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1) Design, Synthesis, Antibacterial Evaluation of Novel Azolylthioether Quinolones as MRSA DNA Intercalators (ChemMedComm) Thursday May 21st 2015
Ling Zhang, Vijaya Kumar Kannekanti, RASHEED SYED, Shao-Lin Zhang, Rong-Xia Geng, Cheng-He Zhou

2) Discovery of novel amino-pyrimidine inhibitors of the insulin-like growth factor 1 (IGF1R) and insulin receptor (INSR) kinases; parallel optimization of cell potency and hERG inhibition (ChemMedComm) Thursday May 21st 2015
Heather Tye, Stephan Zahn, Marco Hofmann, Michael Sanderson, Otmar Schaff, Matthias Troy, Moritz Mayer, Georg Rast, Sandeep Pal, Ulrich Guertler

3) Synthesis and antibacterial activity evaluation of C-5 side chain modified analogues of FYL-66, a potential agent against methicillin-resistant Staphylococcus aureus (ChemMedComm) Thursday May 21st 2015
Xiaoyan Yang, Zicheng Li, Zhenling Wang, Zitai Sang, Haiyue Long, Jianying Tang, Tao Yang, Yuanyuan Liu, Youfu Luo

4) 5-Iodo-2-arylalkylthio-6-aryl pyrimidin-4(3H)-ones as non-nucleoside anti-HBV agents (ChemMedComm) Wednesday May 20th 2015
Yu Zhang, Xuefeng Sun, Ningning Fan, Jianxiong Zhao, Jing Tu, Xiangmei Chen, Junyi Liu, Xiao-wei Wang

5) Alkylamino derivatives of N-benzylpyrazine-2-carboxamide: Synthesis and antimycobacterial evaluation (ChemMedComm) Wednesday May 20th 2015
Barbora Servusova-Vanaskova, Ondrej Jandourek, Pavla Paterova, Jana Kordulakova, Magdalena Plevakova, Vladimir Kubicek, Radim Kucera, Vladimir Garaj, Lieve Naesens, Jiri Kunes, Martin Dolezal, Jan Zitko

6) Synthesis and biological evaluation of potential small molecule inhibitors of Tumor Necrosis Factor (ChemMedComm) Wednesday May 20th 2015
Christos Papaneophytou, Polyxeni Alexiou, Athanasios Papakyriakou, Evangelos Ntougkos, Katerina Tsiliouka, Anna Maranti, Fotini Liepouri, Alexandros Strongilos, Anthi Mettou, Elias Couladouros, Elias Eliopoulos, Eleni Douni, George Kollias, George Kontopidis

7) Chromanones: selective and reversible Monoamine Oxidase B inhibitors with nanomolar potency (ChemMedComm) Wednesday May 20th 2015
Jin-Shuai Lan, Sai-Sai Xie, Ming Huang, Ya-Jian Hu, Ling-Yi Kong, Xiao-Bing Wang

8) Arylsulfonamide derivatives of (aryloxy)ethylpiperidines as 5-HT7 receptor antagonists and their psychotropic properties (ChemMedComm) Tuesday May 19th 2015
Pawel Maria Zajdel, Vittorio Canale, Anna Partyka, Krzysztof Marciniec, Grzegorz Satala, Rafal Kurczab, Agata Siwek, Magdalena Jastrzebska-Wiesek, Anna Wesolowska, Tomasz Kos, Piotr Popik, AJ Bojarski

9) Synthesis and in vitro Assessment of Chemically Modified siRNAs Targeting BCL2 that Contain 2'-Ribose and Triazole-linked Backbone Modifications (ChemMedComm) Monday May 18th 2015
Gord Hagen, Brandon J Peel, John Samis, Jean-Paul Desaulniers

10) Fragment-growing exploiting dynamic combinatorial chemistry of inhibitors of the aspartic protease endothiapepsin (ChemMedComm) Friday May 15th 2015
Milon Mondal, Daphne Groothuis, Anna Katharina Herta Hirsch

11) New selective A2A agonists and A3 antagonists for human adenosine receptors. Synthesis, biological activity and molecular docking studies (ChemMedComm) Wednesday May 13th 2015
Angel Guerrero, Anna Rodriguez, Hugo Gutierrez-de-Teran, David Rodriguez, Jose Brea, Maria Isabel Loza, Gloria Rosell, M. Pilar Bosch

