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1) Discovery of AZD8165 - a Clinical Candidate from a Novel Series of Neutral Thrombin Inhibitors (ChemMedComm) Friday November 27th 2015
Magnus Polla, Jonas Branalt, Joakim Bergman, Maria Olwegard-Halvarsson, Ylva Ortengren, Camilla Wern, Ann-Charlotte Egnell, Patrik Andersson, Ulf Eriksson, David Gustafsson, Kurt.Jurgen Hoffman, Ulf Bredberg, Marie Strimfors, Sofi Nielsen, Kenneth Abrahamsson, Ingemar Nilsson, Tore Skjaeret

2) Targeting microsomal prostaglandin E2 synthase-1 (mPGES-1): the development of inhibitors as an alternative to non-steroidal anti-inflammatory drugs (NSAIDs) (ChemMedComm) Friday November 27th 2015
Yuqing Chen, Huaqing Liu, Shuang Xu, Tianlin Wang, Wei Li

3) Antiprotozoal activity of dehydroabietic acid derivatives against Leishmania donovani and Trypanosoma cruzi (ChemMedComm) Wednesday November 25th 2015
Mikko Vahermo, Sara Krogerus, Abedelmajeed Nasereddin, Marcel Kaiser, Reto Brun, Charles L. Jaffe, Jari Yli-Kauhaluoma, Vania M. Moreira

4) Silver(I) complexes with quinazoline and phthalazine: synthesis, structural characterization and evaluation of biological activities (ChemMedComm) Wednesday November 25th 2015
Nada D Savic, Biljana D Glisic, Hubert Wadepohl, Aleksandar Pavic, Senerovic Lidija, Jasmina Nikodinovic-Runic, Milos I Djuran

5) Isoindole-1,3-dione Derivatives as RSK2 Inhibitors: Synthesis, Molecular Docking Simulation and SAR Analysis (ChemMedComm) Wednesday November 25th 2015
wei zhou, Shiliang Li, Weiqiang Lu, jun yuan, yufang xu, Honglin Li, Jin Huang, Zhenjiang Zhao

6) Correction: Discovery of a potent and highly fluorescent sirtuin inhibitor (ChemMedComm) Friday November 20th 2015
Y. K. Yoon, M. A. Ali, A. C. Wei, T. S. Choon, C. E. Oon, A. N. Shirazi, K. Parang

7) Systematic Assessment of Analog Relationships between Bioactive Compounds and Promiscuity of Analog Sets (ChemMedComm) Thursday November 19th 2015
Dilyana Dimova, Dagmar Stumpfe, J Bajorath

8) Expression of concern: Identifying the inhibitory mechanism of apigenin on the insulin ligand-receptor binding (ChemMedComm) Thursday November 19th 2015
Richard Kelly

9) A review of patents (2011-2015) towards combating resistance to and otoxicity of aminoglycosides (ChemMedComm) Thursday November 19th 2015
Nishad Thamban Chandrika, Sylvie Garneau-Tsodikova

10) Bioorthogonal metabolic labelling with acyl-CoA reporters: targeting protein acylation (ChemMedComm) Thursday November 19th 2015
Maria Eleni Ourailidou, Martijn Zwinderman, Frank Dekker

11) Mechanisms of Resistance to Membrane-Disrupting Antibiotics in Gram-Positive and Gram-Negative Bacteria (ChemMedComm) Thursday November 19th 2015
Micha Fridman, Kfir B. Steinbuch

12) Probing for improved selectivity with dipeptide-derived inhibitors of dipeptidyl peptidases 8 and 9: the impact of P1-variation. (ChemMedComm) Thursday November 19th 2015
Leen Heirbaut, Sebastiaan Van Goethem, Koen Jansen, Hans De Winter, Nicole Lamoen, Jurgen Joossens, Jonathan Cheng, X Chen, Anne-Marie Lambeir, Ingrid De Meester, Koen Augustyns, Pieter Van der Veken

13) Demonstration of the dynamic mass redistribution label-free technology as a useful cell-based pharmacological assay for endogenously expressed GABAA receptors (ChemMedComm) Thursday November 19th 2015
Anders Bue Klein, Mia Nittegaard-Nielsen, Julie Thaulow Christensen, Anas Al-Khawaja, Petrine Wellendorph

