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1) Novel peptidomimetics related to Gonadotropin releasing hormone (GnRH) (ChemMedComm) Tuesday July 28th 2015
Stefania Villa, Arianna Gelain, Luca Rizzi, Laura Legnani, Aurora Pacini, Katerina Spyridaki, Vlasios Karageorgos, George Liapakis

2) Enhanced Antibacterial Activities of Polythionates by Carbonate (ChemMedComm) Thursday July 23rd 2015
Guofang Li, yanbao zhao, Ping Li, Fuqiang Zhang, Peng Qu, Binjie Li, Qingyu Gao, Shaorong Wang

3) Investigating the generation of hydrogen sulfide from the phosphonamidodithioate slow-release donor GYY4137 (ChemMedComm) Thursday July 23rd 2015
Mark E. Wood, Matt Whiteman, Benjamin Edwin Alexander, Bridget Fox, Tahmina Khan, Joseph Maliszewski, Alexis Perry, Simon Coles, Mateusz Pitak

4) Structure-based design of a bisphosphonate 5'(3')-deoxyribonucleotidase inhibitor (ChemMedComm) Thursday July 23rd 2015
Petr Pachl, Ondrej Simak, Pavlina Rezacova, Milan Fabry, Milos Budesinsky, Jiri Brynda, Ivan Rosenberg

5) Inclusion of new 5-fluorouracil derivatives in liposome formulation for cancer treatment (ChemMedComm) Thursday July 23rd 2015
Manuela Petaccia, Maria condello, Luisa Giansanti, Angela La Bella, Francesca Leonelli, stefania Meschini, denise grdella villalva, evelin pellegrini, Francesca Ceccacci, Luciano Galantini, Giovanna Mancini

6) Novel 3-hydroxypyridin-4-one hexadentate ligand-based polymeric iron chelator: synthesis, characterization and antimicrobial evaluation (ChemMedComm) Monday July 20th 2015
Yingjun Zhou, Xiaole Kong, Junpei Li, Yongmin Ma, Robert Hider, Tao Zhou

7) Fragments in bromodomain drug discovery (ChemMedComm) Monday July 20th 2015
Paul Bamborough, Chun-wa Chung

8) Novel benzoxepine-1,2,3-triazole hybrids: Synthesis and pharmacological evaluation as potential antibacterial and anticancer agents (ChemMedComm) Thursday July 16th 2015
Naveen Kuntala, Jhonsee Rani Telu, Venkanna Banothu, N Suresh Babu, Jayashree anireddy, Sarbani Pal

9) GLYCODENDROPEPTIDES STIMULATE DENDRITIC CELL MATURATION AND T CELL PROLIFERATION. A POTENTIAL INFLUENZA A VIRUS IMMUNOTHERAPY. (ChemMedComm) Tuesday July 7th 2015
Ainhoa Mascaraque, Wioleta Kowalczyk, Tahia D Fernandez, Francisca Palomares, Cristobalina Mayorga, David Andreu, Javier Rojo

10) Correction: Identification of a novel class of autotaxin inhibitors through cross-screening (ChemMedComm) Tuesday July 7th 2015
Diana Castagna, Emma L. Duffy, Dima Semaan, Louise C. Young, John M. Pritchard, Simon J. F. Macdonald, David C. Budd, Craig Jamieson, Allan J. B. Watson

11) Design, synthesis and in vivo evaluation of sodium 2-benzyl-chloromalonates as new central nervous system depressants (ChemMedComm) Monday July 6th 2015
Jose Daniel Figueroa-Villar, Andreia Vieira, Bruno Marinho, Luana Souza, Patricia Fernandes

12) Correction: Discovery, synthesis and structure-activity analysis of symmetrical 2,7-disubstituted fluorenones as urea transporter inhibitors (ChemMedComm) Monday July 6th 2015
Sujin Lee, Cristina Esteva-Font, Puay-Wah Phuan, Marc O. Anderson, A. S. Verkman

13) Chemoprevention Effects of Sulindac-Based Compound on TPA-induced skin inflammation in Mice (ChemMedComm) Friday July 3rd 2015
Wenfeng Liu, Yonglian Li, Xi Zheng, kun zhang, Zhiyun Du

