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99) Inhibitor Discovery for the Human GLUT1 from Homology Modeling and Virtual Screening (ACS Chemical Biology) Wednesday May 11th 2016
Peter Man-Un Ung, Wenxin Song, Lili Cheng, Xinbin Zhao, Hailin Hu, Ligong Chen, Avner Schlessinger

100) Deazaflavin Inhibitors of Tyrosyl-DNA Phosphodiesterase 2 (TDP2) Specific for the Human Enzyme and Active against Cellular TDP2 (ACS Chemical Biology) Wednesday May 11th 2016
Christophe Marchand, Monica Abdelmalak, Jayakanth Kankanala, Shar-Yin Huang, Evgeny Kiselev, Katherine Fesen, Kayo Kurahashi, Hiroyuki Sasanuma, Shunichi Takeda, Hideki Aihara, Zhengqiang Wang, Yves Pommier

101) Discovery of a novel NEDD8 Activating Enzyme Inhibitor with Piperidin-4-amine Scaffold by Structure-Based Virtual Screening (ACS Chemical Biology) Friday May 6th 2016
Peng Lu, Xiaoxin Liu, Xinrui Yuan, Minfang He, Yubin Wang, Qi Zhang, Ping-kai Ouyang

102) Bacterial (ACS Chemical Biology) Friday May 6th 2016
Ratana Charoenwattanasatien, Salila Pengthaisong, Imogen Breen, Risa Mutoh, Sompong Sansenya, Yanling Hua, Anupong Tankrathok, Liang Wu, Chomphunuch Songsiriritthigul, Hideaki Tanaka, Spencer J. Williams, Gideon J. Davies, Genji Kurisu, James R. Ketudat Cairns

103) Hepatitis C Virus Selectively Alters the Intracellular Localization of Desmosterol (ACS Chemical Biology) Friday May 6th 2016
Valerie A. Villareal, Dan Fu, Deirdre A. Costello, Xiaoliang Sunney Xie, Priscilla L. Yang

104) ML314: A Biased Neurotensin Receptor Ligand for Methamphetamine Abuse (ACS Chemical Biology) Thursday May 5th 2016
Larry S. Barak, Yushi Bai, Sean Peterson, Tama Evron, Nikhil M. Urs, Satyamaheshwar Peddibhotla, Michael P. Hedrick, Paul Hershberger, Patrick R. Maloney, Thomas D.Y. Chung, Ramona M. Rodriguiz, William C. Wetsel, James B. Thomas, Glen R. Hanson, Anthony B. Pinkerton, Marc G. Caron

105) Clickable Photoaffinity Ligands for Metabotropic Glutamate Receptor 5 Based on Select Acetylenic Negative Allosteric Modulators (ACS Chemical Biology) Wednesday May 4th 2016
Karen J. Gregory, Ranganadh Velagaleti, David M. Thal, Ryan M. Brady, Arthur Christopoulos, P. Jeffrey Conn, David J. Lapinsky

106) Fusion of Ferredoxin and Cytochrome P450 Enables Direct Light-Driven Biosynthesis (ACS Chemical Biology) Wednesday May 4th 2016
Silas Busck Mellor, Agnieszka Zygadlo Nielsen, Meike Burow, Mohammed Saddik Motawia, Dainius Jakubauskas, Birger Lindberg M

107) Elastase-like Activity Is Dominant to Chymotrypsin-like Activity in 20S Proteasome (ACS Chemical Biology) Monday May 2nd 2016
Dennis Bensinger, Theresa Neumann, Christoph Scholz, Constantin Voss, Sabine Knorr, Ulrike Kuckelkorn, Kay Hamacher, Peter-Michael Kloetzel, Boris Schmidt

108) Delivery of Non-Native Cargo into Mammalian Cells Using Anthrax Lethal Toxin (ACS Chemical Biology) Monday May 2nd 2016
Amy E. Rabideau, Bradley Lether Pentelute