14) Novel indole-flutimide heterocycles with activity against influenza PA endonuclease and hepatitis C virus (ChemMedComm) Thursday November 19th 2015
Grigoris Zoidis, Erofili Giannakopoulou, Annelies Stevaert, Efseveia Frakolaki, Vassilios Myrianthopoulos, George Fytas, Penelope Mavromara, E. Mikros, Ralf Bartenshlager, Niki Vassilakic, Lieve Naesens

15) Efficient synthesis of novel disubstituted pyrido[3,4-b]pyrazines for the design of protein kinase inhibitors (ChemMedComm) Thursday November 19th 2015
Maud Antoine, Tilmann Schuster, Irene Seipelt, Babette Aicher, Michael Teifel, Eckhard Gunther, Matthias Gerlach, Pascal Marchand

16) Antimicrobial activity of Levofloxacin - M33 peptide conjugation or combination (ChemMedComm) Thursday November 19th 2015
Federica Ceccherini, Chiara Falciani, Martina Onori, Silvia Scali, Simona Pollini, Gianmaria Rossolini, Luisa Bracci, Alessandro Pini

17) 1,3,4-Oxadiazole derivatives as potential antitumor agents: discovery, optimization and biological activity valuation (ChemMedComm) Thursday November 19th 2015
Yin Luo, Zhi-Jun Liu, Guo Chen, Jing-Ran Li, Jing Shi, Hai-Liang Zhu

18) 6-O-Nucleotidyltransferase: an aminoglycoside-modifying enzyme specific for streptomycin/streptidine (ChemMedComm) Monday November 16th 2015
Montserrat Latorre, Julia Revuelta, Eduardo Garcia-Junceda, Agatha Bastida

19) Integrating Multicomponent Flow Synthesis and Computational Approaches for the Generation of a Tetrahydroquinoline Compound Based Library (ChemMedComm) Monday November 16th 2015
Bruno Cerra, Serena Mostarda, Chiara Custodi, Antonio Macchiarulo, Antimo Gioiello

20) Spirooxadiazoline oxindoles with promising in vitro antitumor activities (ChemMedComm) Monday November 16th 2015
Carlos Ribeiro, Joana Amaral, Cecilia Rodrigues, Rui Moreira, Maria M. M. Santos

21) In-vitro and in-vivo Activity of ML302F: A Thioenolate Inhibitor of VIM-subfamily Metallo β-lactamses (ChemMedComm) Monday November 16th 2015
Jonathan Betts, Lynette Phee, Muhd Abdul Momin, Klaus Umland, Jurgen Brem, Christopher J Schofield, David Wareham

22) Identification of an Inhibitor of the Aminoglycoside 6'-N-Acetyltransferase type Ib [AAC(6′)-Ib] by Glide Molecular Docking (ChemMedComm) Monday November 16th 2015
Kevin Chiem, Saumya Jani, Brooke Fuentes, David Lin, Madeline Rasche, Marcelo Tolmasky

23) Targeting the trehalose utilization pathways of Mycobacterium tuberculosis (ChemMedComm) Monday November 16th 2015
Sandeep Thanna, Steven Joseph Sucheck

24) Structural hybridization of three aminoglycoside antibiotics yields a potent broad-spectrum bactericide that eludes bacterial resistance enzymes (ChemMedComm) Friday November 13th 2015
Juan Pablo Maianti, Stephen Hanessian

25) Insight into the cytotoxicity, DNA binding and cell apoptosis induction of a zinc(II) complex of 5-bromo-8-hydroxylquinoline (HBrQ) (ChemMedComm) Thursday November 12th 2015
Hai-Rong Zhang, Yan-Cheng Liu, Ting Meng, Qi-Pin Qin, Shang-Feng Tang, Zhengfeng Chen, Bi-Qun Zou, You-Nian Liu, Hong Liang

26) Synthesis and evaluation of thieno[2,3-d]pyrimidin-4(3H)-ones as potential antitubercular agents (ChemMedComm) Thursday November 12th 2015
Hanumant Bapurao Borate, Ritesh Annadate, Sandip Vagh, Mahesh Pisal, Sagar Deokate, Manisha Arkile, Nandadeep Jadhav, Laxman Nawale, Dhiman Sarkar

