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1) Correction: Identification of tris-(phenylalkyl)amines as new selective h5-HT2B receptor antagonists (ChemMedComm) Friday January 23rd 2015
Shashikanth Ponnala, Nirav Kapadia, Wayne Wesley Harding

2) Identification of Camphor Derivatives as Novel M2 Ion Channel Inhibitors of Influenza A Virus (ChemMedComm) Monday January 19th 2015
Xin Zhao, Zhen-Wei Zhang, Wei Cui, Shengwei Chen, Yang Zhou, Jianghong Dong, Yanling Jie, Junting Wan, Yong Xu, Wenhui Hu

3) O-Benzoyl Pyridine Aldoxime and Amidoxime Derivatives: Novel Efficient DNA Photo-Cleavage Agents (ChemMedComm) Thursday January 15th 2015
PARASKEVI KARAMTZIOTI, ASTERIOS PAPASTERGIOU, JOHN G. STEFANAKIS, ALEXANDROS E. KOUMBIS, IOANNA ANASTASIOU, MARIA KOFFA, KONSTANTINA C. FYLAKTAKIDOU

4) Nature of the Charged Head Group Dictates the Anticancer Potential of Lithocholic Acid-Tamoxifen Conjugates For Breast Cancer Therapy (ChemMedComm) Wednesday January 14th 2015
Kavita Yadav, Priyanshu Bhargava, Sandhya Bansal, Manish Singh, Siddhi Gupta, Geeta Sandhu, Sandeep Kumar, Vedagopuram Sreekanth, Avinash Bajaj

5) Targeted Photoresponsive TiO2-Coumarin nanoconjugate for efficient Combination therapy in MDA-MB-231 breast cancer cells: Synergic effect of Photodynamic Therapy (PDT) and Anticancer drug Chlorambucil (ChemMedComm) Wednesday January 14th 2015
Moumita Ganguly, Sourav K. Mukhopadhyay, Karthik S, Sharabani Barman, Pradeep N.D. Singh

6) Radiosynthesis of high affinity fluorine-18 labeled GnRH peptide analogues: in vitro studies and in vivo assessment of brain uptake in rats (ChemMedComm) Monday January 12th 2015
Dag Erlend Olberg, Sven H Hausner, Nadine Bauer, Jo Klaveness, Bard Indrevoll, Finn Olav Levy, Kjetil Wessel Andressen, Marie Dahl, Julie L. Sutcliffe, Ira Haraldsen

7) Design, synthesis and biological activity of 4′-[(benzimidazol-1-yl)methyl] biphenyl-2-sulphonamides as dual angiotensin II and endothelin A receptor antagonists (ChemMedComm) Monday January 12th 2015
Liping Hao, Weizhe Xue, Xiaofeng Han, Xing He, Jun Zhang, Zhiming Zhou

8) Activity Based Probes as Molecular Tools for Biomarker Discovery (ChemMedComm) Friday January 9th 2015
Luis Carvalho, Susana Dias Lucas, Eduardo Ruivo, Rui Moreira

9) Cytotoxic potential of di-spirooxindolo/acenaphthoquino andrographolide derivatives against MCF7 cell lines (ChemMedComm) Thursday January 8th 2015
Debanjana Chakraborty, Arindam Maitya, Chetan Kumar Jain, Abhijit Hazra, Yogesh Pandharinath Bharitkar, Tarun Jha, Hemanta Majumder, Susanta Roy Choudhury, Nirup Bikash Mondal

10) Dimethylaminoethyl Methacrylate Copolymer-siRNA nanoparticles for silencing therapeutically relevant gene in macrophages (ChemMedComm) Monday January 5th 2015
Ratnesh Jain, Prajakta Dandekar, Brigitta Loretz, Marcus Koch, C-M. lehr

11) Structure-activity relationship study on senktide for development of novel potent neurokinin-3 receptor selective agonists (ChemMedComm) Monday January 5th 2015
Ryosuke Misu, Koki Yamamoto, Ai Yamada, Taro Noguchi, Hiroaki Ohno, Takashi Yamamura, Hiroaki Okamura, Fuko Matsuda, Satoshi Ohkura, Shinya Oishi, Nobutaka Fujii

