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1) Substituted 4-hydroxy-1,2,3-triazoles: synthesis, characterization and first drug design applications through bioisosteric modulation and scaffold hopping approaches (ChemMedComm) Thursday May 28th 2015
Agnese Chiara Pippione, Franco Dosio, Alex Ducime, Antonella Federico, Katia Martina, Stefano Sainas, Bente Frolund, Major Gooyit, Kim D Janda, Donatella Boschi, Marco Lucio Lolli

2) Identifying the inhibitory mechanism of apigenin on the insulin ligand-receptor binding (ChemMedComm) Wednesday May 27th 2015
Yong Yang

3) Identification of an indole-triazole-amino acid conjugate as highly effective antifungal agent (ChemMedComm) Tuesday May 26th 2015
Kalpana Pawar, Anshuman Yadav, Parteek Prasher, Sahil Mishra, Balwinder Singh, Palwinder Singh, Sneha Komath

4) Synthesis and biological evaluation of novel semi-conservative mono-carbonyl analogs of curcumin as anti-inflammatory agents (ChemMedComm) Tuesday May 26th 2015
Zhe Wang, Peng Zou, Chenglong Li, Wenfei He, Bing Xiao, Qilu Fang, Wenbo Chen, Suqing Zheng, Yunjie Zhao, Yuepiao Cai, Guang Liang

5) Medicinal Organometallic Chemistry - an Emerging Strategy for the Treatment for Neglected Tropical Diseases (ChemMedComm) Tuesday May 26th 2015
Christopher Hyland, Ronald Brown

6) Design, Synthesis, Antibacterial Evaluation of Novel Azolylthioether Quinolones as MRSA DNA Intercalators (ChemMedComm) Thursday May 21st 2015
Ling Zhang, Vijaya Kumar Kannekanti, RASHEED SYED, Shao-Lin Zhang, Rong-Xia Geng, Cheng-He Zhou

7) Discovery of novel amino-pyrimidine inhibitors of the insulin-like growth factor 1 (IGF1R) and insulin receptor (INSR) kinases; parallel optimization of cell potency and hERG inhibition (ChemMedComm) Thursday May 21st 2015
Heather Tye, Stephan Zahn, Marco Hofmann, Michael Sanderson, Otmar Schaff, Matthias Troy, Moritz Mayer, Georg Rast, Sandeep Pal, Ulrich Guertler

8) Synthesis and antibacterial activity evaluation of C-5 side chain modified analogues of FYL-66, a potential agent against methicillin-resistant Staphylococcus aureus (ChemMedComm) Thursday May 21st 2015
Xiaoyan Yang, Zicheng Li, Zhenling Wang, Zitai Sang, Haiyue Long, Jianying Tang, Tao Yang, Yuanyuan Liu, Youfu Luo

9) 5-Iodo-2-arylalkylthio-6-aryl pyrimidin-4(3H)-ones as non-nucleoside anti-HBV agents (ChemMedComm) Wednesday May 20th 2015
Yu Zhang, Xuefeng Sun, Ningning Fan, Jianxiong Zhao, Jing Tu, Xiangmei Chen, Junyi Liu, Xiao-wei Wang

10) Alkylamino derivatives of N-benzylpyrazine-2-carboxamide: Synthesis and antimycobacterial evaluation (ChemMedComm) Wednesday May 20th 2015
Barbora Servusova-Vanaskova, Ondrej Jandourek, Pavla Paterova, Jana Kordulakova, Magdalena Plevakova, Vladimir Kubicek, Radim Kucera, Vladimir Garaj, Lieve Naesens, Jiri Kunes, Martin Dolezal, Jan Zitko

11) Synthesis and biological evaluation of potential small molecule inhibitors of Tumor Necrosis Factor (ChemMedComm) Wednesday May 20th 2015
Christos Papaneophytou, Polyxeni Alexiou, Athanasios Papakyriakou, Evangelos Ntougkos, Katerina Tsiliouka, Anna Maranti, Fotini Liepouri, Alexandros Strongilos, Anthi Mettou, Elias Couladouros, Elias Eliopoulos, Eleni Douni, George Kollias, George Kontopidis

12) Chromanones: selective and reversible Monoamine Oxidase B inhibitors with nanomolar potency (ChemMedComm) Wednesday May 20th 2015
Jin-Shuai Lan, Sai-Sai Xie, Ming Huang, Ya-Jian Hu, Ling-Yi Kong, Xiao-Bing Wang

