, Giulia Coda Zabetta, Roberta Bergo, Barbara Giannelli, Angelo Brunco, Grazia Lombardi, Giovanni Sorba, Tracey Pirali

6) Bisimidazoline arylamides binding to the DNA minor groove. N1-hydroxylation enhances binding affinity and selectivity to AATT sites (ChemMedComm) Thursday October 8th 2015
Carlos H. Rios Martinez, Laura Lagartera, Cristina Trujillo, C Dardonville

7) Synergistic Activity of a Short Lipidated Antimicrobial Peptide (LipoAMP) and Colistin or Tobramycin against Pseudomonas Aeruginosa from Cystic Fibrosis Patients (ChemMedComm) Monday October 5th 2015
Martin de Gier, H. Bauke Albada, Michaele Josten, Rob Willems, Helen Leavis, Rosa Van Mansveld, Fernanda Paganelli, Bertie Dekker, Jan-Willem Lammers, Hans-Georg Sahl, Nils Metzler-Nolte

8) Syntheses and Biological Evaluations of Highly Functionalized Hydroxamate Containing and N-Methylthio Monobactams as Anti-Tuberculosis and β-Lactamase Inhibitory Agents. (ChemMedComm) Monday October 5th 2015
Marvin Miller, Mark Majewski, Kyle Watson, Sanghyun Cho, Patricia Miller, Scott Franzblau

9) Multi-drug delivery nanocarriers for combination therapy (ChemMedComm) Thursday October 1st 2015
Suresh Gadde

10) A Structure-Activity Relationship Study of the Positive Allosteric Modulator LY2033298 at the M4 Muscarinic Acetylcholine Receptor (ChemMedComm) Wednesday September 30th 2015
Monika Szabo, Tracey Huynh, Celine Valent, Robert Lane, Patrick Sexton, Arthur Christopoulos, Ben Capuano

11) Potentiation of Francisella resistance to conventional antibiotics through small molecule adjuvants (ChemMedComm) Wednesday September 30th 2015
Matthew D. Stephens, Veroncia B. Hubble, Robert K. Ernst, Monique L. van Hoek, Roberta J. Melander, John Cavanagh, Christian Melander

12) Discovery of Fluoroquinolone derivatives as potent, selective inhibitors of PI3Kγ (ChemMedComm) Tuesday September 29th 2015
Hai-Liang Zhu, Shao Sha, Hong-Wei Han, Fei Gao, Tian-Bao Liu, zhen li, Chi Xu, Wei-Qing Zhong

13) Ligand-based homology modelling of the human CB2 receptor SR144528 antagonist binding site: a computational approach to explore the 1,5-diaryl pyrazole scaffold (ChemMedComm) Monday September 28th 2015
Elena Cichero, Giulia Menozzi, Sara Guariento, Paola Fossa

14) Semi-synthesis and anti-tumor evaluation of novel 25-hydroxyprotopanaxadiol derivatives as apoptosis inducing agents (ChemMedComm) Friday September 25th 2015
fanzhi qu, chen zhao, yafei liu, jiaqing cao, wei li, yuqing zhao

15) Ionic liquid mediated transcutaneous protein delivery with solid-in-oil nanodispersion (ChemMedComm) Friday September 25th 2015
Shota Araki, Rie Wakabayashi, Muhammad Moniruzzaman, Noriho Kamiya, Masahiro Goto

16) Mode of Action Study of Cationic Anthraquinone Analog: A New Class of Highly Potent Anti-cancer Agent (ChemMedComm) Friday September 25th 2015
Jaya P Shrestha, Yagya Subedi, liaohai chen, Tom Chang

17) Design and synthesis of peptide inhibitor conjugates as probes of the Cytochrome P450s from glycopeptide antibiotic biosynthesis (ChemMedComm) Friday September 25th 2015
Clara Brieke, Theresa Maier, Martin Schroter, Max Cryle