109) Stabilizing the CH2 Domain of an Antibody by Engineering in an Enhanced Aromatic Sequon (ACS Chemical Biology) Friday April 29th 2016
Wentao Chen, Leopold Kong, Stephen Connelly, Julia M. Dendle, Yu Liu, Ian A. Wilson, Evan T. Powers, Jeffery W. Kelly

110) Identification of a Binding Site for Unsaturated Fatty Acids in the Orphan Nuclear Receptor Nurr1 (ACS Chemical Biology) Friday April 29th 2016
Ian Mitchelle S. de Vera, Pankaj K. Giri, Paola Munoz-Tello, Richard Brust, Jakob Fuhrmann, Edna Matta-Camacho, Jinsai Shang, Sean Campbell, Henry D. Wilson, Juan Granados, William J. Gardner, Trevor P. Creamer, Laura. A. Solt, Douglas J. Kojetin

111) Inhibition of Zinc-Dependent Histone Deacetylases with a Chemically Triggered Electrophile (ACS Chemical Biology) Friday April 29th 2016
Zarko V. Boskovic, Melissa M. Kemp, Allyson M. Freedy, Vasanthi S. Viswanathan, Marius S. Pop, Jason H. Fuller, Nicole M. Martinez, Samuel O. Figueroa Lazu

112) Cell Permeable Ratiometric Fluorescent Sensors for Imaging Phosphoinositides (ACS Chemical Biology) Friday April 29th 2016
Samsuzzoha Mondal, Ananya Rakshit, Suranjana Pal, Ankona Datta

113) Dissecting the Multiple Roles of PqsE in Pseudomonas aeruginosa Virulence by Discovery of Small Tool Compounds (ACS Chemical Biology) Friday April 29th 2016
Michael Zender, Florian Witzgall, Steffen L. Drees, Elisabeth Weidel, Christine K. Maurer, Susanne Fetzner, Wulf Blankenfeldt, Martin Empting, Rolf W. Hartmann

114) Pharmacological Chaperones: Design and Development of New Therapeutic Strategies for the Treatment of Conformational Diseases (ACS Chemical Biology) Friday April 29th 2016
Marino Convertino, Jhuma Das, Nikolay V. Dokholyan

115) Identification of MAC1: A Small Molecule That Rescues Spindle Bipolarity in Monastrol-Treated Cells (ACS Chemical Biology) Friday April 29th 2016
Naowras Al-Obaidi, Timothy J. Mitchison, Craig M. Crews, Thomas U. Mayer

116) Synthesis and Characterization of a Promising Novel FFAR1/GPR40 Targeting Fluorescent Probe for (ACS Chemical Biology) Tuesday April 26th 2016
Romain Bertrand, Andrea Wolf, Yuri Ivashchenko, Matthias Lo

117) Production of Sactipeptides in Escherichia coli: Probing the Substrate Promiscuity of Subtilosin A Biosynthesis (ACS Chemical Biology) Monday April 25th 2016
Paul M. Himes, Scott E. Allen, Sungwon Hwang, Albert A. Bowers

118) Structural Basis of Substrate Specificity in Geobacter metallireducens SMUG1 (ACS Chemical Biology) Friday April 22nd 2016
Zhemin Zhang, Jiemin Shen, Ye Yang, Jing Li, Weiguo Cao, Wei Xie

119) Discovery of a Highly Selective STK16 Kinase Inhibitor (ACS Chemical Biology) Friday April 22nd 2016
Feiyang Liu, Jinhua Wang, Xingxing Yang, Binhua Li, Hong Wu, Shuang Qi, Cheng Chen, Xiaochuan Liu, Kailin Yu, Wenchao Wang, Zheng Zhao, Aoli Wang, Yongfei Chen, Li Wang, Nathanael S. Gray, Jing Liu, Xin Zhang, Qingsong Liu

120) Cell-specific Profiling of Nascent Proteomes Using Orthogonal Enzyme-mediated Puromycin Incorporation (ACS Chemical Biology) Thursday April 21st 2016
Ruth M. Barrett, Hui-wen Liu, Haihong Jin, Richard H. Goodman, Michael S. Cohen

