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1) Exploring cinnamic acid scaffold: development of promising neuroprotective lipophilic antioxidants (ChemMedComm) Wednesday April 15th 2015
Fernanda Borges, Daniel Chavarria, Tiago Silva, Teresa Summavielle, Jorge M.P.J. Garrido, Daniel Martins, Joana Bravo

2) Synthesis and Biological Evaluation of N-(4-phenylthiazol-2-yl) Cinnamamide Derivatives as Novel Potential Anti-tumor Agents (ChemMedComm) Monday April 13th 2015
Yong Luo, Yongxia Zhu, Kai Ran, Zhihao Liu, Ningyu Wang, Qiang Feng, Jun Zeng, Lidan Zhang, Bing He, Tinghong Ye, Shirui Zhu, Xiaolong Qiu, Luoting Yu

3) Direct photocapture of bromodomains using tropolone chemical probes (ChemMedComm) Monday April 13th 2015
Erik Hett, Eugene Chekler, Arindrajit Basak, Paul Bonin, Aldrin Denny, Andrew Flick, Kieran F Geoghegan, Shenping Liu, Mathew Pletcher, Parag Sahasrabudhe, Shores Salter, Ingrid Stock, Alex Taylor, Lyn H Jones

4) Discovery of a series of 2-(pyridinyl)pyrimidines as potent antagonists of GPR40 (ChemMedComm) Wednesday April 8th 2015
M J Waring, David Baker, Stuart Bennett, Alastair Dossetter, Mark Fenwick, Rob Garcia, Jennie Georgsson, Sam Groombridge, Sue Loxham, Philip Alexander MacFaul, Katie Maskill, David Morgan, Jenny Morrell, Helen Pointon, Graeme Robb, David Smith, Stephen Stokes, Gary Paul Wilkinson

5) Synthesis and Biological Evaluations of 2,3-Diarylthiophene Analogues of Combretastatin A-4 (ChemMedComm) Thursday April 2nd 2015
Weige Zhang, Zhan Wang, qingkun Yang, Zhaoshi Bai, Jun Sun, xuewei Jiang, Hongrui Song, Yingliang Wu

6) New substituted 9-propyladenine derivatives as adenosine receptor antagonists (ChemMedComm) Thursday April 2nd 2015
Catia Lambertucci, Michela Buccioni, Diego Dal Ben, Sonja Kachler, Gabriella Marucci, Andrea Spinaci, Ajiroghene Thomas, Karl-Norbert Klotz, R Volpini

7) Enantiomeric Diketopiperazines: Getting Insight of the Impact of the Configuration to the Conformation, Nanoimage, u-PA Inhibition and Anti-metastatic Activity (ChemMedComm) Tuesday March 31st 2015
Feng Wang, Shan Li, Yuji Wang, Haimei Zhu, Xiaoyi Zhang, Ming Zhao, Jianhui Wu, Shiqi Peng

8) Chemical genomics reveals novel biological activity of 1,2,3-dithiazoles as potent and reversible melanin synthesis inhibitors (ChemMedComm) Tuesday March 31st 2015
Panayiotis Andreas Koutentis, Paris Skourides, Oleg Alekseevich Rakitin, Anna Charalambous, Maria Koyioni, Ioanna Antoniades, Sophia Michaelidou, Iro Eleftheriou, Stanislav A Amelichev, Lidia S konstantinova, Despoina Pegeioti

9) Correction: Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday March 31st 2015
Taha M. A. Eldebss, Sobhi M. Gomha, Mohamed M. Abdulla, Reem K. Arafa

10) Structure-Based Virtual Screening for Fragment-Like Ligands of the G Protein-Coupled Histamine H4 Receptor (ChemMedComm) Monday March 30th 2015
Enade P. Istyastono, Albert J. Kooistra, Henry Vischer, Martien Kuijer, Luc Roumen, Saskia Nijmeijer, Rogier Smits, Iwan de Esch, Rob Leurs, Chris de Graaf

11) Novel synthesis of fluorochrome-coupled zoledronate with preserved functional activity on gamma/delta T cells and tumor cells (ChemMedComm) Monday March 30th 2015
Vijayanand Chandrasekaran, Shirin Kalyan, Valentina Biehl, Marcus Lettau, Patrik Theodor Nerdal, Hans-Heinrich Oberg, Daniela Wesch, Thisbe K Lindhorst, Dieter Kabelitz