18) Synthesis of indole-derived allocolchicine congeners exhibiting pronounced anti-proliferative and apoptosis-inducing properties (ChemMedComm) Tuesday September 22nd 2015
Nikolay Sitnikov, Alexander Sinzov, Diane Allegro, Pascale Barbier, Sebastien Combes, Liliane Abodo Onambele, Aram Prokop, Hans Gunther Schmalz, Alexey Fedorov

19) A synthesis, in silico, in vitro and in vivo study of thieno[2,3-b]pyridine anticancer analogues (ChemMedComm) Tuesday September 22nd 2015
John Arabshahi, Michelle van Rensburg, Lisa Pilkington, Chae Jeon, Mirae Song, Ling-Mey Gridle, Euphemia Leung, David Barker, Milena Vuica-Ross, Konstantin Volcho, Alexandra Zakharenko, Olga Lavrik, Johannes Reynisson

20) Mechanisms of Resistance to Aminoglycoside Antibiotics: Overview and Perspectives (ChemMedComm) Monday September 21st 2015
Sylvie Garneau-Tsodikova, Kristin J. Labby

21) Discovery of a potent and highly fluorescent sirtuin inhibitor (ChemMedComm) Tuesday September 15th 2015
Y. K. Yoon, M. A. Ali, A. C. Wei, T. S. Choon, A. N. Shirazi, K. Parang

22) Phase II Metabolic Pathways of Spectinamide Antitubercular Agents: A Comparative Study of the Reactivity of 4- Substituted Pyridines to Glutathione Conjugation (ChemMedComm) Monday September 7th 2015
Dora Madhura, Jiuyu Liu, Bernd Meibohm, Richard E. Lee

23) Tabtoxinine-β-Lactam is a "Stealth" β-Lactam Antibiotic that Evades β-Lactamase-mediated Antibiotic Resistance (ChemMedComm) Monday September 7th 2015
Timothy Adam Wencewicz, Kathryn Hart, Margaret Reck, Gregory Bowman

24) Rational design of promiscuous binding modulators of p53 inducing E3(Ub)-ligases (Mdm2 and Pirh2) as anticancer agents: An in silico approach (ChemMedComm) Monday September 7th 2015
Sarfaraj Niazi, Madhusudan Purohit

25) 1-[(2E)-3-phenylprop-2-enoyl]-1H-benzimidazoles as anticancer agents: Synthesis, crystal structure analysis and binding studies of the most potent anticancer molecule with serum albumin (ChemMedComm) Monday September 7th 2015
Seetharamappa J, Veerendra Kumar A Kalalbandi

26) Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement (ChemMedComm) Monday September 7th 2015
Sewan Theeramunkong, Ubaldina Galli, Ambra A Grolla, Antonio Caldarelli, Cristina Travelli, Alberto Massarotti, Maria Pia Troiani, Maria Alessandra Alisi, Giuseppe Orsomando, Armando A Genazzani, Gian Cesare Tron

27) Synthesis and Biological Evaluation of Novel 7-O-Lipophilic Substituted Baicalein Derivatives as Potential Anticancer Agents (ChemMedComm) Monday September 7th 2015
Shao-Hung Wang, C.-H. Chen, CY Lo, Ji-Zhen Feng, Hong-Jhih Lin, Po-Ya Chang, Ling-Ling Yang, Lih-Geeng Chen, Yi-Wen Liu, Cheng-Deng Kuo, Jin-Yi Wu

28) 2-[18F]Fluoroethyl tosylate - a versatile tool for building of 18F based radiotracers for positron emission tomography (ChemMedComm) Thursday September 3rd 2015
Torsten Kniess, Markus Laube, Peter Brust, Jorg Steinbach

29) The first potent diphenyl phosphonate KLK4 inhibitors with unexpected binding kinetics (ChemMedComm) Thursday September 3rd 2015
Jeroen Van Soom, Giuliana Cuzzucoli Crucitti, Rafaela Gladysz, Pieter Van der Veken, Roberto Di Santo, Ingmar Stuyver, Victoria Buck, Anne-Marie Lambeir, Viktor Magdolen, Jurgen Joossens, Koen Augustyns