12) Synthesis and biological evaluation of pentanedioic acid derivatives as farnesyltransferase inhibitors (ChemMedComm) Monday January 5th 2015
liuqing Yang, wei liu, Hanbin Mei, yuan Zhang, Xiaojuan Yu, yufang xu, Honglin Li, Jin Huang, Zhenjiang Zhao

13) Recent discoveries and developments of Androgen Receptor based therapy for Prostate Cancer (ChemMedComm) Monday January 5th 2015
Ramakrishnan Elancheran, V.L Maruthanila, M Ramanathan, S Kabilan, R Devi, A Kunnumakara, Jibon Kotoky

14) Chemical space is big. Really big (ChemMedComm) Monday January 5th 2015
Derek Lowe

15) Discovery of Highly Potent Triazole Antifungal Agents with Piperdine-oxadiazole Side Chains (ChemMedComm) Wednesday December 24th 2014
Xiaomeng He, Yan Jiang, Yongqiang Zhang, Shanchao Wu, Guoqiang Dong, Na Liu, Yang Liu, Jianzhong Yao, Zhenyuan Miao, Yan Wang, Wannian Zhang, Chunquan Sheng

16) The Natural Product Brartemicin is a High Affinity Ligand for the Carbohydrate-Recognition Domain of the Macrophage Receptor Mincle (ChemMedComm) Tuesday December 23rd 2014
Kristian Mark Jacobsen, Ulrik Keiding, Lise Lindkvist Clement, Eva Susanne Schaffert, Neela Rambaruth, Mogens Johannsen, Kurt Drickamer, Thomas Bjornskov Poulsen

17) Inhibition of Influenza H5N1 invasion by modified heparin derivatives (ChemMedComm) Tuesday December 23rd 2014
Mark A. Skidmore, Anna Kajaste-Rudnitski, Nicola Wells, Scott Guimond, Timothy Rudd, Eliza Vicenzi, Edwin Yates

18) Pyrrole- and indole-containing tranylcypromine derivatives as novel lysine-specific demethylase 1 inhibitors active on cancer cells (ChemMedComm) Tuesday December 23rd 2014
Veronica Rodriguez, Sergio Valente, Stefano Rovida, Dante Rotili, Giulia Stazi, Alessia Lucidi, Giuseppe Ciossani, Andrea Mattevi, Oronza Botrugno, Paola Dessanti, Ciro Mercurio, Paola Vianello, Saverio Minucci, mario varasi, Antonello Mai

19) Enantiomeric resolution of [(2,2-diphenyl-1,3-dioxolan-4-yl)methyl](2-phenoxyethyl)amine, a potent α 1 and 5HT1A receptors ligand: an In Vitro and Computational Study (ChemMedComm) Tuesday December 23rd 2014
Livio Brasili, Silvia Franchini, Annamaria Baraldi, Claudia Sorbi, Federica Pellati, Elena Cichero, Umberto M. Battisti, Piero Angeli, Antonio Cilia

20) Synthesis and relationship of stability and biological activity of new DSS and TMP conjugates (ChemMedComm) Monday December 22nd 2014
Yewei Sun, Zicheng Tan, Zhibin Liang, Liang Wang, Luchen Shan, Pei Yu, Simon MingYuen Lee, Yuqiang Wang

21) Synthesis and antibacterial activity of trivalent ultrashort Arg-Trp-based antimicrobial peptides (AMPs) (ChemMedComm) Monday December 22nd 2014
Barbara C. Hoffknecht, H. Bauke Albada, Marina Sturm, Pascal Prochnow, Julia E. Bandow, Nils Metzler-Nolte

22) Non-nucleoside anti-HBV agents: Advances in structural optimization and mechanism of action investigations (ChemMedComm) Tuesday December 16th 2014
Na Liu, Diwakar Rai, Fabao Zhao, Haiyong Jia, Peng Zhan, Xinyong Liu

23) Discovery of a new class of histone deacetylase inhibitors with a novel zinc binding group (ChemMedComm) Tuesday December 16th 2014
Youxuan Li, Patrick M. Woster

24) The chemistry and pharmacology of privileged pyrroloquinazolines (ChemMedComm) Monday December 15th 2014
Bo Chao, Bingbing X Li, Xiangshu Xiao

25) Synthesis of six mexiletine derivatives with isoindolines attached as potential antioxidants and their evaluation as cardioprotective agents (ChemMedComm) Monday December 15th 2014
W Roy Jackson, Anh Chau, Grant Drummond, Bevyn Jarrott, Alyson Miller, Kamani Subasinghe, Christina Yan Ru Tan, Paul J White, Christine E Wright, James Ziogas

