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1) Synthesis and in vitro antiproliferative activity of novel pyrazolo[3,4-d]pyrimidine derivatives (ChemMedComm) Friday July 3rd 2015
Nermin S. Abdou, Rabah A. T. Serya, Ahmed Esmat, Mai F. Tolba, Nasser S. M. Ismail, Khaled A. M. Abouzid

2) Magic molecule modifiers (ChemMedComm) Thursday July 2nd 2015
Derek Lowe

3) The discovery of a novel antibiotic for the treatment of Clostridium difficile infections: a story of an effective academic-industrial partnership (ChemMedComm) Wednesday July 1st 2015
John Mann, Peter Taylor, Colin Dorgan, Peter Johnson, Francis X. Wilson, Richard Vickers, Aaron Dale, Stephen Neidle

4) Synthesis and anti-cancer screening of novel heterocyclic-(2H)-1,2,3-triazoles as potential anti-cancer agents (ChemMedComm) Tuesday June 30th 2015
Narsimha Penthala, Leena Maddukuri, Shraddha Thakkar, Nikhil Reddy Madadi, Gauri Lamture, Robert Eoff, Peter Crooks

5) Correction: Synthesis and biological evaluation of novel semi-conservative monocarbonyl analogs of curcumin as anti-inflammatory agents (ChemMedComm) Monday June 29th 2015
Zhe Wang, Peng Zou, Chenglong Li, Wenfei He, Bing Xiao, Qilu Fang, Wenbo Chen, Suqing Zheng, Yunjie Zhao, Yuepiao Cai, Guang Liang

6) Correction: Design, synthesis, and antibacterial evaluation of novel azolylthioether quinolones as MRSA DNA intercalators (ChemMedComm) Monday June 29th 2015
Ling Zhang, Kannekanti Vijaya Kumar, Syed Rasheed, Shao-Lin Zhang, Rong-Xia Geng, Cheng-He Zhou

7) PEGylated solid lipid nanoparticles: design, methotrexate loading and biological evaluation in animal models (ChemMedComm) Friday June 26th 2015
Dipti Kakkar, Shweta Dumoga, Rohit Kumar, Krishna Chuttani, Anil Kumar Mishra

8) Design, synthesis, and evaluation of semi-conservative mono-carbonyl analogs of curcumin as anti-inflammatory agents against lipopolysaccharide induced acute lung injury (ChemMedComm) Thursday June 25th 2015
Lili Dong, Suqing Zheng, Yali Zhang, Xin Jiang, Jianzhang Wu, Xiaoqing Zhang, Xiaoou Shan, Dandan Liang, Shilong Ying, Jianpeng Feng, Guang Liang

9) Discovery of TRAF-2 and NCK-interacting kinase (TNIK) inhibitors by ligand-based virtual screening methods (ChemMedComm) Wednesday June 24th 2015
Anna Bujak, Filip Stefaniak, Daria Zdzalik, Paulina Grygielewicz, Barbara Dymek, Marcin Zagozda, Pawel Gunerka, Monika Lamparska-Przybysz, Krzysztof Dubiel, Maciej Wieczorek, Karolina Dzwonek

10) Synthesis and anti-tubercular activity of conformationally-constrained and bisquinoline analogs of TMC207 (ChemMedComm) Tuesday June 23rd 2015
Dimpy Kalia, Anil Kumar K.S., Gajanand Meena, Kashmir Prasad Sethi, Rohit Sharma, Priyanka Trivedi, Shaheb Raj Khan, Ajay Singh Verma, Shyam Singh, Sandeep Sharma, Kuldeep K Roy, Ruchir Kant, Manju Yasodha Krishnan, Bhupendra N. Singh, Sudhir Sinha, Vinita Chaturvedi, Anil K Saxena, Dinesh K Dikshit

11) Transition Metal Diamine Complexes with Antimicrobial Activity Against Staphylococcus aureus and Methicillin-Resistant S. aureus (MRSA). (ChemMedComm) Monday June 22nd 2015
Joseph S Merola, George Karpin, David Morris, Mai Ngo, Joseph Falkinham

