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1) Rational design of protein-protein interaction inhibitors (ChemMedComm) Tuesday September 23rd 2014
Didier Rognan

2) Repair of methyl lesions in RNA by oxidative demethylation (ChemMedComm) Tuesday September 23rd 2014
Fei Ye, Liyi Zhang, Lu Jin, Mingyue Zheng, Hualiang Jiang, Cheng Luo

3) Novel isoniazid-amidoether derivatives: Synthesis, characterization and antimycobacterial activity evaluation (ChemMedComm) Tuesday September 23rd 2014
Deepak Kumar, Garima Khare, Beena Negi, Saqib Kidwai, Anil K. Tyagi, Ramandeep Singh, DS Rawat

4) The status of the lysophosphatidic acid receptor type 1 (LPA1R) (ChemMedComm) Monday September 22nd 2014
Ines Gonzalez-Gil, Debora Zian, Henar Vazquez-Villa, Silvia Ortega-Gutierrez, Maria L. Lopez-Rodriguez

5) Synthesis of tetrazole compounds as novel type of potential antimicrobial agents and their synergistic effects with clinical drugs and interaction with calf thymus DNA (ChemMedComm) Monday September 22nd 2014
Ling-Ling Dai, huizhen zhang, Sangaraiah Nagarajan, Syed Rasheed, Cheng-He Zhou

6) A STEP FORWARD IN THE SIGMA ENIGMA: A ROLE FOR CHIRALITY IN THE SIGMA1 RECEPTOR-LIGAND INTERACTION? (ChemMedComm) Friday September 19th 2014
Daniela Rossi, Annamaria Marra, Marta Rui, Erik Laurini, Maurizio Fermeglia, Sabrina Pricl, Dirk Schepmann, Bernhard Wuensch, Marco Peviani, Daniela Curti, Simona Collina

7) Macrocyclic derivatives of 6-methyluracil as ligands of the peripheral anionic site of acetylcholinesterase (ChemMedComm) Friday September 19th 2014
Vyacheslav E. Semenov, Rashit Kh. Giniyatullin, Sofya V. Lushchekina, Ekaterina D. Kots, Konstantin A. Petrov, Alexandra D. Nikitashina, Oksana A. Minnekhanova, Vladimir V. Zobov, Evgeny E. Nikolsky, Patrick Masson, Vladimir S. Reznik

8) Structure-activity relationship studies of SETD8 inhibitors (ChemMedComm) Wednesday September 17th 2014
Anqi Ma, Wenyu Yu, Yan Xiong, Kyle Butler, Peter Brown, Jian Jin

9) 3-propyonyl-thiazoldine-4-carboxylic acid ethyl esters: a Family of Antiproliferative Thiazolidines. (ChemMedComm) Monday September 15th 2014
Esra Filiz ONEN BAYRAM, Kerem Buran, Irem Durmaz, Barkin Berk, Rengul Cetin-Atalay

10) Elucidating new structural features of the triazole scaffold for the development of mPGES-1 inhibitor (ChemMedComm) Monday September 15th 2014
Maria Giovanna Chini, Claudia Ferroni, Vincenza Cantone, Paolo Dambruoso, Greta Varchi, Antonella Pepe, Katrin Fischer, Oliver Werz, Carlo Pergola, Ines Bruno, R Riccio, Giuseppe Bifulco

11) Computationally motivated synthesis and enzyme kinetic evaluation of N-(β-D-glucopyranosyl)-1,2,4-triazolecarboxamides as glycogen phosphorylase inhibitors (ChemMedComm) Monday September 15th 2014
Jaida Begum, Gergely Varga, Tibor Docsa, Pal Gergely, Joseph M Hayes, Laszlo Juhasz, Laszlo Somsak

12) Optimisation of a Triazolopyridine Based Histone Demethylase Inhibitor Yields a Potent and Selective KDM2A (FBXL11) Inhibitor (ChemMedComm) Monday September 15th 2014
Paul Brennan, Katherine England, Anthony Tumber, Tobias Krojer, Giuseppe Scozzafava, Stanley Ng, Michelle Daniel, Aleksandra Szykowska, KaHing Che, Frank von Delft, Nicola A Burgess-Brown, Akane Kawamura, Christopher J Schofield