12) Discovery of 2-(5,6-dimethoxypyridin-3-yl)-4-(2,4,6-trifluorobenzyl)-2H-pyrido[2,3-e][1,2,4]thiadiazin-3(4H)-one 1,1-dioxide (HTL6641), a dual orexin receptor antagonist with differentiated pharmacodynamic properties.[dagger] (ChemMedComm) Monday March 30th 2015
John Andrew Christopher, Sarah Aves, Jason Brown, James Errey, Suki Klair, Christopher Langmead, Oliver Mace, Richard Mould, Jayesh Patel, Ben Tehan, Andrei Zhukov, Fiona Marshall, Miles Congreve

13) Design of pyrazolo-pyrimidines as 11β-HSD1 inhibitors through optimisation of molecular electrostatic potential (ChemMedComm) Monday March 30th 2015
Graeme Robb, Scott Boyd, Christopher Davies, Alexander Dossetter, Frederick W Goldberg, Paul D Kemmitt, James Scott, John Swales

14) Concise Synthesis of Spergualin-Inspired Molecules With Broad-Spectrum Antibiotic Activity (ChemMedComm) Monday March 30th 2015
Victoria Assimon, Hao Shao, Sylvie Garneau-Tsodikova, Jason E. Gestwicki

15) 4-methyl-coumarins with cytotoxic activity against T24 and RT4 human bladder cancer cell lines (ChemMedComm) Thursday March 26th 2015
DAMIANA DA ROCHA VIANNA, LEILA Ruschel, FABRICIA Dietrich, Fabricio Figueiro, Fernanda Morrone, Romulo F. S. Canto, Flavia Corvello, Alice Velho, Allan Crestani, Helder Teixeira, Gilsane Lino von Poser, Ana Maria Oliveira Battastini, Vera Eifler-Lima

16) Tantalising technology (ChemMedComm) Tuesday March 24th 2015
Derek Lowe

17) Synthesis of a new HYNIC-DAPI derivative for labelling with 99mTechnetium and its in vitro evaluation in an FRTL5 cell line (ChemMedComm) Monday March 23rd 2015
Sandra Ferl, Gerd Wunderlich, Rene Smits, Alexander Hoepping, Anne Naumann, Jorg Kotzerke

18) Interactive articles in MedChemComm - connecting readers to a wealth of data and information (ChemMedComm) Thursday March 19th 2015
Richard Kelly

19) Insights into a defined secondary binding region on β-adrenoceptors and putative roles in ligand binding and drug design (ChemMedComm) Thursday March 12th 2015
Marvin Antonio Soriano-Ursua, Jose G Trujillo-Ferrara, Jose A Arias-Montano, Rafael Villalobos-Molina

20) Synthesis and evaluation of anticancer activity of novel andrographolide derivatives (ChemMedComm) Monday March 9th 2015
Devendar Ponnam, Lakshma Nayak V, Dharmendra Yadav, Niranjana Kumar Arigari, Kotesh Kumar Jonnala, Satya Srinivas KVN, Sridhar Balasubramanian, Feroz Khan, Pandu Sastry Kakaraparthi, Ramakrishna Sistla

21) Contributors to 'New Talent: Asia-Pacific' (ChemMedComm) Monday March 9th 2015


22) Membrane-interacting properties of the functionalised fatty acid moiety of muraymycin antibiotics (ChemMedComm) Friday March 6th 2015
Oliver Ries, Christian Carnarius, Claudia Steinem, Christian Ducho

23) In silico study on aging and reactivation processes of tabun conjugated AChE (ChemMedComm) Monday March 2nd 2015
Nellore Bhanu Chandar, Rabindranath Lo, Manoj K Kesharwani, Bishwajit Ganguly

24) Design, synthesis and biological evaluation of thiourea and nicotinamide-containing sorafenib analogs as antitumor agents (ChemMedComm) Monday March 2nd 2015
Xiangkai Kong, Zeyu Yao, Zuopeng He, Wen-Fang Xu, Jianwen Yao

25) Novel non-substrate modulators of the transmembrane efflux pump P-glycoprotein (ABCB1) (ChemMedComm) Friday February 27th 2015
Soren Krawczyk, Christiane Baumert, Josef Molnar, Christoph Ritter, Jens Hopner, Charlotte Kloft, Andreas Hilgeroth

26) Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday February 17th 2015
Taha Eldebss, Sobhi Gomha, Mohamed Abdalla, Reem Arafa

27) Matrix-immobilized yeast for large-scale production of recombinant human lactoferrin (ChemMedComm) Tuesday February 17th 2015
Chun Loong Ho, In Young Hwang, Kathy Loh, Matthew Chang

28) Synthesis and evaluation of amide, sulfonamide and urea - benzisoxazole derivatives as potential atypical antipsychotics (ChemMedComm) Friday February 13th 2015
Yin Chen, Yu Lan, Xudong Cao, Xiangqing Xu, Juecheng Zhang, Minquan Yu, Xin Liu, Bifeng Liu, Guisen Zhang

29) Synthesis and protective effect of new ligustrazine derivatives against CoCl2-induced neurotoxicity in differentiated PC12 cells. Part 2 (ChemMedComm) Thursday February 12th 2015
Bing Xu, Yan Gong, Xin Xu, Chenze Zhang, Yuzhong Zhang, Fuhao Chu, Hongbing Liu, Penglong Wang, Haimin Lei

30) BODIPY appended copper(II) complexes of curcumin showing mitochondria targeted remarkable photocytotoxicity in visible light (ChemMedComm) Thursday February 12th 2015
Akhil R Chakravarty, Arnab Bhattacharyya, Akanksha Dixit, Koushambi Mitra, Samya Banerjee, Anjali A Karande

31) Synthesis and biological evaluation of novel [capital Delta]2-isoxazoline fused cyclopentane derivatives as potential antimicrobial and anticancer agents (ChemMedComm) Wednesday February 11th 2015
Nagendra Babu Bathini, Santosh Kumar Prajapti, Shweta Shrivastava, Umesh Bihade, Ajay Kumar Gupta, V.G. M Naidu, Uttam Chand Banerjee

32) Evaluation of the anti-inflammatory/chondroprotective activity of aldose reductase inhibitors in human chondrocyte cultures (ChemMedComm) Wednesday February 4th 2015
Annamaria Panico, Rosanna Maccari, Venera Cardile, Sergio Avondo, Lucia Crasci, Rosaria Ottana

33) Inhibition of Insulin Amyloid Fibrillization by Glyco-Acridines: In vitro and in silico study (ChemMedComm) Wednesday February 4th 2015
Quan Van Vuong, Zuzana Bednarikova, Andrea Antosova, Huy Dinh Quoc Pham, Katarina Siposova, Nguyen Anh Tuan, Mai Suan Li, Zuzana Gazova

34) Application of QM/MM and QM methods to investigate histone deacetylase 8 (ChemMedComm) Monday February 2nd 2015
Duangkamol Gleeson, M. Paul Gleeson

35) Structure-Based Design, Synthesis by Click Chemistry and in Vivo Activity of Highly Selective A3 Adenosine Receptor Agonists (ChemMedComm) Monday February 2nd 2015
Dilip Tosh, Silvia Paoletta, Zhoumou Chen, Steven Crane, John Lloyd, Zhan-Guo Gao, Elizabeth Gizewski, John Auchampach, Daniela Salvemini, Kenneth A. Jacobson

36) Synthesis and evaluation of a series of resveratrol analogues as potent anticancer agents that target tubulin (ChemMedComm) Friday January 30th 2015
Nikhil Reddy Madadi, Hongliang Zong, Amit Ketkar, Zhen Chen, Narsimha Penthala, Venumadhav Janganati, Shobanbabu Bommagani, Robert Eoff, Monica Guzman, Peter Crooks

37) Design, Facile Synthesis and Anthelmintic Activity of New O-Substituted 6-Methoxybenzothiazole-2-carbamates (ChemMedComm) Tuesday January 27th 2015
A. Mohsen M.E. Omar, Omaima M. Aboulwafa, Doaa A. E. Issa, May M.S. El-Shokrofy, May E. Amr, Ibrahim M. El-Ashmawy