12) A novel aminotriazole-based NHC complex for the design of gold(I) anti-cancer agents: synthesis and biological evaluation (ChemMedComm) Wednesday May 13th 2015
Tatiyana V Serebryanskaya, Andrey A. Zolotarev, Ingo Ott

13) 1,2,3-Triazole derivatives as antitubercular agents: synthesis, biological evaluation and molecular docking study (ChemMedComm) Wednesday May 13th 2015
Mubarak H. Shaikh, Dnyaneshwar D. Subhedar, Laxman Nawale, Dhiman Sarkar, Firoz A. Kalam Khan, Jaiprakash N. Sangshetti, Bapurao B. Shingate

14) Synthesis, Biological Evaluation and Mechanisms Study of a Class of Benzylideneindanone Derivatives as Novel Anticancer Agents (ChemMedComm) Friday May 8th 2015
Jinhui Hu, Jun Yan, Jie Chen, Yanqing Pang, ling huang, Xingshu Li

15) Identification of a novel class of Autotaxin inhibitors through cross-screening (ChemMedComm) Friday May 8th 2015
Diana Castagna, Emma Duffy, Dima Semaan, Louise Young, John Pritchard, simon macdonald, David Budd, Craig Jamieson, Allan John Bell Watson

16) Synthesis and evaluation of novel N-3-benzimidazolephenylbisamide derivatives for antiproliferative and hedgehog pathway inhibitory activity (ChemMedComm) Wednesday May 6th 2015
Chiyu Sun, Yangsheng Li, Ailong Shi, Jingzhou Zhang, Yafei Li, Mingming Zhao, Lijuan Zhang, Huachuan Zheng, Ying Meng, Huaiwei Ding, Hongrui Song

17) Synthesis and biological evaluation of nitric oxide-releasing hybrids from gemcitabine and phenylsulfonyl furoxans as anti-tumor agents (ChemMedComm) Wednesday April 29th 2015
Xianghua Li, Xuemin Wang, Chenjun Xu, Junkai Huang, Chengniu Wang, Xinyang Wang, Yong Ling, Liqin He

18) Synthesis and biodistribution of novel 99mTc labeled 4-nitroimidazole dithiocarbamate complexes as potential agents to target tumor hypoxia (ChemMedComm) Thursday April 23rd 2015
zhenxiang li, Junbo zhang, zhonghui jin, weifang zhang, Yanyan zhang

19) Synthesis and evaluation of [11C]PBD150, a radiolabeled glutaminyl cyclase inhibitor for the potential detection of Alzheimer's disease prior to amyloid β aggregation. (ChemMedComm) Thursday April 23rd 2015
Allen F Brooks, Isaac Jackson, Xia Shao, George Kropog, Phillip Sherman, Carole Quesada, Peter Scott

20) Discovery and optimisation of 1-acyl-2-benzylpyrrolidines as potent dual orexin receptor antagonists (ChemMedComm) Tuesday April 21st 2015
Jodi Williams, John Gatfield, Catherine Roch, Alexander Treiber, Francois Jenck, Martin Bolli, Christine Brotschi, Thierry Sifferlen, Bibia Heidmann, Christoph Boss

21) Novel indole-based sigma-2 receptor ligands: synthesis, structure-affinity relationship and antiproliferative activity (ChemMedComm) Monday April 20th 2015
Fang Xie, Torsten Kniess, Christin Neuber, Winnie Deuther-Conrad, Constantin Mamat, Brian P. Lieberman, BL Liu, Robert Henry Mach, Peter Brust, Jorg Steinbach, Jens Pietzsch, Hongmei Jia

22) Target-based Analysis of Ionization States of Bioactive Compounds (ChemMedComm) Monday April 20th 2015
Shilva Kayastha, Antonio de la Vega de Leon, Dilyana Dimova, J Bajorath

23) Exploring the Recognition Pathway at the Human A2A Adenosine Receptor of the Endogenous Agonist Adenosine using Supervised Molecular Dynamics Simulations. (ChemMedComm) Monday April 20th 2015
Davide Sabbadin, Antonella Ciancetta, Giuseppe Deganutti, Alberto Cuzzolin, Stefano Moro