12) Synthesis and biological evaluation of α-sulfonamido-N-adamantanecarboxamide derivatives as 11β-HSD1 inhibitors (ChemMedComm) Thursday June 18th 2015
Young Hoon Kim, Seung Kyu Kang, Gwi Bin Lee, Kyu Myung Lee, Jaladi Ashok Kumar, Ki Young Kim, Sang Dal Rhee, Jeongmin Joo, Myung Ae Bae, Won Koo Lee, Jin Hee Ahn

13) Design and synthesis of potent and selective inhibitors of BRD9 and BRD7 bromodomains. (ChemMedComm) Monday June 15th 2015
Duncan Hay, Paul Brennan, Oleg Fedorov, Cynthia Tallant, Octovia Monteiro, Susanne Muller-Knapp, Stefan Knapp, Christopher J Schofield, Sarah Martin, Catherine Rogers

14) Identification of new hit scaffolds by INPHARMA-guided virtual screening (ChemMedComm) Monday June 15th 2015
Teresa Carlomagno, Justyna Sikorska, Luca Codutti, Lars Skjaerven, Bettina Elshorst, Rebeca Saez Ameneiro, Andrea Angelini, Peter Monecke

15) Correction: Synthesis and biological evaluation of N-(4-phenylthiazol-2-yl)cinnamamide derivatives as novel potential anti-tumor agents (ChemMedComm) Monday June 15th 2015
Yong Luo, Yongxia Zhu, Kai Ran, Zhihao Liu, Ningyu Wang, Qiang Feng, Jun Zeng, Lidan Zhang, Bing He, Tinghong Ye, Shirui Zhu, Xiaolong Qiu, Luoting Yu

16) Synthesis of novel 1-substituted triazole linked 1,2-benzothiazine 1,1-dioxido propenone derivatives as potent anti-inflammatory agents and inhibitors of monocyte-to-macrophage differentiation (ChemMedComm) Saturday June 13th 2015
B Narsaiah, Malla Reddy GANNARAPU, Sathish Babu Vasamsetti, nagender punna, Srigiridhar Kotamraju

17) Enhanced in vitro and in vivo uptake of a hydrophobic model drug coumarin-6 in the presence of cucurbit[7]uril (ChemMedComm) Friday June 12th 2015
Xiaoqing Miao, Ye Li, Ian Wyman, Simon Ming-Yuen Lee, Donal H Macartney, Ying Zheng, Ruibing Wang

18) Discovery of C-shaped aurone human neutrophil elastase inhibitors (ChemMedComm) Friday June 12th 2015
Susana Dias Lucas, Marta P. Carrasco, Lidia M. Goncalves, Rui Moreira, Rita Cardoso Guedes

19) Synthesis and biological evaluation of 4′-[(benzimidazol-1-yl) methyl] biphenyl-2-amides as dual angiotensin II and endothelin A receptor antagonists (ChemMedComm) Wednesday June 10th 2015
Xiaofeng Han, Weizhe Xue, Liping Hao, Zhiming Zhou

20) Synthesis and biological evaluation of lipid like 5-(2-hydroxyethyl)-4-methyl-1,3-thiazole derivatives as potential anticancer and antimicrobial agents (ChemMedComm) Wednesday June 10th 2015
Alla Zablotskaya, Izolda Segal, Prof. Athina Geronikaki, Galina Kazachonokh, Yuris Popelis, Irina Shestakova, Vizma Prof. Nikolajeva, Daina Eze

21) Discovery of Anilinopyrimidine-Based Naphthamide Derivatives as Potent VEGFR-2 Inhibitors (ChemMedComm) Monday June 8th 2015
Yongcong Lv, Mengyuan Li, Sufen Cao, Linjiang Tong, Ting Peng, Lixin Wei, Hua Xie, Jian Ding, Wenhu Duan

22) Identifying Farnesoid X Receptor Agonists with Naive Bayesian and Recursive Partitioning Approaches (ChemMedComm) Monday June 8th 2015
Qianzhi Ding, Chanjuan Li, Ling Wang, Yali Li, Huihao Zhou, Qiong Gu, Jun Xu

23) Novel Difluoroacetamide Analogues of Agomelatine and Melatonin: Probing the Melatonin Receptors for MT1-Selectivity (ChemMedComm) Monday June 8th 2015
Darius Paul Zlotos, Noura Riad, Mai Osman, Bala R. Dodda, Paula Witt-Enderby