38) BEYOND THE AFFINITY FOR PROTEIN KINASE C: EXPLORING 2-PHENYL-3-HYDROXYPROPYL PIVALATE ANALOGUES AS C1 DOMAIN-TARGETING LIGANDS (ChemMedComm) Monday January 26th 2015
Daniela Rossi, Virpi Talman, Gustav Boije, Annamaria Marra, pietro Picconi, Rita Nasti, Massimo Serra, ANN JIHYAE, Marialaura Amadio, Alessia Pascale, Jeewoo Lee, Raimo Tuominen, Jari Yli-Kauhaluoma, Simona Collina

39) Correction: Identification of tris-(phenylalkyl)amines as new selective h5-HT2B receptor antagonists (ChemMedComm) Friday January 23rd 2015
Shashikanth Ponnala, Nirav Kapadia, Wayne Wesley Harding

40) Identification of Camphor Derivatives as Novel M2 Ion Channel Inhibitors of Influenza A Virus (ChemMedComm) Monday January 19th 2015
Xin Zhao, Zhen-Wei Zhang, Wei Cui, Shengwei Chen, Yang Zhou, Jianghong Dong, Yanling Jie, Junting Wan, Yong Xu, Wenhui Hu

41) O-Benzoyl Pyridine Aldoxime and Amidoxime Derivatives: Novel Efficient DNA Photo-Cleavage Agents (ChemMedComm) Thursday January 15th 2015
PARASKEVI KARAMTZIOTI, ASTERIOS PAPASTERGIOU, JOHN G. STEFANAKIS, ALEXANDROS E. KOUMBIS, IOANNA ANASTASIOU, MARIA KOFFA, KONSTANTINA C. FYLAKTAKIDOU

42) Nature of the Charged Head Group Dictates the Anticancer Potential of Lithocholic Acid-Tamoxifen Conjugates For Breast Cancer Therapy (ChemMedComm) Wednesday January 14th 2015
Kavita Yadav, Priyanshu Bhargava, Sandhya Bansal, Manish Singh, Siddhi Gupta, Geeta Sandhu, Sandeep Kumar, Vedagopuram Sreekanth, Avinash Bajaj

43) Targeted Photoresponsive TiO2-Coumarin nanoconjugate for efficient Combination therapy in MDA-MB-231 breast cancer cells: Synergic effect of Photodynamic Therapy (PDT) and Anticancer drug Chlorambucil (ChemMedComm) Wednesday January 14th 2015
Moumita Ganguly, Sourav K. Mukhopadhyay, Karthik S, Sharabani Barman, Pradeep N.D. Singh

44) Radiosynthesis of high affinity fluorine-18 labeled GnRH peptide analogues: in vitro studies and in vivo assessment of brain uptake in rats (ChemMedComm) Monday January 12th 2015
Dag Erlend Olberg, Sven H Hausner, Nadine Bauer, Jo Klaveness, Bard Indrevoll, Finn Olav Levy, Kjetil Wessel Andressen, Marie Dahl, Julie L. Sutcliffe, Ira Haraldsen

45) Design, synthesis and biological activity of 4′-[(benzimidazol-1-yl)methyl] biphenyl-2-sulphonamides as dual angiotensin II and endothelin A receptor antagonists (ChemMedComm) Monday January 12th 2015
Liping Hao, Weizhe Xue, Xiaofeng Han, Xing He, Jun Zhang, Zhiming Zhou

46) Activity Based Probes as Molecular Tools for Biomarker Discovery (ChemMedComm) Friday January 9th 2015
Luis Carvalho, Susana Dias Lucas, Eduardo Ruivo, Rui Moreira

47) Cytotoxic potential of di-spirooxindolo/acenaphthoquino andrographolide derivatives against MCF7 cell lines (ChemMedComm) Thursday January 8th 2015
Debanjana Chakraborty, Arindam Maitya, Chetan Kumar Jain, Abhijit Hazra, Yogesh Pandharinath Bharitkar, Tarun Jha, Hemanta Majumder, Susanta Roy Choudhury, Nirup Bikash Mondal

48) Dimethylaminoethyl Methacrylate Copolymer-siRNA nanoparticles for silencing therapeutically relevant gene in macrophages (ChemMedComm) Monday January 5th 2015
Ratnesh Jain, Prajakta Dandekar, Brigitta Loretz, Marcus Koch, C-M. lehr