24) 3-Aminooxazolidinone AHL analogs as hydrolytically-stable quorum sensing agonists in Gram-negative bacteria (ChemMedComm) Monday April 20th 2015
Min Guo, Yue Zheng, Clement Opoku-Temeng, Rusty Starks, Xiaochu Ma, Herman O Sintim

25) Synthesis, biological evaluation and QSAR studies of diarylpentanoid analogues as potential nitric oxide inhibitors (ChemMedComm) Monday April 20th 2015
Siti Munirah Mohd Faudzi, Sze Wei Leong, Faridah Abas, Mohd Fadhlizil Fasihi Mohd Aluwi, Kamal Rullah, Kok Wai Lam, Syahida Ahmad, Chau Ling Tham, Khozirah Shaari, Nordin H Lajis

26) Neuronal selective targeting, protection and signaling network analysis via dopamine mediated mesoporous silica nanoparticle (ChemMedComm) Monday April 20th 2015
shupeng li, hailong zhang, Yuhua Jiang, Sheng-gang Zhao, Li-qin Jiang, Yan Meng, Peng Liu, Myeong Ok Kim

27) Exploring cinnamic acid scaffold: development of promising neuroprotective lipophilic antioxidants (ChemMedComm) Wednesday April 15th 2015
Fernanda Borges, Daniel Chavarria, Tiago Silva, Teresa Summavielle, Jorge M.P.J. Garrido, Daniel Martins, Joana Bravo

28) Synthesis and Biological Evaluation of N-(4-phenylthiazol-2-yl) Cinnamamide Derivatives as Novel Potential Anti-tumor Agents (ChemMedComm) Monday April 13th 2015
Yong Luo, Yongxia Zhu, Kai Ran, Zhihao Liu, Ningyu Wang, Qiang Feng, Jun Zeng, Lidan Zhang, Bing He, Tinghong Ye, Shirui Zhu, Xiaolong Qiu, Luoting Yu

29) Direct photocapture of bromodomains using tropolone chemical probes (ChemMedComm) Monday April 13th 2015
Erik Hett, Eugene Chekler, Arindrajit Basak, Paul Bonin, Aldrin Denny, Andrew Flick, Kieran F Geoghegan, Shenping Liu, Mathew Pletcher, Parag Sahasrabudhe, Shores Salter, Ingrid Stock, Alex Taylor, Lyn H Jones

30) Discovery of a series of 2-(pyridinyl)pyrimidines as potent antagonists of GPR40 (ChemMedComm) Wednesday April 8th 2015
M J Waring, David Baker, Stuart Bennett, Alastair Dossetter, Mark Fenwick, Rob Garcia, Jennie Georgsson, Sam Groombridge, Sue Loxham, Philip Alexander MacFaul, Katie Maskill, David Morgan, Jenny Morrell, Helen Pointon, Graeme Robb, David Smith, Stephen Stokes, Gary Paul Wilkinson

31) Synthesis and Biological Evaluations of 2,3-Diarylthiophene Analogues of Combretastatin A-4 (ChemMedComm) Thursday April 2nd 2015
Weige Zhang, Zhan Wang, qingkun Yang, Zhaoshi Bai, Jun Sun, xuewei Jiang, Hongrui Song, Yingliang Wu

32) New substituted 9-propyladenine derivatives as adenosine receptor antagonists (ChemMedComm) Thursday April 2nd 2015
Catia Lambertucci, Michela Buccioni, Diego Dal Ben, Sonja Kachler, Gabriella Marucci, Andrea Spinaci, Ajiroghene Thomas, Karl-Norbert Klotz, R Volpini

33) Enantiomeric Diketopiperazines: Getting Insight of the Impact of the Configuration to the Conformation, Nanoimage, u-PA Inhibition and Anti-metastatic Activity (ChemMedComm) Tuesday March 31st 2015
Feng Wang, Shan Li, Yuji Wang, Haimei Zhu, Xiaoyi Zhang, Ming Zhao, Jianhui Wu, Shiqi Peng

34) Chemical genomics reveals novel biological activity of 1,2,3-dithiazoles as potent and reversible melanin synthesis inhibitors (ChemMedComm) Tuesday March 31st 2015
Panayiotis Andreas Koutentis, Paris Skourides, Oleg Alekseevich Rakitin, Anna Charalambous, Maria Koyioni, Ioanna Antoniades, Sophia Michaelidou, Iro Eleftheriou, Stanislav A Amelichev, Lidia S konstantinova, Despoina Pegeioti

