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1) 2-[18F]Fluoroethyl tosylate - a versatile tool for building of 18F based radiotracers for positron emission tomography (ChemMedComm) Thursday September 3rd 2015
Torsten Kniess, Markus Laube, Peter Brust, Jorg Steinbach

2) The first potent diphenyl phosphonate KLK4 inhibitors with unexpected binding kinetics (ChemMedComm) Thursday September 3rd 2015
Jeroen Van Soom, Giuliana Cuzzucoli Crucitti, Rafaela Gladysz, Pieter Van der Veken, Roberto Di Santo, Ingmar Stuyver, Victoria Buck, Anne-Marie Lambeir, Viktor Magdolen, Jurgen Joossens, Koen Augustyns

3) Evaluation of binding competition and group epitopes of Acetylcholinesterase inhibitors by STD NMR, Tr-NOESY, DOSY and Molecular Docking: An old approach but new findings (ChemMedComm) Thursday September 3rd 2015
Nazish Urooj Tanoli, Sheraz Ahmad Khan Tanoli, Antonio Gilberto Ferreira, Sana Gul, Zaheer Ul Haq

4) Missing the target (ChemMedComm) Wednesday September 2nd 2015
Derek Lowe

5) Property-based characterization of kinase-like ligand space for library design and virtual screening (ChemMedComm) Wednesday September 2nd 2015
David Bajusz, Gyorgy Ferenczy, George M Keseru

6) Design, Synthesis and Bioevaluation of Tacrine Hybrids with Cinnamate and Cinnamylideneacetate Derivatives as Potential Anti-Alzheimer Drug Candidates (ChemMedComm) Wednesday September 2nd 2015
Amelia Santos, Catarina Quintanova, Rangappa S Keri, Sergio Marques, Sandra Cardoso, M L. M. Serralheiro, Maria Goncalves Fernandes

7) Supramolecular, Prodrug-based Micelles with Enzyme Regulated Release Behavior for Controlled Drug Delivery (ChemMedComm) Friday August 28th 2015
Yong-yong Li, Yu-qin Chen, Hai-qing Dong, Chun-yan Dong

8) Sulfasalazine in Ionic Liquid Form with Improved Solubility and Exposure (ChemMedComm) Wednesday August 26th 2015
Mohammad Shadid, Gabriela Gurau, Julia L. Shamshina, Bei-Ching Chuang, Shumet Hailu, Emily Guan, Swapan Chowdhury, Jing-Tao Wu, Syed A. A. Rizvi, Robert Griffin, Robin D. Rogers

9) Aryl- Imidazothiadiazole Analogues as Microtubule Disrupting Agents (ChemMedComm) Wednesday August 26th 2015
Ahmed Kamal, Subba Rao A.V., Srinivasa Reddy Telukutla, Sowjanya Polepalli, chandrakant Bagul, Vishnuvardhan MVPS, Siddiq Pasha Shaik, Nishant Jainb

10) Insights into the impact of N- and O-methylation on aqueous solubility and lipophilicity using matched molecular pair analysis (ChemMedComm) Friday August 21st 2015
Timothy John Ritchie, simon macdonald, Stephen Pickett

11) Inspired by magnolol: design of NSAIDs-based compounds with excellent anti-inflammatory effect (ChemMedComm) Friday August 21st 2015
Wenfeng Liu, Yuan Yue, Yonglian Li, Xi Zheng, Kun Zhang, Zhiyun Du

12) Novel Quinoline Derivatives as Potent In Vitro α-Glucosidase Inhibitors: In Silico Studies and SAR Predictions (ChemMedComm) Friday August 21st 2015
Muhammad Taha, Nor Ismail Ismail, Syahrul Imran, Abdul Wadood, Fazal Rahim, Muhammad Ali, Ahsfaq Rehman

13) Correction: Synthesis and antibacterial activity evaluation of C-5 side chain modified analogues of FYL-66, a potential agent against methicillin-resistant Staphylococcus aureus (ChemMedComm) Friday August 21st 2015
Xiaoyan Yang, Zicheng Li, Zhenling Wang, Zitai Sang, Haiyue Long, Jianying Tang, Tao Yang, Yuanyuan Liu, Youfu Luo