49) Structure-activity relationship study on senktide for development of novel potent neurokinin-3 receptor selective agonists (ChemMedComm) Monday January 5th 2015
Ryosuke Misu, Koki Yamamoto, Ai Yamada, Taro Noguchi, Hiroaki Ohno, Takashi Yamamura, Hiroaki Okamura, Fuko Matsuda, Satoshi Ohkura, Shinya Oishi, Nobutaka Fujii

50) Synthesis and biological evaluation of pentanedioic acid derivatives as farnesyltransferase inhibitors (ChemMedComm) Monday January 5th 2015
liuqing Yang, wei liu, Hanbin Mei, yuan Zhang, Xiaojuan Yu, yufang xu, Honglin Li, Jin Huang, Zhenjiang Zhao

51) Recent discoveries and developments of Androgen Receptor based therapy for Prostate Cancer (ChemMedComm) Monday January 5th 2015
Ramakrishnan Elancheran, V.L Maruthanila, M Ramanathan, S Kabilan, R Devi, A Kunnumakara, Jibon Kotoky

52) Chemical space is big. Really big (ChemMedComm) Monday January 5th 2015
Derek Lowe

53) Discovery of Highly Potent Triazole Antifungal Agents with Piperdine-oxadiazole Side Chains (ChemMedComm) Wednesday December 24th 2014
Xiaomeng He, Yan Jiang, Yongqiang Zhang, Shanchao Wu, Guoqiang Dong, Na Liu, Yang Liu, Jianzhong Yao, Zhenyuan Miao, Yan Wang, Wannian Zhang, Chunquan Sheng

54) The Natural Product Brartemicin is a High Affinity Ligand for the Carbohydrate-Recognition Domain of the Macrophage Receptor Mincle (ChemMedComm) Tuesday December 23rd 2014
Kristian Mark Jacobsen, Ulrik Keiding, Lise Lindkvist Clement, Eva Susanne Schaffert, Neela Rambaruth, Mogens Johannsen, Kurt Drickamer, Thomas Bjornskov Poulsen

55) Inhibition of Influenza H5N1 invasion by modified heparin derivatives (ChemMedComm) Tuesday December 23rd 2014
Mark A. Skidmore, Anna Kajaste-Rudnitski, Nicola Wells, Scott Guimond, Timothy Rudd, Eliza Vicenzi, Edwin Yates

56) Pyrrole- and indole-containing tranylcypromine derivatives as novel lysine-specific demethylase 1 inhibitors active on cancer cells (ChemMedComm) Tuesday December 23rd 2014
Veronica Rodriguez, Sergio Valente, Stefano Rovida, Dante Rotili, Giulia Stazi, Alessia Lucidi, Giuseppe Ciossani, Andrea Mattevi, Oronza Botrugno, Paola Dessanti, Ciro Mercurio, Paola Vianello, Saverio Minucci, mario varasi, Antonello Mai

57) Enantiomeric resolution of [(2,2-diphenyl-1,3-dioxolan-4-yl)methyl](2-phenoxyethyl)amine, a potent α 1 and 5HT1A receptors ligand: an In Vitro and Computational Study (ChemMedComm) Tuesday December 23rd 2014
Livio Brasili, Silvia Franchini, Annamaria Baraldi, Claudia Sorbi, Federica Pellati, Elena Cichero, Umberto M. Battisti, Piero Angeli, Antonio Cilia

58) Synthesis and relationship of stability and biological activity of new DSS and TMP conjugates (ChemMedComm) Monday December 22nd 2014
Yewei Sun, Zicheng Tan, Zhibin Liang, Liang Wang, Luchen Shan, Pei Yu, Simon MingYuen Lee, Yuqiang Wang

59) Synthesis and antibacterial activity of trivalent ultrashort Arg-Trp-based antimicrobial peptides (AMPs) (ChemMedComm) Monday December 22nd 2014
Barbara C. Hoffknecht, H. Bauke Albada, Marina Sturm, Pascal Prochnow, Julia E. Bandow, Nils Metzler-Nolte

60) Non-nucleoside anti-HBV agents: Advances in structural optimization and mechanism of action investigations (ChemMedComm) Tuesday December 16th 2014
Na Liu, Diwakar Rai, Fabao Zhao, Haiyong Jia, Peng Zhan, Xinyong Liu

61) Discovery of a new class of histone deacetylase inhibitors with a novel zinc binding group (ChemMedComm) Tuesday December 16th 2014
Youxuan Li, Patrick M. Woster