35) Correction: Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday March 31st 2015
Taha M. A. Eldebss, Sobhi M. Gomha, Mohamed M. Abdulla, Reem K. Arafa

36) Structure-Based Virtual Screening for Fragment-Like Ligands of the G Protein-Coupled Histamine H4 Receptor (ChemMedComm) Monday March 30th 2015
Enade P. Istyastono, Albert J. Kooistra, Henry Vischer, Martien Kuijer, Luc Roumen, Saskia Nijmeijer, Rogier Smits, Iwan de Esch, Rob Leurs, Chris de Graaf

37) Novel synthesis of fluorochrome-coupled zoledronate with preserved functional activity on gamma/delta T cells and tumor cells (ChemMedComm) Monday March 30th 2015
Vijayanand Chandrasekaran, Shirin Kalyan, Valentina Biehl, Marcus Lettau, Patrik Theodor Nerdal, Hans-Heinrich Oberg, Daniela Wesch, Thisbe K Lindhorst, Dieter Kabelitz

38) Discovery of 2-(5,6-dimethoxypyridin-3-yl)-4-(2,4,6-trifluorobenzyl)-2H-pyrido[2,3-e][1,2,4]thiadiazin-3(4H)-one 1,1-dioxide (HTL6641), a dual orexin receptor antagonist with differentiated pharmacodynamic properties.[dagger] (ChemMedComm) Monday March 30th 2015
John Andrew Christopher, Sarah Aves, Jason Brown, James Errey, Suki Klair, Christopher Langmead, Oliver Mace, Richard Mould, Jayesh Patel, Ben Tehan, Andrei Zhukov, Fiona Marshall, Miles Congreve

39) Design of pyrazolo-pyrimidines as 11β-HSD1 inhibitors through optimisation of molecular electrostatic potential (ChemMedComm) Monday March 30th 2015
Graeme Robb, Scott Boyd, Christopher Davies, Alexander Dossetter, Frederick W Goldberg, Paul D Kemmitt, James Scott, John Swales

40) Concise Synthesis of Spergualin-Inspired Molecules With Broad-Spectrum Antibiotic Activity (ChemMedComm) Monday March 30th 2015
Victoria Assimon, Hao Shao, Sylvie Garneau-Tsodikova, Jason E. Gestwicki

41) 4-methyl-coumarins with cytotoxic activity against T24 and RT4 human bladder cancer cell lines (ChemMedComm) Thursday March 26th 2015
DAMIANA DA ROCHA VIANNA, LEILA Ruschel, FABRICIA Dietrich, Fabricio Figueiro, Fernanda Morrone, Romulo F. S. Canto, Flavia Corvello, Alice Velho, Allan Crestani, Helder Teixeira, Gilsane Lino von Poser, Ana Maria Oliveira Battastini, Vera Eifler-Lima

42) Tantalising technology (ChemMedComm) Tuesday March 24th 2015
Derek Lowe

43) Synthesis of a new HYNIC-DAPI derivative for labelling with 99mTechnetium and its in vitro evaluation in an FRTL5 cell line (ChemMedComm) Monday March 23rd 2015
Sandra Ferl, Gerd Wunderlich, Rene Smits, Alexander Hoepping, Anne Naumann, Jorg Kotzerke

44) Interactive articles in MedChemComm - connecting readers to a wealth of data and information (ChemMedComm) Thursday March 19th 2015
Richard Kelly

45) Insights into a defined secondary binding region on β-adrenoceptors and putative roles in ligand binding and drug design (ChemMedComm) Thursday March 12th 2015
Marvin Antonio Soriano-Ursua, Jose G Trujillo-Ferrara, Jose A Arias-Montano, Rafael Villalobos-Molina

46) Synthesis and evaluation of anticancer activity of novel andrographolide derivatives (ChemMedComm) Monday March 9th 2015
Devendar Ponnam, Lakshma Nayak V, Dharmendra Yadav, Niranjana Kumar Arigari, Kotesh Kumar Jonnala, Satya Srinivas KVN, Sridhar Balasubramanian, Feroz Khan, Pandu Sastry Kakaraparthi, Ramakrishna Sistla

47) Contributors to 'New Talent: Asia-Pacific' (ChemMedComm) Monday March 9th 2015


