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1) Design, synthesis and evaluation of QD-DTC-BisBiotin Nanobioconjugate as a potential Optical-SPECT imaging agent (ChemMedComm) Friday November 21st 2014
Narmada Bag, Rashi Mathur, Sweta Singh, Firasat Hussain, Ramprakash Chauhan, krishna Chuttani, Anil K Mishra

2) 4-Thiazolidinone derivatives as potent antimicrobial agents: microwave-assisted synthesis, biological evaluation and docking studies (ChemMedComm) Wednesday November 19th 2014
Eleni Pitta, Evangelia Tsolaki, Athina Geronikaki, Jovana Petrovic, Jasmina Glamoclija, Marina Sokovic, Emmanuele Crespan, Giovanni Maga, Shome S. Bhunia, Anil K. Saxena

3) Evaluation of aromatic 6-substituted thienopyrimidines as scaffolds against parasites that cause trypanosomiasis, leishmaniasis, and malaria. (ChemMedComm) Friday November 14th 2014
Jennifer Woodring, Gautam Patel, Jessey Erath, Ranjan Behera, Patricia Lee, Susan Leed, Ana Rodriguez, Richard Sciotti, Kojo Mensa-Wilmot, Michael Pollastri

4) Exclusive Formation of Imino [4+4] cycloaddition Products with Biologically Relevant Amines: Plausible Candidates of Acrolein Biomarkers and Biofunctional Modulators (ChemMedComm) Friday November 14th 2014
Ayumi Tsutsui, Ambara R. Pradipta, Elena Saigitbatalova, Almira Kurbangalieva, Katsunori Tanaka

5) Cytotoxic Peptide Conjugates of Dinuclear Arene Ruthenium Trithiolato Complexes (ChemMedComm) Wednesday November 12th 2014
Federico Giannini, Marco Bartoloni, Lydia E. H. Paul, Georg Suss-Fink, Jean-Louis Reymond, Julien Furrer

6) Novel β-carboline-quinazolinone hybrid as inhibitor of Leishmania donovani Trypanothione Reductase: Synthesis, molecular docking and bioevaluation (ChemMedComm) Tuesday November 4th 2014
Shikha S. Chauhan, Shashi pandey, Rahul Shivahare, Karthik Ramalingam, Shagun Krishna, Preeti Vishwakarma, M. I. Siddiqi, Suman Gupta, Neena Goyal, PMS Chauhan

7) Potent chemical chaperone compounds for GM1-gangliosidosis: N-substituted (+)-conduramine F-4 derivatives (ChemMedComm) Tuesday November 4th 2014
Shinichi Kuno, Katsumi Higaki, Atsushi Takahashi, Eiji Namba, Seiichiro Ogawa

8) Decorated 6,6',7,7'-tetrahydro-1H,1'H-2,3'-biindole scaffold as promising candidate for recognition of CDK2 allosteric site (ChemMedComm) Monday November 3rd 2014
Maria Teresa Sciortino, Angela Scala, Antonio Rescifina, Ivana Colao, Gabriel Siracusano, Antonino Mazzaglia, Ugo Chiacchio, Giovanni Grassi

9) Virtual screening for novel Atg5-Atg16 complex inhibitors for autophagy modulation (ChemMedComm) Monday November 3rd 2014
Elizabeth Robinson, Euphemia Leung, Anna Matuszek, Niels Krogsgaard-Larsen, Daniel Furkert, Margaret A Brimble, Alan Richardson, Johannes Reynisson

10) Antimicrobial spine-bone cement with caffeic acid phenethyl ester for controlled release formulation and in vivo biological assessments (ChemMedComm) Monday November 3rd 2014
Hye Sun Lee, Jeong Ho Chang

11) Design, synthesis and anticancer mechanistic studies of linked azoles (ChemMedComm) Friday October 31st 2014
Amirul Islam, Yuqi Zhang, Yao Wang, Shelli Renee McAlpine

12) Probing cytochrome P450-mediated activation with a truncated azinomycin analogue (ChemMedComm) Wednesday October 22nd 2014
Victoria Vinader, Maria Sadiq, Mark Sutherland, Mengying Huang, Paul Loadman, Lina Elsalem, Steve Shnyder, Hongjuan Cui, Kamyar Afarinkia, Mark Searcey, L H Patterson, Klaus Pors