13) Arylsulfonamide derivatives of (aryloxy)ethylpiperidines as 5-HT7 receptor antagonists and their psychotropic properties (ChemMedComm) Tuesday May 19th 2015
Pawel Maria Zajdel, Vittorio Canale, Anna Partyka, Krzysztof Marciniec, Grzegorz Satala, Rafal Kurczab, Agata Siwek, Magdalena Jastrzebska-Wiesek, Anna Wesolowska, Tomasz Kos, Piotr Popik, AJ Bojarski

14) Synthesis and in vitro Assessment of Chemically Modified siRNAs Targeting BCL2 that Contain 2'-Ribose and Triazole-linked Backbone Modifications (ChemMedComm) Monday May 18th 2015
Gord Hagen, Brandon J Peel, John Samis, Jean-Paul Desaulniers

15) Fragment-growing exploiting dynamic combinatorial chemistry of inhibitors of the aspartic protease endothiapepsin (ChemMedComm) Friday May 15th 2015
Milon Mondal, Daphne Groothuis, Anna Katharina Herta Hirsch

16) New selective A2A agonists and A3 antagonists for human adenosine receptors. Synthesis, biological activity and molecular docking studies (ChemMedComm) Wednesday May 13th 2015
Angel Guerrero, Anna Rodriguez, Hugo Gutierrez-de-Teran, David Rodriguez, Jose Brea, Maria Isabel Loza, Gloria Rosell, M. Pilar Bosch

17) A novel aminotriazole-based NHC complex for the design of gold(I) anti-cancer agents: synthesis and biological evaluation (ChemMedComm) Wednesday May 13th 2015
Tatiyana V Serebryanskaya, Andrey A. Zolotarev, Ingo Ott

18) 1,2,3-Triazole derivatives as antitubercular agents: synthesis, biological evaluation and molecular docking study (ChemMedComm) Wednesday May 13th 2015
Mubarak H. Shaikh, Dnyaneshwar D. Subhedar, Laxman Nawale, Dhiman Sarkar, Firoz A. Kalam Khan, Jaiprakash N. Sangshetti, Bapurao B. Shingate

19) Synthesis, Biological Evaluation and Mechanisms Study of a Class of Benzylideneindanone Derivatives as Novel Anticancer Agents (ChemMedComm) Friday May 8th 2015
Jinhui Hu, Jun Yan, Jie Chen, Yanqing Pang, ling huang, Xingshu Li

20) Identification of a novel class of Autotaxin inhibitors through cross-screening (ChemMedComm) Friday May 8th 2015
Diana Castagna, Emma Duffy, Dima Semaan, Louise Young, John Pritchard, simon macdonald, David Budd, Craig Jamieson, Allan John Bell Watson

21) Synthesis and evaluation of novel N-3-benzimidazolephenylbisamide derivatives for antiproliferative and hedgehog pathway inhibitory activity (ChemMedComm) Wednesday May 6th 2015
Chiyu Sun, Yangsheng Li, Ailong Shi, Jingzhou Zhang, Yafei Li, Mingming Zhao, Lijuan Zhang, Huachuan Zheng, Ying Meng, Huaiwei Ding, Hongrui Song

22) Synthesis and biological evaluation of nitric oxide-releasing hybrids from gemcitabine and phenylsulfonyl furoxans as anti-tumor agents (ChemMedComm) Wednesday April 29th 2015
Xianghua Li, Xuemin Wang, Chenjun Xu, Junkai Huang, Chengniu Wang, Xinyang Wang, Yong Ling, Liqin He

23) Synthesis and biodistribution of novel 99mTc labeled 4-nitroimidazole dithiocarbamate complexes as potential agents to target tumor hypoxia (ChemMedComm) Thursday April 23rd 2015
zhenxiang li, Junbo zhang, zhonghui jin, weifang zhang, Yanyan zhang

24) Synthesis and evaluation of [11C]PBD150, a radiolabeled glutaminyl cyclase inhibitor for the potential detection of Alzheimer's disease prior to amyloid β aggregation. (ChemMedComm) Thursday April 23rd 2015
Allen F Brooks, Isaac Jackson, Xia Shao, George Kropog, Phillip Sherman, Carole Quesada, Peter Scott