14) Navigating into chemical space between MGCD0103 and SAHA: Novel Histone Deacetylase Inhibitor as a Promising Lead (ChemMedComm) Monday August 17th 2015
Xin Zhang, Peng-Cheng Lv, Dongdong Li, weiming zhang, Hai-Liang Zhu

15) Discovery of Pyridyl-based inhibitors of Plasmodium falciparum N-myristoyltransferase (ChemMedComm) Monday August 17th 2015
Zhiyong Yu, James A Brannigan, Kaveri Rangachari, William Heal, Anthony J Wilkinson, Tony Holder, Robin J Leatherbarrow, Edward William Tate

16) Discovery of High Affinity Inhibitors of Leishmania donovani N-Myristoyltransferase (ChemMedComm) Monday August 17th 2015
Mark Rackham, Zhiyong Yu, James A Brannigan, William Heal, Daniel Paape, Victoria Barker, Anthony J Wilkinson, Deborah Smith, Robin J Leatherbarrow, Edward William Tate

17) Inhibitory effect of cytotoxic nitrogen-containing heterocyclic stilbene analogues on the VEGF protein secretion and the expression of the VEGF, hTERT and c-Myc genes (ChemMedComm) Wednesday August 12th 2015
Eva Falomir, Rosa Marti-Centelles, Juan Murga, Miguel Carda, J. Alberto Marco

18) Synthesis, in vitro and in vivo anticancer activities of novel 4-substituted 1,2-bis(4-chlorophenyl)-pyrazolidine-3,5-dione derivatives (ChemMedComm) Wednesday August 12th 2015
Xu-Yao Zhang, Yi-Fei Gu, Ting Chen, Dong-Xiao Yang, Xi-Xin Wang, Bai-Ling Jiang, Kun-Peng Shao, Wen Zhao, Cong Wang, Jun-Wei Wang, Qiu-Rong Zhang, Hong-Min Liu

19) Correction: Application of QM/MM and QM methods to investigate histone deacetylase 8 (ChemMedComm) Wednesday August 12th 2015
Duangkamol Gleeson, M. Paul Gleeson

20) Structure activity relationship of C1-C2-linker substituted 1,5-naphthyridine analogues of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-7) (ChemMedComm) Wednesday August 12th 2015
Sheo B Singh, David Kaelin, Jin Wu, Lynn Miesel, Christopher Tan, Peter Meinke, David Olsen, Armando Lagrutta, Changqing Wei, Yonggang Liao, Xuanjia Peng, Xiu Wang, Hideyuki Fukuda, Ryuta Kishii, Masaya Takei, Takeshi Shibata, Tomoko Takeuchi, Kohei Ohata, Akinori Nishimura, Yasumichi Fukuda

21) Inhibition of Phosphatidylinositol-3,4,5-trisphosphate Binding to AKT Pleckstrin Homology Domain by 4-Amino-1,2,5-oxadiazole Derivatives (ChemMedComm) Tuesday August 11th 2015
Debasis Manna, Sukhamoy Gorai, Saurav Paul, Ganga Sankaran, Manas Kumar Santra, Rituparna Borah

22) Design and discovery of 3-aryl-5-substituted-isoquinolin-1-ones as potent tankyrase inhibitors (ChemMedComm) Tuesday August 11th 2015
Richard J.R Elliott, Ashley Jarvis, Mohan B Rajasekaran, Malini Menon, Leandra Bowers, Raymond Boffey, Melanie Bayford, Stuart Firth-Clark, Rebekah Key, Rehan Aqil, Stewart B. Kirton, Dan Niculescu-Duvaz, Laura Fish, Filipa Lopes, Robert McLeary, Ines Trindade, Elisenda Vendrell, Felix Munkonge, Rod Porter, Trevor Perrior, CJ Springer, Antony Oliver, Laurence Pearl, Alan Ashworth, Christopher J. Lord

23) Isothiazolo[4,3-b]pyridines as inhibitors of cyclin G associated kinase : synthesis, structure-activity relationship studies and antiviral activity (ChemMedComm) Friday August 7th 2015
Jiahong Li, Sona Kovackova, Szuyuan Pu, Jef Rozenski, Steven De Jonghe, Shirit Einav, Piet Herdewijn

24) Correction: Design, synthesis, and evaluation of semi-conservative mono-carbonyl analogs of curcumin as anti-inflammatory agents against lipopolysaccharide-induced acute lung injury (ChemMedComm) Friday August 7th 2015
Lili Dong, Suqing Zheng, Yali Zhang, Xin Jiang, Jianzhang Wu, Xiaoqin Zhang, Xiaoou Shan, Dandan Liang, Shilong Ying, Jianpeng Feng, Guang Liang