14) Synthesis and in vitro antiproliferative activity of novel pyrazolo[3,4-d]pyrimidine derivatives (ChemMedComm) Friday July 3rd 2015
Nermin S. Abdou, Rabah A. T. Serya, Ahmed Esmat, Mai F. Tolba, Nasser S. M. Ismail, Khaled A. M. Abouzid

15) Magic molecule modifiers (ChemMedComm) Thursday July 2nd 2015
Derek Lowe

16) The discovery of a novel antibiotic for the treatment of Clostridium difficile infections: a story of an effective academic-industrial partnership (ChemMedComm) Wednesday July 1st 2015
John Mann, Peter Taylor, Colin Dorgan, Peter Johnson, Francis X. Wilson, Richard Vickers, Aaron Dale, Stephen Neidle

17) Synthesis and anti-cancer screening of novel heterocyclic-(2H)-1,2,3-triazoles as potential anti-cancer agents (ChemMedComm) Tuesday June 30th 2015
Narsimha Penthala, Leena Maddukuri, Shraddha Thakkar, Nikhil Reddy Madadi, Gauri Lamture, Robert Eoff, Peter Crooks

18) Correction: Synthesis and biological evaluation of novel semi-conservative monocarbonyl analogs of curcumin as anti-inflammatory agents (ChemMedComm) Monday June 29th 2015
Zhe Wang, Peng Zou, Chenglong Li, Wenfei He, Bing Xiao, Qilu Fang, Wenbo Chen, Suqing Zheng, Yunjie Zhao, Yuepiao Cai, Guang Liang

19) Correction: Design, synthesis, and antibacterial evaluation of novel azolylthioether quinolones as MRSA DNA intercalators (ChemMedComm) Monday June 29th 2015
Ling Zhang, Kannekanti Vijaya Kumar, Syed Rasheed, Shao-Lin Zhang, Rong-Xia Geng, Cheng-He Zhou

20) PEGylated solid lipid nanoparticles: design, methotrexate loading and biological evaluation in animal models (ChemMedComm) Friday June 26th 2015
Dipti Kakkar, Shweta Dumoga, Rohit Kumar, Krishna Chuttani, Anil Kumar Mishra

21) Design, synthesis, and evaluation of semi-conservative mono-carbonyl analogs of curcumin as anti-inflammatory agents against lipopolysaccharide induced acute lung injury (ChemMedComm) Thursday June 25th 2015
Lili Dong, Suqing Zheng, Yali Zhang, Xin Jiang, Jianzhang Wu, Xiaoqing Zhang, Xiaoou Shan, Dandan Liang, Shilong Ying, Jianpeng Feng, Guang Liang

22) Discovery of TRAF-2 and NCK-interacting kinase (TNIK) inhibitors by ligand-based virtual screening methods (ChemMedComm) Wednesday June 24th 2015
Anna Bujak, Filip Stefaniak, Daria Zdzalik, Paulina Grygielewicz, Barbara Dymek, Marcin Zagozda, Pawel Gunerka, Monika Lamparska-Przybysz, Krzysztof Dubiel, Maciej Wieczorek, Karolina Dzwonek

23) Synthesis and anti-tubercular activity of conformationally-constrained and bisquinoline analogs of TMC207 (ChemMedComm) Tuesday June 23rd 2015
Dimpy Kalia, Anil Kumar K.S., Gajanand Meena, Kashmir Prasad Sethi, Rohit Sharma, Priyanka Trivedi, Shaheb Raj Khan, Ajay Singh Verma, Shyam Singh, Sandeep Sharma, Kuldeep K Roy, Ruchir Kant, Manju Yasodha Krishnan, Bhupendra N. Singh, Sudhir Sinha, Vinita Chaturvedi, Anil K Saxena, Dinesh K Dikshit

24) Transition Metal Diamine Complexes with Antimicrobial Activity Against Staphylococcus aureus and Methicillin-Resistant S. aureus (MRSA). (ChemMedComm) Monday June 22nd 2015
Joseph S Merola, George Karpin, David Morris, Mai Ngo, Joseph Falkinham

25) Synthesis and biological evaluation of α-sulfonamido-N-adamantanecarboxamide derivatives as 11β-HSD1 inhibitors (ChemMedComm) Thursday June 18th 2015
Young Hoon Kim, Seung Kyu Kang, Gwi Bin Lee, Kyu Myung Lee, Jaladi Ashok Kumar, Ki Young Kim, Sang Dal Rhee, Jeongmin Joo, Myung Ae Bae, Won Koo Lee, Jin Hee Ahn