25) Discovery and optimisation of 1-acyl-2-benzylpyrrolidines as potent dual orexin receptor antagonists (ChemMedComm) Tuesday April 21st 2015
Jodi Williams, John Gatfield, Catherine Roch, Alexander Treiber, Francois Jenck, Martin Bolli, Christine Brotschi, Thierry Sifferlen, Bibia Heidmann, Christoph Boss

26) Novel indole-based sigma-2 receptor ligands: synthesis, structure-affinity relationship and antiproliferative activity (ChemMedComm) Monday April 20th 2015
Fang Xie, Torsten Kniess, Christin Neuber, Winnie Deuther-Conrad, Constantin Mamat, Brian P. Lieberman, BL Liu, Robert Henry Mach, Peter Brust, Jorg Steinbach, Jens Pietzsch, Hongmei Jia

27) Target-based Analysis of Ionization States of Bioactive Compounds (ChemMedComm) Monday April 20th 2015
Shilva Kayastha, Antonio de la Vega de Leon, Dilyana Dimova, J Bajorath

28) Exploring the Recognition Pathway at the Human A2A Adenosine Receptor of the Endogenous Agonist Adenosine using Supervised Molecular Dynamics Simulations. (ChemMedComm) Monday April 20th 2015
Davide Sabbadin, Antonella Ciancetta, Giuseppe Deganutti, Alberto Cuzzolin, Stefano Moro

29) 3-Aminooxazolidinone AHL analogs as hydrolytically-stable quorum sensing agonists in Gram-negative bacteria (ChemMedComm) Monday April 20th 2015
Min Guo, Yue Zheng, Clement Opoku-Temeng, Rusty Starks, Xiaochu Ma, Herman O Sintim

30) Synthesis, biological evaluation and QSAR studies of diarylpentanoid analogues as potential nitric oxide inhibitors (ChemMedComm) Monday April 20th 2015
Siti Munirah Mohd Faudzi, Sze Wei Leong, Faridah Abas, Mohd Fadhlizil Fasihi Mohd Aluwi, Kamal Rullah, Kok Wai Lam, Syahida Ahmad, Chau Ling Tham, Khozirah Shaari, Nordin H Lajis

31) Neuronal selective targeting, protection and signaling network analysis via dopamine mediated mesoporous silica nanoparticle (ChemMedComm) Monday April 20th 2015
shupeng li, hailong zhang, Yuhua Jiang, Sheng-gang Zhao, Li-qin Jiang, Yan Meng, Peng Liu, Myeong Ok Kim

32) Exploring cinnamic acid scaffold: development of promising neuroprotective lipophilic antioxidants (ChemMedComm) Wednesday April 15th 2015
Fernanda Borges, Daniel Chavarria, Tiago Silva, Teresa Summavielle, Jorge M.P.J. Garrido, Daniel Martins, Joana Bravo

33) Synthesis and Biological Evaluation of N-(4-phenylthiazol-2-yl) Cinnamamide Derivatives as Novel Potential Anti-tumor Agents (ChemMedComm) Monday April 13th 2015
Yong Luo, Yongxia Zhu, Kai Ran, Zhihao Liu, Ningyu Wang, Qiang Feng, Jun Zeng, Lidan Zhang, Bing He, Tinghong Ye, Shirui Zhu, Xiaolong Qiu, Luoting Yu

34) Direct photocapture of bromodomains using tropolone chemical probes (ChemMedComm) Monday April 13th 2015
Erik Hett, Eugene Chekler, Arindrajit Basak, Paul Bonin, Aldrin Denny, Andrew Flick, Kieran F Geoghegan, Shenping Liu, Mathew Pletcher, Parag Sahasrabudhe, Shores Salter, Ingrid Stock, Alex Taylor, Lyn H Jones

35) Discovery of a series of 2-(pyridinyl)pyrimidines as potent antagonists of GPR40 (ChemMedComm) Wednesday April 8th 2015
M J Waring, David Baker, Stuart Bennett, Alastair Dossetter, Mark Fenwick, Rob Garcia, Jennie Georgsson, Sam Groombridge, Sue Loxham, Philip Alexander MacFaul, Katie Maskill, David Morgan, Jenny Morrell, Helen Pointon, Graeme Robb, David Smith, Stephen Stokes, Gary Paul Wilkinson