48) Membrane-interacting properties of the functionalised fatty acid moiety of muraymycin antibiotics (ChemMedComm) Friday March 6th 2015
Oliver Ries, Christian Carnarius, Claudia Steinem, Christian Ducho

49) In silico study on aging and reactivation processes of tabun conjugated AChE (ChemMedComm) Monday March 2nd 2015
Nellore Bhanu Chandar, Rabindranath Lo, Manoj K Kesharwani, Bishwajit Ganguly

50) Design, synthesis and biological evaluation of thiourea and nicotinamide-containing sorafenib analogs as antitumor agents (ChemMedComm) Monday March 2nd 2015
Xiangkai Kong, Zeyu Yao, Zuopeng He, Wen-Fang Xu, Jianwen Yao

51) Novel non-substrate modulators of the transmembrane efflux pump P-glycoprotein (ABCB1) (ChemMedComm) Friday February 27th 2015
Soren Krawczyk, Christiane Baumert, Josef Molnar, Christoph Ritter, Jens Hopner, Charlotte Kloft, Andreas Hilgeroth

52) Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday February 17th 2015
Taha Eldebss, Sobhi Gomha, Mohamed Abdalla, Reem Arafa

53) Matrix-immobilized yeast for large-scale production of recombinant human lactoferrin (ChemMedComm) Tuesday February 17th 2015
Chun Loong Ho, In Young Hwang, Kathy Loh, Matthew Chang

54) Synthesis and evaluation of amide, sulfonamide and urea - benzisoxazole derivatives as potential atypical antipsychotics (ChemMedComm) Friday February 13th 2015
Yin Chen, Yu Lan, Xudong Cao, Xiangqing Xu, Juecheng Zhang, Minquan Yu, Xin Liu, Bifeng Liu, Guisen Zhang

55) Synthesis and protective effect of new ligustrazine derivatives against CoCl2-induced neurotoxicity in differentiated PC12 cells. Part 2 (ChemMedComm) Thursday February 12th 2015
Bing Xu, Yan Gong, Xin Xu, Chenze Zhang, Yuzhong Zhang, Fuhao Chu, Hongbing Liu, Penglong Wang, Haimin Lei

56) BODIPY appended copper(II) complexes of curcumin showing mitochondria targeted remarkable photocytotoxicity in visible light (ChemMedComm) Thursday February 12th 2015
Akhil R Chakravarty, Arnab Bhattacharyya, Akanksha Dixit, Koushambi Mitra, Samya Banerjee, Anjali A Karande

57) Synthesis and biological evaluation of novel [capital Delta]2-isoxazoline fused cyclopentane derivatives as potential antimicrobial and anticancer agents (ChemMedComm) Wednesday February 11th 2015
Nagendra Babu Bathini, Santosh Kumar Prajapti, Shweta Shrivastava, Umesh Bihade, Ajay Kumar Gupta, V.G. M Naidu, Uttam Chand Banerjee

58) Evaluation of the anti-inflammatory/chondroprotective activity of aldose reductase inhibitors in human chondrocyte cultures (ChemMedComm) Wednesday February 4th 2015
Annamaria Panico, Rosanna Maccari, Venera Cardile, Sergio Avondo, Lucia Crasci, Rosaria Ottana

59) Inhibition of Insulin Amyloid Fibrillization by Glyco-Acridines: In vitro and in silico study (ChemMedComm) Wednesday February 4th 2015
Quan Van Vuong, Zuzana Bednarikova, Andrea Antosova, Huy Dinh Quoc Pham, Katarina Siposova, Nguyen Anh Tuan, Mai Suan Li, Zuzana Gazova

60) Application of QM/MM and QM methods to investigate histone deacetylase 8 (ChemMedComm) Monday February 2nd 2015
Duangkamol Gleeson, M. Paul Gleeson

61) Structure-Based Design, Synthesis by Click Chemistry and in Vivo Activity of Highly Selective A3 Adenosine Receptor Agonists (ChemMedComm) Monday February 2nd 2015
Dilip Tosh, Silvia Paoletta, Zhoumou Chen, Steven Crane, John Lloyd, Zhan-Guo Gao, Elizabeth Gizewski, John Auchampach, Daniela Salvemini, Kenneth A. Jacobson