30) Evaluation of binding competition and group epitopes of Acetylcholinesterase inhibitors by STD NMR, Tr-NOESY, DOSY and Molecular Docking: An old approach but new findings (ChemMedComm) Thursday September 3rd 2015
Nazish Urooj Tanoli, Sheraz Ahmad Khan Tanoli, Antonio Gilberto Ferreira, Sana Gul, Zaheer Ul Haq

31) Missing the target (ChemMedComm) Wednesday September 2nd 2015
Derek Lowe

32) Property-based characterization of kinase-like ligand space for library design and virtual screening (ChemMedComm) Wednesday September 2nd 2015
David Bajusz, Gyorgy Ferenczy, George M Keseru

33) Design, Synthesis and Bioevaluation of Tacrine Hybrids with Cinnamate and Cinnamylideneacetate Derivatives as Potential Anti-Alzheimer Drug Candidates (ChemMedComm) Wednesday September 2nd 2015
Amelia Santos, Catarina Quintanova, Rangappa S Keri, Sergio Marques, Sandra Cardoso, M L. M. Serralheiro, Maria Goncalves Fernandes

34) Supramolecular, Prodrug-based Micelles with Enzyme Regulated Release Behavior for Controlled Drug Delivery (ChemMedComm) Friday August 28th 2015
Yong-yong Li, Yu-qin Chen, Hai-qing Dong, Chun-yan Dong

35) Sulfasalazine in Ionic Liquid Form with Improved Solubility and Exposure (ChemMedComm) Wednesday August 26th 2015
Mohammad Shadid, Gabriela Gurau, Julia L. Shamshina, Bei-Ching Chuang, Shumet Hailu, Emily Guan, Swapan Chowdhury, Jing-Tao Wu, Syed A. A. Rizvi, Robert Griffin, Robin D. Rogers

36) Aryl- Imidazothiadiazole Analogues as Microtubule Disrupting Agents (ChemMedComm) Wednesday August 26th 2015
Ahmed Kamal, Subba Rao A.V., Srinivasa Reddy Telukutla, Sowjanya Polepalli, chandrakant Bagul, Vishnuvardhan MVPS, Siddiq Pasha Shaik, Nishant Jainb

37) Insights into the impact of N- and O-methylation on aqueous solubility and lipophilicity using matched molecular pair analysis (ChemMedComm) Friday August 21st 2015
Timothy John Ritchie, simon macdonald, Stephen Pickett

38) Inspired by magnolol: design of NSAIDs-based compounds with excellent anti-inflammatory effect (ChemMedComm) Friday August 21st 2015
Wenfeng Liu, Yuan Yue, Yonglian Li, Xi Zheng, Kun Zhang, Zhiyun Du

39) Novel Quinoline Derivatives as Potent In Vitro α-Glucosidase Inhibitors: In Silico Studies and SAR Predictions (ChemMedComm) Friday August 21st 2015
Muhammad Taha, Nor Ismail Ismail, Syahrul Imran, Abdul Wadood, Fazal Rahim, Muhammad Ali, Ahsfaq Rehman

40) Correction: Synthesis and antibacterial activity evaluation of C-5 side chain modified analogues of FYL-66, a potential agent against methicillin-resistant Staphylococcus aureus (ChemMedComm) Friday August 21st 2015
Xiaoyan Yang, Zicheng Li, Zhenling Wang, Zitai Sang, Haiyue Long, Jianying Tang, Tao Yang, Yuanyuan Liu, Youfu Luo

41) Navigating into chemical space between MGCD0103 and SAHA: Novel Histone Deacetylase Inhibitor as a Promising Lead (ChemMedComm) Monday August 17th 2015
Xin Zhang, Peng-Cheng Lv, Dongdong Li, weiming zhang, Hai-Liang Zhu

42) Discovery of Pyridyl-based inhibitors of Plasmodium falciparum N-myristoyltransferase (ChemMedComm) Monday August 17th 2015
Zhiyong Yu, James A Brannigan, Kaveri Rangachari, William Heal, Anthony J Wilkinson, Tony Holder, Robin J Leatherbarrow, Edward William Tate