36) Synthesis and Biological Evaluations of 2,3-Diarylthiophene Analogues of Combretastatin A-4 (ChemMedComm) Thursday April 2nd 2015
Weige Zhang, Zhan Wang, qingkun Yang, Zhaoshi Bai, Jun Sun, xuewei Jiang, Hongrui Song, Yingliang Wu

37) New substituted 9-propyladenine derivatives as adenosine receptor antagonists (ChemMedComm) Thursday April 2nd 2015
Catia Lambertucci, Michela Buccioni, Diego Dal Ben, Sonja Kachler, Gabriella Marucci, Andrea Spinaci, Ajiroghene Thomas, Karl-Norbert Klotz, R Volpini

38) Enantiomeric Diketopiperazines: Getting Insight of the Impact of the Configuration to the Conformation, Nanoimage, u-PA Inhibition and Anti-metastatic Activity (ChemMedComm) Tuesday March 31st 2015
Feng Wang, Shan Li, Yuji Wang, Haimei Zhu, Xiaoyi Zhang, Ming Zhao, Jianhui Wu, Shiqi Peng

39) Chemical genomics reveals novel biological activity of 1,2,3-dithiazoles as potent and reversible melanin synthesis inhibitors (ChemMedComm) Tuesday March 31st 2015
Panayiotis Andreas Koutentis, Paris Skourides, Oleg Alekseevich Rakitin, Anna Charalambous, Maria Koyioni, Ioanna Antoniades, Sophia Michaelidou, Iro Eleftheriou, Stanislav A Amelichev, Lidia S konstantinova, Despoina Pegeioti

40) Correction: Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday March 31st 2015
Taha M. A. Eldebss, Sobhi M. Gomha, Mohamed M. Abdulla, Reem K. Arafa

41) Structure-Based Virtual Screening for Fragment-Like Ligands of the G Protein-Coupled Histamine H4 Receptor (ChemMedComm) Monday March 30th 2015
Enade P. Istyastono, Albert J. Kooistra, Henry Vischer, Martien Kuijer, Luc Roumen, Saskia Nijmeijer, Rogier Smits, Iwan de Esch, Rob Leurs, Chris de Graaf

42) Novel synthesis of fluorochrome-coupled zoledronate with preserved functional activity on gamma/delta T cells and tumor cells (ChemMedComm) Monday March 30th 2015
Vijayanand Chandrasekaran, Shirin Kalyan, Valentina Biehl, Marcus Lettau, Patrik Theodor Nerdal, Hans-Heinrich Oberg, Daniela Wesch, Thisbe K Lindhorst, Dieter Kabelitz

43) Discovery of 2-(5,6-dimethoxypyridin-3-yl)-4-(2,4,6-trifluorobenzyl)-2H-pyrido[2,3-e][1,2,4]thiadiazin-3(4H)-one 1,1-dioxide (HTL6641), a dual orexin receptor antagonist with differentiated pharmacodynamic properties.[dagger] (ChemMedComm) Monday March 30th 2015
John Andrew Christopher, Sarah Aves, Jason Brown, James Errey, Suki Klair, Christopher Langmead, Oliver Mace, Richard Mould, Jayesh Patel, Ben Tehan, Andrei Zhukov, Fiona Marshall, Miles Congreve

44) Design of pyrazolo-pyrimidines as 11β-HSD1 inhibitors through optimisation of molecular electrostatic potential (ChemMedComm) Monday March 30th 2015
Graeme Robb, Scott Boyd, Christopher Davies, Alexander Dossetter, Frederick W Goldberg, Paul D Kemmitt, James Scott, John Swales

45) Concise Synthesis of Spergualin-Inspired Molecules With Broad-Spectrum Antibiotic Activity (ChemMedComm) Monday March 30th 2015
Victoria Assimon, Hao Shao, Sylvie Garneau-Tsodikova, Jason E. Gestwicki

46) 4-methyl-coumarins with cytotoxic activity against T24 and RT4 human bladder cancer cell lines (ChemMedComm) Thursday March 26th 2015
DAMIANA DA ROCHA VIANNA, LEILA Ruschel, FABRICIA Dietrich, Fabricio Figueiro, Fernanda Morrone, Romulo F. S. Canto, Flavia Corvello, Alice Velho, Allan Crestani, Helder Teixeira, Gilsane Lino von Poser, Ana Maria Oliveira Battastini, Vera Eifler-Lima