24) Transcutaneous immunization against cancer using a solid-in-oil nanodispersion (ChemMedComm) Monday June 8th 2015
Yuya Hirakawa, Rie Wakabayashi, Ayaka Naritomi, Masato Sakuragi, Noriho Kamiya, Masahiro Goto

25) Effect of dibucaine hydrochloride on raft-like lipid domains in model membrane systems (ChemMedComm) Monday June 8th 2015
Kazunari Yoshida, Akito Takashima, Izumi Nishio

26) Discovery, synthesis and structure-activity analysis of symmetrical 2,7-disubstituted fluorenones as urea transporter inhibitors (ChemMedComm) Friday June 5th 2015
Sujin Lee, Cristina Esteva-Font, Puay-wah Phuan, Marc O. Anderson, Alan S. Verkman

27) RGD-peptides modifying dexamethasone: To enhance the efficacy of anti-inflammation and limit the risk of osteoporosis (ChemMedComm) Thursday June 4th 2015
Hualong Yu, Shenghui Mei, Zhao Li, Ming Zhao, Yuji Wang, Haimei Zhu, Yaonan Wang, Jianhui Wu, Chunying Cui, Wenyun Xu, Shiqi Peng

28) Substituted 4-hydroxy-1,2,3-triazoles: synthesis, characterization and first drug design applications through bioisosteric modulation and scaffold hopping approaches (ChemMedComm) Thursday May 28th 2015
Agnese Chiara Pippione, Franco Dosio, Alex Ducime, Antonella Federico, Katia Martina, Stefano Sainas, Bente Frolund, Major Gooyit, Kim D Janda, Donatella Boschi, Marco Lucio Lolli

29) Identifying the inhibitory mechanism of apigenin on the insulin ligand-receptor binding (ChemMedComm) Wednesday May 27th 2015
Yong Yang

30) Identification of an indole-triazole-amino acid conjugate as highly effective antifungal agent (ChemMedComm) Tuesday May 26th 2015
Kalpana Pawar, Anshuman Yadav, Parteek Prasher, Sahil Mishra, Balwinder Singh, Palwinder Singh, Sneha Komath

31) Synthesis and biological evaluation of novel semi-conservative mono-carbonyl analogs of curcumin as anti-inflammatory agents (ChemMedComm) Tuesday May 26th 2015
Zhe Wang, Peng Zou, Chenglong Li, Wenfei He, Bing Xiao, Qilu Fang, Wenbo Chen, Suqing Zheng, Yunjie Zhao, Yuepiao Cai, Guang Liang

32) Medicinal Organometallic Chemistry - an Emerging Strategy for the Treatment for Neglected Tropical Diseases (ChemMedComm) Tuesday May 26th 2015
Christopher Hyland, Ronald Brown

33) Design, Synthesis, Antibacterial Evaluation of Novel Azolylthioether Quinolones as MRSA DNA Intercalators (ChemMedComm) Thursday May 21st 2015
Ling Zhang, Vijaya Kumar Kannekanti, RASHEED SYED, Shao-Lin Zhang, Rong-Xia Geng, Cheng-He Zhou

34) Discovery of novel amino-pyrimidine inhibitors of the insulin-like growth factor 1 (IGF1R) and insulin receptor (INSR) kinases; parallel optimization of cell potency and hERG inhibition (ChemMedComm) Thursday May 21st 2015
Heather Tye, Stephan Zahn, Marco Hofmann, Michael Sanderson, Otmar Schaff, Matthias Troy, Moritz Mayer, Georg Rast, Sandeep Pal, Ulrich Guertler

35) Synthesis and antibacterial activity evaluation of C-5 side chain modified analogues of FYL-66, a potential agent against methicillin-resistant Staphylococcus aureus (ChemMedComm) Thursday May 21st 2015
Xiaoyan Yang, Zicheng Li, Zhenling Wang, Zitai Sang, Haiyue Long, Jianying Tang, Tao Yang, Yuanyuan Liu, Youfu Luo

36) 5-Iodo-2-arylalkylthio-6-aryl pyrimidin-4(3H)-ones as non-nucleoside anti-HBV agents (ChemMedComm) Wednesday May 20th 2015
Yu Zhang, Xuefeng Sun, Ningning Fan, Jianxiong Zhao, Jing Tu, Xiangmei Chen, Junyi Liu, Xiao-wei Wang