26) Solid- and solution-phase-based library of 2β-methyl substituted penicillin derivatives. Effects on growth inhibition of tumor cell lines (ChemMedComm) Monday December 15th 2014
Dora B. Boggian, Patricia Cornier, Ernesto Mata, Viviana Blanck, Mariano Cardenas, LP Roguin

27) Identification of tris-(phenylalkyl)amines as new selective h5-HT2B receptor antagonists (ChemMedComm) Monday December 15th 2014
Wayne Harding, Shashikanth Ponnala, Nirav Kapadia

28) Photoswitching property of hairpin ODNs with azobenzene derivatives in the loop (ChemMedComm) Monday December 15th 2014
Li Wu, Ya Wu, Hongwei Jin, Liangren Zhang, Yujian He, XinJing Tang

29) Synthesis and evaluation of 6-methylcoumarin derivatives as potent and selective Monoamine Oxidase B inhibitors (ChemMedComm) Monday December 15th 2014
Jin-Shuai Lan, Long-Fei Pan, Sai-Sai Xie, Xiao-Bing Wang, Ling-Yi Kong

30) Naturally occurring FANCF-Hes1 complex inhibitors from Wrightia religiosa (ChemMedComm) Thursday December 11th 2014
Midori A. Arai, Kenji Uemura, Nozomi Hamahiga, Naoki Ishikawa, Takashi Koyano, Thaworn Kowithayakorn, Tagrid Kaddar, Madeleine Carreau, Masami Ishibashi

31) Correction: Design and chemoproteomic functional characterization of a chemical probe targeted to bromodomains of BET family proteins (ChemMedComm) Monday December 8th 2014
Jiang Wu, Julia Shin, Cara M. M. Williams, Kieran F. Geoghegan, Stephen W. Wright, David C. Limburg, Parag Sahasrabudhe, Paul D. Bonin, Bruce A. Lefker, Simeon J. Ramsey

32) Relating Caco-2 permeability to molecular properties using block relevance analysis (ChemMedComm) Monday December 8th 2014
Tim Potter, G Caron, Giuseppe Ermondi, Gayle Newbury

33) Design, synthesis and biological evaluation of imidazopyridine/imidazopyrimidine-benzimidazole conjugates as potential anticancer agents (ChemMedComm) Wednesday December 3rd 2014
Ahmed Kamal, Bharath Kumar G, Lakshma Nayak V, Santhosh Reddy Vangala, Anver Basha Shaik, Rajender Rajender, Kashi Reddy Methuku

34) Synthesis and cytostatic activity of 7-arylsulfanyl-7-deazapurine bases and ribonucleosides (ChemMedComm) Tuesday December 2nd 2014
Martin Klecka, Lenka Slavetinska, Eva Tloustova, Petr Dzubak, Marian Hajduch, Michal Hocek

35) Synthesis of 17-membered azalides from a 16-membered macrolide utilizing amide-selective silane reduction (ChemMedComm) Tuesday December 2nd 2014
Atsushi Seki, Toshihiro Mori, Kouji Sasaki, Yoshiaki Takahashi, Toshiaki Miyake, Yuzuru Akamatsu

36) 3-(2,6-Dichloro-benzyloxy)-11-oxo-olean-12-ene-29-oic acid, a semisynthetic derivative of glycyrrhetic acid: Synthesis, antiproliferative, apoptotic and anti-angiogenesis activity (ChemMedComm) Monday December 1st 2014
Rajni Sharma, Santosh Guru, Shreyans K Jain, Anup S Pathania, Ram A Vishwakarma, Shashi Bhushan, Sandip Bibishan Bharate

37) Discovery of novel 5-fluoro-N2,N4-diphenylpyrimidine-2,4-diamines as potent inhibitors against CDK2 and CDK9 (ChemMedComm) Friday November 28th 2014
Jiadi Gao, Cheng Fang, Zhiyan Xiao, Li Huang, Chin Ho Chen, Li-Ting Wang, Kuo-Hsiung Lee

38) Recent advances in molecular imaging probes for β-amyloid plaques (ChemMedComm) Tuesday November 25th 2014
Masahiro Ono, Hideo Saji