13) Stabilization for loop isomers of c-myc G-quadruplex DNA and anticancer activity by ruthenium complexes (ChemMedComm) Monday September 15th 2014
Ying Liu, Yanan Liu, Licong Yang, Chengwen Cao, Yanhui Zhou, Jie Liu

14) Design and chemoproteomic functional characterization of a chemical probe targeted to bromodomains of BET family proteins (ChemMedComm) Friday September 12th 2014
Bruce A Lefker, Julia Shin, Cara Williams, Kieran F Geoghegan, Stephen W Wright, David Limburg, Paul Bonin, Simeon Ramsey, Jiang Wu, Parag Sahasrabudhe

15) Correction: Synthesis, chiral resolution, absolute configuration assignment and pharmacological evaluation of a series of melatoninergic ligands (ChemMedComm) Friday September 12th 2014
Mohamed Ettaoussi, Basile Peres, Christian Jarry, Viviane Pallage, Olivier Nosjean, Jean A. Boutin, Arnaud Gohier, Clotilde Mannoury la Cour, Daniel-Henri Caignard, Philippe Delagrange, Pascal Berthelot, Said Yous

16) Design, synthesis, and biological and docking studies of novel podophyllotoxin-chalcone hybrids as potential anticancer agents (ChemMedComm) Thursday September 11th 2014
Abid H. Banday, Vinod Kulkarni, Victor Hruby

17) Synthesis of α-brominated phosphonates and their application as phosphate bioisosteres (ChemMedComm) Friday September 5th 2014
A. Michael Downey, Christopher W. Cairo

18) Isoxazole derivatives of 6-fluoro-N-(6-methoxybenzo[d]thiazol-2-yl)benzo[d]thiazol-2-amine and N-(pyrimidin-2-yl)benzo[d]thiazol-2-amine: regulation of cell cycle and apoptosis by p53 activation via mitochondrial-dependent pathways (ChemMedComm) Tuesday September 2nd 2014
Ravindra M. Kumbhare, Tulshiram L. Dadmal, T. Anjana Devi, Dinesh Kumar, umesh kosurkar, Debabrata chowdhury chowdhury, killari appalanaidu, Y. Khageswara Rao, janki ramana, Manika Pal Bhadra

19) Amphiphilic designer nano-carriers for controlled release, from drug delivery to diagnostics (ChemMedComm) Tuesday September 2nd 2014
Malinda Salim, Hiroyuki Minamikawa, A Sugimura, Rauzah Hashim

20) Bile Acid Amphiphiles with Tunable Head Groups as Highly Selective Antitubercular Agents (ChemMedComm) Monday September 1st 2014
Sandhya Bansal, Manish Singh, Saqib Kidwai, Priyanshu Bhargava, Ashima Singh, Vedagopuram Sreekanth, Ramandeep Singh, Avinash Bajaj

21) Discovery of an Orally Active Subtype-Selective HDAC Inhibitor, Chidamide, as an Epigenetic Modulator for Cancer Treatment (ChemMedComm) Monday September 1st 2014
Desi Pan, Qian-Jiao Yang, Xin Fu, Song Shan, Jing-Zhong Zhu, Kun Zhang, Zhi-Bing Li, Zhi-Qiang Ning, Xian-ping Lu

22) An imidazole-based derivative shows anti cancer potential by inducing apoptosis and cellular senescence (ChemMedComm) Thursday August 28th 2014
Sharma Gangavaram, Adepu Ramesh, Singh Ashita, Gourishetty Srikanth, Vankudoth Jayaram, Divya Duscharla, Jung Ho Jun, Ummanni Ramesh, Sanjay Malhotra

23) Discovery of Dehydroabietylamine Derivatives as Multifunctional Agents for the Treatment of Alzheimer's Disease (ChemMedComm) Wednesday August 27th 2014
Yingying Cao, Ling Wang, Zhongxiang Lin, FengYin Liang, Zhong Pei, Jun Xu, Qiong Gu