27) Selective inhibitors of phosphodiesterases: therapeutic promise for neurodegenerative disorders (ChemMedComm) Thursday November 12th 2015
Tarana Umar, Nasim ul Hoda

28) Discovery of Trace Amine-Associated Receptor 1 Ligands by Molecular Docking Screening against a Homology Model (ChemMedComm) Thursday November 12th 2015
Vincent Lam, David Rodriguez, Thomas Zhang, Eun Koh, Jens Carlsson, Ali Salahpour

29) Correction: Acetophenone derivatives: novel and potent small molecule inhibitors of monoamine oxidase B (ChemMedComm) Monday November 9th 2015
Zhi-Min Wang, Xue-Mei Li, Wei Xu, Fan Li, Jin Wang, Ling-Yi Kong, Xiao-Bing Wang

30) Correction: Syntheses and biological evaluations of highly functionalized hydroxamate containing and N-methylthio monobactams as anti-tuberculosis and β-lactamase inhibitory agents (ChemMedComm) Friday November 6th 2015
Mark W. Majewski, Kyle D. Watson, Sanghyun Cho, Patricia A. Miller, Scott G. Franzblau, Marvin J. Miller

31) Correction: Discovery of fluoroquinolone derivatives as potent, selective inhibitors of PI3Kγ (ChemMedComm) Friday November 6th 2015
Shao Sha, Hong-Wei Han, Fei Gao, Tian-Bao Liu, Zhen Li, Chi Xu, Wei-Qing Zhong, Hai-Liang Zhu

32) Synthesis of sliver nanoparticles loaded sulfadiazine/polyvinyl alcohol nanorods and their antibacterial activities (ChemMedComm) Friday November 6th 2015
Binjie Li, Ping Li, Xiangmin Xu, Longlong Wu, Yanbao Zhao

33) Development of Subnanomolar Radiofluorinated (2-Pyrrolidin-1-yl)imidazo[1,2-b]pyridazine pan-Trk Inhibitors as Candidate PET Imaging Probes (ChemMedComm) Thursday November 5th 2015
Vadim Bernard-Gauthier, Justin James Bailey, Arturo Aliaga, Alexey Kostikov, Pedro Rosa-Neto, Melinda Wuest, Garrett M. Brodeur, Frank Wuest, Ralf Schirrmacher

34) Endless Resistance. Endless Antibiotics? (ChemMedComm) Tuesday November 3rd 2015
Jed Fisher, Shahriar Mobashery

35) Synthesis of N-cyano-substituted sulfilimine and sulfoximine derivatives of S0859 and their biological evaluation as sodium bicarbonate co-transport inhibitors (ChemMedComm) Tuesday November 3rd 2015
Anne-Dorothee Steinkamp, Nico Seling, Soojung Lee, Ebbe Boedtkjer, Carsten Bolm

36) Antimycobacterial activity of rhodamine 3,4-HPO iron chelators against Mycobacterium avium: analysis of the contribution of functional groups and of chelator (ChemMedComm) Tuesday November 3rd 2015
Tania Moniz, Daniel da Silva, Tania Silva, Maria Salome Gomes, Maria Rangel

37) Arginine-linked neomycin B dimers: synthesis, rRNA binding, and resistance enzyme activity (ChemMedComm) Tuesday November 3rd 2015
Yi Jin, Derrick Watkins, Natalya N Degtyareva, Keith D Green, Meredith N Spano, Sylvie Garneau-Tsodikova, Dev P Arya

38) Synthesis and biological evaluation of piperzaine group linked bivalent β-carbolines as potential antitumor agents (ChemMedComm) Tuesday November 3rd 2015
Rihui Cao, Rongqin Sun, Rui Liu, Chi Zhou, Zhenghua Ren, Liang Guo, Qin Ma, Wenxi Fan, Liqin Qiu, Huijuan Yu, guang shao