26) Design and synthesis of potent and selective inhibitors of BRD9 and BRD7 bromodomains. (ChemMedComm) Monday June 15th 2015
Duncan Hay, Paul Brennan, Oleg Fedorov, Cynthia Tallant, Octovia Monteiro, Susanne Muller-Knapp, Stefan Knapp, Christopher J Schofield, Sarah Martin, Catherine Rogers

27) Identification of new hit scaffolds by INPHARMA-guided virtual screening (ChemMedComm) Monday June 15th 2015
Teresa Carlomagno, Justyna Sikorska, Luca Codutti, Lars Skjaerven, Bettina Elshorst, Rebeca Saez Ameneiro, Andrea Angelini, Peter Monecke

28) Correction: Synthesis and biological evaluation of N-(4-phenylthiazol-2-yl)cinnamamide derivatives as novel potential anti-tumor agents (ChemMedComm) Monday June 15th 2015
Yong Luo, Yongxia Zhu, Kai Ran, Zhihao Liu, Ningyu Wang, Qiang Feng, Jun Zeng, Lidan Zhang, Bing He, Tinghong Ye, Shirui Zhu, Xiaolong Qiu, Luoting Yu

29) Synthesis of novel 1-substituted triazole linked 1,2-benzothiazine 1,1-dioxido propenone derivatives as potent anti-inflammatory agents and inhibitors of monocyte-to-macrophage differentiation (ChemMedComm) Saturday June 13th 2015
B Narsaiah, Malla Reddy GANNARAPU, Sathish Babu Vasamsetti, nagender punna, Srigiridhar Kotamraju

30) Enhanced in vitro and in vivo uptake of a hydrophobic model drug coumarin-6 in the presence of cucurbit[7]uril (ChemMedComm) Friday June 12th 2015
Xiaoqing Miao, Ye Li, Ian Wyman, Simon Ming-Yuen Lee, Donal H Macartney, Ying Zheng, Ruibing Wang

31) Discovery of C-shaped aurone human neutrophil elastase inhibitors (ChemMedComm) Friday June 12th 2015
Susana Dias Lucas, Marta P. Carrasco, Lidia M. Goncalves, Rui Moreira, Rita Cardoso Guedes

32) Synthesis and biological evaluation of 4′-[(benzimidazol-1-yl) methyl] biphenyl-2-amides as dual angiotensin II and endothelin A receptor antagonists (ChemMedComm) Wednesday June 10th 2015
Xiaofeng Han, Weizhe Xue, Liping Hao, Zhiming Zhou

33) Synthesis and biological evaluation of lipid like 5-(2-hydroxyethyl)-4-methyl-1,3-thiazole derivatives as potential anticancer and antimicrobial agents (ChemMedComm) Wednesday June 10th 2015
Alla Zablotskaya, Izolda Segal, Prof. Athina Geronikaki, Galina Kazachonokh, Yuris Popelis, Irina Shestakova, Vizma Prof. Nikolajeva, Daina Eze

34) Discovery of Anilinopyrimidine-Based Naphthamide Derivatives as Potent VEGFR-2 Inhibitors (ChemMedComm) Monday June 8th 2015
Yongcong Lv, Mengyuan Li, Sufen Cao, Linjiang Tong, Ting Peng, Lixin Wei, Hua Xie, Jian Ding, Wenhu Duan

35) Identifying Farnesoid X Receptor Agonists with Naive Bayesian and Recursive Partitioning Approaches (ChemMedComm) Monday June 8th 2015
Qianzhi Ding, Chanjuan Li, Ling Wang, Yali Li, Huihao Zhou, Qiong Gu, Jun Xu

36) Novel Difluoroacetamide Analogues of Agomelatine and Melatonin: Probing the Melatonin Receptors for MT1-Selectivity (ChemMedComm) Monday June 8th 2015
Darius Paul Zlotos, Noura Riad, Mai Osman, Bala R. Dodda, Paula Witt-Enderby