37) Alkylamino derivatives of N-benzylpyrazine-2-carboxamide: Synthesis and antimycobacterial evaluation (ChemMedComm) Wednesday May 20th 2015
Barbora Servusova-Vanaskova, Ondrej Jandourek, Pavla Paterova, Jana Kordulakova, Magdalena Plevakova, Vladimir Kubicek, Radim Kucera, Vladimir Garaj, Lieve Naesens, Jiri Kunes, Martin Dolezal, Jan Zitko

38) Synthesis and biological evaluation of potential small molecule inhibitors of Tumor Necrosis Factor (ChemMedComm) Wednesday May 20th 2015
Christos Papaneophytou, Polyxeni Alexiou, Athanasios Papakyriakou, Evangelos Ntougkos, Katerina Tsiliouka, Anna Maranti, Fotini Liepouri, Alexandros Strongilos, Anthi Mettou, Elias Couladouros, Elias Eliopoulos, Eleni Douni, George Kollias, George Kontopidis

39) Chromanones: selective and reversible Monoamine Oxidase B inhibitors with nanomolar potency (ChemMedComm) Wednesday May 20th 2015
Jin-Shuai Lan, Sai-Sai Xie, Ming Huang, Ya-Jian Hu, Ling-Yi Kong, Xiao-Bing Wang

40) Arylsulfonamide derivatives of (aryloxy)ethylpiperidines as 5-HT7 receptor antagonists and their psychotropic properties (ChemMedComm) Tuesday May 19th 2015
Pawel Maria Zajdel, Vittorio Canale, Anna Partyka, Krzysztof Marciniec, Grzegorz Satala, Rafal Kurczab, Agata Siwek, Magdalena Jastrzebska-Wiesek, Anna Wesolowska, Tomasz Kos, Piotr Popik, AJ Bojarski

41) Synthesis and in vitro Assessment of Chemically Modified siRNAs Targeting BCL2 that Contain 2'-Ribose and Triazole-linked Backbone Modifications (ChemMedComm) Monday May 18th 2015
Gord Hagen, Brandon J Peel, John Samis, Jean-Paul Desaulniers

42) Fragment-growing exploiting dynamic combinatorial chemistry of inhibitors of the aspartic protease endothiapepsin (ChemMedComm) Friday May 15th 2015
Milon Mondal, Daphne Groothuis, Anna Katharina Herta Hirsch

43) New selective A2A agonists and A3 antagonists for human adenosine receptors. Synthesis, biological activity and molecular docking studies (ChemMedComm) Wednesday May 13th 2015
Angel Guerrero, Anna Rodriguez, Hugo Gutierrez-de-Teran, David Rodriguez, Jose Brea, Maria Isabel Loza, Gloria Rosell, M. Pilar Bosch

44) A novel aminotriazole-based NHC complex for the design of gold(I) anti-cancer agents: synthesis and biological evaluation (ChemMedComm) Wednesday May 13th 2015
Tatiyana V Serebryanskaya, Andrey A. Zolotarev, Ingo Ott

45) 1,2,3-Triazole derivatives as antitubercular agents: synthesis, biological evaluation and molecular docking study (ChemMedComm) Wednesday May 13th 2015
Mubarak H. Shaikh, Dnyaneshwar D. Subhedar, Laxman Nawale, Dhiman Sarkar, Firoz A. Kalam Khan, Jaiprakash N. Sangshetti, Bapurao B. Shingate

46) Synthesis, Biological Evaluation and Mechanisms Study of a Class of Benzylideneindanone Derivatives as Novel Anticancer Agents (ChemMedComm) Friday May 8th 2015
Jinhui Hu, Jun Yan, Jie Chen, Yanqing Pang, ling huang, Xingshu Li

47) Identification of a novel class of Autotaxin inhibitors through cross-screening (ChemMedComm) Friday May 8th 2015
Diana Castagna, Emma Duffy, Dima Semaan, Louise Young, John Pritchard, simon macdonald, David Budd, Craig Jamieson, Allan John Bell Watson

48) Synthesis and evaluation of novel N-3-benzimidazolephenylbisamide derivatives for antiproliferative and hedgehog pathway inhibitory activity (ChemMedComm) Wednesday May 6th 2015
Chiyu Sun, Yangsheng Li, Ailong Shi, Jingzhou Zhang, Yafei Li, Mingming Zhao, Lijuan Zhang, Huachuan Zheng, Ying Meng, Huaiwei Ding, Hongrui Song