13) Study of a D-proline peptidomimetic inhibitor of melanoma and endothelial cells invasion through activity towards MMP-2 and MMP-9 (ChemMedComm) Tuesday October 21st 2014
Francesca Bianchini, Chiara Calugi, Jessica Ruzzolini, Gloria Menchi, Lido Calorini, Antonio Guarna, Andrea Trabocchi

14) Polymeric Micelles for Hydrogen Sulfide Delivery (ChemMedComm) Tuesday October 21st 2014
Urara Hasegawa, Andre J van der Vlies

15) Synthesis and Biological Evaluation of novel derivatives of Gambogenic acid as Anticancer Agent (ChemMedComm) Friday October 17th 2014
Liqin He, Peng Huang, Zhong Hu, Xiaoshan Wang, Yaxian Wu

16) Synthesis, 3D pharmacophore, QSAR and docking studies of novel quinazoline derivatives with nitric oxide release moiety as preferential COX-2 inhibitors (ChemMedComm) Friday October 17th 2014
Doaa Boshra Farag, Nahla Ahmed Farag, Ahmed Esmat, Sally A. Abuelezz, Eman Abdel-Salam Ibrahim, Dalal A. Abou El Ella

17) Synthesis, Structure-Activity Relationship, and Mechanistic Investigation of Lithocholic Acid Amphiphiles for Colon Cancer Therapy (ChemMedComm) Wednesday October 15th 2014
Manish Singh, Sandhya Bansal, Somanath Kundu, Priyanshu Bhargava, Ashima Singh, Rajender Motiani, Radhey Shyam, Vedagopuram Sreekanth, Sagar Sengupta, Avinash Bajaj

18) Towards understanding cell penetration by stapled peptides (ChemMedComm) Tuesday October 14th 2014
Qian Chu, Raymond E. Moellering, Gerard J. Hilinski, Young-Woo Kim, Tom N. Grossmann, Johannes T.-H. Yeh, Gregory L. Verdine

19) Synthesis of new betulinic acid-peptide conjugates and in vivo and in silico studies of the influence of peptide moieties on the triterpenoid core activity (ChemMedComm) Monday October 13th 2014
Valentine Nenajdenko, Anastasiya Govdi, Nadezhda Sokolova, Irina Sorokina, Sergey Vasilevsky, Dmitry Baev, Tatyana Tolstikova, Victor Mamatyuk, Dmitry Fadeev

20) Poly-α,β-aspartyl-Arg-Gly-Asp-Phe: A novel polymeric nanomedicine (ChemMedComm) Monday October 13th 2014
Shuangling Chen, Yuji Wang, Shan Li, Yaonan Wang, Ming Zhao, Haimei Zhu, Jianhui Wu, Shiqi Peng

21) Synthesis and biological evaluation of a new class of quinazolinone azoles as potential antimicrobial agents and their interactions with calf thymus DNA and Human Serum Albumin (ChemMedComm) Wednesday October 8th 2014
Cheng-He Zhou, Li-Ping Peng, Nagarajan Sangaraiah, RASHEED SYED

22) Synthesis and Evaluation of Phenoxymethylbenzamide Analogues as Anti-Trypanosomal Agents (ChemMedComm) Wednesday October 8th 2014
Richard James Payne, Alexandra Manos-Turvey, Emma Watson, Vicky Mary Avery, Amy Jones, Melissa Sykes, Jonathan D. Baell, Marcel Kaiser

23) Polypharmacology Modelling Using Proteochemometrics (PCM): Recent Methodological Developments, Applications to Target Families, and Future Prospects (ChemMedComm) Tuesday October 7th 2014
Isidro Cortes-Ciriano, Qurrat ul Ain, Vigneshwari Subramanian, Bart Lenselink, Oscar Mendez-Lucio, AP IJzerman, Gerd Wohlfahrt, Peteris Prusis, Therese E Malliavin, Gerard van Westen, Andreas Bender

24) Can we use the epigenetic bioactivity of caloric restriction and phytochemicals to promote healthy ageing? (ChemMedComm) Friday October 3rd 2014
nadine helene martinet, adeline thomas, Stephane Poulain, Michael Christodoulou, Bertrand Philippe, rachid benhida, Daniele Passarella, melita vidakovic, daumantas matulis, maija .lahtela-kakkonen, eva Bartova, christophe blanquart, E. Mikros, nikolas fokialakis

25) Elucidation of shanorellin biosynthetic pathway and functional analysis of associated enzymes (ChemMedComm) Thursday October 2nd 2014
Michio Sato, Haruka Yamada, Kinya Hotta, Kenji Watanabe