37) Transcutaneous immunization against cancer using a solid-in-oil nanodispersion (ChemMedComm) Monday June 8th 2015
Yuya Hirakawa, Rie Wakabayashi, Ayaka Naritomi, Masato Sakuragi, Noriho Kamiya, Masahiro Goto

38) Effect of dibucaine hydrochloride on raft-like lipid domains in model membrane systems (ChemMedComm) Monday June 8th 2015
Kazunari Yoshida, Akito Takashima, Izumi Nishio

39) Discovery, synthesis and structure-activity analysis of symmetrical 2,7-disubstituted fluorenones as urea transporter inhibitors (ChemMedComm) Friday June 5th 2015
Sujin Lee, Cristina Esteva-Font, Puay-wah Phuan, Marc O. Anderson, Alan S. Verkman

40) RGD-peptides modifying dexamethasone: To enhance the efficacy of anti-inflammation and limit the risk of osteoporosis (ChemMedComm) Thursday June 4th 2015
Hualong Yu, Shenghui Mei, Zhao Li, Ming Zhao, Yuji Wang, Haimei Zhu, Yaonan Wang, Jianhui Wu, Chunying Cui, Wenyun Xu, Shiqi Peng

41) Substituted 4-hydroxy-1,2,3-triazoles: synthesis, characterization and first drug design applications through bioisosteric modulation and scaffold hopping approaches (ChemMedComm) Thursday May 28th 2015
Agnese Chiara Pippione, Franco Dosio, Alex Ducime, Antonella Federico, Katia Martina, Stefano Sainas, Bente Frolund, Major Gooyit, Kim D Janda, Donatella Boschi, Marco Lucio Lolli

42) Identifying the inhibitory mechanism of apigenin on the insulin ligand-receptor binding (ChemMedComm) Wednesday May 27th 2015
Yong Yang

43) Identification of an indole-triazole-amino acid conjugate as highly effective antifungal agent (ChemMedComm) Tuesday May 26th 2015
Kalpana Pawar, Anshuman Yadav, Parteek Prasher, Sahil Mishra, Balwinder Singh, Palwinder Singh, Sneha Komath

44) Synthesis and biological evaluation of novel semi-conservative mono-carbonyl analogs of curcumin as anti-inflammatory agents (ChemMedComm) Tuesday May 26th 2015
Zhe Wang, Peng Zou, Chenglong Li, Wenfei He, Bing Xiao, Qilu Fang, Wenbo Chen, Suqing Zheng, Yunjie Zhao, Yuepiao Cai, Guang Liang

45) Medicinal Organometallic Chemistry - an Emerging Strategy for the Treatment for Neglected Tropical Diseases (ChemMedComm) Tuesday May 26th 2015
Christopher Hyland, Ronald Brown

46) Design, Synthesis, Antibacterial Evaluation of Novel Azolylthioether Quinolones as MRSA DNA Intercalators (ChemMedComm) Thursday May 21st 2015
Ling Zhang, Vijaya Kumar Kannekanti, RASHEED SYED, Shao-Lin Zhang, Rong-Xia Geng, Cheng-He Zhou

47) Discovery of novel amino-pyrimidine inhibitors of the insulin-like growth factor 1 (IGF1R) and insulin receptor (INSR) kinases; parallel optimization of cell potency and hERG inhibition (ChemMedComm) Thursday May 21st 2015
Heather Tye, Stephan Zahn, Marco Hofmann, Michael Sanderson, Otmar Schaff, Matthias Troy, Moritz Mayer, Georg Rast, Sandeep Pal, Ulrich Guertler

48) Synthesis and antibacterial activity evaluation of C-5 side chain modified analogues of FYL-66, a potential agent against methicillin-resistant Staphylococcus aureus (ChemMedComm) Thursday May 21st 2015
Xiaoyan Yang, Zicheng Li, Zhenling Wang, Zitai Sang, Haiyue Long, Jianying Tang, Tao Yang, Yuanyuan Liu, Youfu Luo

49) 5-Iodo-2-arylalkylthio-6-aryl pyrimidin-4(3H)-ones as non-nucleoside anti-HBV agents (ChemMedComm) Wednesday May 20th 2015
Yu Zhang, Xuefeng Sun, Ningning Fan, Jianxiong Zhao, Jing Tu, Xiangmei Chen, Junyi Liu, Xiao-wei Wang