62) The chemistry and pharmacology of privileged pyrroloquinazolines (ChemMedComm) Monday December 15th 2014
Bo Chao, Bingbing X Li, Xiangshu Xiao

63) Synthesis of six mexiletine derivatives with isoindolines attached as potential antioxidants and their evaluation as cardioprotective agents (ChemMedComm) Monday December 15th 2014
W Roy Jackson, Anh Chau, Grant Drummond, Bevyn Jarrott, Alyson Miller, Kamani Subasinghe, Christina Yan Ru Tan, Paul J White, Christine E Wright, James Ziogas

64) Solid- and solution-phase-based library of 2β-methyl substituted penicillin derivatives. Effects on growth inhibition of tumor cell lines (ChemMedComm) Monday December 15th 2014
Dora B. Boggian, Patricia Cornier, Ernesto Mata, Viviana Blanck, Mariano Cardenas, LP Roguin

65) Identification of tris-(phenylalkyl)amines as new selective h5-HT2B receptor antagonists (ChemMedComm) Monday December 15th 2014
Wayne Harding, Shashikanth Ponnala, Nirav Kapadia

66) Photoswitching property of hairpin ODNs with azobenzene derivatives in the loop (ChemMedComm) Monday December 15th 2014
Li Wu, Ya Wu, Hongwei Jin, Liangren Zhang, Yujian He, XinJing Tang

67) Synthesis and evaluation of 6-methylcoumarin derivatives as potent and selective Monoamine Oxidase B inhibitors (ChemMedComm) Monday December 15th 2014
Jin-Shuai Lan, Long-Fei Pan, Sai-Sai Xie, Xiao-Bing Wang, Ling-Yi Kong

68) Naturally occurring FANCF-Hes1 complex inhibitors from Wrightia religiosa (ChemMedComm) Thursday December 11th 2014
Midori A. Arai, Kenji Uemura, Nozomi Hamahiga, Naoki Ishikawa, Takashi Koyano, Thaworn Kowithayakorn, Tagrid Kaddar, Madeleine Carreau, Masami Ishibashi

69) Correction: Design and chemoproteomic functional characterization of a chemical probe targeted to bromodomains of BET family proteins (ChemMedComm) Monday December 8th 2014
Jiang Wu, Julia Shin, Cara M. M. Williams, Kieran F. Geoghegan, Stephen W. Wright, David C. Limburg, Parag Sahasrabudhe, Paul D. Bonin, Bruce A. Lefker, Simeon J. Ramsey

70) Relating Caco-2 permeability to molecular properties using block relevance analysis (ChemMedComm) Monday December 8th 2014
Tim Potter, G Caron, Giuseppe Ermondi, Gayle Newbury

71) Design, synthesis and biological evaluation of imidazopyridine/imidazopyrimidine-benzimidazole conjugates as potential anticancer agents (ChemMedComm) Wednesday December 3rd 2014
Ahmed Kamal, Bharath Kumar G, Lakshma Nayak V, Santhosh Reddy Vangala, Anver Basha Shaik, Rajender Rajender, Kashi Reddy Methuku

72) Synthesis and cytostatic activity of 7-arylsulfanyl-7-deazapurine bases and ribonucleosides (ChemMedComm) Tuesday December 2nd 2014
Martin Klecka, Lenka Slavetinska, Eva Tloustova, Petr Dzubak, Marian Hajduch, Michal Hocek

73) Synthesis of 17-membered azalides from a 16-membered macrolide utilizing amide-selective silane reduction (ChemMedComm) Tuesday December 2nd 2014
Atsushi Seki, Toshihiro Mori, Kouji Sasaki, Yoshiaki Takahashi, Toshiaki Miyake, Yuzuru Akamatsu

74) 3-(2,6-Dichloro-benzyloxy)-11-oxo-olean-12-ene-29-oic acid, a semisynthetic derivative of glycyrrhetic acid: Synthesis, antiproliferative, apoptotic and anti-angiogenesis activity (ChemMedComm) Monday December 1st 2014
Rajni Sharma, Santosh Guru, Shreyans K Jain, Anup S Pathania, Ram A Vishwakarma, Shashi Bhushan, Sandip Bibishan Bharate