121) Inforna 2.0: A Platform for the Sequence-Based Design of Small Molecules Targeting Structured RNAs (ACS Chemical Biology) Wednesday April 20th 2016
Matthew D. Disney, Audrey M. Winkelsas, Sai Pradeep Velagapudi, Mark Southern, Mohammad Fallahi, Jessica L. Childs-Disney

122) Conformational Adaption May Explain the Slow Dissociation Kinetics of Roniciclib (BAY 1000394), a Type I CDK Inhibitor with Kinetic Selectivity for CDK2 and CDK9 (ACS Chemical Biology) Tuesday April 19th 2016
Pelin Ayaz, Dorothee Andres, Dennis A. Kwiatkowski, Carl-Christian Kolbe, Philip Lienau, Gerhard Siemeister, Ulrich Lu

123) Altering the Specificity of the Antibody Response to HIV gp120 with a Glycoconjugate Antigen (ACS Chemical Biology) Monday April 18th 2016
Chang-Cheng Liu, Canjia Zhai, Xiu-Jing Zheng, Xin-Shan Ye

124) The Chemical Ecology of Predatory Soil Bacteria (ACS Chemical Biology) Friday April 15th 2016
Brandon L. Findlay

125) Turnover of Bacterial Cell Wall by SltB3, a Multidomain Lytic Transglycosylase of Pseudomonas aeruginosa (ACS Chemical Biology) Monday April 11th 2016
Mijoon Lee, Teresa Domi

126) Global Isotope Metabolomics Reveals Adaptive Strategies for Nitrogen Assimilation (ACS Chemical Biology) Friday April 8th 2016
Michael E. Kurczy, Erica M. Forsberg, Michael P. Thorgersen, Farris L. Poole, H. Paul Benton, Julijana Ivanisevic, Minerva L. Tran, Judy D. Wall, Dwayne A. Elias, Michael W. W. Adams, Gary Siuzdak

127) Exploring Peptide Ligase Orthologs in Actinobacteria (ACS Chemical Biology) Friday April 8th 2016
Yasushi Ogasawara, Junpei Kawata, Motoyoshi Noike, Yasuharu Satoh, Kazuo Furihata, Tohru Dairi

128) Transition State Structure and Inhibition of Rv0091, a 5 (ACS Chemical Biology) Friday April 8th 2016
Hilda A. Namanja-Magliano, Christopher F. Stratton, Vern L. Schramm

129) Identification of a Novel Mycobacterial Arabinosyltransferase Activity Which Adds an Arabinosyl Residue to (ACS Chemical Biology) Friday April 8th 2016
Shiva kumar Angala, Michael R. McNeil, Lu Zou, Avraham Liav, Junfeng Zhang, Todd L. Lowary, Mary Jackson

130) Six Biophysical Screening Methods Miss a Large Proportion of Crystallographically Discovered Fragment Hits: A Case Study (ACS Chemical Biology) Friday April 8th 2016
Johannes Schiebel, Nedyalka Radeva, Stefan G. Krimmer, Xiaojie Wang, Martin Stieler, Frederik R. Ehrmann, Kan Fu, Alexander Metz, Franziska U. Huschmann, Manfred S. Weiss, Uwe Mueller, Andreas Heine, Gerhard Klebe

131) Synchronous Bioimaging of Intracellular pH and Chloride Based on LSS Fluorescent Protein (ACS Chemical Biology) Thursday April 7th 2016
Jose M. Paredes, Aurora I. Idilli, Letizia Mariotti, Gabriele Losi, Lyaysan R. Arslanbaeva, Sebastian Sulis Sato, Pietro Artoni, Joanna Szczurkowska, Laura Cancedda, Gian Michele Ratto, Giorgio Carmignoto, Daniele Arosio

132) Benzothiazole Sulfinate: a Water-Soluble and Slow-Releasing Sulfur Dioxide Donor (ACS Chemical Biology) Thursday April 7th 2016
Jacob J. Day, Zhenhua Yang, Wei Chen, Armando Pacheco, Ming Xian