50) Alkylamino derivatives of N-benzylpyrazine-2-carboxamide: Synthesis and antimycobacterial evaluation (ChemMedComm) Wednesday May 20th 2015
Barbora Servusova-Vanaskova, Ondrej Jandourek, Pavla Paterova, Jana Kordulakova, Magdalena Plevakova, Vladimir Kubicek, Radim Kucera, Vladimir Garaj, Lieve Naesens, Jiri Kunes, Martin Dolezal, Jan Zitko

51) Synthesis and biological evaluation of potential small molecule inhibitors of Tumor Necrosis Factor (ChemMedComm) Wednesday May 20th 2015
Christos Papaneophytou, Polyxeni Alexiou, Athanasios Papakyriakou, Evangelos Ntougkos, Katerina Tsiliouka, Anna Maranti, Fotini Liepouri, Alexandros Strongilos, Anthi Mettou, Elias Couladouros, Elias Eliopoulos, Eleni Douni, George Kollias, George Kontopidis

52) Chromanones: selective and reversible Monoamine Oxidase B inhibitors with nanomolar potency (ChemMedComm) Wednesday May 20th 2015
Jin-Shuai Lan, Sai-Sai Xie, Ming Huang, Ya-Jian Hu, Ling-Yi Kong, Xiao-Bing Wang

53) Arylsulfonamide derivatives of (aryloxy)ethylpiperidines as 5-HT7 receptor antagonists and their psychotropic properties (ChemMedComm) Tuesday May 19th 2015
Pawel Maria Zajdel, Vittorio Canale, Anna Partyka, Krzysztof Marciniec, Grzegorz Satala, Rafal Kurczab, Agata Siwek, Magdalena Jastrzebska-Wiesek, Anna Wesolowska, Tomasz Kos, Piotr Popik, AJ Bojarski

54) Synthesis and in vitro Assessment of Chemically Modified siRNAs Targeting BCL2 that Contain 2'-Ribose and Triazole-linked Backbone Modifications (ChemMedComm) Monday May 18th 2015
Gord Hagen, Brandon J Peel, John Samis, Jean-Paul Desaulniers

55) Fragment-growing exploiting dynamic combinatorial chemistry of inhibitors of the aspartic protease endothiapepsin (ChemMedComm) Friday May 15th 2015
Milon Mondal, Daphne Groothuis, Anna Katharina Herta Hirsch

56) New selective A2A agonists and A3 antagonists for human adenosine receptors. Synthesis, biological activity and molecular docking studies (ChemMedComm) Wednesday May 13th 2015
Angel Guerrero, Anna Rodriguez, Hugo Gutierrez-de-Teran, David Rodriguez, Jose Brea, Maria Isabel Loza, Gloria Rosell, M. Pilar Bosch

57) A novel aminotriazole-based NHC complex for the design of gold(I) anti-cancer agents: synthesis and biological evaluation (ChemMedComm) Wednesday May 13th 2015
Tatiyana V Serebryanskaya, Andrey A. Zolotarev, Ingo Ott

58) 1,2,3-Triazole derivatives as antitubercular agents: synthesis, biological evaluation and molecular docking study (ChemMedComm) Wednesday May 13th 2015
Mubarak H. Shaikh, Dnyaneshwar D. Subhedar, Laxman Nawale, Dhiman Sarkar, Firoz A. Kalam Khan, Jaiprakash N. Sangshetti, Bapurao B. Shingate

59) Synthesis, Biological Evaluation and Mechanisms Study of a Class of Benzylideneindanone Derivatives as Novel Anticancer Agents (ChemMedComm) Friday May 8th 2015
Jinhui Hu, Jun Yan, Jie Chen, Yanqing Pang, ling huang, Xingshu Li

60) Identification of a novel class of Autotaxin inhibitors through cross-screening (ChemMedComm) Friday May 8th 2015
Diana Castagna, Emma Duffy, Dima Semaan, Louise Young, John Pritchard, simon macdonald, David Budd, Craig Jamieson, Allan John Bell Watson

61) Synthesis and evaluation of novel N-3-benzimidazolephenylbisamide derivatives for antiproliferative and hedgehog pathway inhibitory activity (ChemMedComm) Wednesday May 6th 2015
Chiyu Sun, Yangsheng Li, Ailong Shi, Jingzhou Zhang, Yafei Li, Mingming Zhao, Lijuan Zhang, Huachuan Zheng, Ying Meng, Huaiwei Ding, Hongrui Song