24) Analogues of the Marine Alkaloids Oroidin, Clathrodin, and Hymenidin Induce Apoptosis in Human HepG2 and THP-1 Cancer Cells (ChemMedComm) Tuesday August 26th 2014
Tihomir Tomasic, Dominik Nabergoj, Sanja Vrbek, Nace Zidar, Ziga Jakopin, Ales Zula, Ziga Hodnik, Marko Jukic, Marko Anderluh, JANEZ ILAS, Marija Sollner Dolenc, Jean Peluso, Genevieve Ubeaud-Sequier, Christian D. Muller, Lucija Peterlin Masic, Danijel KIKELJ

25) Identification of 2,4-Diamino-6,7-dimethoxyquinoline derivatives as G9a Inhibitors (ChemMedComm) Tuesday August 26th 2014
Nitipol Srimongkolpithak, Sandeep Sundriyal, Fengling Lu, Masoud Vedadi, Matthew Fuchter

26) Cytoprotective effects of hydrogen sulfide-releasing N-methyl-D-aspartate receptor antagonists mediated by intracellular sulfane sulfur (ChemMedComm) Tuesday August 26th 2014
Eizo Marutani, Masahiro Sakaguchi, Wei Chen, Kiyoshi Sasakura, Jifeng Liu, Ming Xian, Kenjiro Hanaoka, Tetsuo Nagano, Fumito Ichinose

27) 3,5-Diamino-1,3,4-triazoles as a novel scaffold for potent, reversible LSD1 (KDM1A) inhibitors (ChemMedComm) Friday August 22nd 2014
Craig J Kutz, Steven Lee Holshouser, Ethan Marrow, Patrick M. Woster

28) Radiosynthesis and in vivo evaluation of a novel [sigma]1 selective PET ligand (ChemMedComm) Friday August 22nd 2014
Hongjun Jin, Jinda Fan, Xiang Zhang, Junfeng Li, Hubert Flores, Joel S Perlmutter, Stanley Parsons, Zhude Tu

29) Adamantane amine derivatives as dual acting NMDA receptor and voltage-gated calcium channel inhibitors for neuroprotection (ChemMedComm) Friday August 22nd 2014
Yakub Kadernani, Frank Zindo, Erika Kapp, Sarel Malan, Jacques Joubert

30) Structural Biology and Chemistry of Protein Arginine Methyltransferases (ChemMedComm) Thursday August 21st 2014
Matthieu Schapira, Renato Ferreira de Freitas

31) A double effect molecular switch leads to a novel potent negative allosteric modulator of metabotropic glutamate receptor 5 (ChemMedComm) Wednesday August 20th 2014
X. Gomez-Santacana, X. Rovira, J. A. Dalton, C. Goudet, J. P. Pin, P. Gorostiza, J. Giraldo, A. Llebaria

32) Identification and optimisation of 7-azaindole PAK1 inhibitors with improved potency and kinase selectivity (ChemMedComm) Tuesday August 19th 2014
William McCoull, Edward J. Hennessy, Kevin Blades, Matthew R. Box, Claudio Chuaqui, James E. Dowling, Christopher D. Davies, Andrew D. Ferguson, Frederick W. Goldberg, Nicholas J. Howe, Paul D. Kemmitt, Gillian M. Lamont, Katrina Madden, Claire McWhirter, Jeffrey G. Varnes, Richard A. Ward, Jason D. Williams, Bin Yang

33) Synthesis, DNA binding, docking and photocleavage studies of quinolinyl chalcones (ChemMedComm) Monday August 18th 2014
Bindu P.J, Ravikumar Naik, Mahadevan K.M, Harish B.G

34) Synthesis of imidazo[2,1-b][1,3,4]thiadiazole-chalcones as apoptosis inducing anticancer agents (ChemMedComm) Friday August 15th 2014
Ahmed Kamal, Santhosh Reddy Vangala, Santosh Karnewar, Bharath Kumar G, Anver Basha Shaik, Sumit S. Chourasiya, Mahesh Rasala, Ibrahim Bin Sayeed, Srigiridhar Kotamraju