133) An Ancestral Tryptophanyl-tRNA Synthetase Precursor Achieves High Catalytic Rate Enhancement without Ordered Ground-State Tertiary Structures (ACS Chemical Biology) Thursday April 7th 2016
Paul J. Sapienza, Li Li, Tishan Williams, Andrew L. Lee, Charles W. Carter

134) Catch and Release DNA Decoys: Capture and Photochemical Dissociation of NF- (ACS Chemical Biology) Thursday April 7th 2016
Nicholas B. Struntz, Daniel A. Harki

135) Potent Inhibitors of Acetyltransferase Eis Overcome Kanamycin Resistance in Mycobacterium tuberculosis (ACS Chemical Biology) Thursday April 7th 2016
Melisa J. Willby, Keith D. Green, Chathurada S. Gajadeera, Caixia Hou, Oleg V. Tsodikov, James E. Posey, Sylvie Garneau-Tsodikova

136) Traceless Production of Cyclic Peptide Libraries in E. coli (ACS Chemical Biology) Wednesday April 6th 2016
Jaime E. Townend, Ali Tavassoli

137) Chondro-Protective and Antiarthritic Effects of Sulfonamido-Based Gallate (ACS Chemical Biology) Tuesday April 5th 2016
Zhenhui Lu, Huayu Wu, Xiao Lin, Buming Liu, Cuiwu Lin, Li Zheng, Jinmin Zhao

138) Site-Specific Radiofluorination of Biomolecules with 8-[18F]-Fluorooctanoic Acid Catalyzed by Lipoic Acid Ligase (ACS Chemical Biology) Thursday March 31st 2016
Christopher R. Drake, Natalia Sevillano, Charles Truillet, Charles S. Craik, Henry F. VanBrocklin, Michael J. Evans

139) Structure of the Human Protein Kinase ZAK in Complex with Vemurafenib (ACS Chemical Biology) Thursday March 31st 2016
Sebastian Mathea, Kamal R. Abdul Azeez, Eidarus Salah, Cynthia Tallant, Finn Wolfreys, Rebecca Konietzny, Roman Fischer, Hua Jane Lou, Paul E. Brennan, Gisela Schnapp, Alexander Pautsch, Benedikt M. Kessler, Benjamin E. Turk, Stefan Knapp

140) Reprogramming Caspase-7 Specificity by Regio-Specific Mutations and Selection Provides Alternate Solutions for Substrate Recognition (ACS Chemical Biology) Thursday March 31st 2016
Maureen E. Hill, Derek J. MacPherson, Peng Wu, Olivier Julien, James A. Wells, Jeanne A. Hardy

141) Highly Dynamic Interactions Maintain Kinetic Stability of the ClpXP Protease During the ATP-Fueled Mechanical Cycle (ACS Chemical Biology) Wednesday March 30th 2016
Alvaro J. Amor, Karl R. Schmitz, Jason K. Sello, Tania A. Baker, Robert T. Sauer

142) Mass Spectrometry Reveals Protein Kinase CK2 High-Order Oligomerization via the Circular and Linear Assembly (ACS Chemical Biology) Tuesday March 29th 2016
Wei-Guang Seetoh, Daniel Shiu-Hin Chan, Dijana Matak-Vinkovic

143) Nicotinamide Cofactors Suppress Active-Site Labeling of Aldehyde Dehydrogenases (ACS Chemical Biology) Friday March 25th 2016
Naim Stiti, Balakumaran Chandrasekar, Laura Strubl, Shabaz Mohammed, Dorothea Bartels, Renier A. L. van der Hoorn

144) Designing an Antibody-Based Chaperoning System through Programming the Binding and Release of the Folding Intermediate (ACS Chemical Biology) Friday March 25th 2016
Tingting Liu, Caixian Sun, Cong Li, Jinhyuk Lee, Yong-Doo Park, Yixin Zhang, Sen Li