25) Tricyclic phenothiazine and phenoselenazine derivatives as potential multi-targeting agents to treat Alzheimer's disease (ChemMedComm) Friday August 7th 2015
Gary Tin, Tarek Mohamed, Nyasha Gondora, Michael Beazely, Praveen P Nekkar Rao

26) Synthesis of carboxyimidamide-substituted benzo[c][1,2,5]oxadiazoles and their analogs, and evaluation of biological activity against Leishmania donovani (ChemMedComm) Friday August 7th 2015
Leena Keurulainen, Mikko Heiskari, Satu Nenonen, Abedelmajeed Nasereddin, Dmitry Kopelyanskiy, Teppo Leino, Jari Yli-Kauhaluoma, Charles Jaffe, Paula Kiuru

27) D1-like Receptors Distinguishing Thieno-azecine Regioisomers (ChemMedComm) Wednesday August 5th 2015
Mohamed Abdel-Fattah, Ashraf H. Abadi, J Lehmann, P. Schweikert, Christoph Enzensperger

28) C-5 Substituted Pyrido[2,3-d]pyrimidin-7-ones as Highly Specific Kinase Inhibitors Targeting Clinical Resistance related EGFRT790M Mutant (ChemMedComm) Wednesday August 5th 2015
Ke Ding, Jian Ding, Hua Xie, Meiyu Geng, Linjiang Tong, Ting Peng, zhaoyu Huang, Tianfeng Xu, xiaomei Ren, Zhengchao Tu, Lianwen Zhang, zhang zhang, xiaoyun lu, Lei Yu, Jinfeng Luo

29) Induction of apoptosis by cyclobutanones and derived polycyclic γ-lactones: a preliminary analysis of antiproliferative activity (ChemMedComm) Tuesday August 4th 2015
Vishal Sharma, Ashun Chaudhary, Gousia Chashoo, Saroj Arora, Ajit K. Saxena, Mohan Paul S. Ishar

30) Novel peptidomimetics related to Gonadotropin releasing hormone (GnRH) (ChemMedComm) Tuesday July 28th 2015
Stefania Villa, Arianna Gelain, Luca Rizzi, Laura Legnani, Aurora Pacini, Katerina Spyridaki, Vlasios Karageorgos, George Liapakis

31) Enhanced Antibacterial Activities of Polythionates by Carbonate (ChemMedComm) Thursday July 23rd 2015
Guofang Li, yanbao zhao, Ping Li, Fuqiang Zhang, Peng Qu, Binjie Li, Qingyu Gao, Shaorong Wang

32) Investigating the generation of hydrogen sulfide from the phosphonamidodithioate slow-release donor GYY4137 (ChemMedComm) Thursday July 23rd 2015
Mark E. Wood, Matt Whiteman, Benjamin Edwin Alexander, Bridget Fox, Tahmina Khan, Joseph Maliszewski, Alexis Perry, Simon Coles, Mateusz Pitak

33) Structure-based design of a bisphosphonate 5'(3')-deoxyribonucleotidase inhibitor (ChemMedComm) Thursday July 23rd 2015
Petr Pachl, Ondrej Simak, Pavlina Rezacova, Milan Fabry, Milos Budesinsky, Jiri Brynda, Ivan Rosenberg

34) Inclusion of new 5-fluorouracil derivatives in liposome formulation for cancer treatment (ChemMedComm) Thursday July 23rd 2015
Manuela Petaccia, Maria condello, Luisa Giansanti, Angela La Bella, Francesca Leonelli, stefania Meschini, denise grdella villalva, evelin pellegrini, Francesca Ceccacci, Luciano Galantini, Giovanna Mancini

35) Novel 3-hydroxypyridin-4-one hexadentate ligand-based polymeric iron chelator: synthesis, characterization and antimicrobial evaluation (ChemMedComm) Monday July 20th 2015
Yingjun Zhou, Xiaole Kong, Junpei Li, Yongmin Ma, Robert Hider, Tao Zhou

36) Fragments in bromodomain drug discovery (ChemMedComm) Monday July 20th 2015
Paul Bamborough, Chun-wa Chung