39) Synthesis and Preclinical Evaluation of a Novel, Selective 111In-labelled Aminoproline-RGD-peptide For Non-invasive Melanoma Tumor Imaging (ChemMedComm) Tuesday November 3rd 2015
Andrea Sartori, Francesca Bianchini, Silvia Migliari, Paola Burreddu, Claudio Curti, Federica Vacondio, Daniela Arosio, Livia Ruffini, Gloria Rassu, Lido Calorini, Alberto Pupi, Franca Zanardi, Lucia Battistini

40) Spice up your compounds (ChemMedComm) Thursday October 22nd 2015
Derek Lowe

41) Acetophenone derivatives: novel and potent small molecule inhibitors of monoamine oxidase B (ChemMedComm) Wednesday October 21st 2015
Zhi-Min Wang, Xue-Mei Li, Wei Xu, Fan Li, Jin Wang, Ling-Yi Kong, Xiao-Bing Wang

42) Novel N-thiazolyl piperazine-1-carboxamide CCR2 antagonists - investigation of an unexpected reaction with glutathione (ChemMedComm) Monday October 19th 2015
J. G. Cumming, P. A. MacFaul, A. G. Leach

43) Synthesis of fusidic acid bioisosteres as antiplasmodial agents and molecular docking studies in the binding site of elongation factor-G (ChemMedComm) Tuesday October 13th 2015
Gurminder Kaur, Kawaljit Singh, Elumalai Pavadai, Mathew Njoroge, Marlene Espinoza-Moraga, Carmen De Kock, Peter J. Smith, Sergio Wittlin, Kelly Chibale

44) Patterns of Biofilm Structure and Formation Kinetics among Acinetobacter baumannii Clinical Isolates with Different Antibiotic Resistance Profiles (ChemMedComm) Tuesday October 13th 2015
Elias Dahdouh, Belen Orgaz, Rosa Gomez-Gil, Jesus Mingorance, Ziad Daoud, Monica Suarez, Carmen SanJose

45) Molecular Basis for Resistance Against Phosphonate Antibiotics and Herbicides (ChemMedComm) Monday October 12th 2015
Jonathan Chekan, Dillon P Cogan, Satish Nair

46) Thermoresponsive fluorinated small-molecule drugs: a new concept for efficient localized chemotherapy. (ChemMedComm) Thursday October 8th 2015
Paul Dyson, Catherine Clavel, Patrycja Nowak-Sliwinska, Emilia Paunescu

47) In silico-driven multicomponent synthesis of 4,5- and 1,5-disustituted imidazoles as indoleamine 2,3-dioxygenase inhibitors (ChemMedComm) Thursday October 8th 2015
Silvia Fallarini, Alberto Massarotti, Alessandro Gesu, Sara Giovarruscio, Giulia Coda Zabetta, Roberta Bergo, Barbara Giannelli, Angelo Brunco, Grazia Lombardi, Giovanni Sorba, Tracey Pirali

48) Bisimidazoline arylamides binding to the DNA minor groove. N1-hydroxylation enhances binding affinity and selectivity to AATT sites (ChemMedComm) Thursday October 8th 2015
Carlos H. Rios Martinez, Laura Lagartera, Cristina Trujillo, C Dardonville

49) Synergistic Activity of a Short Lipidated Antimicrobial Peptide (LipoAMP) and Colistin or Tobramycin against Pseudomonas Aeruginosa from Cystic Fibrosis Patients (ChemMedComm) Monday October 5th 2015
Martin de Gier, H. Bauke Albada, Michaele Josten, Rob Willems, Helen Leavis, Rosa Van Mansveld, Fernanda Paganelli, Bertie Dekker, Jan-Willem Lammers, Hans-Georg Sahl, Nils Metzler-Nolte

50) Syntheses and Biological Evaluations of Highly Functionalized Hydroxamate Containing and N-Methylthio Monobactams as Anti-Tuberculosis and β-Lactamase Inhibitory Agents. (ChemMedComm) Monday October 5th 2015
Marvin Miller, Mark Majewski, Kyle Watson, Sanghyun Cho, Patricia Miller, Scott Franzblau

51) Multi-drug delivery nanocarriers for combination therapy (ChemMedComm) Thursday October 1st 2015
Suresh Gadde