26) Synthesis and biological evaluation of a series of aryl triazoles as firefly luciferase inhibitors (ChemMedComm) Tuesday September 30th 2014
Haixiu Bai, Peng Zhu, Wenxiao Wu, Jing Li, Zhao Ma, Wei Zhang, Yanna Cheng, Lupei Du, Minyong Li

27) Discovery of novel Sphingosine Kinase 1 inhibitors via structure-based hierarchical virtual screening (ChemMedComm) Tuesday September 30th 2014
Xiaojian Wang, Chenbin Sun, Liang Fang, Dali Yin

28) Discovery of mitochondria-targeting berberine derivatives as inhibitors of proliferation, invasion and migration against rat C6 and human U87 glioma cells (ChemMedComm) Tuesday September 30th 2014
Shengnan Fu, Yanqi Xie, Juo Tuo, Yalong Wang, Wenbo Zhu, Sihan Wu, Guangmei Yan, Haiyan Hu

29) CCK8 peptide-labeled Pluronic[registered sign] F127 micelles as a targeted vehicle of gold-based anticancer chemotherapeutics (ChemMedComm) Tuesday September 30th 2014
Chiara Nardon, Giulia Boscutti, LD Via, Paola Ringhieri, Vito Di Noto, Giancarlo Morelli, Antonella Accardo, Dolores Fregona

30) Attenuation of quorum sensing-mediated virulence in Gram-negative pathogenic bacteria: implications for the post-antibiotic era (ChemMedComm) Tuesday September 30th 2014
Ravindra P Singh

31) Design, synthesis, and biological activity of N-alkylated analogue of NCL1, a selective inhibitor of lysine-specific demethylase 1 (ChemMedComm) Monday September 29th 2014
Mohammed Naseer Ahmed Khan, Hiroki Tsumoto, Yukihiro Itoh, Yosuke Ota, Miki Suzuki, Daisuke Ogasawara, Hidehiko Nakagawa, Tamio Mizukami, N Miyata, Takayoshi Suzuki

32) Design, Synthesis and Biological Evaluation of Novel 1,2,4-Triazolo and 1,2,4-Triazino[4,3-a]quinoxalines as Potential Anticancer and Antimicrobial Agents (ChemMedComm) Monday September 29th 2014
Doaa A. E. Issa, Nargues S. Habib, Abeer E. Abdel Wahab

33) Tetrazole Regioisomers in the Development of Nitro Group-Containing Antitubercular Agents (ChemMedComm) Thursday September 25th 2014
Galina Karabanovich, Jaroslav Roh, Ondrej Soukup, Ivona Pavkova, Marketa Pasdiorova, Vojtech Tambor, Jirina Stolarikova, Marcela Vejsova, Katerina Vavrova, Vera Klimesova, Alexandr Hrabalek

34) Naphthoquinone-based Chalcone Hybrids and Derivatives: Synthesis and Potent Activity Against Cancer Cell Lines (ChemMedComm) Wednesday September 24th 2014
Guilherme Jardim, Tiago Guimaraes, Maria do Carmo Pinto, Bruno Cavalcanti, Kaio Farias, Claudia Pessoa, Claudia C Gatto, Divya K Nair, Irishi Namboothiri, Eufranio Silva Junior

35) Rational design of protein-protein interaction inhibitors (ChemMedComm) Tuesday September 23rd 2014
Didier Rognan

36) Repair of methyl lesions in RNA by oxidative demethylation (ChemMedComm) Tuesday September 23rd 2014
Fei Ye, Liyi Zhang, Lu Jin, Mingyue Zheng, Hualiang Jiang, Cheng Luo

37) Novel isoniazid-amidoether derivatives: Synthesis, characterization and antimycobacterial activity evaluation (ChemMedComm) Tuesday September 23rd 2014
Deepak Kumar, Garima Khare, Beena Negi, Saqib Kidwai, Anil K. Tyagi, Ramandeep Singh, DS Rawat

38) The status of the lysophosphatidic acid receptor type 1 (LPA1R) (ChemMedComm) Monday September 22nd 2014
Ines Gonzalez-Gil, Debora Zian, Henar Vazquez-Villa, Silvia Ortega-Gutierrez, Maria L. Lopez-Rodriguez