43) Discovery of High Affinity Inhibitors of Leishmania donovani N-Myristoyltransferase (ChemMedComm) Monday August 17th 2015
Mark Rackham, Zhiyong Yu, James A Brannigan, William Heal, Daniel Paape, Victoria Barker, Anthony J Wilkinson, Deborah Smith, Robin J Leatherbarrow, Edward William Tate

44) Inhibitory effect of cytotoxic nitrogen-containing heterocyclic stilbene analogues on the VEGF protein secretion and the expression of the VEGF, hTERT and c-Myc genes (ChemMedComm) Wednesday August 12th 2015
Eva Falomir, Rosa Marti-Centelles, Juan Murga, Miguel Carda, J. Alberto Marco

45) Synthesis, in vitro and in vivo anticancer activities of novel 4-substituted 1,2-bis(4-chlorophenyl)-pyrazolidine-3,5-dione derivatives (ChemMedComm) Wednesday August 12th 2015
Xu-Yao Zhang, Yi-Fei Gu, Ting Chen, Dong-Xiao Yang, Xi-Xin Wang, Bai-Ling Jiang, Kun-Peng Shao, Wen Zhao, Cong Wang, Jun-Wei Wang, Qiu-Rong Zhang, Hong-Min Liu

46) Correction: Application of QM/MM and QM methods to investigate histone deacetylase 8 (ChemMedComm) Wednesday August 12th 2015
Duangkamol Gleeson, M. Paul Gleeson

47) Structure activity relationship of C1-C2-linker substituted 1,5-naphthyridine analogues of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-7) (ChemMedComm) Wednesday August 12th 2015
Sheo B Singh, David Kaelin, Jin Wu, Lynn Miesel, Christopher Tan, Peter Meinke, David Olsen, Armando Lagrutta, Changqing Wei, Yonggang Liao, Xuanjia Peng, Xiu Wang, Hideyuki Fukuda, Ryuta Kishii, Masaya Takei, Takeshi Shibata, Tomoko Takeuchi, Kohei Ohata, Akinori Nishimura, Yasumichi Fukuda

48) Inhibition of Phosphatidylinositol-3,4,5-trisphosphate Binding to AKT Pleckstrin Homology Domain by 4-Amino-1,2,5-oxadiazole Derivatives (ChemMedComm) Tuesday August 11th 2015
Debasis Manna, Sukhamoy Gorai, Saurav Paul, Ganga Sankaran, Manas Kumar Santra, Rituparna Borah

49) Design and discovery of 3-aryl-5-substituted-isoquinolin-1-ones as potent tankyrase inhibitors (ChemMedComm) Tuesday August 11th 2015
Richard J.R Elliott, Ashley Jarvis, Mohan B Rajasekaran, Malini Menon, Leandra Bowers, Raymond Boffey, Melanie Bayford, Stuart Firth-Clark, Rebekah Key, Rehan Aqil, Stewart B. Kirton, Dan Niculescu-Duvaz, Laura Fish, Filipa Lopes, Robert McLeary, Ines Trindade, Elisenda Vendrell, Felix Munkonge, Rod Porter, Trevor Perrior, CJ Springer, Antony Oliver, Laurence Pearl, Alan Ashworth, Christopher J. Lord

50) Isothiazolo[4,3-b]pyridines as inhibitors of cyclin G associated kinase : synthesis, structure-activity relationship studies and antiviral activity (ChemMedComm) Friday August 7th 2015
Jiahong Li, Sona Kovackova, Szuyuan Pu, Jef Rozenski, Steven De Jonghe, Shirit Einav, Piet Herdewijn

51) Correction: Design, synthesis, and evaluation of semi-conservative mono-carbonyl analogs of curcumin as anti-inflammatory agents against lipopolysaccharide-induced acute lung injury (ChemMedComm) Friday August 7th 2015
Lili Dong, Suqing Zheng, Yali Zhang, Xin Jiang, Jianzhang Wu, Xiaoqin Zhang, Xiaoou Shan, Dandan Liang, Shilong Ying, Jianpeng Feng, Guang Liang