52) A Structure-Activity Relationship Study of the Positive Allosteric Modulator LY2033298 at the M4 Muscarinic Acetylcholine Receptor (ChemMedComm) Wednesday September 30th 2015
Monika Szabo, Tracey Huynh, Celine Valent, Robert Lane, Patrick Sexton, Arthur Christopoulos, Ben Capuano

53) Potentiation of Francisella resistance to conventional antibiotics through small molecule adjuvants (ChemMedComm) Wednesday September 30th 2015
Matthew D. Stephens, Veroncia B. Hubble, Robert K. Ernst, Monique L. van Hoek, Roberta J. Melander, John Cavanagh, Christian Melander

54) Discovery of Fluoroquinolone derivatives as potent, selective inhibitors of PI3Kγ (ChemMedComm) Tuesday September 29th 2015
Hai-Liang Zhu, Shao Sha, Hong-Wei Han, Fei Gao, Tian-Bao Liu, zhen li, Chi Xu, Wei-Qing Zhong

55) Ligand-based homology modelling of the human CB2 receptor SR144528 antagonist binding site: a computational approach to explore the 1,5-diaryl pyrazole scaffold (ChemMedComm) Monday September 28th 2015
Elena Cichero, Giulia Menozzi, Sara Guariento, Paola Fossa

56) Semi-synthesis and anti-tumor evaluation of novel 25-hydroxyprotopanaxadiol derivatives as apoptosis inducing agents (ChemMedComm) Friday September 25th 2015
fanzhi qu, chen zhao, yafei liu, jiaqing cao, wei li, yuqing zhao

57) Ionic liquid mediated transcutaneous protein delivery with solid-in-oil nanodispersion (ChemMedComm) Friday September 25th 2015
Shota Araki, Rie Wakabayashi, Muhammad Moniruzzaman, Noriho Kamiya, Masahiro Goto

58) Mode of Action Study of Cationic Anthraquinone Analog: A New Class of Highly Potent Anti-cancer Agent (ChemMedComm) Friday September 25th 2015
Jaya P Shrestha, Yagya Subedi, liaohai chen, Tom Chang

59) Design and synthesis of peptide inhibitor conjugates as probes of the Cytochrome P450s from glycopeptide antibiotic biosynthesis (ChemMedComm) Friday September 25th 2015
Clara Brieke, Theresa Maier, Martin Schroter, Max Cryle

60) Synthesis of indole-derived allocolchicine congeners exhibiting pronounced anti-proliferative and apoptosis-inducing properties (ChemMedComm) Tuesday September 22nd 2015
Nikolay Sitnikov, Alexander Sinzov, Diane Allegro, Pascale Barbier, Sebastien Combes, Liliane Abodo Onambele, Aram Prokop, Hans Gunther Schmalz, Alexey Fedorov

61) A synthesis, in silico, in vitro and in vivo study of thieno[2,3-b]pyridine anticancer analogues (ChemMedComm) Tuesday September 22nd 2015
John Arabshahi, Michelle van Rensburg, Lisa Pilkington, Chae Jeon, Mirae Song, Ling-Mey Gridle, Euphemia Leung, David Barker, Milena Vuica-Ross, Konstantin Volcho, Alexandra Zakharenko, Olga Lavrik, Johannes Reynisson

62) Mechanisms of Resistance to Aminoglycoside Antibiotics: Overview and Perspectives (ChemMedComm) Monday September 21st 2015
Sylvie Garneau-Tsodikova, Kristin J. Labby

63) Discovery of a potent and highly fluorescent sirtuin inhibitor (ChemMedComm) Tuesday September 15th 2015
Y. K. Yoon, M. A. Ali, A. C. Wei, T. S. Choon, A. N. Shirazi, K. Parang

64) Phase II Metabolic Pathways of Spectinamide Antitubercular Agents: A Comparative Study of the Reactivity of 4- Substituted Pyridines to Glutathione Conjugation (ChemMedComm) Monday September 7th 2015
Dora Madhura, Jiuyu Liu, Bernd Meibohm, Richard E. Lee

65) Tabtoxinine-β-Lactam is a "Stealth" β-Lactam Antibiotic that Evades β-Lactamase-mediated Antibiotic Resistance (ChemMedComm) Monday September 7th 2015
Timothy Adam Wencewicz, Kathryn Hart, Margaret Reck, Gregory Bowman