47) Tantalising technology (ChemMedComm) Tuesday March 24th 2015
Derek Lowe

48) Synthesis of a new HYNIC-DAPI derivative for labelling with 99mTechnetium and its in vitro evaluation in an FRTL5 cell line (ChemMedComm) Monday March 23rd 2015
Sandra Ferl, Gerd Wunderlich, Rene Smits, Alexander Hoepping, Anne Naumann, Jorg Kotzerke

49) Interactive articles in MedChemComm - connecting readers to a wealth of data and information (ChemMedComm) Thursday March 19th 2015
Richard Kelly

50) Insights into a defined secondary binding region on β-adrenoceptors and putative roles in ligand binding and drug design (ChemMedComm) Thursday March 12th 2015
Marvin Antonio Soriano-Ursua, Jose G Trujillo-Ferrara, Jose A Arias-Montano, Rafael Villalobos-Molina

51) Synthesis and evaluation of anticancer activity of novel andrographolide derivatives (ChemMedComm) Monday March 9th 2015
Devendar Ponnam, Lakshma Nayak V, Dharmendra Yadav, Niranjana Kumar Arigari, Kotesh Kumar Jonnala, Satya Srinivas KVN, Sridhar Balasubramanian, Feroz Khan, Pandu Sastry Kakaraparthi, Ramakrishna Sistla

52) Contributors to 'New Talent: Asia-Pacific' (ChemMedComm) Monday March 9th 2015


53) Membrane-interacting properties of the functionalised fatty acid moiety of muraymycin antibiotics (ChemMedComm) Friday March 6th 2015
Oliver Ries, Christian Carnarius, Claudia Steinem, Christian Ducho

54) In silico study on aging and reactivation processes of tabun conjugated AChE (ChemMedComm) Monday March 2nd 2015
Nellore Bhanu Chandar, Rabindranath Lo, Manoj K Kesharwani, Bishwajit Ganguly

55) Design, synthesis and biological evaluation of thiourea and nicotinamide-containing sorafenib analogs as antitumor agents (ChemMedComm) Monday March 2nd 2015
Xiangkai Kong, Zeyu Yao, Zuopeng He, Wen-Fang Xu, Jianwen Yao

56) Novel non-substrate modulators of the transmembrane efflux pump P-glycoprotein (ABCB1) (ChemMedComm) Friday February 27th 2015
Soren Krawczyk, Christiane Baumert, Josef Molnar, Christoph Ritter, Jens Hopner, Charlotte Kloft, Andreas Hilgeroth

57) Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday February 17th 2015
Taha Eldebss, Sobhi Gomha, Mohamed Abdalla, Reem Arafa

58) Matrix-immobilized yeast for large-scale production of recombinant human lactoferrin (ChemMedComm) Tuesday February 17th 2015
Chun Loong Ho, In Young Hwang, Kathy Loh, Matthew Chang

59) Synthesis and evaluation of amide, sulfonamide and urea - benzisoxazole derivatives as potential atypical antipsychotics (ChemMedComm) Friday February 13th 2015
Yin Chen, Yu Lan, Xudong Cao, Xiangqing Xu, Juecheng Zhang, Minquan Yu, Xin Liu, Bifeng Liu, Guisen Zhang

60) Synthesis and protective effect of new ligustrazine derivatives against CoCl2-induced neurotoxicity in differentiated PC12 cells. Part 2 (ChemMedComm) Thursday February 12th 2015
Bing Xu, Yan Gong, Xin Xu, Chenze Zhang, Yuzhong Zhang, Fuhao Chu, Hongbing Liu, Penglong Wang, Haimin Lei

61) BODIPY appended copper(II) complexes of curcumin showing mitochondria targeted remarkable photocytotoxicity in visible light (ChemMedComm) Thursday February 12th 2015
Akhil R Chakravarty, Arnab Bhattacharyya, Akanksha Dixit, Koushambi Mitra, Samya Banerjee, Anjali A Karande

62) Synthesis and biological evaluation of novel [capital Delta]2-isoxazoline fused cyclopentane derivatives as potential antimicrobial and anticancer agents (ChemMedComm) Wednesday February 11th 2015
Nagendra Babu Bathini, Santosh Kumar Prajapti, Shweta Shrivastava, Umesh Bihade, Ajay Kumar Gupta, V.G. M Naidu, Uttam Chand Banerjee