52) Tricyclic phenothiazine and phenoselenazine derivatives as potential multi-targeting agents to treat Alzheimer's disease (ChemMedComm) Friday August 7th 2015
Gary Tin, Tarek Mohamed, Nyasha Gondora, Michael Beazely, Praveen P Nekkar Rao

53) Synthesis of carboxyimidamide-substituted benzo[c][1,2,5]oxadiazoles and their analogs, and evaluation of biological activity against Leishmania donovani (ChemMedComm) Friday August 7th 2015
Leena Keurulainen, Mikko Heiskari, Satu Nenonen, Abedelmajeed Nasereddin, Dmitry Kopelyanskiy, Teppo Leino, Jari Yli-Kauhaluoma, Charles Jaffe, Paula Kiuru

54) D1-like Receptors Distinguishing Thieno-azecine Regioisomers (ChemMedComm) Wednesday August 5th 2015
Mohamed Abdel-Fattah, Ashraf H. Abadi, J Lehmann, P. Schweikert, Christoph Enzensperger

55) C-5 Substituted Pyrido[2,3-d]pyrimidin-7-ones as Highly Specific Kinase Inhibitors Targeting Clinical Resistance related EGFRT790M Mutant (ChemMedComm) Wednesday August 5th 2015
Ke Ding, Jian Ding, Hua Xie, Meiyu Geng, Linjiang Tong, Ting Peng, zhaoyu Huang, Tianfeng Xu, xiaomei Ren, Zhengchao Tu, Lianwen Zhang, zhang zhang, xiaoyun lu, Lei Yu, Jinfeng Luo

56) Induction of apoptosis by cyclobutanones and derived polycyclic γ-lactones: a preliminary analysis of antiproliferative activity (ChemMedComm) Tuesday August 4th 2015
Vishal Sharma, Ashun Chaudhary, Gousia Chashoo, Saroj Arora, Ajit K. Saxena, Mohan Paul S. Ishar

57) Novel peptidomimetics related to Gonadotropin releasing hormone (GnRH) (ChemMedComm) Tuesday July 28th 2015
Stefania Villa, Arianna Gelain, Luca Rizzi, Laura Legnani, Aurora Pacini, Katerina Spyridaki, Vlasios Karageorgos, George Liapakis

58) Enhanced Antibacterial Activities of Polythionates by Carbonate (ChemMedComm) Thursday July 23rd 2015
Guofang Li, yanbao zhao, Ping Li, Fuqiang Zhang, Peng Qu, Binjie Li, Qingyu Gao, Shaorong Wang

59) Investigating the generation of hydrogen sulfide from the phosphonamidodithioate slow-release donor GYY4137 (ChemMedComm) Thursday July 23rd 2015
Mark E. Wood, Matt Whiteman, Benjamin Edwin Alexander, Bridget Fox, Tahmina Khan, Joseph Maliszewski, Alexis Perry, Simon Coles, Mateusz Pitak

60) Structure-based design of a bisphosphonate 5'(3')-deoxyribonucleotidase inhibitor (ChemMedComm) Thursday July 23rd 2015
Petr Pachl, Ondrej Simak, Pavlina Rezacova, Milan Fabry, Milos Budesinsky, Jiri Brynda, Ivan Rosenberg

61) Inclusion of new 5-fluorouracil derivatives in liposome formulation for cancer treatment (ChemMedComm) Thursday July 23rd 2015
Manuela Petaccia, Maria condello, Luisa Giansanti, Angela La Bella, Francesca Leonelli, stefania Meschini, denise grdella villalva, evelin pellegrini, Francesca Ceccacci, Luciano Galantini, Giovanna Mancini

62) Novel 3-hydroxypyridin-4-one hexadentate ligand-based polymeric iron chelator: synthesis, characterization and antimicrobial evaluation (ChemMedComm) Monday July 20th 2015
Yingjun Zhou, Xiaole Kong, Junpei Li, Yongmin Ma, Robert Hider, Tao Zhou

63) Fragments in bromodomain drug discovery (ChemMedComm) Monday July 20th 2015
Paul Bamborough, Chun-wa Chung