39) Design, synthesis and evaluation of QD-DTC-BisBiotin Nanobioconjugate as a potential Optical-SPECT imaging agent (ChemMedComm) Friday November 21st 2014
Narmada Bag, Rashi Mathur, Sweta Singh, Firasat Hussain, Ramprakash Chauhan, krishna Chuttani, Anil K Mishra

40) 4-Thiazolidinone derivatives as potent antimicrobial agents: microwave-assisted synthesis, biological evaluation and docking studies (ChemMedComm) Wednesday November 19th 2014
Eleni Pitta, Evangelia Tsolaki, Athina Geronikaki, Jovana Petrovic, Jasmina Glamoclija, Marina Sokovic, Emmanuele Crespan, Giovanni Maga, Shome S. Bhunia, Anil K. Saxena

41) Evaluation of aromatic 6-substituted thienopyrimidines as scaffolds against parasites that cause trypanosomiasis, leishmaniasis, and malaria. (ChemMedComm) Friday November 14th 2014
Jennifer Woodring, Gautam Patel, Jessey Erath, Ranjan Behera, Patricia Lee, Susan Leed, Ana Rodriguez, Richard Sciotti, Kojo Mensa-Wilmot, Michael Pollastri

42) Exclusive Formation of Imino [4+4] cycloaddition Products with Biologically Relevant Amines: Plausible Candidates of Acrolein Biomarkers and Biofunctional Modulators (ChemMedComm) Friday November 14th 2014
Ayumi Tsutsui, Ambara R. Pradipta, Elena Saigitbatalova, Almira Kurbangalieva, Katsunori Tanaka

43) Cytotoxic Peptide Conjugates of Dinuclear Arene Ruthenium Trithiolato Complexes (ChemMedComm) Wednesday November 12th 2014
Federico Giannini, Marco Bartoloni, Lydia E. H. Paul, Georg Suss-Fink, Jean-Louis Reymond, Julien Furrer

44) Novel β-carboline-quinazolinone hybrid as inhibitor of Leishmania donovani Trypanothione Reductase: Synthesis, molecular docking and bioevaluation (ChemMedComm) Tuesday November 4th 2014
Shikha S. Chauhan, Shashi pandey, Rahul Shivahare, Karthik Ramalingam, Shagun Krishna, Preeti Vishwakarma, M. I. Siddiqi, Suman Gupta, Neena Goyal, PMS Chauhan

45) Potent chemical chaperone compounds for GM1-gangliosidosis: N-substituted (+)-conduramine F-4 derivatives (ChemMedComm) Tuesday November 4th 2014
Shinichi Kuno, Katsumi Higaki, Atsushi Takahashi, Eiji Namba, Seiichiro Ogawa

46) Decorated 6,6',7,7'-tetrahydro-1H,1'H-2,3'-biindole scaffold as promising candidate for recognition of CDK2 allosteric site (ChemMedComm) Monday November 3rd 2014
Maria Teresa Sciortino, Angela Scala, Antonio Rescifina, Ivana Colao, Gabriel Siracusano, Antonino Mazzaglia, Ugo Chiacchio, Giovanni Grassi

47) Virtual screening for novel Atg5-Atg16 complex inhibitors for autophagy modulation (ChemMedComm) Monday November 3rd 2014
Elizabeth Robinson, Euphemia Leung, Anna Matuszek, Niels Krogsgaard-Larsen, Daniel Furkert, Margaret A Brimble, Alan Richardson, Johannes Reynisson

48) Antimicrobial spine-bone cement with caffeic acid phenethyl ester for controlled release formulation and in vivo biological assessments (ChemMedComm) Monday November 3rd 2014
Hye Sun Lee, Jeong Ho Chang

49) Design, synthesis and anticancer mechanistic studies of linked azoles (ChemMedComm) Friday October 31st 2014
Amirul Islam, Yuqi Zhang, Yao Wang, Shelli Renee McAlpine

50) Probing cytochrome P450-mediated activation with a truncated azinomycin analogue (ChemMedComm) Wednesday October 22nd 2014
Victoria Vinader, Maria Sadiq, Mark Sutherland, Mengying Huang, Paul Loadman, Lina Elsalem, Steve Shnyder, Hongjuan Cui, Kamyar Afarinkia, Mark Searcey, L H Patterson, Klaus Pors