39) Synthesis of tetrazole compounds as novel type of potential antimicrobial agents and their synergistic effects with clinical drugs and interaction with calf thymus DNA (ChemMedComm) Monday September 22nd 2014
Ling-Ling Dai, huizhen zhang, Sangaraiah Nagarajan, Syed Rasheed, Cheng-He Zhou

40) A STEP FORWARD IN THE SIGMA ENIGMA: A ROLE FOR CHIRALITY IN THE SIGMA1 RECEPTOR-LIGAND INTERACTION? (ChemMedComm) Friday September 19th 2014
Daniela Rossi, Annamaria Marra, Marta Rui, Erik Laurini, Maurizio Fermeglia, Sabrina Pricl, Dirk Schepmann, Bernhard Wuensch, Marco Peviani, Daniela Curti, Simona Collina

41) Macrocyclic derivatives of 6-methyluracil as ligands of the peripheral anionic site of acetylcholinesterase (ChemMedComm) Friday September 19th 2014
Vyacheslav E. Semenov, Rashit Kh. Giniyatullin, Sofya V. Lushchekina, Ekaterina D. Kots, Konstantin A. Petrov, Alexandra D. Nikitashina, Oksana A. Minnekhanova, Vladimir V. Zobov, Evgeny E. Nikolsky, Patrick Masson, Vladimir S. Reznik

42) Structure-activity relationship studies of SETD8 inhibitors (ChemMedComm) Wednesday September 17th 2014
Anqi Ma, Wenyu Yu, Yan Xiong, Kyle Butler, Peter Brown, Jian Jin

43) 3-propyonyl-thiazoldine-4-carboxylic acid ethyl esters: a Family of Antiproliferative Thiazolidines. (ChemMedComm) Monday September 15th 2014
Esra Filiz ONEN BAYRAM, Kerem Buran, Irem Durmaz, Barkin Berk, Rengul Cetin-Atalay

44) Elucidating new structural features of the triazole scaffold for the development of mPGES-1 inhibitor (ChemMedComm) Monday September 15th 2014
Maria Giovanna Chini, Claudia Ferroni, Vincenza Cantone, Paolo Dambruoso, Greta Varchi, Antonella Pepe, Katrin Fischer, Oliver Werz, Carlo Pergola, Ines Bruno, R Riccio, Giuseppe Bifulco

45) Computationally motivated synthesis and enzyme kinetic evaluation of N-(β-D-glucopyranosyl)-1,2,4-triazolecarboxamides as glycogen phosphorylase inhibitors (ChemMedComm) Monday September 15th 2014
Jaida Begum, Gergely Varga, Tibor Docsa, Pal Gergely, Joseph M Hayes, Laszlo Juhasz, Laszlo Somsak

46) Optimisation of a Triazolopyridine Based Histone Demethylase Inhibitor Yields a Potent and Selective KDM2A (FBXL11) Inhibitor (ChemMedComm) Monday September 15th 2014
Paul Brennan, Katherine England, Anthony Tumber, Tobias Krojer, Giuseppe Scozzafava, Stanley Ng, Michelle Daniel, Aleksandra Szykowska, KaHing Che, Frank von Delft, Nicola A Burgess-Brown, Akane Kawamura, Christopher J Schofield

47) Stabilization for loop isomers of c-myc G-quadruplex DNA and anticancer activity by ruthenium complexes (ChemMedComm) Monday September 15th 2014
Ying Liu, Yanan Liu, Licong Yang, Chengwen Cao, Yanhui Zhou, Jie Liu

48) Design and chemoproteomic functional characterization of a chemical probe targeted to bromodomains of BET family proteins (ChemMedComm) Friday September 12th 2014
Bruce A Lefker, Julia Shin, Cara Williams, Kieran F Geoghegan, Stephen W Wright, David Limburg, Paul Bonin, Simeon Ramsey, Jiang Wu, Parag Sahasrabudhe

49) Correction: Synthesis, chiral resolution, absolute configuration assignment and pharmacological evaluation of a series of melatoninergic ligands (ChemMedComm) Friday September 12th 2014
Mohamed Ettaoussi, Basile Peres, Christian Jarry, Viviane Pallage, Olivier Nosjean, Jean A. Boutin, Arnaud Gohier, Clotilde Mannoury la Cour, Daniel-Henri Caignard, Philippe Delagrange, Pascal Berthelot, Said Yous

50) Design, synthesis, and biological and docking studies of novel podophyllotoxin-chalcone hybrids as potential anticancer agents (ChemMedComm) Thursday September 11th 2014
Abid H. Banday, Vinod Kulkarni, Victor Hruby