64) Novel benzoxepine-1,2,3-triazole hybrids: Synthesis and pharmacological evaluation as potential antibacterial and anticancer agents (ChemMedComm) Thursday July 16th 2015
Naveen Kuntala, Jhonsee Rani Telu, Venkanna Banothu, N Suresh Babu, Jayashree anireddy, Sarbani Pal

Ainhoa Mascaraque, Wioleta Kowalczyk, Tahia D Fernandez, Francisca Palomares, Cristobalina Mayorga, David Andreu, Javier Rojo

66) Correction: Identification of a novel class of autotaxin inhibitors through cross-screening (ChemMedComm) Tuesday July 7th 2015
Diana Castagna, Emma L. Duffy, Dima Semaan, Louise C. Young, John M. Pritchard, Simon J. F. Macdonald, David C. Budd, Craig Jamieson, Allan J. B. Watson

67) Design, synthesis and in vivo evaluation of sodium 2-benzyl-chloromalonates as new central nervous system depressants (ChemMedComm) Monday July 6th 2015
Jose Daniel Figueroa-Villar, Andreia Vieira, Bruno Marinho, Luana Souza, Patricia Fernandes

68) Correction: Discovery, synthesis and structure-activity analysis of symmetrical 2,7-disubstituted fluorenones as urea transporter inhibitors (ChemMedComm) Monday July 6th 2015
Sujin Lee, Cristina Esteva-Font, Puay-Wah Phuan, Marc O. Anderson, A. S. Verkman

69) Chemoprevention Effects of Sulindac-Based Compound on TPA-induced skin inflammation in Mice (ChemMedComm) Friday July 3rd 2015
Wenfeng Liu, Yonglian Li, Xi Zheng, kun zhang, Zhiyun Du

70) Synthesis and in vitro antiproliferative activity of novel pyrazolo[3,4-d]pyrimidine derivatives (ChemMedComm) Friday July 3rd 2015
Nermin S. Abdou, Rabah A. T. Serya, Ahmed Esmat, Mai F. Tolba, Nasser S. M. Ismail, Khaled A. M. Abouzid

71) Magic molecule modifiers (ChemMedComm) Thursday July 2nd 2015
Derek Lowe

72) The discovery of a novel antibiotic for the treatment of Clostridium difficile infections: a story of an effective academic-industrial partnership (ChemMedComm) Wednesday July 1st 2015
John Mann, Peter Taylor, Colin Dorgan, Peter Johnson, Francis X. Wilson, Richard Vickers, Aaron Dale, Stephen Neidle

73) Synthesis and anti-cancer screening of novel heterocyclic-(2H)-1,2,3-triazoles as potential anti-cancer agents (ChemMedComm) Tuesday June 30th 2015
Narsimha Penthala, Leena Maddukuri, Shraddha Thakkar, Nikhil Reddy Madadi, Gauri Lamture, Robert Eoff, Peter Crooks

74) Correction: Synthesis and biological evaluation of novel semi-conservative monocarbonyl analogs of curcumin as anti-inflammatory agents (ChemMedComm) Monday June 29th 2015
Zhe Wang, Peng Zou, Chenglong Li, Wenfei He, Bing Xiao, Qilu Fang, Wenbo Chen, Suqing Zheng, Yunjie Zhao, Yuepiao Cai, Guang Liang

75) Correction: Design, synthesis, and antibacterial evaluation of novel azolylthioether quinolones as MRSA DNA intercalators (ChemMedComm) Monday June 29th 2015
Ling Zhang, Kannekanti Vijaya Kumar, Syed Rasheed, Shao-Lin Zhang, Rong-Xia Geng, Cheng-He Zhou

76) PEGylated solid lipid nanoparticles: design, methotrexate loading and biological evaluation in animal models (ChemMedComm) Friday June 26th 2015
Dipti Kakkar, Shweta Dumoga, Rohit Kumar, Krishna Chuttani, Anil Kumar Mishra