51) Study of a D-proline peptidomimetic inhibitor of melanoma and endothelial cells invasion through activity towards MMP-2 and MMP-9 (ChemMedComm) Tuesday October 21st 2014
Francesca Bianchini, Chiara Calugi, Jessica Ruzzolini, Gloria Menchi, Lido Calorini, Antonio Guarna, Andrea Trabocchi

52) Polymeric Micelles for Hydrogen Sulfide Delivery (ChemMedComm) Tuesday October 21st 2014
Urara Hasegawa, Andre J van der Vlies

53) Synthesis and Biological Evaluation of novel derivatives of Gambogenic acid as Anticancer Agent (ChemMedComm) Friday October 17th 2014
Liqin He, Peng Huang, Zhong Hu, Xiaoshan Wang, Yaxian Wu

54) Synthesis, 3D pharmacophore, QSAR and docking studies of novel quinazoline derivatives with nitric oxide release moiety as preferential COX-2 inhibitors (ChemMedComm) Friday October 17th 2014
Doaa Boshra Farag, Nahla Ahmed Farag, Ahmed Esmat, Sally A. Abuelezz, Eman Abdel-Salam Ibrahim, Dalal A. Abou El Ella

55) Synthesis, Structure-Activity Relationship, and Mechanistic Investigation of Lithocholic Acid Amphiphiles for Colon Cancer Therapy (ChemMedComm) Wednesday October 15th 2014
Manish Singh, Sandhya Bansal, Somanath Kundu, Priyanshu Bhargava, Ashima Singh, Rajender Motiani, Radhey Shyam, Vedagopuram Sreekanth, Sagar Sengupta, Avinash Bajaj

56) Towards understanding cell penetration by stapled peptides (ChemMedComm) Tuesday October 14th 2014
Qian Chu, Raymond E. Moellering, Gerard J. Hilinski, Young-Woo Kim, Tom N. Grossmann, Johannes T.-H. Yeh, Gregory L. Verdine

57) Synthesis of new betulinic acid-peptide conjugates and in vivo and in silico studies of the influence of peptide moieties on the triterpenoid core activity (ChemMedComm) Monday October 13th 2014
Valentine Nenajdenko, Anastasiya Govdi, Nadezhda Sokolova, Irina Sorokina, Sergey Vasilevsky, Dmitry Baev, Tatyana Tolstikova, Victor Mamatyuk, Dmitry Fadeev

58) Poly-α,β-aspartyl-Arg-Gly-Asp-Phe: A novel polymeric nanomedicine (ChemMedComm) Monday October 13th 2014
Shuangling Chen, Yuji Wang, Shan Li, Yaonan Wang, Ming Zhao, Haimei Zhu, Jianhui Wu, Shiqi Peng

59) Synthesis and biological evaluation of a new class of quinazolinone azoles as potential antimicrobial agents and their interactions with calf thymus DNA and Human Serum Albumin (ChemMedComm) Wednesday October 8th 2014
Cheng-He Zhou, Li-Ping Peng, Nagarajan Sangaraiah, RASHEED SYED

60) Synthesis and Evaluation of Phenoxymethylbenzamide Analogues as Anti-Trypanosomal Agents (ChemMedComm) Wednesday October 8th 2014
Richard James Payne, Alexandra Manos-Turvey, Emma Watson, Vicky Mary Avery, Amy Jones, Melissa Sykes, Jonathan D. Baell, Marcel Kaiser

61) Polypharmacology Modelling Using Proteochemometrics (PCM): Recent Methodological Developments, Applications to Target Families, and Future Prospects (ChemMedComm) Tuesday October 7th 2014
Isidro Cortes-Ciriano, Qurrat ul Ain, Vigneshwari Subramanian, Bart Lenselink, Oscar Mendez-Lucio, AP IJzerman, Gerd Wohlfahrt, Peteris Prusis, Therese E Malliavin, Gerard van Westen, Andreas Bender

62) Can we use the epigenetic bioactivity of caloric restriction and phytochemicals to promote healthy ageing? (ChemMedComm) Friday October 3rd 2014
nadine helene martinet, adeline thomas, Stephane Poulain, Michael Christodoulou, Bertrand Philippe, rachid benhida, Daniele Passarella, melita vidakovic, daumantas matulis, maija .lahtela-kakkonen, eva Bartova, christophe blanquart, E. Mikros, nikolas fokialakis