62) Synthesis and biological evaluation of nitric oxide-releasing hybrids from gemcitabine and phenylsulfonyl furoxans as anti-tumor agents (ChemMedComm) Wednesday April 29th 2015
Xianghua Li, Xuemin Wang, Chenjun Xu, Junkai Huang, Chengniu Wang, Xinyang Wang, Yong Ling, Liqin He

63) Synthesis and biodistribution of novel 99mTc labeled 4-nitroimidazole dithiocarbamate complexes as potential agents to target tumor hypoxia (ChemMedComm) Thursday April 23rd 2015
zhenxiang li, Junbo zhang, zhonghui jin, weifang zhang, Yanyan zhang

64) Synthesis and evaluation of [11C]PBD150, a radiolabeled glutaminyl cyclase inhibitor for the potential detection of Alzheimer's disease prior to amyloid β aggregation. (ChemMedComm) Thursday April 23rd 2015
Allen F Brooks, Isaac Jackson, Xia Shao, George Kropog, Phillip Sherman, Carole Quesada, Peter Scott

65) Discovery and optimisation of 1-acyl-2-benzylpyrrolidines as potent dual orexin receptor antagonists (ChemMedComm) Tuesday April 21st 2015
Jodi Williams, John Gatfield, Catherine Roch, Alexander Treiber, Francois Jenck, Martin Bolli, Christine Brotschi, Thierry Sifferlen, Bibia Heidmann, Christoph Boss

66) Novel indole-based sigma-2 receptor ligands: synthesis, structure-affinity relationship and antiproliferative activity (ChemMedComm) Monday April 20th 2015
Fang Xie, Torsten Kniess, Christin Neuber, Winnie Deuther-Conrad, Constantin Mamat, Brian P. Lieberman, BL Liu, Robert Henry Mach, Peter Brust, Jorg Steinbach, Jens Pietzsch, Hongmei Jia

67) Target-based Analysis of Ionization States of Bioactive Compounds (ChemMedComm) Monday April 20th 2015
Shilva Kayastha, Antonio de la Vega de Leon, Dilyana Dimova, J Bajorath

68) Exploring the Recognition Pathway at the Human A2A Adenosine Receptor of the Endogenous Agonist Adenosine using Supervised Molecular Dynamics Simulations. (ChemMedComm) Monday April 20th 2015
Davide Sabbadin, Antonella Ciancetta, Giuseppe Deganutti, Alberto Cuzzolin, Stefano Moro

69) 3-Aminooxazolidinone AHL analogs as hydrolytically-stable quorum sensing agonists in Gram-negative bacteria (ChemMedComm) Monday April 20th 2015
Min Guo, Yue Zheng, Clement Opoku-Temeng, Rusty Starks, Xiaochu Ma, Herman O Sintim

70) Synthesis, biological evaluation and QSAR studies of diarylpentanoid analogues as potential nitric oxide inhibitors (ChemMedComm) Monday April 20th 2015
Siti Munirah Mohd Faudzi, Sze Wei Leong, Faridah Abas, Mohd Fadhlizil Fasihi Mohd Aluwi, Kamal Rullah, Kok Wai Lam, Syahida Ahmad, Chau Ling Tham, Khozirah Shaari, Nordin H Lajis

71) Neuronal selective targeting, protection and signaling network analysis via dopamine mediated mesoporous silica nanoparticle (ChemMedComm) Monday April 20th 2015
shupeng li, hailong zhang, Yuhua Jiang, Sheng-gang Zhao, Li-qin Jiang, Yan Meng, Peng Liu, Myeong Ok Kim

72) Exploring cinnamic acid scaffold: development of promising neuroprotective lipophilic antioxidants (ChemMedComm) Wednesday April 15th 2015
Fernanda Borges, Daniel Chavarria, Tiago Silva, Teresa Summavielle, Jorge M.P.J. Garrido, Daniel Martins, Joana Bravo