37) Novel benzoxepine-1,2,3-triazole hybrids: Synthesis and pharmacological evaluation as potential antibacterial and anticancer agents (ChemMedComm) Thursday July 16th 2015
Naveen Kuntala, Jhonsee Rani Telu, Venkanna Banothu, N Suresh Babu, Jayashree anireddy, Sarbani Pal

38) GLYCODENDROPEPTIDES STIMULATE DENDRITIC CELL MATURATION AND T CELL PROLIFERATION. A POTENTIAL INFLUENZA A VIRUS IMMUNOTHERAPY. (ChemMedComm) Tuesday July 7th 2015
Ainhoa Mascaraque, Wioleta Kowalczyk, Tahia D Fernandez, Francisca Palomares, Cristobalina Mayorga, David Andreu, Javier Rojo

39) Correction: Identification of a novel class of autotaxin inhibitors through cross-screening (ChemMedComm) Tuesday July 7th 2015
Diana Castagna, Emma L. Duffy, Dima Semaan, Louise C. Young, John M. Pritchard, Simon J. F. Macdonald, David C. Budd, Craig Jamieson, Allan J. B. Watson

40) Design, synthesis and in vivo evaluation of sodium 2-benzyl-chloromalonates as new central nervous system depressants (ChemMedComm) Monday July 6th 2015
Jose Daniel Figueroa-Villar, Andreia Vieira, Bruno Marinho, Luana Souza, Patricia Fernandes

41) Correction: Discovery, synthesis and structure-activity analysis of symmetrical 2,7-disubstituted fluorenones as urea transporter inhibitors (ChemMedComm) Monday July 6th 2015
Sujin Lee, Cristina Esteva-Font, Puay-Wah Phuan, Marc O. Anderson, A. S. Verkman

42) Chemoprevention Effects of Sulindac-Based Compound on TPA-induced skin inflammation in Mice (ChemMedComm) Friday July 3rd 2015
Wenfeng Liu, Yonglian Li, Xi Zheng, kun zhang, Zhiyun Du

43) Synthesis and in vitro antiproliferative activity of novel pyrazolo[3,4-d]pyrimidine derivatives (ChemMedComm) Friday July 3rd 2015
Nermin S. Abdou, Rabah A. T. Serya, Ahmed Esmat, Mai F. Tolba, Nasser S. M. Ismail, Khaled A. M. Abouzid

44) Magic molecule modifiers (ChemMedComm) Thursday July 2nd 2015
Derek Lowe

45) The discovery of a novel antibiotic for the treatment of Clostridium difficile infections: a story of an effective academic-industrial partnership (ChemMedComm) Wednesday July 1st 2015
John Mann, Peter Taylor, Colin Dorgan, Peter Johnson, Francis X. Wilson, Richard Vickers, Aaron Dale, Stephen Neidle

46) Synthesis and anti-cancer screening of novel heterocyclic-(2H)-1,2,3-triazoles as potential anti-cancer agents (ChemMedComm) Tuesday June 30th 2015
Narsimha Penthala, Leena Maddukuri, Shraddha Thakkar, Nikhil Reddy Madadi, Gauri Lamture, Robert Eoff, Peter Crooks

47) Correction: Synthesis and biological evaluation of novel semi-conservative monocarbonyl analogs of curcumin as anti-inflammatory agents (ChemMedComm) Monday June 29th 2015
Zhe Wang, Peng Zou, Chenglong Li, Wenfei He, Bing Xiao, Qilu Fang, Wenbo Chen, Suqing Zheng, Yunjie Zhao, Yuepiao Cai, Guang Liang

48) Correction: Design, synthesis, and antibacterial evaluation of novel azolylthioether quinolones as MRSA DNA intercalators (ChemMedComm) Monday June 29th 2015
Ling Zhang, Kannekanti Vijaya Kumar, Syed Rasheed, Shao-Lin Zhang, Rong-Xia Geng, Cheng-He Zhou

49) PEGylated solid lipid nanoparticles: design, methotrexate loading and biological evaluation in animal models (ChemMedComm) Friday June 26th 2015
Dipti Kakkar, Shweta Dumoga, Rohit Kumar, Krishna Chuttani, Anil Kumar Mishra