62) Synthesis and evaluation of a series of resveratrol analogues as potent anticancer agents that target tubulin (ChemMedComm) Friday January 30th 2015
Nikhil Reddy Madadi, Hongliang Zong, Amit Ketkar, Zhen Chen, Narsimha Penthala, Venumadhav Janganati, Shobanbabu Bommagani, Robert Eoff, Monica Guzman, Peter Crooks

63) Design, Facile Synthesis and Anthelmintic Activity of New O-Substituted 6-Methoxybenzothiazole-2-carbamates (ChemMedComm) Tuesday January 27th 2015
A. Mohsen M.E. Omar, Omaima M. Aboulwafa, Doaa A. E. Issa, May M.S. El-Shokrofy, May E. Amr, Ibrahim M. El-Ashmawy

64) BEYOND THE AFFINITY FOR PROTEIN KINASE C: EXPLORING 2-PHENYL-3-HYDROXYPROPYL PIVALATE ANALOGUES AS C1 DOMAIN-TARGETING LIGANDS (ChemMedComm) Monday January 26th 2015
Daniela Rossi, Virpi Talman, Gustav Boije, Annamaria Marra, pietro Picconi, Rita Nasti, Massimo Serra, ANN JIHYAE, Marialaura Amadio, Alessia Pascale, Jeewoo Lee, Raimo Tuominen, Jari Yli-Kauhaluoma, Simona Collina

65) Correction: Identification of tris-(phenylalkyl)amines as new selective h5-HT2B receptor antagonists (ChemMedComm) Friday January 23rd 2015
Shashikanth Ponnala, Nirav Kapadia, Wayne Wesley Harding

66) Identification of Camphor Derivatives as Novel M2 Ion Channel Inhibitors of Influenza A Virus (ChemMedComm) Monday January 19th 2015
Xin Zhao, Zhen-Wei Zhang, Wei Cui, Shengwei Chen, Yang Zhou, Jianghong Dong, Yanling Jie, Junting Wan, Yong Xu, Wenhui Hu

67) O-Benzoyl Pyridine Aldoxime and Amidoxime Derivatives: Novel Efficient DNA Photo-Cleavage Agents (ChemMedComm) Thursday January 15th 2015
PARASKEVI KARAMTZIOTI, ASTERIOS PAPASTERGIOU, JOHN G. STEFANAKIS, ALEXANDROS E. KOUMBIS, IOANNA ANASTASIOU, MARIA KOFFA, KONSTANTINA C. FYLAKTAKIDOU

68) Nature of the Charged Head Group Dictates the Anticancer Potential of Lithocholic Acid-Tamoxifen Conjugates For Breast Cancer Therapy (ChemMedComm) Wednesday January 14th 2015
Kavita Yadav, Priyanshu Bhargava, Sandhya Bansal, Manish Singh, Siddhi Gupta, Geeta Sandhu, Sandeep Kumar, Vedagopuram Sreekanth, Avinash Bajaj

69) Targeted Photoresponsive TiO2-Coumarin nanoconjugate for efficient Combination therapy in MDA-MB-231 breast cancer cells: Synergic effect of Photodynamic Therapy (PDT) and Anticancer drug Chlorambucil (ChemMedComm) Wednesday January 14th 2015
Moumita Ganguly, Sourav K. Mukhopadhyay, Karthik S, Sharabani Barman, Pradeep N.D. Singh

70) Radiosynthesis of high affinity fluorine-18 labeled GnRH peptide analogues: in vitro studies and in vivo assessment of brain uptake in rats (ChemMedComm) Monday January 12th 2015
Dag Erlend Olberg, Sven H Hausner, Nadine Bauer, Jo Klaveness, Bard Indrevoll, Finn Olav Levy, Kjetil Wessel Andressen, Marie Dahl, Julie L. Sutcliffe, Ira Haraldsen

71) Design, synthesis and biological activity of 4′-[(benzimidazol-1-yl)methyl] biphenyl-2-sulphonamides as dual angiotensin II and endothelin A receptor antagonists (ChemMedComm) Monday January 12th 2015
Liping Hao, Weizhe Xue, Xiaofeng Han, Xing He, Jun Zhang, Zhiming Zhou

72) Activity Based Probes as Molecular Tools for Biomarker Discovery (ChemMedComm) Friday January 9th 2015
Luis Carvalho, Susana Dias Lucas, Eduardo Ruivo, Rui Moreira