49) Synthesis and biological evaluation of nitric oxide-releasing hybrids from gemcitabine and phenylsulfonyl furoxans as anti-tumor agents (ChemMedComm) Wednesday April 29th 2015
Xianghua Li, Xuemin Wang, Chenjun Xu, Junkai Huang, Chengniu Wang, Xinyang Wang, Yong Ling, Liqin He

50) Synthesis and biodistribution of novel 99mTc labeled 4-nitroimidazole dithiocarbamate complexes as potential agents to target tumor hypoxia (ChemMedComm) Thursday April 23rd 2015
zhenxiang li, Junbo zhang, zhonghui jin, weifang zhang, Yanyan zhang

51) Synthesis and evaluation of [11C]PBD150, a radiolabeled glutaminyl cyclase inhibitor for the potential detection of Alzheimer's disease prior to amyloid β aggregation. (ChemMedComm) Thursday April 23rd 2015
Allen F Brooks, Isaac Jackson, Xia Shao, George Kropog, Phillip Sherman, Carole Quesada, Peter Scott

52) Discovery and optimisation of 1-acyl-2-benzylpyrrolidines as potent dual orexin receptor antagonists (ChemMedComm) Tuesday April 21st 2015
Jodi Williams, John Gatfield, Catherine Roch, Alexander Treiber, Francois Jenck, Martin Bolli, Christine Brotschi, Thierry Sifferlen, Bibia Heidmann, Christoph Boss

53) Novel indole-based sigma-2 receptor ligands: synthesis, structure-affinity relationship and antiproliferative activity (ChemMedComm) Monday April 20th 2015
Fang Xie, Torsten Kniess, Christin Neuber, Winnie Deuther-Conrad, Constantin Mamat, Brian P. Lieberman, BL Liu, Robert Henry Mach, Peter Brust, Jorg Steinbach, Jens Pietzsch, Hongmei Jia

54) Target-based Analysis of Ionization States of Bioactive Compounds (ChemMedComm) Monday April 20th 2015
Shilva Kayastha, Antonio de la Vega de Leon, Dilyana Dimova, J Bajorath

55) Exploring the Recognition Pathway at the Human A2A Adenosine Receptor of the Endogenous Agonist Adenosine using Supervised Molecular Dynamics Simulations. (ChemMedComm) Monday April 20th 2015
Davide Sabbadin, Antonella Ciancetta, Giuseppe Deganutti, Alberto Cuzzolin, Stefano Moro

56) 3-Aminooxazolidinone AHL analogs as hydrolytically-stable quorum sensing agonists in Gram-negative bacteria (ChemMedComm) Monday April 20th 2015
Min Guo, Yue Zheng, Clement Opoku-Temeng, Rusty Starks, Xiaochu Ma, Herman O Sintim

57) Synthesis, biological evaluation and QSAR studies of diarylpentanoid analogues as potential nitric oxide inhibitors (ChemMedComm) Monday April 20th 2015
Siti Munirah Mohd Faudzi, Sze Wei Leong, Faridah Abas, Mohd Fadhlizil Fasihi Mohd Aluwi, Kamal Rullah, Kok Wai Lam, Syahida Ahmad, Chau Ling Tham, Khozirah Shaari, Nordin H Lajis

58) Neuronal selective targeting, protection and signaling network analysis via dopamine mediated mesoporous silica nanoparticle (ChemMedComm) Monday April 20th 2015
shupeng li, hailong zhang, Yuhua Jiang, Sheng-gang Zhao, Li-qin Jiang, Yan Meng, Peng Liu, Myeong Ok Kim

59) Exploring cinnamic acid scaffold: development of promising neuroprotective lipophilic antioxidants (ChemMedComm) Wednesday April 15th 2015
Fernanda Borges, Daniel Chavarria, Tiago Silva, Teresa Summavielle, Jorge M.P.J. Garrido, Daniel Martins, Joana Bravo

60) Synthesis and Biological Evaluation of N-(4-phenylthiazol-2-yl) Cinnamamide Derivatives as Novel Potential Anti-tumor Agents (ChemMedComm) Monday April 13th 2015
Yong Luo, Yongxia Zhu, Kai Ran, Zhihao Liu, Ningyu Wang, Qiang Feng, Jun Zeng, Lidan Zhang, Bing He, Tinghong Ye, Shirui Zhu, Xiaolong Qiu, Luoting Yu