66) Rational design of promiscuous binding modulators of p53 inducing E3(Ub)-ligases (Mdm2 and Pirh2) as anticancer agents: An in silico approach (ChemMedComm) Monday September 7th 2015
Sarfaraj Niazi, Madhusudan Purohit

67) 1-[(2E)-3-phenylprop-2-enoyl]-1H-benzimidazoles as anticancer agents: Synthesis, crystal structure analysis and binding studies of the most potent anticancer molecule with serum albumin (ChemMedComm) Monday September 7th 2015
Seetharamappa J, Veerendra Kumar A Kalalbandi

68) Identification of a novel NAMPT inhibitor by combinatorial click chemistry and chemical refinement (ChemMedComm) Monday September 7th 2015
Sewan Theeramunkong, Ubaldina Galli, Ambra A Grolla, Antonio Caldarelli, Cristina Travelli, Alberto Massarotti, Maria Pia Troiani, Maria Alessandra Alisi, Giuseppe Orsomando, Armando A Genazzani, Gian Cesare Tron

69) Synthesis and Biological Evaluation of Novel 7-O-Lipophilic Substituted Baicalein Derivatives as Potential Anticancer Agents (ChemMedComm) Monday September 7th 2015
Shao-Hung Wang, C.-H. Chen, CY Lo, Ji-Zhen Feng, Hong-Jhih Lin, Po-Ya Chang, Ling-Ling Yang, Lih-Geeng Chen, Yi-Wen Liu, Cheng-Deng Kuo, Jin-Yi Wu

70) 2-[18F]Fluoroethyl tosylate - a versatile tool for building of 18F based radiotracers for positron emission tomography (ChemMedComm) Thursday September 3rd 2015
Torsten Kniess, Markus Laube, Peter Brust, Jorg Steinbach

71) The first potent diphenyl phosphonate KLK4 inhibitors with unexpected binding kinetics (ChemMedComm) Thursday September 3rd 2015
Jeroen Van Soom, Giuliana Cuzzucoli Crucitti, Rafaela Gladysz, Pieter Van der Veken, Roberto Di Santo, Ingmar Stuyver, Victoria Buck, Anne-Marie Lambeir, Viktor Magdolen, Jurgen Joossens, Koen Augustyns

72) Evaluation of binding competition and group epitopes of Acetylcholinesterase inhibitors by STD NMR, Tr-NOESY, DOSY and Molecular Docking: An old approach but new findings (ChemMedComm) Thursday September 3rd 2015
Nazish Urooj Tanoli, Sheraz Ahmad Khan Tanoli, Antonio Gilberto Ferreira, Sana Gul, Zaheer Ul Haq

73) Missing the target (ChemMedComm) Wednesday September 2nd 2015
Derek Lowe

74) Property-based characterization of kinase-like ligand space for library design and virtual screening (ChemMedComm) Wednesday September 2nd 2015
David Bajusz, Gyorgy Ferenczy, George M Keseru

75) Design, Synthesis and Bioevaluation of Tacrine Hybrids with Cinnamate and Cinnamylideneacetate Derivatives as Potential Anti-Alzheimer Drug Candidates (ChemMedComm) Wednesday September 2nd 2015
Amelia Santos, Catarina Quintanova, Rangappa S Keri, Sergio Marques, Sandra Cardoso, M L. M. Serralheiro, Maria Goncalves Fernandes

76) Supramolecular, Prodrug-based Micelles with Enzyme Regulated Release Behavior for Controlled Drug Delivery (ChemMedComm) Friday August 28th 2015
Yong-yong Li, Yu-qin Chen, Hai-qing Dong, Chun-yan Dong

77) Sulfasalazine in Ionic Liquid Form with Improved Solubility and Exposure (ChemMedComm) Wednesday August 26th 2015
Mohammad Shadid, Gabriela Gurau, Julia L. Shamshina, Bei-Ching Chuang, Shumet Hailu, Emily Guan, Swapan Chowdhury, Jing-Tao Wu, Syed A. A. Rizvi, Robert Griffin, Robin D. Rogers