35) Paclitaxel loaded human serum albumin nanoparticles stabilized with intermolecular disulfide bonds (ChemMedComm) Wednesday August 13th 2014
Shufang Zhao, Wentan Wang, Yanbin Huang, Yuhang Fu, Yi Cheng

36) Selective inhibitors of fibroblast activation protein (FAP) with a xanthine scaffold (ChemMedComm) Tuesday August 12th 2014
Koen Jansen, Hans De Winter, Leen Heirbaut, Jonathan Cheng, Jurgen Joossens, Anne-Marie Lambeir, Ingrid De Meester, Koen Augustyns, Pieter Van der Veken

37) An azumamide C analogue without the zinc-binding carboxylate functionality (ChemMedComm) Tuesday August 12th 2014
Jesper Villadsen, Betul Kitir, Kathrine Wich, Tina Friis, Andreas S Madsen, Christian Adam Olsen

38) Non-classical β-carbonic anhydrase inhibitors - Towards novel anti-mycobacterials (ChemMedComm) Tuesday August 12th 2014
Natascha von Gnielinski, Lisa Nienaber, Lyndel Mason, Samantha Ellis, James Triccas, Rohan A Davis, Andreas Hofmann

39) Synthesis of 1-O-acetylbritannilactone analogues from Inula britannica and in vitro Evaluation of their Anticancer Potential (ChemMedComm) Tuesday August 12th 2014
Jiang-Jiang Tang, Shuai Dong, Yang-Yang Han, Ming Lei, J.-M. Gao

40) Identification of pyrazine-based TrkA inhibitors: design, synthesis, evaluation, and computational modeling studies (ChemMedComm) Monday August 11th 2014
Brendan Frett, Nick McConnell, Yuanxiang Wang, Zhigang Xu, Andrew Ambrose, Hong-yu Li

41) Pyrido- and benzisothiazolones as inhibitors of histone acetyltransferases (HATs) (ChemMedComm) Monday August 11th 2014
Silviya Furdas, Inga Hoffmann, Dina Robaa, Benjamin Herquel, Wieslaw Malinka, Piotr Swiatek, Asifa Akhtar, Wolfgang Sippl, Manfred Jung

42) Novel Anti-HIV-1 NNRTIs Based on a Pyrazolo[4,3-d]isoxazole Backbone Scaffold: Design, Synthesis and Insights into the Molecular Basis of Action (ChemMedComm) Friday August 8th 2014
Sobhi Gomha, Mohamed Badrey, Mohamed Abdalla, Reem Arafa

43) Influence of water-soluble derivatives of [60]fullerene on therapeutically important targets related to neurodegenerative diseases (ChemMedComm) Friday August 8th 2014
Raisa A. Kotelnikova, Anastasiya V Smolina, A A Grigoryev, Irina Faingold, Denis Mischenko, Alexander A. Rybkin, Darya troshin2003@inbox.ru Poletaeva, G. I. Vankin, V. L. Zamoyskiy, Ilya I. Voronov, Pavel Troshin, Alexander Kotelnikov, Sergey O. Bachurin

44) Synthesis of imidazothiadiazole-benzimidazole conjugates as mitochondrial apoptosis inducers (ChemMedComm) Monday August 4th 2014
Ahmed Kamal, Swapna Ponnampalli, Vishnuvardhan MVPS, M P Narasimha Rao, Kishore Mullagiri, Lakshma Nayak, chandrakant Bagul

45) Antisense Oligonucleotides: Modifications and Clinical Trials (ChemMedComm) Friday August 1st 2014
Vivek Sharma, Raman Kumar Sharma, Sunil Singh

46) Naphtahlene and 2,3-dihydrobenzo[b][1,4]dioxin Derivatives With Extended Side Chains as New Scaffolds of CB2 Selective Ligands (ChemMedComm) Thursday July 31st 2014
Ashraf H. Abadi, Noha Osman, Amr Mahmoud, Christian Klein, Vincenzo Di Marzo, Khaled A. M. Abouzid, Marco Allara