51) Synthesis of α-brominated phosphonates and their application as phosphate bioisosteres (ChemMedComm) Friday September 5th 2014
A. Michael Downey, Christopher W. Cairo

52) Isoxazole derivatives of 6-fluoro-N-(6-methoxybenzo[d]thiazol-2-yl)benzo[d]thiazol-2-amine and N-(pyrimidin-2-yl)benzo[d]thiazol-2-amine: regulation of cell cycle and apoptosis by p53 activation via mitochondrial-dependent pathways (ChemMedComm) Tuesday September 2nd 2014
Ravindra M. Kumbhare, Tulshiram L. Dadmal, T. Anjana Devi, Dinesh Kumar, umesh kosurkar, Debabrata chowdhury chowdhury, killari appalanaidu, Y. Khageswara Rao, janki ramana, Manika Pal Bhadra

53) Amphiphilic designer nano-carriers for controlled release, from drug delivery to diagnostics (ChemMedComm) Tuesday September 2nd 2014
Malinda Salim, Hiroyuki Minamikawa, A Sugimura, Rauzah Hashim

54) Bile Acid Amphiphiles with Tunable Head Groups as Highly Selective Antitubercular Agents (ChemMedComm) Monday September 1st 2014
Sandhya Bansal, Manish Singh, Saqib Kidwai, Priyanshu Bhargava, Ashima Singh, Vedagopuram Sreekanth, Ramandeep Singh, Avinash Bajaj

55) Discovery of an Orally Active Subtype-Selective HDAC Inhibitor, Chidamide, as an Epigenetic Modulator for Cancer Treatment (ChemMedComm) Monday September 1st 2014
Desi Pan, Qian-Jiao Yang, Xin Fu, Song Shan, Jing-Zhong Zhu, Kun Zhang, Zhi-Bing Li, Zhi-Qiang Ning, Xian-ping Lu

56) An imidazole-based derivative shows anti cancer potential by inducing apoptosis and cellular senescence (ChemMedComm) Thursday August 28th 2014
Sharma Gangavaram, Adepu Ramesh, Singh Ashita, Gourishetty Srikanth, Vankudoth Jayaram, Divya Duscharla, Jung Ho Jun, Ummanni Ramesh, Sanjay Malhotra

57) Discovery of Dehydroabietylamine Derivatives as Multifunctional Agents for the Treatment of Alzheimer's Disease (ChemMedComm) Wednesday August 27th 2014
Yingying Cao, Ling Wang, Zhongxiang Lin, FengYin Liang, Zhong Pei, Jun Xu, Qiong Gu

58) Analogues of the Marine Alkaloids Oroidin, Clathrodin, and Hymenidin Induce Apoptosis in Human HepG2 and THP-1 Cancer Cells (ChemMedComm) Tuesday August 26th 2014
Tihomir Tomasic, Dominik Nabergoj, Sanja Vrbek, Nace Zidar, Ziga Jakopin, Ales Zula, Ziga Hodnik, Marko Jukic, Marko Anderluh, JANEZ ILAS, Marija Sollner Dolenc, Jean Peluso, Genevieve Ubeaud-Sequier, Christian D. Muller, Lucija Peterlin Masic, Danijel KIKELJ

59) Identification of 2,4-Diamino-6,7-dimethoxyquinoline derivatives as G9a Inhibitors (ChemMedComm) Tuesday August 26th 2014
Nitipol Srimongkolpithak, Sandeep Sundriyal, Fengling Lu, Masoud Vedadi, Matthew Fuchter

60) Cytoprotective effects of hydrogen sulfide-releasing N-methyl-D-aspartate receptor antagonists mediated by intracellular sulfane sulfur (ChemMedComm) Tuesday August 26th 2014
Eizo Marutani, Masahiro Sakaguchi, Wei Chen, Kiyoshi Sasakura, Jifeng Liu, Ming Xian, Kenjiro Hanaoka, Tetsuo Nagano, Fumito Ichinose

61) 3,5-Diamino-1,3,4-triazoles as a novel scaffold for potent, reversible LSD1 (KDM1A) inhibitors (ChemMedComm) Friday August 22nd 2014
Craig J Kutz, Steven Lee Holshouser, Ethan Marrow, Patrick M. Woster

62) Radiosynthesis and in vivo evaluation of a novel [sigma]1 selective PET ligand (ChemMedComm) Friday August 22nd 2014
Hongjun Jin, Jinda Fan, Xiang Zhang, Junfeng Li, Hubert Flores, Joel S Perlmutter, Stanley Parsons, Zhude Tu