75) Discovery of novel 5-fluoro-N2,N4-diphenylpyrimidine-2,4-diamines as potent inhibitors against CDK2 and CDK9 (ChemMedComm) Friday November 28th 2014
Jiadi Gao, Cheng Fang, Zhiyan Xiao, Li Huang, Chin Ho Chen, Li-Ting Wang, Kuo-Hsiung Lee

76) Recent advances in molecular imaging probes for β-amyloid plaques (ChemMedComm) Tuesday November 25th 2014
Masahiro Ono, Hideo Saji

77) Design, synthesis and evaluation of QD-DTC-BisBiotin Nanobioconjugate as a potential Optical-SPECT imaging agent (ChemMedComm) Friday November 21st 2014
Narmada Bag, Rashi Mathur, Sweta Singh, Firasat Hussain, Ramprakash Chauhan, krishna Chuttani, Anil K Mishra

78) 4-Thiazolidinone derivatives as potent antimicrobial agents: microwave-assisted synthesis, biological evaluation and docking studies (ChemMedComm) Wednesday November 19th 2014
Eleni Pitta, Evangelia Tsolaki, Athina Geronikaki, Jovana Petrovic, Jasmina Glamoclija, Marina Sokovic, Emmanuele Crespan, Giovanni Maga, Shome S. Bhunia, Anil K. Saxena

79) Evaluation of aromatic 6-substituted thienopyrimidines as scaffolds against parasites that cause trypanosomiasis, leishmaniasis, and malaria. (ChemMedComm) Friday November 14th 2014
Jennifer Woodring, Gautam Patel, Jessey Erath, Ranjan Behera, Patricia Lee, Susan Leed, Ana Rodriguez, Richard Sciotti, Kojo Mensa-Wilmot, Michael Pollastri

80) Exclusive Formation of Imino [4+4] cycloaddition Products with Biologically Relevant Amines: Plausible Candidates of Acrolein Biomarkers and Biofunctional Modulators (ChemMedComm) Friday November 14th 2014
Ayumi Tsutsui, Ambara R. Pradipta, Elena Saigitbatalova, Almira Kurbangalieva, Katsunori Tanaka

81) Cytotoxic Peptide Conjugates of Dinuclear Arene Ruthenium Trithiolato Complexes (ChemMedComm) Wednesday November 12th 2014
Federico Giannini, Marco Bartoloni, Lydia E. H. Paul, Georg Suss-Fink, Jean-Louis Reymond, Julien Furrer

82) Novel β-carboline-quinazolinone hybrid as inhibitor of Leishmania donovani Trypanothione Reductase: Synthesis, molecular docking and bioevaluation (ChemMedComm) Tuesday November 4th 2014
Shikha S. Chauhan, Shashi pandey, Rahul Shivahare, Karthik Ramalingam, Shagun Krishna, Preeti Vishwakarma, M. I. Siddiqi, Suman Gupta, Neena Goyal, PMS Chauhan

83) Potent chemical chaperone compounds for GM1-gangliosidosis: N-substituted (+)-conduramine F-4 derivatives (ChemMedComm) Tuesday November 4th 2014
Shinichi Kuno, Katsumi Higaki, Atsushi Takahashi, Eiji Namba, Seiichiro Ogawa

84) Decorated 6,6',7,7'-tetrahydro-1H,1'H-2,3'-biindole scaffold as promising candidate for recognition of CDK2 allosteric site (ChemMedComm) Monday November 3rd 2014
Maria Teresa Sciortino, Angela Scala, Antonio Rescifina, Ivana Colao, Gabriel Siracusano, Antonino Mazzaglia, Ugo Chiacchio, Giovanni Grassi

85) Virtual screening for novel Atg5-Atg16 complex inhibitors for autophagy modulation (ChemMedComm) Monday November 3rd 2014
Elizabeth Robinson, Euphemia Leung, Anna Matuszek, Niels Krogsgaard-Larsen, Daniel Furkert, Margaret A Brimble, Alan Richardson, Johannes Reynisson

86) Antimicrobial spine-bone cement with caffeic acid phenethyl ester for controlled release formulation and in vivo biological assessments (ChemMedComm) Monday November 3rd 2014
Hye Sun Lee, Jeong Ho Chang

87) Design, synthesis and anticancer mechanistic studies of linked azoles (ChemMedComm) Friday October 31st 2014
Amirul Islam, Yuqi Zhang, Yao Wang, Shelli Renee McAlpine