47) Design, synthesis and molecular docking of novel bipyrazolyl thiazolone scaffold as a new class of antibacterial agents (ChemMedComm) Thursday July 31st 2014
Piyush N. Kalaria, Jigar A. Makawana, Shailesh Satasia, Dipak K. Raval, Hai-Liang Zhu

48) Exploring the substrate promiscuity of an antibiotic inactivating enzyme (ChemMedComm) Wednesday July 30th 2014
Vinayak Agarwal, Gaston Vondenhoff, Bharat Gadakh, Konstantin Severinov, Arthur van Aerschot, Satish Nair

49) Peptide HIV Fusion Inhibitors: modifications and conjugations (ChemMedComm) Tuesday July 29th 2014
Wei Liu, Jianjun Tan, Mohammadreza Mohammadzad Mehryar, Zhiping Teng, Yi Zeng

50) Discovery of Novel Guanidinophenylpyrazole Human Acrosin Inhibitors by Molecular Hybridization (ChemMedComm) Monday July 28th 2014
Juntao Zhao, Nuannuan Sun, Yue Gao, Diya Lv, Yang Liu, Yan Jiang, Guoqiang Dong, Qianqian Chen, Wei Li, Youjun Zhou, Ju Zhu, Jiaguo Lv, Chunquan Sheng

51) Osthol and curcumin as inhibitors of human Pgp and multidrug efflux pumps of Staphylococcus aureus: Reversing the resistance against frontline antibacterial drugs (ChemMedComm) Wednesday July 23rd 2014
Prashant Joshi, Samsher Singh, Abubakar Wani, Sadhana Sharma, Shreyans K Jain, Baljinder Singh, Bishan Gupta, Naresh Satti, S Koul, Inshad A Khan, Ajay Kumar, Sandip Bibishan Bharate, Ram A Vishwakarma

52) A novel surface-coated nanocarrier for efficient encapsulation and delivery of Camptothecin to cells (ChemMedComm) Wednesday July 23rd 2014
Rie Wakabayashi, Ryutaro Ishiyama, Noriho Kamiya, Masahiro Goto

53) A Critical Evaluation of Pyrrolo[2,3-d]pyrimidine-4-amines as Plasmodium falciparum Apical Membrane Antigen 1 (AMA1) Inhibitors (ChemMedComm) Wednesday July 23rd 2014
Shane Devine, San Lim, Indu Chandrashekaran, Christopher MacRaild, Damien Drew, Cael Debono, Raymond Lam, Robin Anders, James Beeson, Martin Scanlon, Peter J. Scammells, Ray Norton

54) Gold compounds as aquaporin inhibitors: new opportunities for therapy and imaging (ChemMedComm) Tuesday July 22nd 2014
Andreia de Almeida, Graca Soveral, Angela Casini

55) Diversity-Oriented Synthesis for Novel, Selective and Drug-like Inhibitors for a Phosphatase from Mycobacterium Tuberculosis (ChemMedComm) Tuesday July 22nd 2014
Rongjun He, Yunpeng Bai, Zhi-Hong Yu, Li Wu, Andrea M. Gunawan, Zhong-Yin Zhang

56) Gold(I) compounds with lansoprazole-type ligands: synthesis, characterization and anticancer properties in vitro (ChemMedComm) Monday July 21st 2014
Maria Serratrice, Benoit Bertrand, Esmee F. J. Janssen, Eline Hemelt, Antonio Zucca, Fabio Cocco, Maria A. Cinellu, Angela Casini

57) Synthesis of a novel series of 2,3,4-trisubstituted oxazolidines designed by isosteric replacement or rigidification of the structure and cytotoxic evaluation (ChemMedComm) Monday July 21st 2014
Saulo Andrade, Claudia Teixeira, Jonas Ramos, Marcela Lopes, Rodrigo Padua, Monica Oliveira, Elaine Souza-Fagundes, Ricardo Alves

58) Anaplastic lymphoma kinase (ALK) inhibitors: a review of design and discovery (ChemMedComm) Monday July 21st 2014
Wen-Chieh Wang, Hui-Yi Shiao, Chieh-Chien Lee, Ka-Shu Fung, Hsing-Pang Hsieh