78) Aryl- Imidazothiadiazole Analogues as Microtubule Disrupting Agents (ChemMedComm) Wednesday August 26th 2015
Ahmed Kamal, Subba Rao A.V., Srinivasa Reddy Telukutla, Sowjanya Polepalli, chandrakant Bagul, Vishnuvardhan MVPS, Siddiq Pasha Shaik, Nishant Jainb

79) Insights into the impact of N- and O-methylation on aqueous solubility and lipophilicity using matched molecular pair analysis (ChemMedComm) Friday August 21st 2015
Timothy John Ritchie, simon macdonald, Stephen Pickett

80) Inspired by magnolol: design of NSAIDs-based compounds with excellent anti-inflammatory effect (ChemMedComm) Friday August 21st 2015
Wenfeng Liu, Yuan Yue, Yonglian Li, Xi Zheng, Kun Zhang, Zhiyun Du

81) Novel Quinoline Derivatives as Potent In Vitro α-Glucosidase Inhibitors: In Silico Studies and SAR Predictions (ChemMedComm) Friday August 21st 2015
Muhammad Taha, Nor Ismail Ismail, Syahrul Imran, Abdul Wadood, Fazal Rahim, Muhammad Ali, Ahsfaq Rehman

82) Correction: Synthesis and antibacterial activity evaluation of C-5 side chain modified analogues of FYL-66, a potential agent against methicillin-resistant Staphylococcus aureus (ChemMedComm) Friday August 21st 2015
Xiaoyan Yang, Zicheng Li, Zhenling Wang, Zitai Sang, Haiyue Long, Jianying Tang, Tao Yang, Yuanyuan Liu, Youfu Luo

83) Navigating into chemical space between MGCD0103 and SAHA: Novel Histone Deacetylase Inhibitor as a Promising Lead (ChemMedComm) Monday August 17th 2015
Xin Zhang, Peng-Cheng Lv, Dongdong Li, weiming zhang, Hai-Liang Zhu

84) Discovery of Pyridyl-based inhibitors of Plasmodium falciparum N-myristoyltransferase (ChemMedComm) Monday August 17th 2015
Zhiyong Yu, James A Brannigan, Kaveri Rangachari, William Heal, Anthony J Wilkinson, Tony Holder, Robin J Leatherbarrow, Edward William Tate

85) Discovery of High Affinity Inhibitors of Leishmania donovani N-Myristoyltransferase (ChemMedComm) Monday August 17th 2015
Mark Rackham, Zhiyong Yu, James A Brannigan, William Heal, Daniel Paape, Victoria Barker, Anthony J Wilkinson, Deborah Smith, Robin J Leatherbarrow, Edward William Tate

86) Inhibitory effect of cytotoxic nitrogen-containing heterocyclic stilbene analogues on the VEGF protein secretion and the expression of the VEGF, hTERT and c-Myc genes (ChemMedComm) Wednesday August 12th 2015
Eva Falomir, Rosa Marti-Centelles, Juan Murga, Miguel Carda, J. Alberto Marco

87) Synthesis, in vitro and in vivo anticancer activities of novel 4-substituted 1,2-bis(4-chlorophenyl)-pyrazolidine-3,5-dione derivatives (ChemMedComm) Wednesday August 12th 2015
Xu-Yao Zhang, Yi-Fei Gu, Ting Chen, Dong-Xiao Yang, Xi-Xin Wang, Bai-Ling Jiang, Kun-Peng Shao, Wen Zhao, Cong Wang, Jun-Wei Wang, Qiu-Rong Zhang, Hong-Min Liu

88) Correction: Application of QM/MM and QM methods to investigate histone deacetylase 8 (ChemMedComm) Wednesday August 12th 2015
Duangkamol Gleeson, M. Paul Gleeson

89) Structure activity relationship of C1-C2-linker substituted 1,5-naphthyridine analogues of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-7) (ChemMedComm) Wednesday August 12th 2015
Sheo B Singh, David Kaelin, Jin Wu, Lynn Miesel, Christopher Tan, Peter Meinke, David Olsen, Armando Lagrutta, Changqing Wei, Yonggang Liao, Xuanjia Peng, Xiu Wang, Hideyuki Fukuda, Ryuta Kishii, Masaya Takei, Takeshi Shibata, Tomoko Takeuchi, Kohei Ohata, Akinori Nishimura, Yasumichi Fukuda