73) Cytotoxic potential of di-spirooxindolo/acenaphthoquino andrographolide derivatives against MCF7 cell lines (ChemMedComm) Thursday January 8th 2015
Debanjana Chakraborty, Arindam Maitya, Chetan Kumar Jain, Abhijit Hazra, Yogesh Pandharinath Bharitkar, Tarun Jha, Hemanta Majumder, Susanta Roy Choudhury, Nirup Bikash Mondal

74) Dimethylaminoethyl Methacrylate Copolymer-siRNA nanoparticles for silencing therapeutically relevant gene in macrophages (ChemMedComm) Monday January 5th 2015
Ratnesh Jain, Prajakta Dandekar, Brigitta Loretz, Marcus Koch, C-M. lehr

75) Structure-activity relationship study on senktide for development of novel potent neurokinin-3 receptor selective agonists (ChemMedComm) Monday January 5th 2015
Ryosuke Misu, Koki Yamamoto, Ai Yamada, Taro Noguchi, Hiroaki Ohno, Takashi Yamamura, Hiroaki Okamura, Fuko Matsuda, Satoshi Ohkura, Shinya Oishi, Nobutaka Fujii

76) Synthesis and biological evaluation of pentanedioic acid derivatives as farnesyltransferase inhibitors (ChemMedComm) Monday January 5th 2015
liuqing Yang, wei liu, Hanbin Mei, yuan Zhang, Xiaojuan Yu, yufang xu, Honglin Li, Jin Huang, Zhenjiang Zhao

77) Recent discoveries and developments of Androgen Receptor based therapy for Prostate Cancer (ChemMedComm) Monday January 5th 2015
Ramakrishnan Elancheran, V.L Maruthanila, M Ramanathan, S Kabilan, R Devi, A Kunnumakara, Jibon Kotoky

78) Chemical space is big. Really big (ChemMedComm) Monday January 5th 2015
Derek Lowe

79) Discovery of Highly Potent Triazole Antifungal Agents with Piperdine-oxadiazole Side Chains (ChemMedComm) Wednesday December 24th 2014
Xiaomeng He, Yan Jiang, Yongqiang Zhang, Shanchao Wu, Guoqiang Dong, Na Liu, Yang Liu, Jianzhong Yao, Zhenyuan Miao, Yan Wang, Wannian Zhang, Chunquan Sheng

80) The Natural Product Brartemicin is a High Affinity Ligand for the Carbohydrate-Recognition Domain of the Macrophage Receptor Mincle (ChemMedComm) Tuesday December 23rd 2014
Kristian Mark Jacobsen, Ulrik Keiding, Lise Lindkvist Clement, Eva Susanne Schaffert, Neela Rambaruth, Mogens Johannsen, Kurt Drickamer, Thomas Bjornskov Poulsen

81) Inhibition of Influenza H5N1 invasion by modified heparin derivatives (ChemMedComm) Tuesday December 23rd 2014
Mark A. Skidmore, Anna Kajaste-Rudnitski, Nicola Wells, Scott Guimond, Timothy Rudd, Eliza Vicenzi, Edwin Yates

82) Pyrrole- and indole-containing tranylcypromine derivatives as novel lysine-specific demethylase 1 inhibitors active on cancer cells (ChemMedComm) Tuesday December 23rd 2014
Veronica Rodriguez, Sergio Valente, Stefano Rovida, Dante Rotili, Giulia Stazi, Alessia Lucidi, Giuseppe Ciossani, Andrea Mattevi, Oronza Botrugno, Paola Dessanti, Ciro Mercurio, Paola Vianello, Saverio Minucci, mario varasi, Antonello Mai

83) Enantiomeric resolution of [(2,2-diphenyl-1,3-dioxolan-4-yl)methyl](2-phenoxyethyl)amine, a potent α 1 and 5HT1A receptors ligand: an In Vitro and Computational Study (ChemMedComm) Tuesday December 23rd 2014
Livio Brasili, Silvia Franchini, Annamaria Baraldi, Claudia Sorbi, Federica Pellati, Elena Cichero, Umberto M. Battisti, Piero Angeli, Antonio Cilia

84) Synthesis and relationship of stability and biological activity of new DSS and TMP conjugates (ChemMedComm) Monday December 22nd 2014
Yewei Sun, Zicheng Tan, Zhibin Liang, Liang Wang, Luchen Shan, Pei Yu, Simon MingYuen Lee, Yuqiang Wang