59) Structure-based approaches towards identification of fragments for the low-druggability ATAD2 bromodomain (ChemMedComm) Tuesday July 15th 2014
Apirat Chaikuada, Andrew Petros, Oleg Fedorov, Jing Xu, Stefan Knapp

60) Carbohydrates themed issue (ChemMedComm) Tuesday July 15th 2014
Sylvie Garneau-Tsodikova, Timor Baasov

61) Beyond substrate analogues: new inhibitor chemotypes for glycosyltransferases (ChemMedComm) Friday July 11th 2014
Lauren Tedaldi, Gerd K. Wagner

62) Benzylidene-linked thiohydantoin derivatives as inhibitors of tyrosinase and melanogenesis: Importance of β-phenyl-α,β-unsaturated carbonyl functionality (ChemMedComm) Wednesday July 2nd 2014
Hye Rim Kim, Hye Jin Lee, Yeon Ja Choi, Yun Jung Park, Youngwoo Woo, Seong Jin Kim, Min Hi Park, Hee Won Lee, Pusoon Chun, H.Y. Chung, Hyung Ryong Moon

63) N-Arylalkylbenzo[d]thiazole-2-carboxamides as anti-mycobacterial agents: Design, new methods of synthesis and biological evaluation (ChemMedComm) Monday June 30th 2014
Asit Kumar Chakraborti, Parth Shah, Tejas Dhameliya, Rohit Bansal, Manesh Nautiyal, Damodara Naidu Kommi, Pradeep S. Jadhavar, Jonnalagadda Padma Sridevi, Yogeeswari Sriram, Dharmarajan Sriram

64) Triazole containing novobiocin and biphenyl amides as Hsp90 C-terminal inhibitors (ChemMedComm) Friday June 27th 2014
Jinbo Zhao, Huiping Zhao, Jessica A. Hall, Douglas Brown, Eileen Brandes, Joseph Bazzill, Patrick T. Grogan, Chitra Subramanian, George Vielhauer, Mark S. Cohen, Brian S. J. Blagg

65) Mechanism of forming trimer, self-assembling nano-particle and inhibiting tumor growth of small molecule CIPPCT (ChemMedComm) Wednesday June 25th 2014
Fengxiang Du, Xiaoyi Zhang, Shan Li, Yaonan Wang, Meiqing Zheng, Yuji Wang, Shurui Zhao, Jianhui Wu, Lin Gui, Ming Zhao, Shiqi Peng

66) Prekinamycin and an Isosteric-Isoelectronic Analogue Exhibit Comparable Cytotoxicity Towards K562 Human Leukemia Cells (ChemMedComm) Wednesday June 25th 2014
Gary I Dmitrienko, Glenn Abbott, Brian Hasinoff, Xing Wu, Vladimir Birman, zhufeng zhao, Lei Guo

67) In vitro selection of a peptide aptamer that potentiates inhibition of cyclin-dependent kinase by purvalanol (ChemMedComm) Wednesday June 25th 2014
Wei Wang, Yoshinori Hirano, Takanori Uzawa, Mingzhe Liu, Makoto Taiji, Yoshihiro Ito

68) Optimization of the anti-cancer activity of phopshotidylinositol-3 kinase pathway inhibitor PITENIN-1: switching a thiourea with 1,2,3-triazole (ChemMedComm) Tuesday June 24th 2014
Yadagiri Kommagalla, Sinziana Cornea, Robert Riehle, Vladimir Torchilin, Alexei Degterev, Cherupi Ramana

69) Imidazolium derived ionic salts induce inhibition of cancerous cell growth through apoptosis (ChemMedComm) Tuesday June 24th 2014
Sanjay Malhotra, Vineet Kumar, Christian E Velez Gerena, Beatriz Zayas

70) Identification of Tanshinone IIA as a Natural Monoacylglycerol Lipase Inhibitor by Combined in silico and in vitro Approach (ChemMedComm) Monday June 23rd 2014
Jianhua Liu, Ruolin Yang, Yang Lu