90) Inhibition of Phosphatidylinositol-3,4,5-trisphosphate Binding to AKT Pleckstrin Homology Domain by 4-Amino-1,2,5-oxadiazole Derivatives (ChemMedComm) Tuesday August 11th 2015
Debasis Manna, Sukhamoy Gorai, Saurav Paul, Ganga Sankaran, Manas Kumar Santra, Rituparna Borah

91) Design and discovery of 3-aryl-5-substituted-isoquinolin-1-ones as potent tankyrase inhibitors (ChemMedComm) Tuesday August 11th 2015
Richard J.R Elliott, Ashley Jarvis, Mohan B Rajasekaran, Malini Menon, Leandra Bowers, Raymond Boffey, Melanie Bayford, Stuart Firth-Clark, Rebekah Key, Rehan Aqil, Stewart B. Kirton, Dan Niculescu-Duvaz, Laura Fish, Filipa Lopes, Robert McLeary, Ines Trindade, Elisenda Vendrell, Felix Munkonge, Rod Porter, Trevor Perrior, CJ Springer, Antony Oliver, Laurence Pearl, Alan Ashworth, Christopher J. Lord

92) Isothiazolo[4,3-b]pyridines as inhibitors of cyclin G associated kinase : synthesis, structure-activity relationship studies and antiviral activity (ChemMedComm) Friday August 7th 2015
Jiahong Li, Sona Kovackova, Szuyuan Pu, Jef Rozenski, Steven De Jonghe, Shirit Einav, Piet Herdewijn

93) Correction: Design, synthesis, and evaluation of semi-conservative mono-carbonyl analogs of curcumin as anti-inflammatory agents against lipopolysaccharide-induced acute lung injury (ChemMedComm) Friday August 7th 2015
Lili Dong, Suqing Zheng, Yali Zhang, Xin Jiang, Jianzhang Wu, Xiaoqin Zhang, Xiaoou Shan, Dandan Liang, Shilong Ying, Jianpeng Feng, Guang Liang

94) Tricyclic phenothiazine and phenoselenazine derivatives as potential multi-targeting agents to treat Alzheimer's disease (ChemMedComm) Friday August 7th 2015
Gary Tin, Tarek Mohamed, Nyasha Gondora, Michael Beazely, Praveen P Nekkar Rao

95) Synthesis of carboxyimidamide-substituted benzo[c][1,2,5]oxadiazoles and their analogs, and evaluation of biological activity against Leishmania donovani (ChemMedComm) Friday August 7th 2015
Leena Keurulainen, Mikko Heiskari, Satu Nenonen, Abedelmajeed Nasereddin, Dmitry Kopelyanskiy, Teppo Leino, Jari Yli-Kauhaluoma, Charles Jaffe, Paula Kiuru

96) D1-like Receptors Distinguishing Thieno-azecine Regioisomers (ChemMedComm) Wednesday August 5th 2015
Mohamed Abdel-Fattah, Ashraf H. Abadi, J Lehmann, P. Schweikert, Christoph Enzensperger

97) C-5 Substituted Pyrido[2,3-d]pyrimidin-7-ones as Highly Specific Kinase Inhibitors Targeting Clinical Resistance related EGFRT790M Mutant (ChemMedComm) Wednesday August 5th 2015
Ke Ding, Jian Ding, Hua Xie, Meiyu Geng, Linjiang Tong, Ting Peng, zhaoyu Huang, Tianfeng Xu, xiaomei Ren, Zhengchao Tu, Lianwen Zhang, zhang zhang, xiaoyun lu, Lei Yu, Jinfeng Luo

98) Induction of apoptosis by cyclobutanones and derived polycyclic γ-lactones: a preliminary analysis of antiproliferative activity (ChemMedComm) Tuesday August 4th 2015
Vishal Sharma, Ashun Chaudhary, Gousia Chashoo, Saroj Arora, Ajit K. Saxena, Mohan Paul S. Ishar

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Mitch Andre Garcia's Chem Feeds 2008-present

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