63) Evaluation of the anti-inflammatory/chondroprotective activity of aldose reductase inhibitors in human chondrocyte cultures (ChemMedComm) Wednesday February 4th 2015
Annamaria Panico, Rosanna Maccari, Venera Cardile, Sergio Avondo, Lucia Crasci, Rosaria Ottana

64) Inhibition of Insulin Amyloid Fibrillization by Glyco-Acridines: In vitro and in silico study (ChemMedComm) Wednesday February 4th 2015
Quan Van Vuong, Zuzana Bednarikova, Andrea Antosova, Huy Dinh Quoc Pham, Katarina Siposova, Nguyen Anh Tuan, Mai Suan Li, Zuzana Gazova

65) Application of QM/MM and QM methods to investigate histone deacetylase 8 (ChemMedComm) Monday February 2nd 2015
Duangkamol Gleeson, M. Paul Gleeson

66) Structure-Based Design, Synthesis by Click Chemistry and in Vivo Activity of Highly Selective A3 Adenosine Receptor Agonists (ChemMedComm) Monday February 2nd 2015
Dilip Tosh, Silvia Paoletta, Zhoumou Chen, Steven Crane, John Lloyd, Zhan-Guo Gao, Elizabeth Gizewski, John Auchampach, Daniela Salvemini, Kenneth A. Jacobson

67) Synthesis and evaluation of a series of resveratrol analogues as potent anticancer agents that target tubulin (ChemMedComm) Friday January 30th 2015
Nikhil Reddy Madadi, Hongliang Zong, Amit Ketkar, Zhen Chen, Narsimha Penthala, Venumadhav Janganati, Shobanbabu Bommagani, Robert Eoff, Monica Guzman, Peter Crooks

68) Design, Facile Synthesis and Anthelmintic Activity of New O-Substituted 6-Methoxybenzothiazole-2-carbamates (ChemMedComm) Tuesday January 27th 2015
A. Mohsen M.E. Omar, Omaima M. Aboulwafa, Doaa A. E. Issa, May M.S. El-Shokrofy, May E. Amr, Ibrahim M. El-Ashmawy

69) BEYOND THE AFFINITY FOR PROTEIN KINASE C: EXPLORING 2-PHENYL-3-HYDROXYPROPYL PIVALATE ANALOGUES AS C1 DOMAIN-TARGETING LIGANDS (ChemMedComm) Monday January 26th 2015
Daniela Rossi, Virpi Talman, Gustav Boije, Annamaria Marra, pietro Picconi, Rita Nasti, Massimo Serra, ANN JIHYAE, Marialaura Amadio, Alessia Pascale, Jeewoo Lee, Raimo Tuominen, Jari Yli-Kauhaluoma, Simona Collina

70) Correction: Identification of tris-(phenylalkyl)amines as new selective h5-HT2B receptor antagonists (ChemMedComm) Friday January 23rd 2015
Shashikanth Ponnala, Nirav Kapadia, Wayne Wesley Harding

71) Identification of Camphor Derivatives as Novel M2 Ion Channel Inhibitors of Influenza A Virus (ChemMedComm) Monday January 19th 2015
Xin Zhao, Zhen-Wei Zhang, Wei Cui, Shengwei Chen, Yang Zhou, Jianghong Dong, Yanling Jie, Junting Wan, Yong Xu, Wenhui Hu

72) O-Benzoyl Pyridine Aldoxime and Amidoxime Derivatives: Novel Efficient DNA Photo-Cleavage Agents (ChemMedComm) Thursday January 15th 2015
PARASKEVI KARAMTZIOTI, ASTERIOS PAPASTERGIOU, JOHN G. STEFANAKIS, ALEXANDROS E. KOUMBIS, IOANNA ANASTASIOU, MARIA KOFFA, KONSTANTINA C. FYLAKTAKIDOU

73) Nature of the Charged Head Group Dictates the Anticancer Potential of Lithocholic Acid-Tamoxifen Conjugates For Breast Cancer Therapy (ChemMedComm) Wednesday January 14th 2015
Kavita Yadav, Priyanshu Bhargava, Sandhya Bansal, Manish Singh, Siddhi Gupta, Geeta Sandhu, Sandeep Kumar, Vedagopuram Sreekanth, Avinash Bajaj