63) Adamantane amine derivatives as dual acting NMDA receptor and voltage-gated calcium channel inhibitors for neuroprotection (ChemMedComm) Friday August 22nd 2014
Yakub Kadernani, Frank Zindo, Erika Kapp, Sarel Malan, Jacques Joubert

64) Structural Biology and Chemistry of Protein Arginine Methyltransferases (ChemMedComm) Thursday August 21st 2014
Matthieu Schapira, Renato Ferreira de Freitas

65) A double effect molecular switch leads to a novel potent negative allosteric modulator of metabotropic glutamate receptor 5 (ChemMedComm) Wednesday August 20th 2014
X. Gomez-Santacana, X. Rovira, J. A. Dalton, C. Goudet, J. P. Pin, P. Gorostiza, J. Giraldo, A. Llebaria

66) Identification and optimisation of 7-azaindole PAK1 inhibitors with improved potency and kinase selectivity (ChemMedComm) Tuesday August 19th 2014
William McCoull, Edward J. Hennessy, Kevin Blades, Matthew R. Box, Claudio Chuaqui, James E. Dowling, Christopher D. Davies, Andrew D. Ferguson, Frederick W. Goldberg, Nicholas J. Howe, Paul D. Kemmitt, Gillian M. Lamont, Katrina Madden, Claire McWhirter, Jeffrey G. Varnes, Richard A. Ward, Jason D. Williams, Bin Yang

67) Synthesis, DNA binding, docking and photocleavage studies of quinolinyl chalcones (ChemMedComm) Monday August 18th 2014
Bindu P.J, Ravikumar Naik, Mahadevan K.M, Harish B.G

68) Synthesis of imidazo[2,1-b][1,3,4]thiadiazole-chalcones as apoptosis inducing anticancer agents (ChemMedComm) Friday August 15th 2014
Ahmed Kamal, Santhosh Reddy Vangala, Santosh Karnewar, Bharath Kumar G, Anver Basha Shaik, Sumit S. Chourasiya, Mahesh Rasala, Ibrahim Bin Sayeed, Srigiridhar Kotamraju

69) Paclitaxel loaded human serum albumin nanoparticles stabilized with intermolecular disulfide bonds (ChemMedComm) Wednesday August 13th 2014
Shufang Zhao, Wentan Wang, Yanbin Huang, Yuhang Fu, Yi Cheng

70) Selective inhibitors of fibroblast activation protein (FAP) with a xanthine scaffold (ChemMedComm) Tuesday August 12th 2014
Koen Jansen, Hans De Winter, Leen Heirbaut, Jonathan Cheng, Jurgen Joossens, Anne-Marie Lambeir, Ingrid De Meester, Koen Augustyns, Pieter Van der Veken

71) An azumamide C analogue without the zinc-binding carboxylate functionality (ChemMedComm) Tuesday August 12th 2014
Jesper Villadsen, Betul Kitir, Kathrine Wich, Tina Friis, Andreas S Madsen, Christian Adam Olsen

72) Non-classical β-carbonic anhydrase inhibitors - Towards novel anti-mycobacterials (ChemMedComm) Tuesday August 12th 2014
Natascha von Gnielinski, Lisa Nienaber, Lyndel Mason, Samantha Ellis, James Triccas, Rohan A Davis, Andreas Hofmann

73) Synthesis of 1-O-acetylbritannilactone analogues from Inula britannica and in vitro Evaluation of their Anticancer Potential (ChemMedComm) Tuesday August 12th 2014
Jiang-Jiang Tang, Shuai Dong, Yang-Yang Han, Ming Lei, J.-M. Gao

74) Identification of pyrazine-based TrkA inhibitors: design, synthesis, evaluation, and computational modeling studies (ChemMedComm) Monday August 11th 2014
Brendan Frett, Nick McConnell, Yuanxiang Wang, Zhigang Xu, Andrew Ambrose, Hong-yu Li

75) Pyrido- and benzisothiazolones as inhibitors of histone acetyltransferases (HATs) (ChemMedComm) Monday August 11th 2014
Silviya Furdas, Inga Hoffmann, Dina Robaa, Benjamin Herquel, Wieslaw Malinka, Piotr Swiatek, Asifa Akhtar, Wolfgang Sippl, Manfred Jung