145) Directed Evolution of a Cyclized Peptoid (ACS Chemical Biology) Thursday March 24th 2016
Takashi Kawakami, Koji Ogawa, Tomohisa Hatta, Naoki Goshima, Tohru Natsume

146) Bacterial Riboswitches and Ribozymes Potently Activate the Human Innate Immune Sensor PKR (ACS Chemical Biology) Thursday March 24th 2016
Chelsea M. Hull, Ananya Anmangandla, Philip C. Bevilacqua

147) Thymidylate Limitation Potentiates Cephalosporin Activity toward Enterococci via an Exopolysaccharide-Based Mechanism (ACS Chemical Biology) Wednesday March 23rd 2016
Jessica S. Hoff, Christopher J. Kristich

148) Mixing Up the Pieces of the Desferrioxamine B Jigsaw Defines the Biosynthetic Sequence Catalyzed by DesD (ACS Chemical Biology) Wednesday March 23rd 2016
Thomas J. Telfer, Michael P. Gotsbacher, Cho Zin Soe, Rachel Codd

149) Chemically Modifying Viruses for Diverse Applications (ACS Chemical Biology) Monday March 21st 2016
Kritika Mohan, Gregory A. Weiss

150) Why Nature Chose Selenium (ACS Chemical Biology) Monday March 21st 2016
Hans J. Reich, Robert J. Hondal

151) Targeting Tumor Cells by Natural Anti-Carbohydrate Antibodies Using Rhamnose-Functionalized Liposomes (ACS Chemical Biology) Friday March 18th 2016
Xuexia Li, Xiongjian Rao, Li Cai, Xuling Liu, Huixia Wang, Weinan Wu, Chenggang Zhu, Min Chen, Peng G. Wang, Wen Yi

152) Reaction of PerR with Molecular Oxygen May Assist H2O2 Sensing in Anaerobes (ACS Chemical Biology) Wednesday March 16th 2016
Ramakrishnan Sethu, Eric Goure

153) Orthogonal Assays Clarify the Oxidative Biochemistry of Taxol P450 CYP725A4 (ACS Chemical Biology) Wednesday March 16th 2016
Bradley Walters Biggs, John Edward Rouck, Amogh Kambalyal, William Arnold, Chin Giaw Lim, Marjan De Mey, Mark O

154) A Small Molecule Screen Exposes mTOR Signaling Pathway Involvement in Radiation-Induced Apoptosis (ACS Chemical Biology) Monday March 14th 2016
Elizabeth R. Sharlow, Stephanie Leimgruber, Ana Lira, Michael J. McConnell, Andre

155) Vectorization of Nucleic Acids for Therapeutic Approach: Tutorial Review (ACS Chemical Biology) Friday March 11th 2016
Frederic Geinguenaud, Erwann Guenin, Yoann Lalatonne, Laurence Motte

156) Phage Selection of Chemically Stabilized (ACS Chemical Biology) Friday March 11th 2016
Philippe Diderich, Davide Bertoldo, Pierre Dessen, Maola M. Khan, Irene Pizzitola, Werner Held, Joerg Huelsken, Christian Heinis

157) Mapping and Exploring the Collagen-I Proteostasis Network (ACS Chemical Biology) Wednesday March 9th 2016
Andrew S. DiChiara, Rebecca J. Taylor, Madeline Y. Wong, Ngoc-Duc Doan, Amanda M. Del Rosario, Matthew D. Shoulders

158) Chemically Induced Cryptic Sesquiterpenoids and Expression of Sesquiterpene Cyclases in Botrytis cinerea Revealed New Sporogenic (+)-4-Epieremophil-9-en-11-ols (ACS Chemical Biology) Tuesday March 8th 2016
Cristina Pinedo, Javier Moraga, Javier Barua, Victoria E. Gonza

159) Key Players in I-DmoI Endonuclease Catalysis Revealed from Structure and Dynamics (ACS Chemical Biology) Tuesday March 8th 2016
Rafael Molina, Neva Besker, Maria Jose Marcaida, Guillermo Montoya, Jesu