77) Design, synthesis, and evaluation of semi-conservative mono-carbonyl analogs of curcumin as anti-inflammatory agents against lipopolysaccharide induced acute lung injury (ChemMedComm) Thursday June 25th 2015
Lili Dong, Suqing Zheng, Yali Zhang, Xin Jiang, Jianzhang Wu, Xiaoqing Zhang, Xiaoou Shan, Dandan Liang, Shilong Ying, Jianpeng Feng, Guang Liang

78) Discovery of TRAF-2 and NCK-interacting kinase (TNIK) inhibitors by ligand-based virtual screening methods (ChemMedComm) Wednesday June 24th 2015
Anna Bujak, Filip Stefaniak, Daria Zdzalik, Paulina Grygielewicz, Barbara Dymek, Marcin Zagozda, Pawel Gunerka, Monika Lamparska-Przybysz, Krzysztof Dubiel, Maciej Wieczorek, Karolina Dzwonek

79) Synthesis and anti-tubercular activity of conformationally-constrained and bisquinoline analogs of TMC207 (ChemMedComm) Tuesday June 23rd 2015
Dimpy Kalia, Anil Kumar K.S., Gajanand Meena, Kashmir Prasad Sethi, Rohit Sharma, Priyanka Trivedi, Shaheb Raj Khan, Ajay Singh Verma, Shyam Singh, Sandeep Sharma, Kuldeep K Roy, Ruchir Kant, Manju Yasodha Krishnan, Bhupendra N. Singh, Sudhir Sinha, Vinita Chaturvedi, Anil K Saxena, Dinesh K Dikshit

80) Transition Metal Diamine Complexes with Antimicrobial Activity Against Staphylococcus aureus and Methicillin-Resistant S. aureus (MRSA). (ChemMedComm) Monday June 22nd 2015
Joseph S Merola, George Karpin, David Morris, Mai Ngo, Joseph Falkinham

81) Synthesis and biological evaluation of α-sulfonamido-N-adamantanecarboxamide derivatives as 11β-HSD1 inhibitors (ChemMedComm) Thursday June 18th 2015
Young Hoon Kim, Seung Kyu Kang, Gwi Bin Lee, Kyu Myung Lee, Jaladi Ashok Kumar, Ki Young Kim, Sang Dal Rhee, Jeongmin Joo, Myung Ae Bae, Won Koo Lee, Jin Hee Ahn

82) Design and synthesis of potent and selective inhibitors of BRD9 and BRD7 bromodomains. (ChemMedComm) Monday June 15th 2015
Duncan Hay, Paul Brennan, Oleg Fedorov, Cynthia Tallant, Octovia Monteiro, Susanne Muller-Knapp, Stefan Knapp, Christopher J Schofield, Sarah Martin, Catherine Rogers

83) Identification of new hit scaffolds by INPHARMA-guided virtual screening (ChemMedComm) Monday June 15th 2015
Teresa Carlomagno, Justyna Sikorska, Luca Codutti, Lars Skjaerven, Bettina Elshorst, Rebeca Saez Ameneiro, Andrea Angelini, Peter Monecke

84) Correction: Synthesis and biological evaluation of N-(4-phenylthiazol-2-yl)cinnamamide derivatives as novel potential anti-tumor agents (ChemMedComm) Monday June 15th 2015
Yong Luo, Yongxia Zhu, Kai Ran, Zhihao Liu, Ningyu Wang, Qiang Feng, Jun Zeng, Lidan Zhang, Bing He, Tinghong Ye, Shirui Zhu, Xiaolong Qiu, Luoting Yu

85) Synthesis of novel 1-substituted triazole linked 1,2-benzothiazine 1,1-dioxido propenone derivatives as potent anti-inflammatory agents and inhibitors of monocyte-to-macrophage differentiation (ChemMedComm) Saturday June 13th 2015
B Narsaiah, Malla Reddy GANNARAPU, Sathish Babu Vasamsetti, nagender punna, Srigiridhar Kotamraju