50) Design, synthesis, and evaluation of semi-conservative mono-carbonyl analogs of curcumin as anti-inflammatory agents against lipopolysaccharide induced acute lung injury (ChemMedComm) Thursday June 25th 2015
Lili Dong, Suqing Zheng, Yali Zhang, Xin Jiang, Jianzhang Wu, Xiaoqing Zhang, Xiaoou Shan, Dandan Liang, Shilong Ying, Jianpeng Feng, Guang Liang

51) Discovery of TRAF-2 and NCK-interacting kinase (TNIK) inhibitors by ligand-based virtual screening methods (ChemMedComm) Wednesday June 24th 2015
Anna Bujak, Filip Stefaniak, Daria Zdzalik, Paulina Grygielewicz, Barbara Dymek, Marcin Zagozda, Pawel Gunerka, Monika Lamparska-Przybysz, Krzysztof Dubiel, Maciej Wieczorek, Karolina Dzwonek

52) Synthesis and anti-tubercular activity of conformationally-constrained and bisquinoline analogs of TMC207 (ChemMedComm) Tuesday June 23rd 2015
Dimpy Kalia, Anil Kumar K.S., Gajanand Meena, Kashmir Prasad Sethi, Rohit Sharma, Priyanka Trivedi, Shaheb Raj Khan, Ajay Singh Verma, Shyam Singh, Sandeep Sharma, Kuldeep K Roy, Ruchir Kant, Manju Yasodha Krishnan, Bhupendra N. Singh, Sudhir Sinha, Vinita Chaturvedi, Anil K Saxena, Dinesh K Dikshit

53) Transition Metal Diamine Complexes with Antimicrobial Activity Against Staphylococcus aureus and Methicillin-Resistant S. aureus (MRSA). (ChemMedComm) Monday June 22nd 2015
Joseph S Merola, George Karpin, David Morris, Mai Ngo, Joseph Falkinham

54) Synthesis and biological evaluation of α-sulfonamido-N-adamantanecarboxamide derivatives as 11β-HSD1 inhibitors (ChemMedComm) Thursday June 18th 2015
Young Hoon Kim, Seung Kyu Kang, Gwi Bin Lee, Kyu Myung Lee, Jaladi Ashok Kumar, Ki Young Kim, Sang Dal Rhee, Jeongmin Joo, Myung Ae Bae, Won Koo Lee, Jin Hee Ahn

55) Design and synthesis of potent and selective inhibitors of BRD9 and BRD7 bromodomains. (ChemMedComm) Monday June 15th 2015
Duncan Hay, Paul Brennan, Oleg Fedorov, Cynthia Tallant, Octovia Monteiro, Susanne Muller-Knapp, Stefan Knapp, Christopher J Schofield, Sarah Martin, Catherine Rogers

56) Identification of new hit scaffolds by INPHARMA-guided virtual screening (ChemMedComm) Monday June 15th 2015
Teresa Carlomagno, Justyna Sikorska, Luca Codutti, Lars Skjaerven, Bettina Elshorst, Rebeca Saez Ameneiro, Andrea Angelini, Peter Monecke

57) Correction: Synthesis and biological evaluation of N-(4-phenylthiazol-2-yl)cinnamamide derivatives as novel potential anti-tumor agents (ChemMedComm) Monday June 15th 2015
Yong Luo, Yongxia Zhu, Kai Ran, Zhihao Liu, Ningyu Wang, Qiang Feng, Jun Zeng, Lidan Zhang, Bing He, Tinghong Ye, Shirui Zhu, Xiaolong Qiu, Luoting Yu

58) Synthesis of novel 1-substituted triazole linked 1,2-benzothiazine 1,1-dioxido propenone derivatives as potent anti-inflammatory agents and inhibitors of monocyte-to-macrophage differentiation (ChemMedComm) Saturday June 13th 2015
B Narsaiah, Malla Reddy GANNARAPU, Sathish Babu Vasamsetti, nagender punna, Srigiridhar Kotamraju

59) Enhanced in vitro and in vivo uptake of a hydrophobic model drug coumarin-6 in the presence of cucurbit[7]uril (ChemMedComm) Friday June 12th 2015
Xiaoqing Miao, Ye Li, Ian Wyman, Simon Ming-Yuen Lee, Donal H Macartney, Ying Zheng, Ruibing Wang

60) Discovery of C-shaped aurone human neutrophil elastase inhibitors (ChemMedComm) Friday June 12th 2015
Susana Dias Lucas, Marta P. Carrasco, Lidia M. Goncalves, Rui Moreira, Rita Cardoso Guedes