73) Synthesis and Biological Evaluation of N-(4-phenylthiazol-2-yl) Cinnamamide Derivatives as Novel Potential Anti-tumor Agents (ChemMedComm) Monday April 13th 2015
Yong Luo, Yongxia Zhu, Kai Ran, Zhihao Liu, Ningyu Wang, Qiang Feng, Jun Zeng, Lidan Zhang, Bing He, Tinghong Ye, Shirui Zhu, Xiaolong Qiu, Luoting Yu

74) Direct photocapture of bromodomains using tropolone chemical probes (ChemMedComm) Monday April 13th 2015
Erik Hett, Eugene Chekler, Arindrajit Basak, Paul Bonin, Aldrin Denny, Andrew Flick, Kieran F Geoghegan, Shenping Liu, Mathew Pletcher, Parag Sahasrabudhe, Shores Salter, Ingrid Stock, Alex Taylor, Lyn H Jones

75) Discovery of a series of 2-(pyridinyl)pyrimidines as potent antagonists of GPR40 (ChemMedComm) Wednesday April 8th 2015
M J Waring, David Baker, Stuart Bennett, Alastair Dossetter, Mark Fenwick, Rob Garcia, Jennie Georgsson, Sam Groombridge, Sue Loxham, Philip Alexander MacFaul, Katie Maskill, David Morgan, Jenny Morrell, Helen Pointon, Graeme Robb, David Smith, Stephen Stokes, Gary Paul Wilkinson

76) Synthesis and Biological Evaluations of 2,3-Diarylthiophene Analogues of Combretastatin A-4 (ChemMedComm) Thursday April 2nd 2015
Weige Zhang, Zhan Wang, qingkun Yang, Zhaoshi Bai, Jun Sun, xuewei Jiang, Hongrui Song, Yingliang Wu

77) New substituted 9-propyladenine derivatives as adenosine receptor antagonists (ChemMedComm) Thursday April 2nd 2015
Catia Lambertucci, Michela Buccioni, Diego Dal Ben, Sonja Kachler, Gabriella Marucci, Andrea Spinaci, Ajiroghene Thomas, Karl-Norbert Klotz, R Volpini

78) Enantiomeric Diketopiperazines: Getting Insight of the Impact of the Configuration to the Conformation, Nanoimage, u-PA Inhibition and Anti-metastatic Activity (ChemMedComm) Tuesday March 31st 2015
Feng Wang, Shan Li, Yuji Wang, Haimei Zhu, Xiaoyi Zhang, Ming Zhao, Jianhui Wu, Shiqi Peng

79) Chemical genomics reveals novel biological activity of 1,2,3-dithiazoles as potent and reversible melanin synthesis inhibitors (ChemMedComm) Tuesday March 31st 2015
Panayiotis Andreas Koutentis, Paris Skourides, Oleg Alekseevich Rakitin, Anna Charalambous, Maria Koyioni, Ioanna Antoniades, Sophia Michaelidou, Iro Eleftheriou, Stanislav A Amelichev, Lidia S konstantinova, Despoina Pegeioti

80) Correction: Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday March 31st 2015
Taha M. A. Eldebss, Sobhi M. Gomha, Mohamed M. Abdulla, Reem K. Arafa

81) Structure-Based Virtual Screening for Fragment-Like Ligands of the G Protein-Coupled Histamine H4 Receptor (ChemMedComm) Monday March 30th 2015
Enade P. Istyastono, Albert J. Kooistra, Henry Vischer, Martien Kuijer, Luc Roumen, Saskia Nijmeijer, Rogier Smits, Iwan de Esch, Rob Leurs, Chris de Graaf

82) Novel synthesis of fluorochrome-coupled zoledronate with preserved functional activity on gamma/delta T cells and tumor cells (ChemMedComm) Monday March 30th 2015
Vijayanand Chandrasekaran, Shirin Kalyan, Valentina Biehl, Marcus Lettau, Patrik Theodor Nerdal, Hans-Heinrich Oberg, Daniela Wesch, Thisbe K Lindhorst, Dieter Kabelitz

83) Discovery of 2-(5,6-dimethoxypyridin-3-yl)-4-(2,4,6-trifluorobenzyl)-2H-pyrido[2,3-e][1,2,4]thiadiazin-3(4H)-one 1,1-dioxide (HTL6641), a dual orexin receptor antagonist with differentiated pharmacodynamic properties.[dagger] (ChemMedComm) Monday March 30th 2015
John Andrew Christopher, Sarah Aves, Jason Brown, James Errey, Suki Klair, Christopher Langmead, Oliver Mace, Richard Mould, Jayesh Patel, Ben Tehan, Andrei Zhukov, Fiona Marshall, Miles Congreve