71) Evaluation of Functional Groups as Acetyl-Lysine Mimetics for BET Bromodomain Inhibition (ChemMedComm) Monday June 23rd 2014
Phillip Patrick Sharp, Jean-Marc Garnier, David C.S. Huang, Christopher J Burns

72) Benzothiazolyl Substituted Iminothiazolidinones and Benzamido-oxothiazolidines as Potent and Partly Selective Aldose Reductase Inhibitors (ChemMedComm) Friday June 20th 2014
Jamshed Iqbal, Aamer Saeed, Yildiz Tehseen, Humera Raffique, Norbert Furtmann, J Bajorath, Ulrich Floerke

73) Conformational Analysis of Peramivir Reveals Critical Differences Between Free and Enzyme-Bound States (ChemMedComm) Thursday June 19th 2014
Michele R Richards, Michael G Brant, Martin Boulanger, Christopher W. Cairo, Jeremy E Wulff

74) Understanding the Structural Requirements of Hybrid (S)-6-((2-(4-Phenylpiperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-1-ol and its Analogs as D2/D3 Receptor Ligands: A Three-Dimensional Quantitative Structure-Activity Relationship (3D QSAR) Investigation (ChemMedComm) Thursday June 19th 2014
Gyan Prakash Modi, Horrick Sharma, Prashant Suresh Kharkar, Aloke K. Dutta

75) Characterization of a selective inhibitor for matrix metalloproteinase-8 (MMP-8) (ChemMedComm) Wednesday June 18th 2014
Derong Ding, Katerina Lichtenwalter, Hualiang Pi, Shahriar Mobashery, Mayland Chang

76) Synthesis of Hybrid Anticancer Agents Based on Kinase and Histone Deacetylase Inhibitors (ChemMedComm) Wednesday June 18th 2014
Hiren Patel, Irina Chuckowree, Peter Coxhead, Matthew Guille, Minghua Wang, Alexandra Zuckerman, Robin Williams, Mariangela Librizzi, Ronald Paranal, James Bradner, John Spencer

77) Inhibitors of the human neuraminidase enzymes (ChemMedComm) Wednesday June 18th 2014
Christopher W. Cairo

78) A fundamental view of enthalpy-entropy compensation (ChemMedComm) Tuesday June 17th 2014
Ulf Ryde

79) NMR and Molecular recognition. The application of ligand-based NMR methods to monitor molecular interactions (ChemMedComm) Tuesday June 17th 2014
Unione Luca, Galante Silvia, Diaz Dolores, Javier Canada, Jesus Barbero

80) A versatile acid-labile linker for antibody-drug conjugates (ChemMedComm) Tuesday June 17th 2014
Mathew Finniss, Kevin Chu, Charles Bowerman, James Luft, Zishan Haroon, J. M. Desimone

81) Theoretical and experimental investigation on clarithromycin, erythromycin A and azithromycin and descladinosyl derivatives of clarithromycin and azithromycin with 3-O substitution as anti-bacterial agents (ChemMedComm) Wednesday June 11th 2014
Jill Barber, Biljana Arsic, Abida Awan, Richard Brennan, Juan Aguilar, Ruth Ledder, Andrew J McBain, Andrew Charles Regan

82) Branched α-D-mannopyranosides; a new class of potent FimH antagonists (ChemMedComm) Wednesday June 11th 2014
Tihomir Tomasic, Said Rabbani, Martina Gobec, Irena Mlinaric Rascan, Crtomir Podlipnik, B Ernst, Marko Anderluh

83) Species differences in drug plasma protein binding (ChemMedComm) Tuesday June 10th 2014
Nicola Colclough, Linette Ruston, J. Matthew Wood, Philip A. MacFaul

84) Synthesis of 3'-Deoxy-3'-fluorothymidine (FLT) 5'-O-Glucuronide: A Reference Standard for Imaging Studies with [18F]FLT (ChemMedComm) Tuesday June 3rd 2014
Bernard Thomas Golding, Suzannah Harnor, Tommy Rennison, Martin Galler, Celine Cano, Roger J Griffin, David Newell