61) Direct photocapture of bromodomains using tropolone chemical probes (ChemMedComm) Monday April 13th 2015
Erik Hett, Eugene Chekler, Arindrajit Basak, Paul Bonin, Aldrin Denny, Andrew Flick, Kieran F Geoghegan, Shenping Liu, Mathew Pletcher, Parag Sahasrabudhe, Shores Salter, Ingrid Stock, Alex Taylor, Lyn H Jones

62) Discovery of a series of 2-(pyridinyl)pyrimidines as potent antagonists of GPR40 (ChemMedComm) Wednesday April 8th 2015
M J Waring, David Baker, Stuart Bennett, Alastair Dossetter, Mark Fenwick, Rob Garcia, Jennie Georgsson, Sam Groombridge, Sue Loxham, Philip Alexander MacFaul, Katie Maskill, David Morgan, Jenny Morrell, Helen Pointon, Graeme Robb, David Smith, Stephen Stokes, Gary Paul Wilkinson

63) Synthesis and Biological Evaluations of 2,3-Diarylthiophene Analogues of Combretastatin A-4 (ChemMedComm) Thursday April 2nd 2015
Weige Zhang, Zhan Wang, qingkun Yang, Zhaoshi Bai, Jun Sun, xuewei Jiang, Hongrui Song, Yingliang Wu

64) New substituted 9-propyladenine derivatives as adenosine receptor antagonists (ChemMedComm) Thursday April 2nd 2015
Catia Lambertucci, Michela Buccioni, Diego Dal Ben, Sonja Kachler, Gabriella Marucci, Andrea Spinaci, Ajiroghene Thomas, Karl-Norbert Klotz, R Volpini

65) Enantiomeric Diketopiperazines: Getting Insight of the Impact of the Configuration to the Conformation, Nanoimage, u-PA Inhibition and Anti-metastatic Activity (ChemMedComm) Tuesday March 31st 2015
Feng Wang, Shan Li, Yuji Wang, Haimei Zhu, Xiaoyi Zhang, Ming Zhao, Jianhui Wu, Shiqi Peng

66) Chemical genomics reveals novel biological activity of 1,2,3-dithiazoles as potent and reversible melanin synthesis inhibitors (ChemMedComm) Tuesday March 31st 2015
Panayiotis Andreas Koutentis, Paris Skourides, Oleg Alekseevich Rakitin, Anna Charalambous, Maria Koyioni, Ioanna Antoniades, Sophia Michaelidou, Iro Eleftheriou, Stanislav A Amelichev, Lidia S konstantinova, Despoina Pegeioti

67) Correction: Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday March 31st 2015
Taha M. A. Eldebss, Sobhi M. Gomha, Mohamed M. Abdulla, Reem K. Arafa

68) Structure-Based Virtual Screening for Fragment-Like Ligands of the G Protein-Coupled Histamine H4 Receptor (ChemMedComm) Monday March 30th 2015
Enade P. Istyastono, Albert J. Kooistra, Henry Vischer, Martien Kuijer, Luc Roumen, Saskia Nijmeijer, Rogier Smits, Iwan de Esch, Rob Leurs, Chris de Graaf

69) Novel synthesis of fluorochrome-coupled zoledronate with preserved functional activity on gamma/delta T cells and tumor cells (ChemMedComm) Monday March 30th 2015
Vijayanand Chandrasekaran, Shirin Kalyan, Valentina Biehl, Marcus Lettau, Patrik Theodor Nerdal, Hans-Heinrich Oberg, Daniela Wesch, Thisbe K Lindhorst, Dieter Kabelitz

70) Discovery of 2-(5,6-dimethoxypyridin-3-yl)-4-(2,4,6-trifluorobenzyl)-2H-pyrido[2,3-e][1,2,4]thiadiazin-3(4H)-one 1,1-dioxide (HTL6641), a dual orexin receptor antagonist with differentiated pharmacodynamic properties.[dagger] (ChemMedComm) Monday March 30th 2015
John Andrew Christopher, Sarah Aves, Jason Brown, James Errey, Suki Klair, Christopher Langmead, Oliver Mace, Richard Mould, Jayesh Patel, Ben Tehan, Andrei Zhukov, Fiona Marshall, Miles Congreve