63) Elucidation of shanorellin biosynthetic pathway and functional analysis of associated enzymes (ChemMedComm) Thursday October 2nd 2014
Michio Sato, Haruka Yamada, Kinya Hotta, Kenji Watanabe

64) Synthesis and biological evaluation of a series of aryl triazoles as firefly luciferase inhibitors (ChemMedComm) Tuesday September 30th 2014
Haixiu Bai, Peng Zhu, Wenxiao Wu, Jing Li, Zhao Ma, Wei Zhang, Yanna Cheng, Lupei Du, Minyong Li

65) Discovery of novel Sphingosine Kinase 1 inhibitors via structure-based hierarchical virtual screening (ChemMedComm) Tuesday September 30th 2014
Xiaojian Wang, Chenbin Sun, Liang Fang, Dali Yin

66) Discovery of mitochondria-targeting berberine derivatives as inhibitors of proliferation, invasion and migration against rat C6 and human U87 glioma cells (ChemMedComm) Tuesday September 30th 2014
Shengnan Fu, Yanqi Xie, Juo Tuo, Yalong Wang, Wenbo Zhu, Sihan Wu, Guangmei Yan, Haiyan Hu

67) CCK8 peptide-labeled Pluronic[registered sign] F127 micelles as a targeted vehicle of gold-based anticancer chemotherapeutics (ChemMedComm) Tuesday September 30th 2014
Chiara Nardon, Giulia Boscutti, LD Via, Paola Ringhieri, Vito Di Noto, Giancarlo Morelli, Antonella Accardo, Dolores Fregona

68) Attenuation of quorum sensing-mediated virulence in Gram-negative pathogenic bacteria: implications for the post-antibiotic era (ChemMedComm) Tuesday September 30th 2014
Ravindra P Singh

69) Design, synthesis, and biological activity of N-alkylated analogue of NCL1, a selective inhibitor of lysine-specific demethylase 1 (ChemMedComm) Monday September 29th 2014
Mohammed Naseer Ahmed Khan, Hiroki Tsumoto, Yukihiro Itoh, Yosuke Ota, Miki Suzuki, Daisuke Ogasawara, Hidehiko Nakagawa, Tamio Mizukami, N Miyata, Takayoshi Suzuki

70) Design, Synthesis and Biological Evaluation of Novel 1,2,4-Triazolo and 1,2,4-Triazino[4,3-a]quinoxalines as Potential Anticancer and Antimicrobial Agents (ChemMedComm) Monday September 29th 2014
Doaa A. E. Issa, Nargues S. Habib, Abeer E. Abdel Wahab

71) Tetrazole Regioisomers in the Development of Nitro Group-Containing Antitubercular Agents (ChemMedComm) Thursday September 25th 2014
Galina Karabanovich, Jaroslav Roh, Ondrej Soukup, Ivona Pavkova, Marketa Pasdiorova, Vojtech Tambor, Jirina Stolarikova, Marcela Vejsova, Katerina Vavrova, Vera Klimesova, Alexandr Hrabalek

72) Naphthoquinone-based Chalcone Hybrids and Derivatives: Synthesis and Potent Activity Against Cancer Cell Lines (ChemMedComm) Wednesday September 24th 2014
Guilherme Jardim, Tiago Guimaraes, Maria do Carmo Pinto, Bruno Cavalcanti, Kaio Farias, Claudia Pessoa, Claudia C Gatto, Divya K Nair, Irishi Namboothiri, Eufranio Silva Junior

73) Rational design of protein-protein interaction inhibitors (ChemMedComm) Tuesday September 23rd 2014
Didier Rognan

74) Repair of methyl lesions in RNA by oxidative demethylation (ChemMedComm) Tuesday September 23rd 2014
Fei Ye, Liyi Zhang, Lu Jin, Mingyue Zheng, Hualiang Jiang, Cheng Luo

75) Novel isoniazid-amidoether derivatives: Synthesis, characterization and antimycobacterial activity evaluation (ChemMedComm) Tuesday September 23rd 2014
Deepak Kumar, Garima Khare, Beena Negi, Saqib Kidwai, Anil K. Tyagi, Ramandeep Singh, DS Rawat

76) The status of the lysophosphatidic acid receptor type 1 (LPA1R) (ChemMedComm) Monday September 22nd 2014
Ines Gonzalez-Gil, Debora Zian, Henar Vazquez-Villa, Silvia Ortega-Gutierrez, Maria L. Lopez-Rodriguez