88) Probing cytochrome P450-mediated activation with a truncated azinomycin analogue (ChemMedComm) Wednesday October 22nd 2014
Victoria Vinader, Maria Sadiq, Mark Sutherland, Mengying Huang, Paul Loadman, Lina Elsalem, Steve Shnyder, Hongjuan Cui, Kamyar Afarinkia, Mark Searcey, L H Patterson, Klaus Pors

89) Study of a D-proline peptidomimetic inhibitor of melanoma and endothelial cells invasion through activity towards MMP-2 and MMP-9 (ChemMedComm) Tuesday October 21st 2014
Francesca Bianchini, Chiara Calugi, Jessica Ruzzolini, Gloria Menchi, Lido Calorini, Antonio Guarna, Andrea Trabocchi

90) Polymeric Micelles for Hydrogen Sulfide Delivery (ChemMedComm) Tuesday October 21st 2014
Urara Hasegawa, Andre J van der Vlies

91) Synthesis and Biological Evaluation of novel derivatives of Gambogenic acid as Anticancer Agent (ChemMedComm) Friday October 17th 2014
Liqin He, Peng Huang, Zhong Hu, Xiaoshan Wang, Yaxian Wu

92) Synthesis, 3D pharmacophore, QSAR and docking studies of novel quinazoline derivatives with nitric oxide release moiety as preferential COX-2 inhibitors (ChemMedComm) Friday October 17th 2014
Doaa Boshra Farag, Nahla Ahmed Farag, Ahmed Esmat, Sally A. Abuelezz, Eman Abdel-Salam Ibrahim, Dalal A. Abou El Ella

93) Synthesis, Structure-Activity Relationship, and Mechanistic Investigation of Lithocholic Acid Amphiphiles for Colon Cancer Therapy (ChemMedComm) Wednesday October 15th 2014
Manish Singh, Sandhya Bansal, Somanath Kundu, Priyanshu Bhargava, Ashima Singh, Rajender Motiani, Radhey Shyam, Vedagopuram Sreekanth, Sagar Sengupta, Avinash Bajaj

94) Towards understanding cell penetration by stapled peptides (ChemMedComm) Tuesday October 14th 2014
Qian Chu, Raymond E. Moellering, Gerard J. Hilinski, Young-Woo Kim, Tom N. Grossmann, Johannes T.-H. Yeh, Gregory L. Verdine

95) Synthesis of new betulinic acid-peptide conjugates and in vivo and in silico studies of the influence of peptide moieties on the triterpenoid core activity (ChemMedComm) Monday October 13th 2014
Valentine Nenajdenko, Anastasiya Govdi, Nadezhda Sokolova, Irina Sorokina, Sergey Vasilevsky, Dmitry Baev, Tatyana Tolstikova, Victor Mamatyuk, Dmitry Fadeev

96) Poly-α,β-aspartyl-Arg-Gly-Asp-Phe: A novel polymeric nanomedicine (ChemMedComm) Monday October 13th 2014
Shuangling Chen, Yuji Wang, Shan Li, Yaonan Wang, Ming Zhao, Haimei Zhu, Jianhui Wu, Shiqi Peng

97) Synthesis and biological evaluation of a new class of quinazolinone azoles as potential antimicrobial agents and their interactions with calf thymus DNA and Human Serum Albumin (ChemMedComm) Wednesday October 8th 2014
Cheng-He Zhou, Li-Ping Peng, Nagarajan Sangaraiah, RASHEED SYED

98) Synthesis and Evaluation of Phenoxymethylbenzamide Analogues as Anti-Trypanosomal Agents (ChemMedComm) Wednesday October 8th 2014
Richard James Payne, Alexandra Manos-Turvey, Emma Watson, Vicky Mary Avery, Amy Jones, Melissa Sykes, Jonathan D. Baell, Marcel Kaiser

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04/17/15 PHD comic: 'Teaching Pet Peeves, Part 1'

A Farewell To Messenger

Check out our trailer of CHF’s new video about Gordon Moore and...

Stopped For Efficacy - Again

You Have One Minute

UC Berkeley’s Graham Fleming Resigns Vice Chancellor Post

Draft Bill May Pave Path For Reform Of Federal Chemical Control Law

That Can't Be Right


Mitch Andre Garcia's Chem Feeds 2008-present

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