61) Synthesis and biological evaluation of 4′-[(benzimidazol-1-yl) methyl] biphenyl-2-amides as dual angiotensin II and endothelin A receptor antagonists (ChemMedComm) Wednesday June 10th 2015
Xiaofeng Han, Weizhe Xue, Liping Hao, Zhiming Zhou

62) Synthesis and biological evaluation of lipid like 5-(2-hydroxyethyl)-4-methyl-1,3-thiazole derivatives as potential anticancer and antimicrobial agents (ChemMedComm) Wednesday June 10th 2015
Alla Zablotskaya, Izolda Segal, Prof. Athina Geronikaki, Galina Kazachonokh, Yuris Popelis, Irina Shestakova, Vizma Prof. Nikolajeva, Daina Eze

63) Discovery of Anilinopyrimidine-Based Naphthamide Derivatives as Potent VEGFR-2 Inhibitors (ChemMedComm) Monday June 8th 2015
Yongcong Lv, Mengyuan Li, Sufen Cao, Linjiang Tong, Ting Peng, Lixin Wei, Hua Xie, Jian Ding, Wenhu Duan

64) Identifying Farnesoid X Receptor Agonists with Naive Bayesian and Recursive Partitioning Approaches (ChemMedComm) Monday June 8th 2015
Qianzhi Ding, Chanjuan Li, Ling Wang, Yali Li, Huihao Zhou, Qiong Gu, Jun Xu

65) Novel Difluoroacetamide Analogues of Agomelatine and Melatonin: Probing the Melatonin Receptors for MT1-Selectivity (ChemMedComm) Monday June 8th 2015
Darius Paul Zlotos, Noura Riad, Mai Osman, Bala R. Dodda, Paula Witt-Enderby

66) Transcutaneous immunization against cancer using a solid-in-oil nanodispersion (ChemMedComm) Monday June 8th 2015
Yuya Hirakawa, Rie Wakabayashi, Ayaka Naritomi, Masato Sakuragi, Noriho Kamiya, Masahiro Goto

67) Effect of dibucaine hydrochloride on raft-like lipid domains in model membrane systems (ChemMedComm) Monday June 8th 2015
Kazunari Yoshida, Akito Takashima, Izumi Nishio

68) Discovery, synthesis and structure-activity analysis of symmetrical 2,7-disubstituted fluorenones as urea transporter inhibitors (ChemMedComm) Friday June 5th 2015
Sujin Lee, Cristina Esteva-Font, Puay-wah Phuan, Marc O. Anderson, Alan S. Verkman

69) RGD-peptides modifying dexamethasone: To enhance the efficacy of anti-inflammation and limit the risk of osteoporosis (ChemMedComm) Thursday June 4th 2015
Hualong Yu, Shenghui Mei, Zhao Li, Ming Zhao, Yuji Wang, Haimei Zhu, Yaonan Wang, Jianhui Wu, Chunying Cui, Wenyun Xu, Shiqi Peng

70) Substituted 4-hydroxy-1,2,3-triazoles: synthesis, characterization and first drug design applications through bioisosteric modulation and scaffold hopping approaches (ChemMedComm) Thursday May 28th 2015
Agnese Chiara Pippione, Franco Dosio, Alex Ducime, Antonella Federico, Katia Martina, Stefano Sainas, Bente Frolund, Major Gooyit, Kim D Janda, Donatella Boschi, Marco Lucio Lolli

71) Identifying the inhibitory mechanism of apigenin on the insulin ligand-receptor binding (ChemMedComm) Wednesday May 27th 2015
Yong Yang

72) Identification of an indole-triazole-amino acid conjugate as highly effective antifungal agent (ChemMedComm) Tuesday May 26th 2015
Kalpana Pawar, Anshuman Yadav, Parteek Prasher, Sahil Mishra, Balwinder Singh, Palwinder Singh, Sneha Komath

73) Synthesis and biological evaluation of novel semi-conservative mono-carbonyl analogs of curcumin as anti-inflammatory agents (ChemMedComm) Tuesday May 26th 2015
Zhe Wang, Peng Zou, Chenglong Li, Wenfei He, Bing Xiao, Qilu Fang, Wenbo Chen, Suqing Zheng, Yunjie Zhao, Yuepiao Cai, Guang Liang