71) Design of pyrazolo-pyrimidines as 11β-HSD1 inhibitors through optimisation of molecular electrostatic potential (ChemMedComm) Monday March 30th 2015
Graeme Robb, Scott Boyd, Christopher Davies, Alexander Dossetter, Frederick W Goldberg, Paul D Kemmitt, James Scott, John Swales

72) Concise Synthesis of Spergualin-Inspired Molecules With Broad-Spectrum Antibiotic Activity (ChemMedComm) Monday March 30th 2015
Victoria Assimon, Hao Shao, Sylvie Garneau-Tsodikova, Jason E. Gestwicki

73) 4-methyl-coumarins with cytotoxic activity against T24 and RT4 human bladder cancer cell lines (ChemMedComm) Thursday March 26th 2015
DAMIANA DA ROCHA VIANNA, LEILA Ruschel, FABRICIA Dietrich, Fabricio Figueiro, Fernanda Morrone, Romulo F. S. Canto, Flavia Corvello, Alice Velho, Allan Crestani, Helder Teixeira, Gilsane Lino von Poser, Ana Maria Oliveira Battastini, Vera Eifler-Lima

74) Tantalising technology (ChemMedComm) Tuesday March 24th 2015
Derek Lowe

75) Synthesis of a new HYNIC-DAPI derivative for labelling with 99mTechnetium and its in vitro evaluation in an FRTL5 cell line (ChemMedComm) Monday March 23rd 2015
Sandra Ferl, Gerd Wunderlich, Rene Smits, Alexander Hoepping, Anne Naumann, Jorg Kotzerke

76) Interactive articles in MedChemComm - connecting readers to a wealth of data and information (ChemMedComm) Thursday March 19th 2015
Richard Kelly

77) Insights into a defined secondary binding region on β-adrenoceptors and putative roles in ligand binding and drug design (ChemMedComm) Thursday March 12th 2015
Marvin Antonio Soriano-Ursua, Jose G Trujillo-Ferrara, Jose A Arias-Montano, Rafael Villalobos-Molina

78) Synthesis and evaluation of anticancer activity of novel andrographolide derivatives (ChemMedComm) Monday March 9th 2015
Devendar Ponnam, Lakshma Nayak V, Dharmendra Yadav, Niranjana Kumar Arigari, Kotesh Kumar Jonnala, Satya Srinivas KVN, Sridhar Balasubramanian, Feroz Khan, Pandu Sastry Kakaraparthi, Ramakrishna Sistla

79) Contributors to 'New Talent: Asia-Pacific' (ChemMedComm) Monday March 9th 2015


80) Membrane-interacting properties of the functionalised fatty acid moiety of muraymycin antibiotics (ChemMedComm) Friday March 6th 2015
Oliver Ries, Christian Carnarius, Claudia Steinem, Christian Ducho

81) In silico study on aging and reactivation processes of tabun conjugated AChE (ChemMedComm) Monday March 2nd 2015
Nellore Bhanu Chandar, Rabindranath Lo, Manoj K Kesharwani, Bishwajit Ganguly

82) Design, synthesis and biological evaluation of thiourea and nicotinamide-containing sorafenib analogs as antitumor agents (ChemMedComm) Monday March 2nd 2015
Xiangkai Kong, Zeyu Yao, Zuopeng He, Wen-Fang Xu, Jianwen Yao

83) Novel non-substrate modulators of the transmembrane efflux pump P-glycoprotein (ABCB1) (ChemMedComm) Friday February 27th 2015
Soren Krawczyk, Christiane Baumert, Josef Molnar, Christoph Ritter, Jens Hopner, Charlotte Kloft, Andreas Hilgeroth

84) Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday February 17th 2015
Taha Eldebss, Sobhi Gomha, Mohamed Abdalla, Reem Arafa

85) Matrix-immobilized yeast for large-scale production of recombinant human lactoferrin (ChemMedComm) Tuesday February 17th 2015
Chun Loong Ho, In Young Hwang, Kathy Loh, Matthew Chang

86) Synthesis and evaluation of amide, sulfonamide and urea - benzisoxazole derivatives as potential atypical antipsychotics (ChemMedComm) Friday February 13th 2015
Yin Chen, Yu Lan, Xudong Cao, Xiangqing Xu, Juecheng Zhang, Minquan Yu, Xin Liu, Bifeng Liu, Guisen Zhang