77) Synthesis of tetrazole compounds as novel type of potential antimicrobial agents and their synergistic effects with clinical drugs and interaction with calf thymus DNA (ChemMedComm) Monday September 22nd 2014
Ling-Ling Dai, huizhen zhang, Sangaraiah Nagarajan, Syed Rasheed, Cheng-He Zhou

78) A STEP FORWARD IN THE SIGMA ENIGMA: A ROLE FOR CHIRALITY IN THE SIGMA1 RECEPTOR-LIGAND INTERACTION? (ChemMedComm) Friday September 19th 2014
Daniela Rossi, Annamaria Marra, Marta Rui, Erik Laurini, Maurizio Fermeglia, Sabrina Pricl, Dirk Schepmann, Bernhard Wuensch, Marco Peviani, Daniela Curti, Simona Collina

79) Macrocyclic derivatives of 6-methyluracil as ligands of the peripheral anionic site of acetylcholinesterase (ChemMedComm) Friday September 19th 2014
Vyacheslav E. Semenov, Rashit Kh. Giniyatullin, Sofya V. Lushchekina, Ekaterina D. Kots, Konstantin A. Petrov, Alexandra D. Nikitashina, Oksana A. Minnekhanova, Vladimir V. Zobov, Evgeny E. Nikolsky, Patrick Masson, Vladimir S. Reznik

80) Structure-activity relationship studies of SETD8 inhibitors (ChemMedComm) Wednesday September 17th 2014
Anqi Ma, Wenyu Yu, Yan Xiong, Kyle Butler, Peter Brown, Jian Jin

81) 3-propyonyl-thiazoldine-4-carboxylic acid ethyl esters: a Family of Antiproliferative Thiazolidines. (ChemMedComm) Monday September 15th 2014
Esra Filiz ONEN BAYRAM, Kerem Buran, Irem Durmaz, Barkin Berk, Rengul Cetin-Atalay

82) Elucidating new structural features of the triazole scaffold for the development of mPGES-1 inhibitor (ChemMedComm) Monday September 15th 2014
Maria Giovanna Chini, Claudia Ferroni, Vincenza Cantone, Paolo Dambruoso, Greta Varchi, Antonella Pepe, Katrin Fischer, Oliver Werz, Carlo Pergola, Ines Bruno, R Riccio, Giuseppe Bifulco

83) Computationally motivated synthesis and enzyme kinetic evaluation of N-(β-D-glucopyranosyl)-1,2,4-triazolecarboxamides as glycogen phosphorylase inhibitors (ChemMedComm) Monday September 15th 2014
Jaida Begum, Gergely Varga, Tibor Docsa, Pal Gergely, Joseph M Hayes, Laszlo Juhasz, Laszlo Somsak

84) Optimisation of a Triazolopyridine Based Histone Demethylase Inhibitor Yields a Potent and Selective KDM2A (FBXL11) Inhibitor (ChemMedComm) Monday September 15th 2014
Paul Brennan, Katherine England, Anthony Tumber, Tobias Krojer, Giuseppe Scozzafava, Stanley Ng, Michelle Daniel, Aleksandra Szykowska, KaHing Che, Frank von Delft, Nicola A Burgess-Brown, Akane Kawamura, Christopher J Schofield

85) Stabilization for loop isomers of c-myc G-quadruplex DNA and anticancer activity by ruthenium complexes (ChemMedComm) Monday September 15th 2014
Ying Liu, Yanan Liu, Licong Yang, Chengwen Cao, Yanhui Zhou, Jie Liu

86) Design and chemoproteomic functional characterization of a chemical probe targeted to bromodomains of BET family proteins (ChemMedComm) Friday September 12th 2014
Bruce A Lefker, Julia Shin, Cara Williams, Kieran F Geoghegan, Stephen W Wright, David Limburg, Paul Bonin, Simeon Ramsey, Jiang Wu, Parag Sahasrabudhe

87) Correction: Synthesis, chiral resolution, absolute configuration assignment and pharmacological evaluation of a series of melatoninergic ligands (ChemMedComm) Friday September 12th 2014
Mohamed Ettaoussi, Basile Peres, Christian Jarry, Viviane Pallage, Olivier Nosjean, Jean A. Boutin, Arnaud Gohier, Clotilde Mannoury la Cour, Daniel-Henri Caignard, Philippe Delagrange, Pascal Berthelot, Said Yous