160) Transition State Structure of RNA Depurination by Saporin L3 (ACS Chemical Biology) Tuesday March 8th 2016
Hongling Yuan, Christopher F. Stratton, Vern L. Schramm

161) Application of an Integrated GPCR SAR-Modeling Platform To Explain the Activation Selectivity of Human 5-HT2C over 5-HT2B (ACS Chemical Biology) Monday March 7th 2016
Alexander Heifetz, R. Ian Storer, Gordon McMurray, Tim James, Inaki Morao, Matteo Aldeghi, Mike J. Bodkin, Philip C. Biggin

162) Decoupling Activation of Heme Biosynthesis from Anaerobic Toxicity in a Molecule Active in Staphylococcus aureus (ACS Chemical Biology) Friday March 4th 2016
Brendan F. Dutter, Laura A. Mike, Paul R. Reid, Katherine M. Chong, Susan J. Ramos-Hunter, Eric P. Skaar, Gary A. Sulikowski

163) Structures of Trypanosome Vacuolar Soluble Pyrophosphatases: Antiparasitic Drug Targets (ACS Chemical Biology) Friday March 4th 2016
Yunyun Yang, Tzu-Ping Ko, Chun-Chi Chen, Guozhong Huang, Yingying Zheng, Weidong Liu, Iren Wang, Meng-Ru Ho, Shang-Te Danny Hsu, Bing O

164) Roles of Aag, Alkbh2, and Alkbh3 in the Repair of Carboxymethylated and Ethylated Thymidine Lesions (ACS Chemical Biology) Friday March 4th 2016
Changjun You, Pengcheng Wang, Stephanie L. Nay, Jianshuang Wang, Xiaoxia Dai, Timothy R. O

165) Structural Analysis of the Tobramycin and Gentamicin Clinical Resistome Reveals Limitations for Next-generation Aminoglycoside Design (ACS Chemical Biology) Friday March 4th 2016
Angelia V. Bassenden, Dmitry Rodionov, Kun Shi, Albert M. Berghuis

166) FRET Characterization of Complex Conformational Changes in a Large 16S Ribosomal RNA Fragment Site-Specifically Labeled Using Unnatural Base Pairs (ACS Chemical Biology) Friday March 4th 2016
Thomas Lavergne, Rajan Lamichhane, Denis A. Malyshev, Zhengtao Li, Lingjun Li, Edit Sperling, James R. Williamson, David P. Millar, Floyd E. Romesberg

167) Multidimensional Screening Platform for Simultaneously Targeting Oncogenic KRAS and Hypoxia-Inducible Factors Pathways in Colorectal Cancer (ACS Chemical Biology) Thursday March 3rd 2016
Michelle S. Bousquet, Jia Jia Ma, Ranjala Ratnayake, Pamela A. Havre, Jin Yao, Nam H. Dang, Valerie J. Paul, Thomas J. Carney, Long H. Dang, Hendrik Luesch

168) SIRT7 Is Activated by DNA and Deacetylates Histone H3 in the Chromatin Context (ACS Chemical Biology) Thursday March 3rd 2016
Zhen Tong, Yi Wang, Xiaoyu Zhang, David D. Kim, Sushabhan Sadhukhan, Quan Hao, Hening Lin

169) The Competitive Interplay between Allosteric HIV-1 Integrase Inhibitor BI/D and LEDGF/p75 during the Early Stage of HIV-1 Replication Adversely Affects Inhibitor Potency (ACS Chemical Biology) Wednesday March 2nd 2016
Lei Feng, Venkatasubramanian Dharmarajan, Erik Serrao, Ashley Hoyte, Ross C. Larue, Alison Slaughter, Amit Sharma, Matthew R. Plumb, Jacques J. Kessl, James R. Fuchs, Frederic D. Bushman, Alan N. Engelman, Patrick R. Griffin, Mamuka Kvaratskhelia