84) Design of pyrazolo-pyrimidines as 11β-HSD1 inhibitors through optimisation of molecular electrostatic potential (ChemMedComm) Monday March 30th 2015
Graeme Robb, Scott Boyd, Christopher Davies, Alexander Dossetter, Frederick W Goldberg, Paul D Kemmitt, James Scott, John Swales

85) Concise Synthesis of Spergualin-Inspired Molecules With Broad-Spectrum Antibiotic Activity (ChemMedComm) Monday March 30th 2015
Victoria Assimon, Hao Shao, Sylvie Garneau-Tsodikova, Jason E. Gestwicki

86) 4-methyl-coumarins with cytotoxic activity against T24 and RT4 human bladder cancer cell lines (ChemMedComm) Thursday March 26th 2015
DAMIANA DA ROCHA VIANNA, LEILA Ruschel, FABRICIA Dietrich, Fabricio Figueiro, Fernanda Morrone, Romulo F. S. Canto, Flavia Corvello, Alice Velho, Allan Crestani, Helder Teixeira, Gilsane Lino von Poser, Ana Maria Oliveira Battastini, Vera Eifler-Lima

87) Tantalising technology (ChemMedComm) Tuesday March 24th 2015
Derek Lowe

88) Synthesis of a new HYNIC-DAPI derivative for labelling with 99mTechnetium and its in vitro evaluation in an FRTL5 cell line (ChemMedComm) Monday March 23rd 2015
Sandra Ferl, Gerd Wunderlich, Rene Smits, Alexander Hoepping, Anne Naumann, Jorg Kotzerke

89) Interactive articles in MedChemComm - connecting readers to a wealth of data and information (ChemMedComm) Thursday March 19th 2015
Richard Kelly

90) Insights into a defined secondary binding region on β-adrenoceptors and putative roles in ligand binding and drug design (ChemMedComm) Thursday March 12th 2015
Marvin Antonio Soriano-Ursua, Jose G Trujillo-Ferrara, Jose A Arias-Montano, Rafael Villalobos-Molina

91) Synthesis and evaluation of anticancer activity of novel andrographolide derivatives (ChemMedComm) Monday March 9th 2015
Devendar Ponnam, Lakshma Nayak V, Dharmendra Yadav, Niranjana Kumar Arigari, Kotesh Kumar Jonnala, Satya Srinivas KVN, Sridhar Balasubramanian, Feroz Khan, Pandu Sastry Kakaraparthi, Ramakrishna Sistla

92) Contributors to 'New Talent: Asia-Pacific' (ChemMedComm) Monday March 9th 2015


93) Membrane-interacting properties of the functionalised fatty acid moiety of muraymycin antibiotics (ChemMedComm) Friday March 6th 2015
Oliver Ries, Christian Carnarius, Claudia Steinem, Christian Ducho

94) In silico study on aging and reactivation processes of tabun conjugated AChE (ChemMedComm) Monday March 2nd 2015
Nellore Bhanu Chandar, Rabindranath Lo, Manoj K Kesharwani, Bishwajit Ganguly

95) Design, synthesis and biological evaluation of thiourea and nicotinamide-containing sorafenib analogs as antitumor agents (ChemMedComm) Monday March 2nd 2015
Xiangkai Kong, Zeyu Yao, Zuopeng He, Wen-Fang Xu, Jianwen Yao

96) Novel non-substrate modulators of the transmembrane efflux pump P-glycoprotein (ABCB1) (ChemMedComm) Friday February 27th 2015
Soren Krawczyk, Christiane Baumert, Josef Molnar, Christoph Ritter, Jens Hopner, Charlotte Kloft, Andreas Hilgeroth

97) Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling (ChemMedComm) Tuesday February 17th 2015
Taha Eldebss, Sobhi Gomha, Mohamed Abdalla, Reem Arafa

98) Matrix-immobilized yeast for large-scale production of recombinant human lactoferrin (ChemMedComm) Tuesday February 17th 2015
Chun Loong Ho, In Young Hwang, Kathy Loh, Matthew Chang

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