86) Enhanced in vitro and in vivo uptake of a hydrophobic model drug coumarin-6 in the presence of cucurbit[7]uril (ChemMedComm) Friday June 12th 2015
Xiaoqing Miao, Ye Li, Ian Wyman, Simon Ming-Yuen Lee, Donal H Macartney, Ying Zheng, Ruibing Wang

87) Discovery of C-shaped aurone human neutrophil elastase inhibitors (ChemMedComm) Friday June 12th 2015
Susana Dias Lucas, Marta P. Carrasco, Lidia M. Goncalves, Rui Moreira, Rita Cardoso Guedes

88) Synthesis and biological evaluation of 4′-[(benzimidazol-1-yl) methyl] biphenyl-2-amides as dual angiotensin II and endothelin A receptor antagonists (ChemMedComm) Wednesday June 10th 2015
Xiaofeng Han, Weizhe Xue, Liping Hao, Zhiming Zhou

89) Synthesis and biological evaluation of lipid like 5-(2-hydroxyethyl)-4-methyl-1,3-thiazole derivatives as potential anticancer and antimicrobial agents (ChemMedComm) Wednesday June 10th 2015
Alla Zablotskaya, Izolda Segal, Prof. Athina Geronikaki, Galina Kazachonokh, Yuris Popelis, Irina Shestakova, Vizma Prof. Nikolajeva, Daina Eze

90) Discovery of Anilinopyrimidine-Based Naphthamide Derivatives as Potent VEGFR-2 Inhibitors (ChemMedComm) Monday June 8th 2015
Yongcong Lv, Mengyuan Li, Sufen Cao, Linjiang Tong, Ting Peng, Lixin Wei, Hua Xie, Jian Ding, Wenhu Duan

91) Identifying Farnesoid X Receptor Agonists with Naive Bayesian and Recursive Partitioning Approaches (ChemMedComm) Monday June 8th 2015
Qianzhi Ding, Chanjuan Li, Ling Wang, Yali Li, Huihao Zhou, Qiong Gu, Jun Xu

92) Novel Difluoroacetamide Analogues of Agomelatine and Melatonin: Probing the Melatonin Receptors for MT1-Selectivity (ChemMedComm) Monday June 8th 2015
Darius Paul Zlotos, Noura Riad, Mai Osman, Bala R. Dodda, Paula Witt-Enderby

93) Transcutaneous immunization against cancer using a solid-in-oil nanodispersion (ChemMedComm) Monday June 8th 2015
Yuya Hirakawa, Rie Wakabayashi, Ayaka Naritomi, Masato Sakuragi, Noriho Kamiya, Masahiro Goto

94) Effect of dibucaine hydrochloride on raft-like lipid domains in model membrane systems (ChemMedComm) Monday June 8th 2015
Kazunari Yoshida, Akito Takashima, Izumi Nishio

95) Discovery, synthesis and structure-activity analysis of symmetrical 2,7-disubstituted fluorenones as urea transporter inhibitors (ChemMedComm) Friday June 5th 2015
Sujin Lee, Cristina Esteva-Font, Puay-wah Phuan, Marc O. Anderson, Alan S. Verkman

96) RGD-peptides modifying dexamethasone: To enhance the efficacy of anti-inflammation and limit the risk of osteoporosis (ChemMedComm) Thursday June 4th 2015
Hualong Yu, Shenghui Mei, Zhao Li, Ming Zhao, Yuji Wang, Haimei Zhu, Yaonan Wang, Jianhui Wu, Chunying Cui, Wenyun Xu, Shiqi Peng

97) Substituted 4-hydroxy-1,2,3-triazoles: synthesis, characterization and first drug design applications through bioisosteric modulation and scaffold hopping approaches (ChemMedComm) Thursday May 28th 2015
Agnese Chiara Pippione, Franco Dosio, Alex Ducime, Antonella Federico, Katia Martina, Stefano Sainas, Bente Frolund, Major Gooyit, Kim D Janda, Donatella Boschi, Marco Lucio Lolli

98) Identifying the inhibitory mechanism of apigenin on the insulin ligand-receptor binding (ChemMedComm) Wednesday May 27th 2015
Yong Yang

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