76) Novel Anti-HIV-1 NNRTIs Based on a Pyrazolo[4,3-d]isoxazole Backbone Scaffold: Design, Synthesis and Insights into the Molecular Basis of Action (ChemMedComm) Friday August 8th 2014
Sobhi Gomha, Mohamed Badrey, Mohamed Abdalla, Reem Arafa

77) Influence of water-soluble derivatives of [60]fullerene on therapeutically important targets related to neurodegenerative diseases (ChemMedComm) Friday August 8th 2014
Raisa A. Kotelnikova, Anastasiya V Smolina, A A Grigoryev, Irina Faingold, Denis Mischenko, Alexander A. Rybkin, Darya troshin2003@inbox.ru Poletaeva, G. I. Vankin, V. L. Zamoyskiy, Ilya I. Voronov, Pavel Troshin, Alexander Kotelnikov, Sergey O. Bachurin

78) Synthesis of imidazothiadiazole-benzimidazole conjugates as mitochondrial apoptosis inducers (ChemMedComm) Monday August 4th 2014
Ahmed Kamal, Swapna Ponnampalli, Vishnuvardhan MVPS, M P Narasimha Rao, Kishore Mullagiri, Lakshma Nayak, chandrakant Bagul

79) Antisense Oligonucleotides: Modifications and Clinical Trials (ChemMedComm) Friday August 1st 2014
Vivek Sharma, Raman Kumar Sharma, Sunil Singh

80) Naphtahlene and 2,3-dihydrobenzo[b][1,4]dioxin Derivatives With Extended Side Chains as New Scaffolds of CB2 Selective Ligands (ChemMedComm) Thursday July 31st 2014
Ashraf H. Abadi, Noha Osman, Amr Mahmoud, Christian Klein, Vincenzo Di Marzo, Khaled A. M. Abouzid, Marco Allara

81) Design, synthesis and molecular docking of novel bipyrazolyl thiazolone scaffold as a new class of antibacterial agents (ChemMedComm) Thursday July 31st 2014
Piyush N. Kalaria, Jigar A. Makawana, Shailesh Satasia, Dipak K. Raval, Hai-Liang Zhu

82) Exploring the substrate promiscuity of an antibiotic inactivating enzyme (ChemMedComm) Wednesday July 30th 2014
Vinayak Agarwal, Gaston Vondenhoff, Bharat Gadakh, Konstantin Severinov, Arthur van Aerschot, Satish Nair

83) Peptide HIV Fusion Inhibitors: modifications and conjugations (ChemMedComm) Tuesday July 29th 2014
Wei Liu, Jianjun Tan, Mohammadreza Mohammadzad Mehryar, Zhiping Teng, Yi Zeng

84) Discovery of Novel Guanidinophenylpyrazole Human Acrosin Inhibitors by Molecular Hybridization (ChemMedComm) Monday July 28th 2014
Juntao Zhao, Nuannuan Sun, Yue Gao, Diya Lv, Yang Liu, Yan Jiang, Guoqiang Dong, Qianqian Chen, Wei Li, Youjun Zhou, Ju Zhu, Jiaguo Lv, Chunquan Sheng

85) Osthol and curcumin as inhibitors of human Pgp and multidrug efflux pumps of Staphylococcus aureus: Reversing the resistance against frontline antibacterial drugs (ChemMedComm) Wednesday July 23rd 2014
Prashant Joshi, Samsher Singh, Abubakar Wani, Sadhana Sharma, Shreyans K Jain, Baljinder Singh, Bishan Gupta, Naresh Satti, S Koul, Inshad A Khan, Ajay Kumar, Sandip Bibishan Bharate, Ram A Vishwakarma

86) A novel surface-coated nanocarrier for efficient encapsulation and delivery of Camptothecin to cells (ChemMedComm) Wednesday July 23rd 2014
Rie Wakabayashi, Ryutaro Ishiyama, Noriho Kamiya, Masahiro Goto

87) A Critical Evaluation of Pyrrolo[2,3-d]pyrimidine-4-amines as Plasmodium falciparum Apical Membrane Antigen 1 (AMA1) Inhibitors (ChemMedComm) Wednesday July 23rd 2014
Shane Devine, San Lim, Indu Chandrashekaran, Christopher MacRaild, Damien Drew, Cael Debono, Raymond Lam, Robin Anders, James Beeson, Martin Scanlon, Peter J. Scammells, Ray Norton