74) Targeted Photoresponsive TiO2-Coumarin nanoconjugate for efficient Combination therapy in MDA-MB-231 breast cancer cells: Synergic effect of Photodynamic Therapy (PDT) and Anticancer drug Chlorambucil (ChemMedComm) Wednesday January 14th 2015
Moumita Ganguly, Sourav K. Mukhopadhyay, Karthik S, Sharabani Barman, Pradeep N.D. Singh

75) Radiosynthesis of high affinity fluorine-18 labeled GnRH peptide analogues: in vitro studies and in vivo assessment of brain uptake in rats (ChemMedComm) Monday January 12th 2015
Dag Erlend Olberg, Sven H Hausner, Nadine Bauer, Jo Klaveness, Bard Indrevoll, Finn Olav Levy, Kjetil Wessel Andressen, Marie Dahl, Julie L. Sutcliffe, Ira Haraldsen

76) Design, synthesis and biological activity of 4′-[(benzimidazol-1-yl)methyl] biphenyl-2-sulphonamides as dual angiotensin II and endothelin A receptor antagonists (ChemMedComm) Monday January 12th 2015
Liping Hao, Weizhe Xue, Xiaofeng Han, Xing He, Jun Zhang, Zhiming Zhou

77) Activity Based Probes as Molecular Tools for Biomarker Discovery (ChemMedComm) Friday January 9th 2015
Luis Carvalho, Susana Dias Lucas, Eduardo Ruivo, Rui Moreira

78) Cytotoxic potential of di-spirooxindolo/acenaphthoquino andrographolide derivatives against MCF7 cell lines (ChemMedComm) Thursday January 8th 2015
Debanjana Chakraborty, Arindam Maitya, Chetan Kumar Jain, Abhijit Hazra, Yogesh Pandharinath Bharitkar, Tarun Jha, Hemanta Majumder, Susanta Roy Choudhury, Nirup Bikash Mondal

79) Dimethylaminoethyl Methacrylate Copolymer-siRNA nanoparticles for silencing therapeutically relevant gene in macrophages (ChemMedComm) Monday January 5th 2015
Ratnesh Jain, Prajakta Dandekar, Brigitta Loretz, Marcus Koch, C-M. lehr

80) Structure-activity relationship study on senktide for development of novel potent neurokinin-3 receptor selective agonists (ChemMedComm) Monday January 5th 2015
Ryosuke Misu, Koki Yamamoto, Ai Yamada, Taro Noguchi, Hiroaki Ohno, Takashi Yamamura, Hiroaki Okamura, Fuko Matsuda, Satoshi Ohkura, Shinya Oishi, Nobutaka Fujii

81) Synthesis and biological evaluation of pentanedioic acid derivatives as farnesyltransferase inhibitors (ChemMedComm) Monday January 5th 2015
liuqing Yang, wei liu, Hanbin Mei, yuan Zhang, Xiaojuan Yu, yufang xu, Honglin Li, Jin Huang, Zhenjiang Zhao

82) Recent discoveries and developments of Androgen Receptor based therapy for Prostate Cancer (ChemMedComm) Monday January 5th 2015
Ramakrishnan Elancheran, V.L Maruthanila, M Ramanathan, S Kabilan, R Devi, A Kunnumakara, Jibon Kotoky

83) Chemical space is big. Really big (ChemMedComm) Monday January 5th 2015
Derek Lowe

84) Discovery of Highly Potent Triazole Antifungal Agents with Piperdine-oxadiazole Side Chains (ChemMedComm) Wednesday December 24th 2014
Xiaomeng He, Yan Jiang, Yongqiang Zhang, Shanchao Wu, Guoqiang Dong, Na Liu, Yang Liu, Jianzhong Yao, Zhenyuan Miao, Yan Wang, Wannian Zhang, Chunquan Sheng

85) The Natural Product Brartemicin is a High Affinity Ligand for the Carbohydrate-Recognition Domain of the Macrophage Receptor Mincle (ChemMedComm) Tuesday December 23rd 2014
Kristian Mark Jacobsen, Ulrik Keiding, Lise Lindkvist Clement, Eva Susanne Schaffert, Neela Rambaruth, Mogens Johannsen, Kurt Drickamer, Thomas Bjornskov Poulsen