74) Medicinal Organometallic Chemistry - an Emerging Strategy for the Treatment for Neglected Tropical Diseases (ChemMedComm) Tuesday May 26th 2015
Christopher Hyland, Ronald Brown

75) Design, Synthesis, Antibacterial Evaluation of Novel Azolylthioether Quinolones as MRSA DNA Intercalators (ChemMedComm) Thursday May 21st 2015
Ling Zhang, Vijaya Kumar Kannekanti, RASHEED SYED, Shao-Lin Zhang, Rong-Xia Geng, Cheng-He Zhou

76) Discovery of novel amino-pyrimidine inhibitors of the insulin-like growth factor 1 (IGF1R) and insulin receptor (INSR) kinases; parallel optimization of cell potency and hERG inhibition (ChemMedComm) Thursday May 21st 2015
Heather Tye, Stephan Zahn, Marco Hofmann, Michael Sanderson, Otmar Schaff, Matthias Troy, Moritz Mayer, Georg Rast, Sandeep Pal, Ulrich Guertler

77) Synthesis and antibacterial activity evaluation of C-5 side chain modified analogues of FYL-66, a potential agent against methicillin-resistant Staphylococcus aureus (ChemMedComm) Thursday May 21st 2015
Xiaoyan Yang, Zicheng Li, Zhenling Wang, Zitai Sang, Haiyue Long, Jianying Tang, Tao Yang, Yuanyuan Liu, Youfu Luo

78) 5-Iodo-2-arylalkylthio-6-aryl pyrimidin-4(3H)-ones as non-nucleoside anti-HBV agents (ChemMedComm) Wednesday May 20th 2015
Yu Zhang, Xuefeng Sun, Ningning Fan, Jianxiong Zhao, Jing Tu, Xiangmei Chen, Junyi Liu, Xiao-wei Wang

79) Alkylamino derivatives of N-benzylpyrazine-2-carboxamide: Synthesis and antimycobacterial evaluation (ChemMedComm) Wednesday May 20th 2015
Barbora Servusova-Vanaskova, Ondrej Jandourek, Pavla Paterova, Jana Kordulakova, Magdalena Plevakova, Vladimir Kubicek, Radim Kucera, Vladimir Garaj, Lieve Naesens, Jiri Kunes, Martin Dolezal, Jan Zitko

80) Synthesis and biological evaluation of potential small molecule inhibitors of Tumor Necrosis Factor (ChemMedComm) Wednesday May 20th 2015
Christos Papaneophytou, Polyxeni Alexiou, Athanasios Papakyriakou, Evangelos Ntougkos, Katerina Tsiliouka, Anna Maranti, Fotini Liepouri, Alexandros Strongilos, Anthi Mettou, Elias Couladouros, Elias Eliopoulos, Eleni Douni, George Kollias, George Kontopidis

81) Chromanones: selective and reversible Monoamine Oxidase B inhibitors with nanomolar potency (ChemMedComm) Wednesday May 20th 2015
Jin-Shuai Lan, Sai-Sai Xie, Ming Huang, Ya-Jian Hu, Ling-Yi Kong, Xiao-Bing Wang

82) Arylsulfonamide derivatives of (aryloxy)ethylpiperidines as 5-HT7 receptor antagonists and their psychotropic properties (ChemMedComm) Tuesday May 19th 2015
Pawel Maria Zajdel, Vittorio Canale, Anna Partyka, Krzysztof Marciniec, Grzegorz Satala, Rafal Kurczab, Agata Siwek, Magdalena Jastrzebska-Wiesek, Anna Wesolowska, Tomasz Kos, Piotr Popik, AJ Bojarski

83) Synthesis and in vitro Assessment of Chemically Modified siRNAs Targeting BCL2 that Contain 2'-Ribose and Triazole-linked Backbone Modifications (ChemMedComm) Monday May 18th 2015
Gord Hagen, Brandon J Peel, John Samis, Jean-Paul Desaulniers

84) Fragment-growing exploiting dynamic combinatorial chemistry of inhibitors of the aspartic protease endothiapepsin (ChemMedComm) Friday May 15th 2015
Milon Mondal, Daphne Groothuis, Anna Katharina Herta Hirsch