87) Synthesis and protective effect of new ligustrazine derivatives against CoCl2-induced neurotoxicity in differentiated PC12 cells. Part 2 (ChemMedComm) Thursday February 12th 2015
Bing Xu, Yan Gong, Xin Xu, Chenze Zhang, Yuzhong Zhang, Fuhao Chu, Hongbing Liu, Penglong Wang, Haimin Lei

88) BODIPY appended copper(II) complexes of curcumin showing mitochondria targeted remarkable photocytotoxicity in visible light (ChemMedComm) Thursday February 12th 2015
Akhil R Chakravarty, Arnab Bhattacharyya, Akanksha Dixit, Koushambi Mitra, Samya Banerjee, Anjali A Karande

89) Synthesis and biological evaluation of novel [capital Delta]2-isoxazoline fused cyclopentane derivatives as potential antimicrobial and anticancer agents (ChemMedComm) Wednesday February 11th 2015
Nagendra Babu Bathini, Santosh Kumar Prajapti, Shweta Shrivastava, Umesh Bihade, Ajay Kumar Gupta, V.G. M Naidu, Uttam Chand Banerjee

90) Evaluation of the anti-inflammatory/chondroprotective activity of aldose reductase inhibitors in human chondrocyte cultures (ChemMedComm) Wednesday February 4th 2015
Annamaria Panico, Rosanna Maccari, Venera Cardile, Sergio Avondo, Lucia Crasci, Rosaria Ottana

91) Inhibition of Insulin Amyloid Fibrillization by Glyco-Acridines: In vitro and in silico study (ChemMedComm) Wednesday February 4th 2015
Quan Van Vuong, Zuzana Bednarikova, Andrea Antosova, Huy Dinh Quoc Pham, Katarina Siposova, Nguyen Anh Tuan, Mai Suan Li, Zuzana Gazova

92) Application of QM/MM and QM methods to investigate histone deacetylase 8 (ChemMedComm) Monday February 2nd 2015
Duangkamol Gleeson, M. Paul Gleeson

93) Structure-Based Design, Synthesis by Click Chemistry and in Vivo Activity of Highly Selective A3 Adenosine Receptor Agonists (ChemMedComm) Monday February 2nd 2015
Dilip Tosh, Silvia Paoletta, Zhoumou Chen, Steven Crane, John Lloyd, Zhan-Guo Gao, Elizabeth Gizewski, John Auchampach, Daniela Salvemini, Kenneth A. Jacobson

94) Synthesis and evaluation of a series of resveratrol analogues as potent anticancer agents that target tubulin (ChemMedComm) Friday January 30th 2015
Nikhil Reddy Madadi, Hongliang Zong, Amit Ketkar, Zhen Chen, Narsimha Penthala, Venumadhav Janganati, Shobanbabu Bommagani, Robert Eoff, Monica Guzman, Peter Crooks

95) Design, Facile Synthesis and Anthelmintic Activity of New O-Substituted 6-Methoxybenzothiazole-2-carbamates (ChemMedComm) Tuesday January 27th 2015
A. Mohsen M.E. Omar, Omaima M. Aboulwafa, Doaa A. E. Issa, May M.S. El-Shokrofy, May E. Amr, Ibrahim M. El-Ashmawy

96) BEYOND THE AFFINITY FOR PROTEIN KINASE C: EXPLORING 2-PHENYL-3-HYDROXYPROPYL PIVALATE ANALOGUES AS C1 DOMAIN-TARGETING LIGANDS (ChemMedComm) Monday January 26th 2015
Daniela Rossi, Virpi Talman, Gustav Boije, Annamaria Marra, pietro Picconi, Rita Nasti, Massimo Serra, ANN JIHYAE, Marialaura Amadio, Alessia Pascale, Jeewoo Lee, Raimo Tuominen, Jari Yli-Kauhaluoma, Simona Collina

97) Correction: Identification of tris-(phenylalkyl)amines as new selective h5-HT2B receptor antagonists (ChemMedComm) Friday January 23rd 2015
Shashikanth Ponnala, Nirav Kapadia, Wayne Wesley Harding

98) Identification of Camphor Derivatives as Novel M2 Ion Channel Inhibitors of Influenza A Virus (ChemMedComm) Monday January 19th 2015
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