86) Inhibition of Influenza H5N1 invasion by modified heparin derivatives (ChemMedComm) Tuesday December 23rd 2014
Mark A. Skidmore, Anna Kajaste-Rudnitski, Nicola Wells, Scott Guimond, Timothy Rudd, Eliza Vicenzi, Edwin Yates

87) Pyrrole- and indole-containing tranylcypromine derivatives as novel lysine-specific demethylase 1 inhibitors active on cancer cells (ChemMedComm) Tuesday December 23rd 2014
Veronica Rodriguez, Sergio Valente, Stefano Rovida, Dante Rotili, Giulia Stazi, Alessia Lucidi, Giuseppe Ciossani, Andrea Mattevi, Oronza Botrugno, Paola Dessanti, Ciro Mercurio, Paola Vianello, Saverio Minucci, mario varasi, Antonello Mai

88) Enantiomeric resolution of [(2,2-diphenyl-1,3-dioxolan-4-yl)methyl](2-phenoxyethyl)amine, a potent α 1 and 5HT1A receptors ligand: an In Vitro and Computational Study (ChemMedComm) Tuesday December 23rd 2014
Livio Brasili, Silvia Franchini, Annamaria Baraldi, Claudia Sorbi, Federica Pellati, Elena Cichero, Umberto M. Battisti, Piero Angeli, Antonio Cilia

89) Synthesis and relationship of stability and biological activity of new DSS and TMP conjugates (ChemMedComm) Monday December 22nd 2014
Yewei Sun, Zicheng Tan, Zhibin Liang, Liang Wang, Luchen Shan, Pei Yu, Simon MingYuen Lee, Yuqiang Wang

90) Synthesis and antibacterial activity of trivalent ultrashort Arg-Trp-based antimicrobial peptides (AMPs) (ChemMedComm) Monday December 22nd 2014
Barbara C. Hoffknecht, H. Bauke Albada, Marina Sturm, Pascal Prochnow, Julia E. Bandow, Nils Metzler-Nolte

91) Non-nucleoside anti-HBV agents: Advances in structural optimization and mechanism of action investigations (ChemMedComm) Tuesday December 16th 2014
Na Liu, Diwakar Rai, Fabao Zhao, Haiyong Jia, Peng Zhan, Xinyong Liu

92) Discovery of a new class of histone deacetylase inhibitors with a novel zinc binding group (ChemMedComm) Tuesday December 16th 2014
Youxuan Li, Patrick M. Woster

93) The chemistry and pharmacology of privileged pyrroloquinazolines (ChemMedComm) Monday December 15th 2014
Bo Chao, Bingbing X Li, Xiangshu Xiao

94) Synthesis of six mexiletine derivatives with isoindolines attached as potential antioxidants and their evaluation as cardioprotective agents (ChemMedComm) Monday December 15th 2014
W Roy Jackson, Anh Chau, Grant Drummond, Bevyn Jarrott, Alyson Miller, Kamani Subasinghe, Christina Yan Ru Tan, Paul J White, Christine E Wright, James Ziogas

95) Solid- and solution-phase-based library of 2β-methyl substituted penicillin derivatives. Effects on growth inhibition of tumor cell lines (ChemMedComm) Monday December 15th 2014
Dora B. Boggian, Patricia Cornier, Ernesto Mata, Viviana Blanck, Mariano Cardenas, LP Roguin

96) Identification of tris-(phenylalkyl)amines as new selective h5-HT2B receptor antagonists (ChemMedComm) Monday December 15th 2014
Wayne Harding, Shashikanth Ponnala, Nirav Kapadia

97) Photoswitching property of hairpin ODNs with azobenzene derivatives in the loop (ChemMedComm) Monday December 15th 2014
Li Wu, Ya Wu, Hongwei Jin, Liangren Zhang, Yujian He, XinJing Tang

98) Synthesis and evaluation of 6-methylcoumarin derivatives as potent and selective Monoamine Oxidase B inhibitors (ChemMedComm) Monday December 15th 2014
Jin-Shuai Lan, Long-Fei Pan, Sai-Sai Xie, Xiao-Bing Wang, Ling-Yi Kong

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Mitch Andre Garcia's Chem Feeds 2008-present

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