88) Gold compounds as aquaporin inhibitors: new opportunities for therapy and imaging (ChemMedComm) Tuesday July 22nd 2014
Andreia de Almeida, Graca Soveral, Angela Casini

89) Diversity-Oriented Synthesis for Novel, Selective and Drug-like Inhibitors for a Phosphatase from Mycobacterium Tuberculosis (ChemMedComm) Tuesday July 22nd 2014
Rongjun He, Yunpeng Bai, Zhi-Hong Yu, Li Wu, Andrea M. Gunawan, Zhong-Yin Zhang

90) Gold(I) compounds with lansoprazole-type ligands: synthesis, characterization and anticancer properties in vitro (ChemMedComm) Monday July 21st 2014
Maria Serratrice, Benoit Bertrand, Esmee F. J. Janssen, Eline Hemelt, Antonio Zucca, Fabio Cocco, Maria A. Cinellu, Angela Casini

91) Synthesis of a novel series of 2,3,4-trisubstituted oxazolidines designed by isosteric replacement or rigidification of the structure and cytotoxic evaluation (ChemMedComm) Monday July 21st 2014
Saulo Andrade, Claudia Teixeira, Jonas Ramos, Marcela Lopes, Rodrigo Padua, Monica Oliveira, Elaine Souza-Fagundes, Ricardo Alves

92) Anaplastic lymphoma kinase (ALK) inhibitors: a review of design and discovery (ChemMedComm) Monday July 21st 2014
Wen-Chieh Wang, Hui-Yi Shiao, Chieh-Chien Lee, Ka-Shu Fung, Hsing-Pang Hsieh

93) Structure-based approaches towards identification of fragments for the low-druggability ATAD2 bromodomain (ChemMedComm) Tuesday July 15th 2014
Apirat Chaikuada, Andrew Petros, Oleg Fedorov, Jing Xu, Stefan Knapp

94) Carbohydrates themed issue (ChemMedComm) Tuesday July 15th 2014
Sylvie Garneau-Tsodikova, Timor Baasov

95) Beyond substrate analogues: new inhibitor chemotypes for glycosyltransferases (ChemMedComm) Friday July 11th 2014
Lauren Tedaldi, Gerd K. Wagner

96) Benzylidene-linked thiohydantoin derivatives as inhibitors of tyrosinase and melanogenesis: Importance of β-phenyl-α,β-unsaturated carbonyl functionality (ChemMedComm) Wednesday July 2nd 2014
Hye Rim Kim, Hye Jin Lee, Yeon Ja Choi, Yun Jung Park, Youngwoo Woo, Seong Jin Kim, Min Hi Park, Hee Won Lee, Pusoon Chun, H.Y. Chung, Hyung Ryong Moon

97) N-Arylalkylbenzo[d]thiazole-2-carboxamides as anti-mycobacterial agents: Design, new methods of synthesis and biological evaluation (ChemMedComm) Monday June 30th 2014
Asit Kumar Chakraborti, Parth Shah, Tejas Dhameliya, Rohit Bansal, Manesh Nautiyal, Damodara Naidu Kommi, Pradeep S. Jadhavar, Jonnalagadda Padma Sridevi, Yogeeswari Sriram, Dharmarajan Sriram

98) Triazole containing novobiocin and biphenyl amides as Hsp90 C-terminal inhibitors (ChemMedComm) Friday June 27th 2014
Jinbo Zhao, Huiping Zhao, Jessica A. Hall, Douglas Brown, Eileen Brandes, Joseph Bazzill, Patrick T. Grogan, Chitra Subramanian, George Vielhauer, Mark S. Cohen, Brian S. J. Blagg

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Third Point, Dow Come To Terms

11/21/14 PHD comic: 'Research I Problems'

Synthetic Self-Assembling Nanococoons Mimic Natural Viruses

Daily Pump Trap: 11/20/14 edition

Arrays Aid Scale-Up Of Drug-Candidate Syntheses

Distillations Podcast: Babies on Demand: Reproduction in a Technological Age

Virtual Covalent Screening

Amgen Claims It All

Eye Test Might One Day Diagnose Alzheimer’s Before Symptoms Appear

Tufts Study Finds Big Rise 
In Cost Of Drug Development


House Of Representatives Passes Bills Targeting Environmental Protection Agency

Twisted By Design

Four Killed At DuPont Plant

Nelson Wins ACS President-Elect

Political Figures European Commission President Axes Science Adviser Position


Mitch Andre Garcia's Chem Feeds 2008-present

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