170) Characterization of Polyketide Synthase Machinery from the pks Island Facilitates Isolation of a Candidate Precolibactin (ACS Chemical Biology) Tuesday March 1st 2016
Li Zha, Matthew R. Wilson, Carolyn A. Brotherton, Emily P. Balskus

171) Five-Membered Ring Peroxide Selectively Initiates Ferroptosis in Cancer Cells (ACS Chemical Biology) Tuesday March 1st 2016
Rachel P. Abrams, William L. Carroll, K. A. Woerpel

172) Recent Advance in Tumor-associated Carbohydrate Antigens (TACAs)-based Antitumor Vaccines (ACS Chemical Biology) Tuesday March 1st 2016
Danyang Feng, Abdul Sami Shaikh, Fengshan Wang

173) Conformation-Selective Analogues of Dasatinib Reveal Insight into Kinase Inhibitor Binding and Selectivity (ACS Chemical Biology) Tuesday March 1st 2016
Frank E. Kwarcinski, Kristoffer R. Brandvold, Sameer Phadke, Omar M. Beleh, Taylor K. Johnson, Jennifer L. Meagher, Markus A. Seeliger, Jeanne A. Stuckey, Matthew B. Soellner

174) Application of Dual Inhibition Concept within Looped Autoregulatory Systems toward Antivirulence Agents against Pseudomonas aeruginosa Infections (ACS Chemical Biology) Tuesday March 1st 2016
Andreas Thomann, Antonio G. G. de Mello Martins, Christian Brengel, Martin Empting, Rolf W. Hartmann

175) Visible Light-Controlled Nitric Oxide Release from Hindered Nitrobenzene Derivatives for Specific Modulation of Mitochondrial Dynamics (ACS Chemical Biology) Monday February 29th 2016
Kai Kitamura, Mitsuyasu Kawaguchi, Naoya Ieda, Naoki Miyata, Hidehiko Nakagawa

176) Analysis of Iterative Screening with Stepwise Compound Selection Based on Novartis In-house HTS Data (ACS Chemical Biology) Friday February 26th 2016
Shardul Paricharak, Adriaan P. IJzerman, Andreas Bender, Florian Nigsch

177) Imaging Pseudomonas aeruginosa Biofilm Extracellular Polymer Scaffolds with Amphiphilic Carbon Dots (ACS Chemical Biology) Friday February 26th 2016
Margarita Ritenberg, Sukhendu Nandi, Sofiya Kolusheva, Rambabu Dandela, Michael M. Meijler, Raz Jelinek

178) Chemical Proteomics Reveals Ferrochelatase as a Common Off-target of Kinase Inhibitors (ACS Chemical Biology) Thursday February 25th 2016
Susan Klaeger, Bjoern Gohlke, Jessica Perrin, Vipul Gupta, Stephanie Heinzlmeir, Dominic Helm, Huichao Qiao, Giovanna Bergamini, Hiroshi Handa, Mikhail M Savitski, Marcus Bantscheff, Guillaume Me

179) The O-Carbamoyl-Transferase Alb15 Is Responsible for the Modification of Albicidin (ACS Chemical Biology) Tuesday February 23rd 2016
Daniel Petras, Dennis Kerwat, Alexander Pesic, Benjamin-F Hempel, Leonard von Eckardstein, Siamak Semsary, Julie Araste

180) Rapid Optimization of Mcl-1 Inhibitors using Stapled Peptide Libraries Including Non-Natural Side Chains (ACS Chemical Biology) Friday February 19th 2016
Raheleh Rezaei Araghi, Jeremy A. Ryan, Anthony Letai, Amy E. Keating

181) Hydroxyphenylation of Histone Lysines: Post-translational Modification by Quinone Imines (ACS Chemical Biology) Thursday February 18th 2016
Kodihalli C. Ravindra, Laura J. Trudel, John S. Wishnok, Gerald N. Wogan, Steven R. Tannenbaum, Paul L. Skipper