85) Recognition of diazirine-modified O-GlcNAc by human O-GlcNAcase (ChemMedComm) Monday June 2nd 2014
Andrea Rodriguez, Jennifer Kohler

86) Multivalent Amino Sugars to Recognize Different TAR RNA Conformations (ChemMedComm) Friday May 30th 2014
Dev P Arya, Patrick Kellish, Mirko Hennig, Meredith Newby, Todd Mack, Sunil Kumar

87) Exploring the meaning of sugar configuration in a supramolecular environment: Comparison of six octyl glycoside micelles by ITC and NMR spectroscopy (ChemMedComm) Friday May 30th 2014
Thisbe K Lindhorst, Jorn Schmidt-Lassen

88) Synthesis, complex stability and small animal PET imaging of a novel 64Cu-labelled cryptand molecule (ChemMedComm) Friday May 30th 2014
Christian Foerster, James Christopher Knight, Melinda Wuest, Brendan Rowan, Suzanne E. Lapi, Angelo J. Amoroso, Peter G Edwards, Frank Wuest

89) Synthesis and biological evaluation of panitumumab-IRDye800 conjugate as a fluorescence imaging probe for EGFR-expressing cancers (ChemMedComm) Friday May 30th 2014
Sibaprasad Bhattacharyya, Nimit Patel, Ling Wei, Lisa A Riffle, Joseph D Kalen, G Craig Hill, Paula M Jacobs, Kurt R Zinn, Eben Rosenthal

90) Tetracycline analogues with a selective inhibitory effect on HIF-1α (ChemMedComm) Friday May 30th 2014
Y. Bendiabdellah, K. M. Rahman, B. Uranchimeg, K. S. Nahar, D. Antonow, R. H. Shoemaker, G. Melillo, G. Zinzalla, D. E. Thurston

91) Synthesis, chiral resolution, absolute configuration assignment and pharmacological evaluation of a series of melatoninergic ligands (ChemMedComm) Wednesday May 28th 2014
Mohamed Ettaoussi, Basile Peres, Christian Jarry, Olivier Nosjean, Jean Boutin, Arnaud Gohier, Clotilde Mannoury la Cour, Daniel Caignard, Philippe Delagrange, Pascal Berthelot, Said Yous

92) A practical glycosyltransferase assay for the identification of new inhibitor chemotypes (ChemMedComm) Friday May 23rd 2014
Lauren Tedaldi, Andrew Evitt, Niina Goos, Jingqian Jiang, Gerd K. Wagner

93) Synthesis of Isoxazole Moiety Containing Ferrocene Derivatives and Preliminarily in vitro Anticancer Activity (ChemMedComm) Thursday May 22nd 2014
Yong Jianping, Can-Zhong Lu, Xiao-Yuan Wu

94) Structure of the Cannabinoid Receptor 1: Homology Modeling of Its Inactive State and Enrichment Study Based on CB1 Antagonist Docking (ChemMedComm) Tuesday May 20th 2014
Haining Liu, Ronak Patel, Robert J. Doerksen

95) When Proteins Start to Make Sense: Fine-tuning Aminoglycosides for PTC Suppression Therapy (ChemMedComm) Friday May 16th 2014
Moran Shalev, Timor BAASOV

96) [small omega]-Heteroarylalkylcarbamates as inhibitors of fatty acid amide hydrolase (FAAH) (ChemMedComm) Friday May 16th 2014
Tobias Terwege, Helmut Dahlhaus, Walburga Hanekamp, M Lehr

97) Small-Molecule Phosphodiesterase Probes: Discovery of Potent and Selective CNS-Penetrable Quinazoline Inhibitors of PDE1 (ChemMedComm) Friday May 16th 2014
John M Humphrey, Eddie Yang, Christopher W. am Ende, Eric Arnold, Jenna Head, Stephen Jenkinson, Spiros Liras, jayvardhan Pandit, Brian Samas, Frank Menniti, Felix Vajdos, Lorraine Lebel

98) Multivalent Glycoconjugates as Vaccines and Potential Drug Candidates (ChemMedComm) Friday May 16th 2014
Rainer Haag, Sumati Bhatia, Mathias Dimde

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