85) Synthesis and antibacterial activity of trivalent ultrashort Arg-Trp-based antimicrobial peptides (AMPs) (ChemMedComm) Monday December 22nd 2014
Barbara C. Hoffknecht, H. Bauke Albada, Marina Sturm, Pascal Prochnow, Julia E. Bandow, Nils Metzler-Nolte

86) Non-nucleoside anti-HBV agents: Advances in structural optimization and mechanism of action investigations (ChemMedComm) Tuesday December 16th 2014
Na Liu, Diwakar Rai, Fabao Zhao, Haiyong Jia, Peng Zhan, Xinyong Liu

87) Discovery of a new class of histone deacetylase inhibitors with a novel zinc binding group (ChemMedComm) Tuesday December 16th 2014
Youxuan Li, Patrick M. Woster

88) The chemistry and pharmacology of privileged pyrroloquinazolines (ChemMedComm) Monday December 15th 2014
Bo Chao, Bingbing X Li, Xiangshu Xiao

89) Synthesis of six mexiletine derivatives with isoindolines attached as potential antioxidants and their evaluation as cardioprotective agents (ChemMedComm) Monday December 15th 2014
W Roy Jackson, Anh Chau, Grant Drummond, Bevyn Jarrott, Alyson Miller, Kamani Subasinghe, Christina Yan Ru Tan, Paul J White, Christine E Wright, James Ziogas

90) Solid- and solution-phase-based library of 2β-methyl substituted penicillin derivatives. Effects on growth inhibition of tumor cell lines (ChemMedComm) Monday December 15th 2014
Dora B. Boggian, Patricia Cornier, Ernesto Mata, Viviana Blanck, Mariano Cardenas, LP Roguin

91) Identification of tris-(phenylalkyl)amines as new selective h5-HT2B receptor antagonists (ChemMedComm) Monday December 15th 2014
Wayne Harding, Shashikanth Ponnala, Nirav Kapadia

92) Photoswitching property of hairpin ODNs with azobenzene derivatives in the loop (ChemMedComm) Monday December 15th 2014
Li Wu, Ya Wu, Hongwei Jin, Liangren Zhang, Yujian He, XinJing Tang

93) Synthesis and evaluation of 6-methylcoumarin derivatives as potent and selective Monoamine Oxidase B inhibitors (ChemMedComm) Monday December 15th 2014
Jin-Shuai Lan, Long-Fei Pan, Sai-Sai Xie, Xiao-Bing Wang, Ling-Yi Kong

94) Naturally occurring FANCF-Hes1 complex inhibitors from Wrightia religiosa (ChemMedComm) Thursday December 11th 2014
Midori A. Arai, Kenji Uemura, Nozomi Hamahiga, Naoki Ishikawa, Takashi Koyano, Thaworn Kowithayakorn, Tagrid Kaddar, Madeleine Carreau, Masami Ishibashi

95) Correction: Design and chemoproteomic functional characterization of a chemical probe targeted to bromodomains of BET family proteins (ChemMedComm) Monday December 8th 2014
Jiang Wu, Julia Shin, Cara M. M. Williams, Kieran F. Geoghegan, Stephen W. Wright, David C. Limburg, Parag Sahasrabudhe, Paul D. Bonin, Bruce A. Lefker, Simeon J. Ramsey

96) Relating Caco-2 permeability to molecular properties using block relevance analysis (ChemMedComm) Monday December 8th 2014
Tim Potter, G Caron, Giuseppe Ermondi, Gayle Newbury

97) Design, synthesis and biological evaluation of imidazopyridine/imidazopyrimidine-benzimidazole conjugates as potential anticancer agents (ChemMedComm) Wednesday December 3rd 2014
Ahmed Kamal, Bharath Kumar G, Lakshma Nayak V, Santhosh Reddy Vangala, Anver Basha Shaik, Rajender Rajender, Kashi Reddy Methuku

98) Synthesis and cytostatic activity of 7-arylsulfanyl-7-deazapurine bases and ribonucleosides (ChemMedComm) Tuesday December 2nd 2014
Martin Klecka, Lenka Slavetinska, Eva Tloustova, Petr Dzubak, Marian Hajduch, Michal Hocek

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Mitch Andre Garcia's Chem Feeds 2008-present

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