182) Leveraging Large-scale Behavioral Profiling in Zebrafish to Explore Neuroactive Polypharmacology (ACS Chemical Biology) Wednesday February 17th 2016
Matthew N. McCarroll, Leo Gendelev, Michael J. Keiser, David Kokel

183) Improving Polymerase Activity with Unnatural Substrates by Sampling Mutations in Homologous Protein Architectures (ACS Chemical Biology) Wednesday February 17th 2016
Matthew R. Dunn, Carine Otto, Kathryn E. Fenton, John C. Chaput

184) Proposed Mode of Binding and Action of Positive Allosteric Modulators at Opioid Receptors (ACS Chemical Biology) Wednesday February 17th 2016
Yi Shang, Holly R. Yeatman, Davide Provasi, Andrew Alt, Arthur Christopoulos, Meritxell Canals, Marta Filizola

185) Therapeutics Targeting Protein Acetylation Perturb Latency of Human Viruses (ACS Chemical Biology) Monday February 15th 2016
Ryan J. Conrad, Melanie Ott

186) A Strategy for Direct Chemical Activation of the Retinoblastoma Protein (ACS Chemical Biology) Thursday February 11th 2016
Cameron R. Pye, Walter M. Bray, Elise R. Brown, Jason R. Burke, R. Scott Lokey, Seth M. Rubin

187) Isoxazole Alters Metabolites and Gene Expression, Decreasing Proliferation and Promoting a Neuroendocrine Phenotype in (ACS Chemical Biology) Wednesday February 10th 2016
Michael A. Kalwat, Zhimin Huang, Chonlarat Wichaidit, Kathleen McGlynn, Svetlana Earnest, Claudia Savoia, Elhadji M. Dioum, Jay W. Schneider, Michele R. Hutchison, Melanie H. Cobb

188) Insights into Complex Oxidation during BE-7585A Biosynthesis: Structural Determination and Analysis of the Polyketide Monooxygenase BexE (ACS Chemical Biology) Wednesday February 10th 2016
David R. Jackson, Xia Yu, Guojung Wang, Avinash B. Patel, Jordi Calveras, Jesus F. Barajas, Eita Sasaki, Mikko Metsa

189) Profiling of Multiple Targets of Artemisinin Activated by Hemin in Cancer Cell Proteome (ACS Chemical Biology) Wednesday February 10th 2016
Yiqing Zhou, Weichao Li, Youli Xiao

190) Bioorthogonal Chemistry for the Isolation and Study of Newly Synthesized Histones and Their Modifications (ACS Chemical Biology) Wednesday February 10th 2016
Anna M. Arnaudo, A. James Link, Benjamin A. Garcia

191) Chemical Inhibition of Kynureninase Reduces Pseudomonas aeruginosa Quorum Sensing and Virulence Factor Expression (ACS Chemical Biology) Wednesday February 10th 2016
Stephen H. Kasper, Richard P. Bonocora, Joseph T. Wade, Rabi Ann Musah, Nathaniel C. Cady

192) Sequential Inactivation of Gliotoxin by the S-Methyltransferase TmtA (ACS Chemical Biology) Tuesday February 9th 2016
Elke R. Duell, Manuel Glaser, Camille Le Chapelain, Iris Antes, Michael Groll, Eva M. Huber

193) Naphthalimide Scaffold Provides Versatile Platform for Selective Thiol Sensing and Protein Labeling (ACS Chemical Biology) Tuesday February 9th 2016
Pengcheng Zhou, Juan Yao, Guodong Hu, Jianguo Fang

194) Chemical and Biophysical Modulation of Cas9 for Tunable Genome Engineering (ACS Chemical Biology) Tuesday February 9th 2016
James K. Nun

195) A Stable Pyrophosphoserine Analog for Incorporation into Peptides and Proteins (ACS Chemical Biology) Friday February 5th 2016
Lisa M. Yates, Dorothea Fiedler

196) Sirtuins 1 and 2 Are Universal Histone Deacetylases (ACS Chemical Biology) Friday February 5th 2016
Willie W. Hsu, Bo Wu, Wenshe R. Liu

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