85) New selective A2A agonists and A3 antagonists for human adenosine receptors. Synthesis, biological activity and molecular docking studies (ChemMedComm) Wednesday May 13th 2015
Angel Guerrero, Anna Rodriguez, Hugo Gutierrez-de-Teran, David Rodriguez, Jose Brea, Maria Isabel Loza, Gloria Rosell, M. Pilar Bosch

86) A novel aminotriazole-based NHC complex for the design of gold(I) anti-cancer agents: synthesis and biological evaluation (ChemMedComm) Wednesday May 13th 2015
Tatiyana V Serebryanskaya, Andrey A. Zolotarev, Ingo Ott

87) 1,2,3-Triazole derivatives as antitubercular agents: synthesis, biological evaluation and molecular docking study (ChemMedComm) Wednesday May 13th 2015
Mubarak H. Shaikh, Dnyaneshwar D. Subhedar, Laxman Nawale, Dhiman Sarkar, Firoz A. Kalam Khan, Jaiprakash N. Sangshetti, Bapurao B. Shingate

88) Synthesis, Biological Evaluation and Mechanisms Study of a Class of Benzylideneindanone Derivatives as Novel Anticancer Agents (ChemMedComm) Friday May 8th 2015
Jinhui Hu, Jun Yan, Jie Chen, Yanqing Pang, ling huang, Xingshu Li

89) Identification of a novel class of Autotaxin inhibitors through cross-screening (ChemMedComm) Friday May 8th 2015
Diana Castagna, Emma Duffy, Dima Semaan, Louise Young, John Pritchard, simon macdonald, David Budd, Craig Jamieson, Allan John Bell Watson

90) Synthesis and evaluation of novel N-3-benzimidazolephenylbisamide derivatives for antiproliferative and hedgehog pathway inhibitory activity (ChemMedComm) Wednesday May 6th 2015
Chiyu Sun, Yangsheng Li, Ailong Shi, Jingzhou Zhang, Yafei Li, Mingming Zhao, Lijuan Zhang, Huachuan Zheng, Ying Meng, Huaiwei Ding, Hongrui Song

91) Synthesis and biological evaluation of nitric oxide-releasing hybrids from gemcitabine and phenylsulfonyl furoxans as anti-tumor agents (ChemMedComm) Wednesday April 29th 2015
Xianghua Li, Xuemin Wang, Chenjun Xu, Junkai Huang, Chengniu Wang, Xinyang Wang, Yong Ling, Liqin He

92) Synthesis and biodistribution of novel 99mTc labeled 4-nitroimidazole dithiocarbamate complexes as potential agents to target tumor hypoxia (ChemMedComm) Thursday April 23rd 2015
zhenxiang li, Junbo zhang, zhonghui jin, weifang zhang, Yanyan zhang

93) Synthesis and evaluation of [11C]PBD150, a radiolabeled glutaminyl cyclase inhibitor for the potential detection of Alzheimer's disease prior to amyloid β aggregation. (ChemMedComm) Thursday April 23rd 2015
Allen F Brooks, Isaac Jackson, Xia Shao, George Kropog, Phillip Sherman, Carole Quesada, Peter Scott

94) Discovery and optimisation of 1-acyl-2-benzylpyrrolidines as potent dual orexin receptor antagonists (ChemMedComm) Tuesday April 21st 2015
Jodi Williams, John Gatfield, Catherine Roch, Alexander Treiber, Francois Jenck, Martin Bolli, Christine Brotschi, Thierry Sifferlen, Bibia Heidmann, Christoph Boss

95) Novel indole-based sigma-2 receptor ligands: synthesis, structure-affinity relationship and antiproliferative activity (ChemMedComm) Monday April 20th 2015
Fang Xie, Torsten Kniess, Christin Neuber, Winnie Deuther-Conrad, Constantin Mamat, Brian P. Lieberman, BL Liu, Robert Henry Mach, Peter Brust, Jorg Steinbach, Jens Pietzsch, Hongmei Jia

96) Target-based Analysis of Ionization States of Bioactive Compounds (ChemMedComm) Monday April 20th 2015
Shilva Kayastha, Antonio de la Vega de Leon, Dilyana Dimova, J Bajorath

97) Exploring the Recognition Pathway at the Human A2A Adenosine Receptor of the Endogenous Agonist Adenosine using Supervised Molecular Dynamics Simulations. (ChemMedComm) Monday April 20th 2015
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