88) Design, synthesis, and biological and docking studies of novel podophyllotoxin-chalcone hybrids as potential anticancer agents (ChemMedComm) Thursday September 11th 2014
Abid H. Banday, Vinod Kulkarni, Victor Hruby

89) Synthesis of α-brominated phosphonates and their application as phosphate bioisosteres (ChemMedComm) Friday September 5th 2014
A. Michael Downey, Christopher W. Cairo

90) Isoxazole derivatives of 6-fluoro-N-(6-methoxybenzo[d]thiazol-2-yl)benzo[d]thiazol-2-amine and N-(pyrimidin-2-yl)benzo[d]thiazol-2-amine: regulation of cell cycle and apoptosis by p53 activation via mitochondrial-dependent pathways (ChemMedComm) Tuesday September 2nd 2014
Ravindra M. Kumbhare, Tulshiram L. Dadmal, T. Anjana Devi, Dinesh Kumar, umesh kosurkar, Debabrata chowdhury chowdhury, killari appalanaidu, Y. Khageswara Rao, janki ramana, Manika Pal Bhadra

91) Amphiphilic designer nano-carriers for controlled release, from drug delivery to diagnostics (ChemMedComm) Tuesday September 2nd 2014
Malinda Salim, Hiroyuki Minamikawa, A Sugimura, Rauzah Hashim

92) Bile Acid Amphiphiles with Tunable Head Groups as Highly Selective Antitubercular Agents (ChemMedComm) Monday September 1st 2014
Sandhya Bansal, Manish Singh, Saqib Kidwai, Priyanshu Bhargava, Ashima Singh, Vedagopuram Sreekanth, Ramandeep Singh, Avinash Bajaj

93) Discovery of an Orally Active Subtype-Selective HDAC Inhibitor, Chidamide, as an Epigenetic Modulator for Cancer Treatment (ChemMedComm) Monday September 1st 2014
Desi Pan, Qian-Jiao Yang, Xin Fu, Song Shan, Jing-Zhong Zhu, Kun Zhang, Zhi-Bing Li, Zhi-Qiang Ning, Xian-ping Lu

94) An imidazole-based derivative shows anti cancer potential by inducing apoptosis and cellular senescence (ChemMedComm) Thursday August 28th 2014
Sharma Gangavaram, Adepu Ramesh, Singh Ashita, Gourishetty Srikanth, Vankudoth Jayaram, Divya Duscharla, Jung Ho Jun, Ummanni Ramesh, Sanjay Malhotra

95) Discovery of Dehydroabietylamine Derivatives as Multifunctional Agents for the Treatment of Alzheimer's Disease (ChemMedComm) Wednesday August 27th 2014
Yingying Cao, Ling Wang, Zhongxiang Lin, FengYin Liang, Zhong Pei, Jun Xu, Qiong Gu

96) Analogues of the Marine Alkaloids Oroidin, Clathrodin, and Hymenidin Induce Apoptosis in Human HepG2 and THP-1 Cancer Cells (ChemMedComm) Tuesday August 26th 2014
Tihomir Tomasic, Dominik Nabergoj, Sanja Vrbek, Nace Zidar, Ziga Jakopin, Ales Zula, Ziga Hodnik, Marko Jukic, Marko Anderluh, JANEZ ILAS, Marija Sollner Dolenc, Jean Peluso, Genevieve Ubeaud-Sequier, Christian D. Muller, Lucija Peterlin Masic, Danijel KIKELJ

97) Identification of 2,4-Diamino-6,7-dimethoxyquinoline derivatives as G9a Inhibitors (ChemMedComm) Tuesday August 26th 2014
Nitipol Srimongkolpithak, Sandeep Sundriyal, Fengling Lu, Masoud Vedadi, Matthew Fuchter

98) Cytoprotective effects of hydrogen sulfide-releasing N-methyl-D-aspartate receptor antagonists mediated by intracellular sulfane sulfur (ChemMedComm) Tuesday August 26th 2014
Eizo Marutani, Masahiro Sakaguchi, Wei Chen, Kiyoshi Sasakura, Jifeng Liu, Ming Xian, Kenjiro Hanaoka, Tetsuo Nagano, Fumito Ichinose

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